recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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UCSF678
CAS:<p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>Formula:C15H18N2O2SColore e forma:SolidPeso molecolare:290.385-HT4 antagonist 1
CAS:<p>5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).</p>Formula:C23H36N4O5SPurezza:99.75%Colore e forma:SolidPeso molecolare:480.62Pridefine
CAS:<p>Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.</p>Formula:C19H21NPurezza:99.15% - 99.66%Colore e forma:SolidPeso molecolare:263.38E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formula:C20H27Cl2N3O2Purezza:98.88% - 98.88%Colore e forma:SolidPeso molecolare:412.35T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Formula:C56H62N6O8Purezza:98%Colore e forma:SolidPeso molecolare:947.146SKF-83566 hydrobromide
CAS:<p>D1-like dopamine receptor antagonist</p>Formula:C17H19BrClNOPurezza:98%Colore e forma:SolidPeso molecolare:368.7GR 55562 dihydrochloride
CAS:<p>5-HT1B (5-HT1Dβ) silent antagonist</p>Formula:C23H27Cl2N3O2Purezza:99.45%Colore e forma:SolidPeso molecolare:448.39MS 245 oxalate
CAS:MS 245 oxalate is a 5-HT6 antagonist.Formula:C21H24N2O7SPurezza:98%Colore e forma:SolidPeso molecolare:448.49EGIS-7625
CAS:<p>EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.</p>Formula:C18H24Cl2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:399.32Glemanserin
CAS:<p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>Formula:C20H25NOPurezza:99.93%Colore e forma:SolidPeso molecolare:295.42DV 7028 hydrochloride
CAS:<p>DV 7028 hydrochloride is a 5-HT2A receptor antagonist.</p>Formula:C21H26ClFN4O3Purezza:98%Colore e forma:SolidPeso molecolare:436.91L-775,606
CAS:<p>L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.</p>Formula:C25H29FN6Purezza:98%Colore e forma:SolidPeso molecolare:432.54Ro 60-0175 fumarate
CAS:<p>5-HT2 receptor agonist</p>Formula:C15H16ClFN2O4Purezza:98%Colore e forma:SolidPeso molecolare:342.75PNU-96415E
CAS:dopamine D4 and serotonergic 5-HT2A receptor antagonistFormula:C21H27Cl2FN2OPurezza:98%Colore e forma:SolidPeso molecolare:413.36Alaproclate (hydrochloride)
CAS:<p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>Formula:C13H19Cl2NO2Colore e forma:SolidPeso molecolare:292.2(R)-Praziquantel
CAS:(R)-Praziquantel is an active enantiomer of praziquantel.Formula:C19H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:312.41F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Formula:C25H29ClF2N4O5Purezza:98.86%Colore e forma:SolidPeso molecolare:538.975-HT3 antagonist 2
CAS:<p>5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.</p>Formula:C18H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.38Donitriptan
CAS:<p>Donitriptan 是一种 5-HT 受体激动剂，对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>Formula:C23H25N5O2Purezza:98.76%Colore e forma:SolidPeso molecolare:403.48AR-A 2
CAS:<p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>Formula:C27H36N4O2Purezza:98%Colore e forma:SolidPeso molecolare:448.6Org37684
CAS:<p>5-HT2 receptors agonist</p>Formula:C14H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:269.77Methiothepin maleate
CAS:<p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>Formula:C24H28N2O4S2Purezza:98%Colore e forma:SolidPeso molecolare:472.62AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Formula:C17H20ClN5O2SPurezza:>99.99%Colore e forma:SolidPeso molecolare:393.89Ro 04-6790
CAS:<p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>Formula:C12H16N6O2SPurezza:98%Colore e forma:SolidPeso molecolare:308.36ST1936
CAS:<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Formula:C13H17ClN2Purezza:98%Colore e forma:SolidPeso molecolare:236.742-Methyl-5-HT maleate
CAS:<p>2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.</p>Formula:C15H18N2O5Purezza:98%Colore e forma:SolidPeso molecolare:306.31Ampreloxetine
CAS:<p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>Formula:C18H18F3NOPurezza:98%Colore e forma:SolidPeso molecolare:321.34RG-12915
CAS:<p>RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).</p>Formula:C20H25ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:360.88Org-13011 fumarate
CAS:<p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>Formula:C22H29F3N4O5Purezza:98.92%Colore e forma:SolidPeso molecolare:486.48Enciprazine
CAS:<p>Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.</p>Formula:C23H32N2O6Purezza:98.63%Colore e forma:SolidPeso molecolare:432.51Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Formula:C23H31N5O6Colore e forma:SolidPeso molecolare:473.53Deramciclane fumarate
CAS:<p>Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.</p>Formula:C24H35NO5Colore e forma:SolidPeso molecolare:417.54Bopindolol
CAS:<p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>Formula:C23H28N2O3Colore e forma:SolidPeso molecolare:380.485-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Formula:C21H23N7Colore e forma:SolidPeso molecolare:373.45MK-212
CAS:<p>MK-212 is a 5HT2C agonist; boosts corticosterone and lowers activity at 0.5-1mg/kg; reduces anxiety without affecting movement at 0.1-0.2mg/kg in mice.</p>Formula:C8H11ClN4Colore e forma:SolidPeso molecolare:198.65RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Formula:C16H24Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:363.28Eplivanserin hemifumarate
CAS:<p>Eplivanserin is an inverse agonist of 5-HT2A.</p>Formula:C23H25FN2O6Colore e forma:SolidPeso molecolare:444.45OSU 6162 hydrochloride
CAS:Dopamine stabilizerFormula:C15H24ClNO2SPurezza:98%Colore e forma:SolidPeso molecolare:317.88S-15535
CAS:<p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>Formula:C21H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:336.43Fonazine
CAS:<p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>Formula:C19H25N3O2S2Colore e forma:SolidPeso molecolare:391.55Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Formula:C26H31FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:454.53GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Formula:C23H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:411.93ATC0065 HCl
CAS:<p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>Formula:C25H31BrCl2F3N5OColore e forma:SolidPeso molecolare:625.35LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Formula:C20H24N4O3Colore e forma:SolidPeso molecolare:368.43SGS518 oxalate
CAS:<p>SGS518 oxalate is a 5-HT6 antagonist.</p>Formula:C23H24F2N2O7SPurezza:98%Colore e forma:SolidPeso molecolare:510.51(Rac)-SEP-363856
CAS:<p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>Formula:C9H13NOSPurezza:98%Colore e forma:SolidPeso molecolare:183.27AP521
CAS:<p>AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).</p>Formula:C20H19ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:402.89SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Colore e forma:SolidPeso molecolare:474.33WAY 161503 hydrochloride
CAS:<p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>Formula:C11H12Cl3N3OPurezza:98%Colore e forma:SolidPeso molecolare:308.59SUN-C5174
CAS:<p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>Formula:C22H29FN4O2Purezza:98%Colore e forma:SolidPeso molecolare:400.49
