
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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Repinotan HCl
CAS:<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Formula:C21H25ClN2O4SPurezza:99.57%Colore e forma:SolidPeso molecolare:436.95CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Formula:C19H28ClN5OPurezza:99.72%Colore e forma:SolidPeso molecolare:377.91Isamoltane hemifumarate
CAS:<p>5-HT1B antagonist</p>Formula:C16H22N202C4H404Purezza:98%Colore e forma:SolidPeso molecolare:332.4WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Formula:C14H18N2Purezza:98%Colore e forma:SolidPeso molecolare:214.31UCSF648
CAS:<p>UCSF648 (Compound 5A6-48) weakly activates MTNR1A and ADRA2A. UCSF648 is a chemical probe for the serotonin receptor 5-HT 5A [1].</p>Formula:C15H19ClN2O2SColore e forma:SolidPeso molecolare:326.84SB 258719 hydrochloride
CAS:<p>Selective 5-HT7 receptor antagonist</p>Formula:C18H31ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:374.97NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Formula:C25H27Cl2N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:504.47Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purezza:98%Colore e forma:SolidPeso molecolare:310.78(R)-DOI hydrochloride
CAS:<p>(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.</p>Formula:C11H17ClINO2Purezza:99.88% - >99.99%Colore e forma:SolidPeso molecolare:357.62OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Formula:C23H28ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:413.94S 14506 hydrochloride
CAS:<p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>Formula:C24H27ClFN3O2Purezza:99.92%Colore e forma:SolidPeso molecolare:443.94PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Formula:C15H20Cl2N2OPurezza:98.67%Colore e forma:SolidPeso molecolare:315.24PNU-96391
CAS:<p>PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.</p>Formula:C15H23NO2SPurezza:99.53%Colore e forma:SolidPeso molecolare:281.41S 32212 hydrochloride
CAS:<p>S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .</p>Formula:C25H29ClN4O2Purezza:97.11% - 99.57%Colore e forma:SolidPeso molecolare:452.98Org-12962 hydrochloride
CAS:<p>Org-12962 hydrochloride is a 5-HT2C receptor agonist.</p>Formula:C10H12Cl2F3N3Purezza:98%Colore e forma:SolidPeso molecolare:302.12Org-12962
CAS:<p>Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).</p>Formula:C10H11ClF3N3Purezza:98.34%Colore e forma:SolidPeso molecolare:265.66Zatosetron maleate
CAS:<p>Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.</p>Formula:C23H29ClN2O6Purezza:98.07%Colore e forma:SolidPeso molecolare:464.94LY 344864 S-enantiomer
CAS:<p>LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.</p>Formula:C21H22FN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.42PRX-08066 Maleic acid
CAS:<p>PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.</p>Formula:C23H21ClFN5O4SPurezza:97.59%Colore e forma:SolidPeso molecolare:517.96Bopindolol fumarate
CAS:<p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>Formula:C27H32N2O7Colore e forma:SolidPeso molecolare:496.56DR4485 hydrochloride
CAS:<p>5-HT7 antagonist</p>Formula:C26H29Cl3N2OPurezza:98%Colore e forma:SolidPeso molecolare:491.88SLV-310
CAS:<p>SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.</p>Formula:C25H24FN3O2Purezza:99.39%Colore e forma:SolidPeso molecolare:417.48Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purezza:98%Colore e forma:SolidPeso molecolare:393.74(R)-Viloxazine Hydrochloride
CAS:<p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>Formula:C13H20ClNO3Purezza:99.88% - 99.94%Colore e forma:SolidPeso molecolare:273.76Trimipramine
CAS:<p>Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.</p>Formula:C20H26N2Purezza:98%Colore e forma:SolidPeso molecolare:294.43OPC-14523 hydrochloride
CAS:<p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>Formula:C23H29Cl2N3O2Purezza:99.60%Colore e forma:SolidPeso molecolare:450.4CGS-12066 maleate salt
CAS:<p>CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.</p>Formula:C21H21F3N4O4Colore e forma:SolidPeso molecolare:450.41GTS-21
CAS:<p>GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.</p>Formula:C19H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:308.37LY320135
CAS:CB1 receptor antagonist/inverse agonistFormula:C24H17NO4Purezza:98%Colore e forma:SolidPeso molecolare:383.4Nexopamil racemate
CAS:<p>Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.</p>Formula:C24H40N2O3Purezza:98.61%Colore e forma:SolidPeso molecolare:404.59Oxetorone fumarate
CAS:<p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>Formula:C25H25NO6Purezza:99.809%Colore e forma:SolidPeso molecolare:435.48Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Formula:C25H27N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:481.56SDZ 21009
CAS:<p>β-adrenoceptor and 5-HT1A/1B receptor antagonist</p>Formula:C19H28N2O4Purezza:98%Colore e forma:SolidPeso molecolare:348.44SEP-363856
CAS:<p>SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.</p>Formula:C9H13NOSPurezza:98%Colore e forma:SolidPeso molecolare:183.27Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formula:C18H22BrNSPurezza:99.65%Colore e forma:SolidPeso molecolare:364.34LY 393558
CAS:<p>Dual 5-HT1B/1D receptor antagonist</p>Formula:C26H31FN4O4S2Purezza:98%Colore e forma:SolidPeso molecolare:546.68Amitifadine hydrochloride
CAS:<p>Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).</p>Formula:C11H12Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:264.58Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Formula:C18H29NO2Purezza:98%Colore e forma:SolidPeso molecolare:291.43Bemesetron
CAS:<p>Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.</p>Formula:C15H17Cl2NO2Purezza:99.77%Colore e forma:SolidPeso molecolare:314.21SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Formula:C21H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:403.86Opiranserin
CAS:<p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>Formula:C21H34N2O5Purezza:98%Colore e forma:SolidPeso molecolare:394.51Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Formula:C19H24N2OPurezza:98%Colore e forma:SolidPeso molecolare:296.41Pancopride
CAS:<p>Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced</p>Formula:C18H24ClN3O2Purezza:93.64%Colore e forma:SolidPeso molecolare:349.86Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Formula:C18H20ClNPurezza:98%Colore e forma:SolidPeso molecolare:285.81PF-4479745
CAS:<p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>Formula:C17H22N4Purezza:98%Colore e forma:SolidPeso molecolare:282.38Masupirdine mesylate
CAS:<p>Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's disease</p>Formula:C23H32BrN3O9S3Purezza:99.57%Colore e forma:SolidPeso molecolare:670.61Ipsapirone
CAS:<p>Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.</p>Formula:C19H23N5O3SPurezza:99.51%Colore e forma:SolidPeso molecolare:401.48SB357134
CAS:<p>SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.</p>Formula:C17H18Br2FN3O3SPurezza:98%Colore e forma:SolidPeso molecolare:523.21Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Formula:C23H31ClN2Purezza:98%Colore e forma:SolidPeso molecolare:370.96SB 206553 hydrochloride
CAS:<p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>Formula:C17H17ClN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:328.8UCSF678
CAS:<p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>Formula:C15H18N2O2SColore e forma:SolidPeso molecolare:290.385-HT4 antagonist 1
CAS:<p>5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).</p>Formula:C23H36N4O5SPurezza:99.75%Colore e forma:SolidPeso molecolare:480.62Pridefine
CAS:<p>Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.</p>Formula:C19H21NPurezza:99.15% - 99.66%Colore e forma:SolidPeso molecolare:263.38E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formula:C20H27Cl2N3O2Purezza:98.88% - 98.88%Colore e forma:SolidPeso molecolare:412.35T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Formula:C56H62N6O8Purezza:98%Colore e forma:SolidPeso molecolare:947.146SKF-83566 hydrobromide
CAS:<p>D1-like dopamine receptor antagonist</p>Formula:C17H19BrClNOPurezza:98%Colore e forma:SolidPeso molecolare:368.7GR 55562 dihydrochloride
CAS:<p>5-HT1B (5-HT1Dβ) silent antagonist</p>Formula:C23H27Cl2N3O2Purezza:99.45%Colore e forma:SolidPeso molecolare:448.39MS 245 oxalate
CAS:MS 245 oxalate is a 5-HT6 antagonist.Formula:C21H24N2O7SPurezza:98%Colore e forma:SolidPeso molecolare:448.49EGIS-7625
CAS:<p>EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.</p>Formula:C18H24Cl2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:399.32Glemanserin
CAS:<p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>Formula:C20H25NOPurezza:99.93%Colore e forma:SolidPeso molecolare:295.42DV 7028 hydrochloride
CAS:<p>DV 7028 hydrochloride is a 5-HT2A receptor antagonist.</p>Formula:C21H26ClFN4O3Purezza:98%Colore e forma:SolidPeso molecolare:436.91L-775,606
CAS:<p>L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.</p>Formula:C25H29FN6Purezza:98%Colore e forma:SolidPeso molecolare:432.54Ro 60-0175 fumarate
CAS:<p>5-HT2 receptor agonist</p>Formula:C15H16ClFN2O4Purezza:98%Colore e forma:SolidPeso molecolare:342.75PNU-96415E
CAS:dopamine D4 and serotonergic 5-HT2A receptor antagonistFormula:C21H27Cl2FN2OPurezza:98%Colore e forma:SolidPeso molecolare:413.36Alaproclate (hydrochloride)
CAS:<p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>Formula:C13H19Cl2NO2Colore e forma:SolidPeso molecolare:292.2(R)-Praziquantel
CAS:(R)-Praziquantel is an active enantiomer of praziquantel.Formula:C19H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:312.41F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Formula:C25H29ClF2N4O5Purezza:98.86%Colore e forma:SolidPeso molecolare:538.975-HT3 antagonist 2
CAS:<p>5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.</p>Formula:C18H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.38Donitriptan
CAS:<p>Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>Formula:C23H25N5O2Purezza:98.76%Colore e forma:SolidPeso molecolare:403.48AR-A 2
CAS:<p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>Formula:C27H36N4O2Purezza:98%Colore e forma:SolidPeso molecolare:448.6Org37684
CAS:<p>5-HT2 receptors agonist</p>Formula:C14H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:269.77Methiothepin maleate
CAS:<p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>Formula:C24H28N2O4S2Purezza:98%Colore e forma:SolidPeso molecolare:472.62AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Formula:C17H20ClN5O2SPurezza:>99.99%Colore e forma:SolidPeso molecolare:393.89Ro 04-6790
CAS:<p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>Formula:C12H16N6O2SPurezza:98%Colore e forma:SolidPeso molecolare:308.36ST1936
CAS:<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Formula:C13H17ClN2Purezza:98%Colore e forma:SolidPeso molecolare:236.742-Methyl-5-HT maleate
CAS:<p>2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.</p>Formula:C15H18N2O5Purezza:98%Colore e forma:SolidPeso molecolare:306.31Ampreloxetine
CAS:<p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>Formula:C18H18F3NOPurezza:98%Colore e forma:SolidPeso molecolare:321.34RG-12915
CAS:<p>RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).</p>Formula:C20H25ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:360.88Org-13011 fumarate
CAS:<p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>Formula:C22H29F3N4O5Purezza:98.92%Colore e forma:SolidPeso molecolare:486.48Enciprazine
CAS:<p>Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.</p>Formula:C23H32N2O6Purezza:98.63%Colore e forma:SolidPeso molecolare:432.51Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Formula:C23H31N5O6Colore e forma:SolidPeso molecolare:473.53Deramciclane fumarate
CAS:<p>Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.</p>Formula:C24H35NO5Colore e forma:SolidPeso molecolare:417.54Bopindolol
CAS:<p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>Formula:C23H28N2O3Colore e forma:SolidPeso molecolare:380.485-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Formula:C21H23N7Colore e forma:SolidPeso molecolare:373.45MK-212
CAS:<p>MK-212 is a 5HT2C agonist; boosts corticosterone and lowers activity at 0.5-1mg/kg; reduces anxiety without affecting movement at 0.1-0.2mg/kg in mice.</p>Formula:C8H11ClN4Colore e forma:SolidPeso molecolare:198.65RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Formula:C16H24Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:363.28Eplivanserin hemifumarate
CAS:<p>Eplivanserin is an inverse agonist of 5-HT2A.</p>Formula:C23H25FN2O6Colore e forma:SolidPeso molecolare:444.45OSU 6162 hydrochloride
CAS:Dopamine stabilizerFormula:C15H24ClNO2SPurezza:98%Colore e forma:SolidPeso molecolare:317.88S-15535
CAS:<p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>Formula:C21H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:336.43Fonazine
CAS:<p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>Formula:C19H25N3O2S2Colore e forma:SolidPeso molecolare:391.55Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Formula:C26H31FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:454.53GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Formula:C23H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:411.93ATC0065 HCl
CAS:<p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>Formula:C25H31BrCl2F3N5OColore e forma:SolidPeso molecolare:625.35LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Formula:C20H24N4O3Colore e forma:SolidPeso molecolare:368.43SGS518 oxalate
CAS:<p>SGS518 oxalate is a 5-HT6 antagonist.</p>Formula:C23H24F2N2O7SPurezza:98%Colore e forma:SolidPeso molecolare:510.51(Rac)-SEP-363856
CAS:<p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>Formula:C9H13NOSPurezza:98%Colore e forma:SolidPeso molecolare:183.27AP521
CAS:<p>AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).</p>Formula:C20H19ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:402.89SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Colore e forma:SolidPeso molecolare:474.33WAY 161503 hydrochloride
CAS:<p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>Formula:C11H12Cl3N3OPurezza:98%Colore e forma:SolidPeso molecolare:308.59SUN-C5174
CAS:<p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>Formula:C22H29FN4O2Purezza:98%Colore e forma:SolidPeso molecolare:400.49Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Formula:C22H27ClN2Colore e forma:SolidPeso molecolare:354.92EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Formula:C24H31N3O2Purezza:95.64% - 99.39%Colore e forma:SolidPeso molecolare:393.522PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purezza:98%Colore e forma:SolidPeso molecolare:267.37FR260010
CAS:<p>FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.</p>Formula:C22H19N5Colore e forma:SolidPeso molecolare:353.42TC-2153
CAS:<p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>Formula:C7H5ClF3NS5Colore e forma:SolidPeso molecolare:355.89Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Formula:C13H18ClNO2Purezza:98.29% - 98.64%Colore e forma:SolidPeso molecolare:255.74LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Formula:C27H38ClN3OSPurezza:98.06%Colore e forma:SolidPeso molecolare:488.13Belaperidone
CAS:<p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>Formula:C22H22FN3O2Colore e forma:SolidPeso molecolare:379.43CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Formula:C12H14ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:251.71CGS 12066B dimaleate
CAS:<p>5-HT1B full agonist</p>Formula:C25H25F3N4O8Purezza:98%Colore e forma:SolidPeso molecolare:566.485-HT6/5-HT2A receptor ligand-2
CAS:<p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>Formula:C20H18FN3O2Colore e forma:SolidPeso molecolare:351.37CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Formula:C19H21N5O2Purezza:98%Colore e forma:SolidPeso molecolare:351.45-HT7 agonist 2
CAS:<p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>Formula:C23H29N3OColore e forma:SolidPeso molecolare:363.5Prucalopride hydrochloride
CAS:<p>Prucalopride hydrochloride is a selective agonist of the 5-HT4.</p>Formula:C18H27Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:404.33WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Formula:C17H20Cl2FN3O2SPurezza:98.43%Colore e forma:SolidPeso molecolare:420.33LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Formula:C19H23FN4Purezza:98%Colore e forma:SolidPeso molecolare:326.41UCSF686
CAS:<p>UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.</p>Formula:C14H19N3O2SColore e forma:SolidPeso molecolare:293.38ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Formula:C25H29BrF3N5OColore e forma:SolidPeso molecolare:552.43ZM 169369
CAS:<p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>Formula:C19H20N2SColore e forma:SolidPeso molecolare:308.44(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Formula:C16H26BrNOPurezza:98%Colore e forma:SolidPeso molecolare:328.29FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Formula:C27H29F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:465.53S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Formula:C22H29Cl2N3O2SColore e forma:SolidPeso molecolare:470.45Tertatolol
CAS:<p>Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.</p>Formula:C16H25NO2SPurezza:98%Colore e forma:SolidPeso molecolare:295.44Piclozotan
CAS:<p>Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)</p>Formula:C23H24ClN3O2Purezza:98.59%Colore e forma:SolidPeso molecolare:409.91Alniditan
CAS:<p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>Formula:C17H26N4OPurezza:98%Colore e forma:SolidPeso molecolare:302.415-HT2A receptor agonist-2
CAS:<p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>Formula:C20H21ClN2O3Colore e forma:SolidPeso molecolare:372.85AP-521 (Free base)
CAS:<p>AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.</p>Formula:C20H18N2O3SColore e forma:SolidPeso molecolare:366.43Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Formula:C26H32N2O7Colore e forma:SolidPeso molecolare:484.549RS 39604
CAS:<p>potent and selective 5-HT4 antagonist</p>Formula:C26H37Cl2N3O6SPurezza:98%Colore e forma:SolidPeso molecolare:590.56Naronapride
CAS:<p>Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.</p>Formula:C27H41ClN4O5Colore e forma:SolidPeso molecolare:537.09Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Formula:C24H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:385.46TMPPAA
CAS:<p>TMPPAA is an allosteric agonist of 5-HT3 receptor.</p>Formula:C15H21NO2Purezza:98%Colore e forma:SolidPeso molecolare:247.33Ziprasidone mesylate trihydrate
CAS:<p>Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.</p>Formula:C22H31ClN4O7S2Colore e forma:SolidPeso molecolare:563.085-HT7 agonist 1
CAS:<p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>Formula:C19H20ClN3Purezza:98.61%Colore e forma:SolidPeso molecolare:325.84Pruvanserin hydrochloride
CAS:<p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>Formula:C22H22ClFN4OPurezza:99.6%Colore e forma:SolidPeso molecolare:412.89Eplivanserin
CAS:<p>Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.</p>Formula:C19H21FN2O2Purezza:97.04%Colore e forma:SolidPeso molecolare:328.38SB-737050A
CAS:<p>SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.</p>Formula:C22H23ClN2O3S2Colore e forma:SolidPeso molecolare:463.01EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Formula:C15H22N2OPurezza:97.66% - 99.78%Colore e forma:SolidPeso molecolare:246.35GR 113808
CAS:<p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>Formula:C19H27N3O4SPurezza:98.16%Colore e forma:SolidPeso molecolare:393.5PNU-142633
CAS:<p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.</p>Formula:C24H30N4O3Purezza:98%Colore e forma:SolidPeso molecolare:422.52SB-221284
CAS:5-HT2C/2B receptor antagonistFormula:C16H14F3N3OSPurezza:98%Colore e forma:SolidPeso molecolare:353.36Adatanserin
CAS:<p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>Formula:C21H31N5OPurezza:99.33%Colore e forma:SolidPeso molecolare:369.5Alniditan dihydrochloride
CAS:<p>Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.</p>Formula:C17H28Cl2N4OColore e forma:SolidPeso molecolare:375.34TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Formula:C14H17ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:280.75LY 125180
CAS:LY 125180 is a serotonin antagonist.Formula:C18H24ClNOPurezza:98%Colore e forma:SolidPeso molecolare:305.84RS 56812 hydrochloride
CAS:<p>5-HT3 partial agonist</p>Formula:C18H22ClN3O2Purezza:98.62%Colore e forma:SolidPeso molecolare:347.84Iprindole
CAS:<p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>Formula:C19H28N2Purezza:99.54%Colore e forma:SolidPeso molecolare:284.44LY 334370 hydrochloride
CAS:5-HT1F receptor agonistFormula:C21H23ClFN3OPurezza:98%Colore e forma:SolidPeso molecolare:387.88Irindalone
CAS:<p>IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.</p>Formula:C24H29FN4OPurezza:98%Colore e forma:SolidPeso molecolare:408.51PNU-282987 S enantiomer hydrochloride
CAS:<p>(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.</p>Formula:C14H18Cl2N2OPurezza:98%Colore e forma:SolidPeso molecolare:301.21Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Formula:C24H27FN4O2Purezza:98.04%Colore e forma:SolidPeso molecolare:422.5Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Formula:C26H32N2O5Purezza:99.17% - 99.67%Colore e forma:SolidPeso molecolare:452.54LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:372.89Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purezza:99.77%Colore e forma:SolidPeso molecolare:304.43Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Formula:C28H30ClN5O3Purezza:99.04%Colore e forma:SolidPeso molecolare:520.02ML 10302 hydrochloride
CAS:<p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>Formula:C15H22Cl2N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:349.25LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purezza:98.58%Colore e forma:SolidPeso molecolare:407.33GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formula:C23H27N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:377.48Itasetron
CAS:<p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>Formula:C16H20N4O2Purezza:98.58% - 99.33%Colore e forma:SolidPeso molecolare:300.36ADR-851 free base
CAS:ADR-851 free base is an antagonist of the HT3 receptor.Formula:C14H18ClN3O2Purezza:97.88% - 98.39%Colore e forma:SolidPeso molecolare:295.77Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59Cianopramine
CAS:<p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>Formula:C20H23N3Purezza:99.92% - 99.92%Colore e forma:SolidPeso molecolare:305.42Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Formula:C15H23NOPurezza:98.09% - 98.77%Colore e forma:SolidPeso molecolare:233.35BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Formula:C28H45ClN4O11S4Purezza:>99.99%Colore e forma:SolidPeso molecolare:777.39Tedatioxetine
CAS:<p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>Formula:C18H21NSPurezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:283.438-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Formula:C16H25NOPurezza:98%Colore e forma:SolidPeso molecolare:247.38SB 699551 dihydrochloride
CAS:<p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>Formula:C34H47Cl2N3OPurezza:99.83%Colore e forma:SolidPeso molecolare:584.66Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Formula:C13H19NO3Purezza:99.67%Colore e forma:SolidPeso molecolare:237.29RS 67333 hydrochloride
CAS:<p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>Formula:C19H30Cl2N2O2Purezza:98.78%Colore e forma:SolidPeso molecolare:389.36CP 96021
CAS:<p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>Formula:C29H21FN4OSPurezza:97.81% - 99.62%Colore e forma:SoildPeso molecolare:492.57Landipirdine
CAS:<p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>Formula:C18H19FN2O3SPurezza:97.61% - 99.37%Colore e forma:SolidPeso molecolare:362.42Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Formula:C20H21N3OPurezza:99.82% - 99.98%Colore e forma:SolidPeso molecolare:319.4RS 42358-197
CAS:<p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>Formula:C19H23ClN2OPurezza:99.70%Colore e forma:SolidPeso molecolare:330.85E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Formula:C17H18ClN5O2S2Purezza:96.32% - 99.53%Colore e forma:SolidPeso molecolare:423.94Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurezza:97.01%Colore e forma:SolidPeso molecolare:323.46MM 77 dihydrochloride
CAS:<p>MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.</p>Formula:C19H29Cl2N3O3Purezza:99.91%Colore e forma:SolidPeso molecolare:418.36(Z)-Thiothixene
CAS:<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Formula:C23H29N3O2S2Purezza:99.21%Colore e forma:Yellow To Yellow With A Tan Cast PowderPeso molecolare:443.63Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Formula:C20H26ClNO2Purezza:99.63%Colore e forma:SolidPeso molecolare:347.88SB-215505
CAS:<p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>Formula:C19H16ClN3OPurezza:98.33%Colore e forma:SolidPeso molecolare:337.85-HT2 antagonist 1
CAS:<p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>Formula:C22H29FN4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:400.49SB228357
CAS:<p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>Formula:C22H17F4N3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:431.38Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Formula:C14H20ClN3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:313.785HT6-ligand-1
CAS:<p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>Formula:C20H22BrN3O2SPurezza:99.24% - 99.93%Colore e forma:SolidPeso molecolare:448.38SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Formula:C23H31Cl2NO8SPurezza:99.37%Colore e forma:SolidPeso molecolare:552.47LY-2624803
CAS:<p>LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.</p>Formula:C22H25N3O3Purezza:99.78% - 99.97%Colore e forma:SolidPeso molecolare:379.45Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:346.47Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formula:C22H22N2O7Purezza:99.66%Colore e forma:SolidPeso molecolare:426.42Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Formula:C24H40N2O3Purezza:97.87% - >99.99%Colore e forma:SolidPeso molecolare:404.59ATC 0175 hydrochloride
CAS:<p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>Formula:C23H26ClF2N5OPurezza:99.98%Colore e forma:SolidPeso molecolare:461.93Perphenazine dihydrochloride
CAS:Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formula:C21H28Cl3N3OSPurezza:99.67%Colore e forma:SolidPeso molecolare:476.89Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Formula:C24H22N4Purezza:99.91%Colore e forma:SolidPeso molecolare:366.46Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Formula:C21H24BrN3O3SPurezza:98.36% - 99.65%Colore e forma:SolidPeso molecolare:478.4Teniloxazine
CAS:<p>Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.</p>Formula:C16H19NO2SPurezza:99.23%Colore e forma:SolidPeso molecolare:289.39Piromelatine
CAS:<p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>Formula:C17H16N2O4Purezza:99.89%Colore e forma:SolidPeso molecolare:312.32H-9 dihydrochloride
CAS:<p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>Formula:C11H15Cl2N3O2SPurezza:97.3%Colore e forma:SolidPeso molecolare:324.235-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Formula:C22H20FN3O3Purezza:98.78% - 99.26%Colore e forma:SolidPeso molecolare:393.41Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Formula:C16H19NOPurezza:99.47%Colore e forma:SolidPeso molecolare:241.33BMY-14802 hydrochloride
CAS:<p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>Formula:C18H23ClF2N4OPurezza:99.97%Colore e forma:SolidPeso molecolare:384.85Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Formula:C24H32N4O2SPurezza:99.74%Colore e forma:SolidPeso molecolare:440.65-HT1A modulator 1
CAS:<p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>Formula:C21H25N3O2SPurezza:99.68%Colore e forma:SolidPeso molecolare:383.51
