recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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Repinotan HCl
CAS:<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Formula:C21H25ClN2O4SPurezza:99.57%Colore e forma:SolidPeso molecolare:436.95CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Formula:C19H28ClN5OPurezza:99.72%Colore e forma:SolidPeso molecolare:377.91Isamoltane hemifumarate
CAS:<p>5-HT1B antagonist</p>Formula:C16H22N202C4H404Purezza:98%Colore e forma:SolidPeso molecolare:332.4WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Formula:C14H18N2Purezza:98%Colore e forma:SolidPeso molecolare:214.31UCSF648
CAS:<p>UCSF648 (Compound 5A6-48) weakly activates MTNR1A and ADRA2A. UCSF648 is a chemical probe for the serotonin receptor 5-HT 5A [1].</p>Formula:C15H19ClN2O2SColore e forma:SolidPeso molecolare:326.84SB 258719 hydrochloride
CAS:<p>Selective 5-HT7 receptor antagonist</p>Formula:C18H31ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:374.97NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Formula:C25H27Cl2N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:504.47Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purezza:98%Colore e forma:SolidPeso molecolare:310.78(R)-DOI hydrochloride
CAS:<p>(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.</p>Formula:C11H17ClINO2Purezza:99.88% - >99.99%Colore e forma:SolidPeso molecolare:357.62OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Formula:C23H28ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:413.94S 14506 hydrochloride
CAS:<p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>Formula:C24H27ClFN3O2Purezza:99.92%Colore e forma:SolidPeso molecolare:443.94PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Formula:C15H20Cl2N2OPurezza:98.67%Colore e forma:SolidPeso molecolare:315.24PNU-96391
CAS:<p>PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.</p>Formula:C15H23NO2SPurezza:99.53%Colore e forma:SolidPeso molecolare:281.41S 32212 hydrochloride
CAS:<p>S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .</p>Formula:C25H29ClN4O2Purezza:97.11% - 99.57%Colore e forma:SolidPeso molecolare:452.98Org-12962 hydrochloride
CAS:<p>Org-12962 hydrochloride is a 5-HT2C receptor agonist.</p>Formula:C10H12Cl2F3N3Purezza:98%Colore e forma:SolidPeso molecolare:302.12Org-12962
CAS:<p>Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).</p>Formula:C10H11ClF3N3Purezza:98.34%Colore e forma:SolidPeso molecolare:265.66Zatosetron maleate
CAS:<p>Zatosetron maleate（LY 277359 maleate） is a potent and selective serotonin 5HT3 receptor antagonist for the study of acute migraine.</p>Formula:C23H29ClN2O6Purezza:98.07%Colore e forma:SolidPeso molecolare:464.94LY 344864 S-enantiomer
CAS:<p>LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.</p>Formula:C21H22FN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.42PRX-08066 Maleic acid
CAS:<p>PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.</p>Formula:C23H21ClFN5O4SPurezza:97.59%Colore e forma:SolidPeso molecolare:517.96Bopindolol fumarate
CAS:<p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>Formula:C27H32N2O7Colore e forma:SolidPeso molecolare:496.56DR4485 hydrochloride
CAS:<p>5-HT7 antagonist</p>Formula:C26H29Cl3N2OPurezza:98%Colore e forma:SolidPeso molecolare:491.88SLV-310
CAS:<p>SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.</p>Formula:C25H24FN3O2Purezza:99.39%Colore e forma:SolidPeso molecolare:417.48Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purezza:98%Colore e forma:SolidPeso molecolare:393.74(R)-Viloxazine Hydrochloride
CAS:<p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>Formula:C13H20ClNO3Purezza:99.88% - 99.94%Colore e forma:SolidPeso molecolare:273.76Trimipramine
CAS:<p>Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.</p>Formula:C20H26N2Purezza:98%Colore e forma:SolidPeso molecolare:294.43OPC-14523 hydrochloride
CAS:<p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>Formula:C23H29Cl2N3O2Purezza:99.60%Colore e forma:SolidPeso molecolare:450.4CGS-12066 maleate salt
CAS:<p>CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.</p>Formula:C21H21F3N4O4Colore e forma:SolidPeso molecolare:450.41GTS-21
CAS:<p>GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.</p>Formula:C19H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:308.37LY320135
CAS:CB1 receptor antagonist/inverse agonistFormula:C24H17NO4Purezza:98%Colore e forma:SolidPeso molecolare:383.4Nexopamil racemate
CAS:<p>Nexopamil racemate（(Rac)-Nexopamil） is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.</p>Formula:C24H40N2O3Purezza:98.61%Colore e forma:SolidPeso molecolare:404.59Oxetorone fumarate
CAS:<p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>Formula:C25H25NO6Purezza:99.809%Colore e forma:SolidPeso molecolare:435.48Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Formula:C25H27N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:481.56SDZ 21009
CAS:β-adrenoceptor and 5-HT1A/1B receptor antagonistFormula:C19H28N2O4Purezza:98%Colore e forma:SolidPeso molecolare:348.44SEP-363856
CAS:<p>SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.</p>Formula:C9H13NOSPurezza:98%Colore e forma:SolidPeso molecolare:183.27Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formula:C18H22BrNSPurezza:99.65%Colore e forma:SolidPeso molecolare:364.34LY 393558
CAS:<p>Dual 5-HT1B/1D receptor antagonist</p>Formula:C26H31FN4O4S2Purezza:98%Colore e forma:SolidPeso molecolare:546.68Amitifadine hydrochloride
CAS:<p>Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).</p>Formula:C11H12Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:264.58Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Formula:C18H29NO2Purezza:98%Colore e forma:SolidPeso molecolare:291.43Bemesetron
CAS:<p>Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.</p>Formula:C15H17Cl2NO2Purezza:99.77%Colore e forma:SolidPeso molecolare:314.21SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Formula:C21H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:403.86Opiranserin
CAS:<p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>Formula:C21H34N2O5Purezza:98%Colore e forma:SolidPeso molecolare:394.51Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Formula:C19H24N2OPurezza:98%Colore e forma:SolidPeso molecolare:296.41Pancopride
CAS:<p>Pancopride（LAS 30451） is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced</p>Formula:C18H24ClN3O2Purezza:93.64%Colore e forma:SolidPeso molecolare:349.86Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Formula:C18H20ClNPurezza:98%Colore e forma:SolidPeso molecolare:285.81PF-4479745
CAS:<p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>Formula:C17H22N4Purezza:98%Colore e forma:SolidPeso molecolare:282.38Masupirdine mesylate
CAS:<p>Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's disease</p>Formula:C23H32BrN3O9S3Purezza:99.57%Colore e forma:SolidPeso molecolare:670.61Ipsapirone
CAS:<p>Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.</p>Formula:C19H23N5O3SPurezza:99.51%Colore e forma:SolidPeso molecolare:401.48SB357134
CAS:<p>SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.</p>Formula:C17H18Br2FN3O3SPurezza:98%Colore e forma:SolidPeso molecolare:523.21Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Formula:C23H31ClN2Purezza:98%Colore e forma:SolidPeso molecolare:370.96SB 206553 hydrochloride
CAS:<p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>Formula:C17H17ClN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:328.8
