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recettore 5-HT

recettore 5-HT

I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.

Trovati 993 prodotti di "recettore 5-HT"

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  • Risperidone Mesylate

    CAS:
    Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.
    Formula:C24H31FN4O5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:506.59
  • N-Methyl amisulpride

    CAS:
    N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.
    Formula:C18H29N3O4S
    Colore e forma:Solid
    Peso molecolare:383.51
  • Escitalopram

    CAS:
    Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.
    Formula:C20H21FN2O
    Purezza:99.82%
    Colore e forma:White Or White Crystalline Powder
    Peso molecolare:324.39
  • Brexpiprazole-d8

    CAS:
    <p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>
    Formula:C25H27N3O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:441.62
  • Mirtazapine D3

    CAS:
    Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .
    Formula:C17H19N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:268.37
  • Amitriptyline-d6 Hydrochloride

    CAS:
    <p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>
    Formula:C20H18D6ClN
    Colore e forma:Solid
    Peso molecolare:319.90
  • Penbutolol sulfate

    CAS:
    <p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>
    Formula:C18H29NO2H2O4S
    Purezza:98.55%
    Colore e forma:Solid
    Peso molecolare:340.47
  • Pardoprunox

    CAS:
    Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.
    Formula:C12H15N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:233.27
  • SB 271046 hydrochloride

    CAS:
    <p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is &gt; 200-fold selective over 55 other receptors, enzymes and ion channels.</p>
    Formula:C20H22ClN3O3S2·HCl
    Purezza:99.77%
    Colore e forma:Solid
    Peso molecolare:488.45
  • 5-Methyltryptamine hydrochloride

    CAS:
    <p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>
    Formula:C11H15ClN2
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:210.703
  • 7-Desmethyl-3-hydroxyagomelatine

    CAS:
    <p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>
    Formula:C14H15NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:245.27
  • Ketanserinol

    CAS:
    <p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>
    Formula:C22H24FN3O3
    Colore e forma:Solid
    Peso molecolare:397.44
  • Hydroxy ziprasidone

    CAS:
    <p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>
    Formula:C21H21ClN4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:428.94
  • Diclofensine

    CAS:
    <p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>
    Formula:C17H17Cl2NO
    Purezza:97.01% - 98.13%
    Colore e forma:Solid
    Peso molecolare:322.23
  • LY 344864

    CAS:
    LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.
    Formula:C21H22FN3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:351.42
  • Paroxetine hydrochloride hemihydrate

    CAS:
    <p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>
    Formula:C38H44Cl2F2N2O7
    Purezza:99.949%
    Colore e forma:Solid
    Peso molecolare:749.67
  • Dolasetron Mesylate

    CAS:
    <p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>
    Formula:C20H24N2O6S
    Purezza:99.05%
    Colore e forma:White Powder
    Peso molecolare:420.48
  • TC-2153

    CAS:
    TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.
    Formula:C7H5ClF3NS5
    Colore e forma:Solid
    Peso molecolare:355.89
  • Lofepramine hydrochloride

    CAS:
    Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.
    Formula:C26H28Cl2N2O
    Purezza:98%
    Colore e forma:Off-White Solid
    Peso molecolare:455.42
  • Ifoxetine sulfate

    CAS:
    Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.
    Formula:C13H19NO2H2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:270.34