
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Formula:C28H30N2O8Purezza:99.7% - >99.99%Colore e forma:PowderPeso molecolare:522.55Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Formula:C19H20N2C10H8O6S2Purezza:99.35% - 99.96%Colore e forma:White Or Almost White CrystallinePeso molecolare:420.52Aripiprazole
CAS:<p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>Formula:C23H27Cl2N3O2Purezza:99.43% - 99.62%Colore e forma:Colourless Flake Crystalline SolidPeso molecolare:448.39CP-809101 hydrochloride
CAS:<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Formula:C15H18Cl2N4OPurezza:99.5%Colore e forma:SolidPeso molecolare:341.24Cisapride
CAS:<p>Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.</p>Formula:C23H29ClFN3O4Purezza:99.77%Colore e forma:White To Slightly Biege Powder SolidPeso molecolare:465.95Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Formula:C19H23Cl2N5OPurezza:99.5% - 99.52%Colore e forma:SolidPeso molecolare:408.33Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Formula:C19H21N·HClPurezza:98.54% - 99.98%Colore e forma:SolidPeso molecolare:299.84Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Formula:C17H19ClN4OPurezza:99.90%Colore e forma:Off-White PowderPeso molecolare:330.81Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formula:C21H21ClN4OSPurezza:99.55%Colore e forma:Tan SolidPeso molecolare:412.94Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurezza:99.84% - 99.92%Colore e forma:White SolidPeso molecolare:332.87Ondansetron hydrochloride dihydrate
CAS:<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Formula:C18H19N3O·HCl·2H2OPurezza:99.92%Colore e forma:White Crystal PowderPeso molecolare:365.862-Bromo-6-methoxynaphthalene
CAS:<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Formula:C11H9BrOPurezza:98.51%Colore e forma:White To Off-White PowderPeso molecolare:237.09Vilazodone
CAS:<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Formula:C26H27N5O2Purezza:99.61%Colore e forma:Light Yellow SolidPeso molecolare:441.52Asenapine Maleate
CAS:Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Formula:C21H20ClNO5Purezza:99.28%Colore e forma:SolidPeso molecolare:401.84Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Formula:C15H17NO2Purezza:99.92%Colore e forma:White SolidPeso molecolare:243.3Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formula:C21H26ClN3OSPurezza:99.3% - 99.99%Colore e forma:SolidPeso molecolare:403.97Naftidrofuryl oxalate
CAS:<p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>Formula:C26H35NO7Purezza:97.12% - 98.38%Colore e forma:SolidPeso molecolare:473.56Ziprasidone hydrochloride
CAS:<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Formula:C21H22CL2N4OSPurezza:97.97% - 99.82%Colore e forma:SolidPeso molecolare:449.4Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purezza:98.76% - 99.75%Colore e forma:SolidPeso molecolare:471.67Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formula:C16H24N2O2·HClPurezza:99% - 99.99%Colore e forma:SolidPeso molecolare:312.84
