recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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Geissoschizine methyl ether
CAS:<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Formula:C22H26N2O3Purezza:99.24% - 99.68%Colore e forma:SolidPeso molecolare:366.45Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formula:C4H3F7OPurezza:98%Colore e forma:Less Oil Colorless OilPeso molecolare:200.05Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Formula:C20H20N2O3Purezza:99.27% - 99.80%Colore e forma:SolidPeso molecolare:336.38SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formula:C18H21Cl2N3O4SPurezza:98.94%Colore e forma:SolidPeso molecolare:446.35m-Chlorophenylbiguanide hydrochloride
CAS:<p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>Formula:C8H11Cl2N5Purezza:99.43% - 99.87%Colore e forma:SolidPeso molecolare:248.11LY334370
CAS:<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Formula:C21H22FN3OPurezza:99.32%Colore e forma:SolidPeso molecolare:351.42Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formula:C24H32ClNO3Purezza:99.57% - 99.77%Colore e forma:SolidPeso molecolare:417.97Tropisetron
CAS:Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.Formula:C17H20N2O2Purezza:99.68%Colore e forma:White SolidPeso molecolare:284.35Piboserod hydrochloride
CAS:<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Formula:C22H32ClN3O2Colore e forma:SolidPeso molecolare:405.96SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurezza:99.83%Colore e forma:SolidPeso molecolare:286.35Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Formula:C28H33ClN2·2HClPurezza:98.05%Colore e forma:Off-White PowderPeso molecolare:505.95Sumatriptan hydrochloride
CAS:<p>Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.</p>Formula:C14H22ClN3O2SColore e forma:SolidPeso molecolare:331.86Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formula:C27H37N5O9Purezza:97.84% - 99.90%Colore e forma:SolidPeso molecolare:575.61ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Formula:C24H29N3O3Colore e forma:SolidPeso molecolare:407.51Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formula:C23H30N4O2SPurezza:99.23%Colore e forma:White PowderPeso molecolare:426.57Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Formula:C35H47FN10O8Purezza:97.97%Colore e forma:SolidPeso molecolare:754.85Serotonin hydrochloride
CAS:<p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>Formula:C10H13ClN2OPurezza:98.05% - 99.93%Colore e forma:White To Cream PowderPeso molecolare:212.6764F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formula:C22H26FNO·C2H2O4Purezza:97.34%Colore e forma:SolidPeso molecolare:429.49Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formula:C22H23FN2O5Purezza:97.39% - 99.73%Colore e forma:White SolidPeso molecolare:414.43Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurezza:97.62%Colore e forma:SolidPeso molecolare:370.28Ondansetron
CAS:<p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>Formula:C18H19N3OPurezza:99.92%Colore e forma:White To Yellow CrystalsPeso molecolare:293.36SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formula:C21H21Cl3N4O2Colore e forma:SolidPeso molecolare:467.78S1RA hydrochloride
CAS:<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Formula:C20H24ClN3O2Purezza:98% - 99.84%Colore e forma:SolidPeso molecolare:373.87Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Formula:C22H31N3O2Purezza:97.21% - 99.49%Colore e forma:SolidPeso molecolare:369.57-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formula:C10H6F3NO2Purezza:97.31% - 97.84%Colore e forma:Yellow PowderPeso molecolare:229.16Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41SKF-83566
CAS:<p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>Formula:C17H18BrNOPurezza:95.00% - 99.82%Colore e forma:SolidPeso molecolare:332.23Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Formula:C17H25N3O2S·C4H6O5Purezza:99.95%Colore e forma:Pale Yellow SolidPeso molecolare:469.55Eltoprazine
CAS:<p>Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.</p>Formula:C12H16N2O2Colore e forma:SolidPeso molecolare:220.27BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Formula:C22H33Cl2N3O3Purezza:97.32% - 99.08%Colore e forma:SolidPeso molecolare:458.42ML 10302
CAS:<p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>Formula:C15H21ClN2O3Colore e forma:SolidPeso molecolare:312.79SAX-187
CAS:<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Formula:C15H13ClN4O2S2Purezza:97.82% - 98%Colore e forma:SolidPeso molecolare:380.87Rotundine
CAS:<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Formula:C21H25NO4Purezza:99.8% - 99.91%Colore e forma:Off-White SolidPeso molecolare:355.43F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Formula:C19H21ClF2N4OPurezza:98.72%Colore e forma:SolidPeso molecolare:394.85Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formula:C18H18ClNOSPurezza:99.78%Colore e forma:SolidPeso molecolare:331.86Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68Metoclopramide
CAS:<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Formula:C22H25ClN4O4S2Colore e forma:SolidPeso molecolare:509.04RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Formula:C17H16FN3Purezza:99.32%Colore e forma:SolidPeso molecolare:281.33Harmine
CAS:<p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>Formula:C13H12N2OPurezza:98.29% - 99.92%Colore e forma:Off-White SolidPeso molecolare:212.25Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Formula:C23H27ClFN3O2Purezza:98%Colore e forma:SolidPeso molecolare:431.93Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Formula:C17H18ClN3OPurezza:99.95%Colore e forma:SolidPeso molecolare:315.8Methiothepin mesylate
CAS:<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Formula:C21H28N2O3S3Purezza:98% - 99.92%Colore e forma:SolidPeso molecolare:452.65Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Formula:C23H24FN3O2Purezza:99.2%Colore e forma:SolidPeso molecolare:393.45Trazodone
CAS:<p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>Formula:C19H22ClN5OPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:371.861-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Formula:C14H17ClN2Purezza:98.27%Colore e forma:SolidPeso molecolare:248.75A-582941 dihydrochloride
CAS:<p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>Formula:C17H22Cl2N4Purezza:99.55%Colore e forma:SolidPeso molecolare:353.29Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Formula:C24H26ClFN4OPurezza:99.87% - 99.92%Colore e forma:Off-White To Pale Yellow SolidPeso molecolare:440.94Rizatriptan benzoate
CAS:<p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>Formula:C22H25N5O2Purezza:99% - 99.79%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:391.47PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurezza:99.35%Colore e forma:SolidPeso molecolare:292.36
