recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Formula:C24H27FN4O2Purezza:98.04%Colore e forma:SolidPeso molecolare:422.5Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Formula:C26H32N2O5Purezza:99.17% - 99.67%Colore e forma:SolidPeso molecolare:452.54LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:372.89Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purezza:99.77%Colore e forma:SolidPeso molecolare:304.43Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Formula:C28H30ClN5O3Purezza:99.04%Colore e forma:SolidPeso molecolare:520.02ML 10302 hydrochloride
CAS:<p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>Formula:C15H22Cl2N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:349.25LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purezza:98.58%Colore e forma:SolidPeso molecolare:407.33GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formula:C23H27N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:377.48Itasetron
CAS:<p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>Formula:C16H20N4O2Purezza:98.58% - 99.33%Colore e forma:SolidPeso molecolare:300.36ADR-851 free base
CAS:ADR-851 free base is an antagonist of the HT3 receptor.Formula:C14H18ClN3O2Purezza:97.88% - 98.39%Colore e forma:SolidPeso molecolare:295.77Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59Cianopramine
CAS:<p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>Formula:C20H23N3Purezza:99.92% - 99.92%Colore e forma:SolidPeso molecolare:305.42Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Formula:C15H23NOPurezza:98.09% - 98.77%Colore e forma:SolidPeso molecolare:233.35BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Formula:C28H45ClN4O11S4Purezza:>99.99%Colore e forma:SolidPeso molecolare:777.39Tedatioxetine
CAS:<p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>Formula:C18H21NSPurezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:283.438-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Formula:C16H25NOPurezza:98%Colore e forma:SolidPeso molecolare:247.38SB 699551 dihydrochloride
CAS:<p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>Formula:C34H47Cl2N3OPurezza:99.83%Colore e forma:SolidPeso molecolare:584.66Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Formula:C13H19NO3Purezza:99.67%Colore e forma:SolidPeso molecolare:237.29RS 67333 hydrochloride
CAS:<p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>Formula:C19H30Cl2N2O2Purezza:98.78%Colore e forma:SolidPeso molecolare:389.36CP 96021
CAS:<p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>Formula:C29H21FN4OSPurezza:97.81% - 99.62%Colore e forma:SoildPeso molecolare:492.57Landipirdine
CAS:<p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>Formula:C18H19FN2O3SPurezza:97.61% - 99.37%Colore e forma:SolidPeso molecolare:362.42Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Formula:C20H21N3OPurezza:99.82% - 99.98%Colore e forma:SolidPeso molecolare:319.4RS 42358-197
CAS:<p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>Formula:C19H23ClN2OPurezza:99.70%Colore e forma:SolidPeso molecolare:330.85E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Formula:C17H18ClN5O2S2Purezza:96.32% - 99.53%Colore e forma:SolidPeso molecolare:423.94Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurezza:97.01%Colore e forma:SolidPeso molecolare:323.46MM 77 dihydrochloride
CAS:<p>MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.</p>Formula:C19H29Cl2N3O3Purezza:99.91%Colore e forma:SolidPeso molecolare:418.36(Z)-Thiothixene
CAS:<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Formula:C23H29N3O2S2Purezza:99.21%Colore e forma:Yellow To Yellow With A Tan Cast PowderPeso molecolare:443.63Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Formula:C20H26ClNO2Purezza:99.63%Colore e forma:SolidPeso molecolare:347.88SB-215505
CAS:<p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>Formula:C19H16ClN3OPurezza:98.33%Colore e forma:SolidPeso molecolare:337.85-HT2 antagonist 1
CAS:<p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>Formula:C22H29FN4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:400.49SB228357
CAS:<p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>Formula:C22H17F4N3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:431.38Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Formula:C14H20ClN3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:313.785HT6-ligand-1
CAS:<p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>Formula:C20H22BrN3O2SPurezza:99.24% - 99.93%Colore e forma:SolidPeso molecolare:448.38SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Formula:C23H31Cl2NO8SPurezza:99.37%Colore e forma:SolidPeso molecolare:552.47LY-2624803
CAS:<p>LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.</p>Formula:C22H25N3O3Purezza:99.78% - 99.97%Colore e forma:SolidPeso molecolare:379.45Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:346.47Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formula:C22H22N2O7Purezza:99.66%Colore e forma:SolidPeso molecolare:426.42Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Formula:C24H40N2O3Purezza:97.87% - >99.99%Colore e forma:SolidPeso molecolare:404.59ATC 0175 hydrochloride
CAS:<p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>Formula:C23H26ClF2N5OPurezza:99.98%Colore e forma:SolidPeso molecolare:461.93Perphenazine dihydrochloride
CAS:Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formula:C21H28Cl3N3OSPurezza:99.67%Colore e forma:SolidPeso molecolare:476.89Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Formula:C24H22N4Purezza:99.91%Colore e forma:SolidPeso molecolare:366.46Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Formula:C21H24BrN3O3SPurezza:98.36% - 99.65%Colore e forma:SolidPeso molecolare:478.4Teniloxazine
CAS:<p>Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.</p>Formula:C16H19NO2SPurezza:99.23%Colore e forma:SolidPeso molecolare:289.39Piromelatine
CAS:<p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>Formula:C17H16N2O4Purezza:99.89%Colore e forma:SolidPeso molecolare:312.32H-9 dihydrochloride
CAS:<p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>Formula:C11H15Cl2N3O2SPurezza:97.3%Colore e forma:SolidPeso molecolare:324.235-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Formula:C22H20FN3O3Purezza:98.78% - 99.26%Colore e forma:SolidPeso molecolare:393.41Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Formula:C16H19NOPurezza:99.47%Colore e forma:SolidPeso molecolare:241.33BMY-14802 hydrochloride
CAS:<p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>Formula:C18H23ClF2N4OPurezza:99.97%Colore e forma:SolidPeso molecolare:384.85Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Formula:C24H32N4O2SPurezza:99.74%Colore e forma:SolidPeso molecolare:440.65-HT1A modulator 1
CAS:<p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>Formula:C21H25N3O2SPurezza:99.68%Colore e forma:SolidPeso molecolare:383.51
