
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 993 prodotti di "recettore 5-HT"
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Risperidone Mesylate
CAS:Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formula:C24H31FN4O5SPurezza:98%Colore e forma:SolidPeso molecolare:506.59N-Methyl amisulpride
CAS:N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formula:C18H29N3O4SColore e forma:SolidPeso molecolare:383.51Escitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formula:C20H21FN2OPurezza:99.82%Colore e forma:White Or White Crystalline PowderPeso molecolare:324.39Brexpiprazole-d8
CAS:<p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>Formula:C25H27N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:441.62Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purezza:98%Colore e forma:SolidPeso molecolare:268.37Amitriptyline-d6 Hydrochloride
CAS:<p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>Formula:C20H18D6ClNColore e forma:SolidPeso molecolare:319.90Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Formula:C18H29NO2H2O4SPurezza:98.55%Colore e forma:SolidPeso molecolare:340.47Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.27SB 271046 hydrochloride
CAS:<p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.</p>Formula:C20H22ClN3O3S2·HClPurezza:99.77%Colore e forma:SolidPeso molecolare:488.455-Methyltryptamine hydrochloride
CAS:<p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>Formula:C11H15ClN2Purezza:99.45%Colore e forma:SolidPeso molecolare:210.7037-Desmethyl-3-hydroxyagomelatine
CAS:<p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>Formula:C14H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:245.27Ketanserinol
CAS:<p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>Formula:C22H24FN3O3Colore e forma:SolidPeso molecolare:397.44Hydroxy ziprasidone
CAS:<p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>Formula:C21H21ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:428.94Diclofensine
CAS:<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Formula:C17H17Cl2NOPurezza:97.01% - 98.13%Colore e forma:SolidPeso molecolare:322.23LY 344864
CAS:LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formula:C21H22FN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.42Paroxetine hydrochloride hemihydrate
CAS:<p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>Formula:C38H44Cl2F2N2O7Purezza:99.949%Colore e forma:SolidPeso molecolare:749.67Dolasetron Mesylate
CAS:<p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>Formula:C20H24N2O6SPurezza:99.05%Colore e forma:White PowderPeso molecolare:420.48TC-2153
CAS:TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.Formula:C7H5ClF3NS5Colore e forma:SolidPeso molecolare:355.89Lofepramine hydrochloride
CAS:Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.Formula:C26H28Cl2N2OPurezza:98%Colore e forma:Off-White SolidPeso molecolare:455.42Ifoxetine sulfate
CAS:Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.Formula:C13H19NO2H2O4SPurezza:98%Colore e forma:SolidPeso molecolare:270.34
