Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 728 prodotti di "Recettore adrenergico"
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Ulimorelin
CAS:Ulimorelin, ghrelin receptor agonist (EC50: 29 nM, Ki: 16 nM), is a prokinetic and vasorelaxant via α1-adrenoceptor antagonism.Formula:C30H39FN4O4Purezza:98%Colore e forma:SolidPeso molecolare:538.65(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Colore e forma:SolidPeso molecolare:367.44Metoprolol HCl
CAS:Metoprolol: a β1 blocker for high blood pressure, chest pain, fast heart rate, post-heart attack care, and migraine prevention.Formula:C15H26ClNO3Colore e forma:SolidPeso molecolare:303.827Carbuterol hydrochloride
CAS:Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.Formula:C13H22ClN3O3Colore e forma:SolidPeso molecolare:303.79Afurolol Hydrochloride
CAS:Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.Formula:C15H22ClNO4Purezza:98.86%Colore e forma:SolidPeso molecolare:315.79Amosulalol, (+)-
CAS:Amosulalol, (+)-, is an adrenergic agent.Formula:C18H24N2O5SColore e forma:SolidPeso molecolare:380.46YM-430
CAS:YM-430: β1 blocker & Ca²⁺ channel antagonist; antianginal & antihypertensive; IC50: 59.2 nM (rhythmic contractions), 36.6 mg/kg in rats (ST depression).Formula:C29H35N3O8Purezza:98%Colore e forma:SolidPeso molecolare:553.6Pirepemat fumarate
CAS:Pirepemat fumarate (IRL752), aids Parkinson's research, boosts cognition and cortical catecholamine transmission.Formula:C15H17F2NO5Colore e forma:SolidPeso molecolare:329.3Trimazosin hydrochloride
CAS:Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.Formula:C20H32ClN5O7Colore e forma:SolidPeso molecolare:489.95RX821002
CAS:RX821002: potent α2-adrenoceptor antagonist, selective for α2D (pKd 9.7) over α2A (pKd 8.2), low affinity for imidazoline.Formula:C12H14N2O3Purezza:98%Colore e forma:SolidPeso molecolare:234.25SNAP-5089
CAS:SNAP-5089 is a highly selective alpha1A-adrenoceptor antagonist.Formula:C36H41ClN4O5Colore e forma:SolidPeso molecolare:645.2Amibegron
CAS:Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formula:C22H26ClNO4Colore e forma:SolidPeso molecolare:403.9Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purezza:97.15% - 98.85%Colore e forma:SolidPeso molecolare:251.33Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purezza:99.89%Colore e forma:SolidPeso molecolare:483.56Ref: TM-T11148
1mg369,00€5mg735,00€10mg938,00€25mg1.473,00€50mg1.882,00€100mg2.670,00€1mL*10mM (DMSO)929,00€Palatrigine
CAS:Palatrigine (BW-A 256C) is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.Formula:C12H13Cl2N5Purezza:98.87%Colore e forma:SolidPeso molecolare:298.17Bisaramil hydrochloride
CAS:Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.Formula:C17H24Cl2N2O2Purezza:98.64% - 99.48%Colore e forma:SolidPeso molecolare:359.29GP2-114
CAS:GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.Formula:C19H24N2O4Purezza:99.32%Colore e forma:SolidPeso molecolare:344.4Bedoradrine
CAS:Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5Purezza:>99.99%Colore e forma:SolidPeso molecolare:428.52Butofilolol
CAS:Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Formula:C17H26FNO3Purezza:98.96% - >99.99%Colore e forma:SolidPeso molecolare:311.392Imiloxan
CAS:Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formula:C14H16N2O2Purezza:98.13% - 99.8%Colore e forma:SolidPeso molecolare:244.29Taprizosin
CAS:Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.Formula:C25H26N6O4SPurezza:98.10% - 99.11%Colore e forma:SolidPeso molecolare:506.58Rezatomidine
CAS:Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.Formula:C13H16N2SPurezza:98.34%Colore e forma:SolidPeso molecolare:232.34Oxyfedrine L-form HCl
CAS:Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.Formula:C19H24ClNO3Purezza:99.5% - 99.57%Colore e forma:SolidPeso molecolare:349.85Ref: TM-T24579
1mg96,00€5mg188,00€10mg329,00€25mg512,00€50mg740,00€100mg944,00€200mg1.264,00€1mL*10mM (DMSO)215,00€Midaglizole hydrochloride
CAS:Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Formula:C16H19Cl2N3Purezza:99.39% - 99.82%Colore e forma:SolidPeso molecolare:324.25Ref: TM-T11015
1mg57,00€5mg126,00€10mg198,00€25mg324,00€50mg439,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)160,00€Neldazosin
CAS:Neldazosin is used as a potent α1-adrenoceptor antagonist.Formula:C18H25N5O4Purezza:99.76% - 99.97%Colore e forma:SolidPeso molecolare:375.42Soquinolol
CAS:Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a longFormula:C17H26N2O3Purezza:97.48% - 98.63%Colore e forma:SolidPeso molecolare:306.4Xamoterol hemifumarate
CAS:Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationshipFormula:C36H54N6O14Purezza:99.79%Colore e forma:White SolidPeso molecolare:794.37Nemazoline Free Base
CAS:Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Formula:C10H11Cl2N3Purezza:98.06% - 98.83%Colore e forma:SolidPeso molecolare:244.12Dabelotine
CAS:<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Formula:C15H22N2O2Purezza:98.55%Colore e forma:SolidPeso molecolare:262.35JP1302
CAS:JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formula:C24H24N4Purezza:99.96%Colore e forma:SolidPeso molecolare:368.47Rafabegron
CAS:Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Formula:C21H23ClN2O4Purezza:99.81%Colore e forma:SolidPeso molecolare:402.87Pipoxazole
CAS:Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Formula:C14H20N4OPurezza:98.58% - 99.53%Colore e forma:SolidPeso molecolare:260.33Egis-11150
CAS:Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formula:C19H21ClFN5O2Purezza:97.49% - >99.99%Colore e forma:SolidPeso molecolare:405.85(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purezza:98.27%Colore e forma:SolidPeso molecolare:646.17Fipamezole
CAS:Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.Formula:C14H15FN2Purezza:99.32% - 99.97%Colore e forma:SolidPeso molecolare:230.28CL 316243
CAS:CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Formula:C20H18ClNNa2O7Purezza:98.00% - 99.68%Colore e forma:SolidPeso molecolare:465.79Ref: TM-T10830
1mg52,00€5mg111,00€10mg169,00€25mg329,00€50mg527,00€100mgPrezzo su richiesta500mgPrezzo su richiestaMilveterol HCl
CAS:Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formula:C25H30ClN3O4Purezza:99.9%Colore e forma:SolidPeso molecolare:471.98Vadocaine
CAS:Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.Formula:C18H28N2O2Purezza:99.7%Colore e forma:SolidPeso molecolare:304.43Amosulalol
CAS:<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Formula:C18H24N2O5SPurezza:99.5%Colore e forma:SolidPeso molecolare:380.46ST 91
CAS:ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.Formula:C13H20ClN3Purezza:99.83%Colore e forma:SolidPeso molecolare:253.77Ref: TM-T23397
5mg52,00€10mg75,00€25mg150,00€50mg259,00€100mg374,00€200mg525,00€1mL*10mM (DMSO)52,00€Bedoradrine sulfate
CAS:Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5H2O4SPurezza:99.31%Colore e forma:SolidPeso molecolare:477.56ORM-10921
CAS:ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formula:C18H23NO2Purezza:99.46% - 99.98%Colore e forma:SolidPeso molecolare:285.38BMS-194449
CAS:BMS-194449 is a full beta 3 agonist.Formula:C24H24F4N2O6SColore e forma:SolidPeso molecolare:544.52Abediterol
CAS:Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.Formula:C25H30F2N2O4Colore e forma:SolidPeso molecolare:460.51β3-AR agonist 2
CAS:β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Formula:C27H38N4O7SPurezza:98%Colore e forma:SolidPeso molecolare:562.68Pronetalol
CAS:Pronethalol ((±)-Pronethalol), a non-selective β-adrenergic antagonist, effectively inhibits Sox2 expression and offers protection against Digitalis-induced ventricular arrhythmias. Additionally, it can reverse such arrhythmias and limit the development of cerebral arteriovenous malformations (AVMs) [1] [2].Formula:C15H19NOColore e forma:SolidPeso molecolare:229.32(±)-N-Methylcoclaurine
CAS:N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].Formula:C18H21NO3Purezza:98%Colore e forma:SolidPeso molecolare:299.36Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurezza:99.73%Colore e forma:SolidPeso molecolare:555.65Nolomirole HCl
CAS:Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to studyFormula:C19H28ClNO4Purezza:99.03% - >99.99%Colore e forma:SolidPeso molecolare:369.88β3-AR agonist 1
CAS:β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/Formula:C22H28N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:444.55Mefenidil
CAS:Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.Formula:C12H11N3Purezza:98.27%Colore e forma:SolidPeso molecolare:197.24L-796568 dihydrochloride
CAS:L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.Formula:C31H29Cl2F3N4O3S2Colore e forma:SolidPeso molecolare:697.62N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Formula:C20H23Cl2NO5Colore e forma:SolidPeso molecolare:428.31SDZ-NVI-085
CAS:SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.Formula:C15H21NO2SColore e forma:SolidPeso molecolare:279.4Lidamidine
CAS:Lidamidine (Lidamidinum) is an effective antidiarrheal agent that inhibits intestinal secretion, reduces intestinal transit, and inhibits smooth muscleFormula:C11H16N4OPurezza:99.98%Colore e forma:SolidPeso molecolare:220.27Ref: TM-T25719
1mg115,00€2mg162,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€AR-08
CAS:<p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>Formula:C12H12N6Purezza:99.7%Colore e forma:SolidPeso molecolare:240.26Ro-70-0004
CAS:Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.Formula:C20H24F4N4O3Colore e forma:SolidPeso molecolare:444.42RS100329 hydrochloride
CAS:RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.Formula:C20H26ClF3N4O3Purezza:99.95%Colore e forma:SolidPeso molecolare:462.89Ref: TM-T23253
1mg35,00€5mg64,00€10mg104,00€25mg220,00€50mg328,00€100mg469,00€500mgPrezzo su richiestaRitodrine
CAS:Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].Formula:C17H21NO3Colore e forma:SolidPeso molecolare:287.35Phentolamine Analogue 1
CAS:Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formula:C17H19N3OPurezza:99.96%Colore e forma:SolidPeso molecolare:281.35Ref: TM-T12444
1mg86,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)172,00€Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formula:C30H30ClN5O4SColore e forma:SolidPeso molecolare:592.11Bufuralol (hydrochloride)
CAS:Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.Formula:C16H24ClNO2Colore e forma:SolidPeso molecolare:297.82Binedaline
CAS:Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formula:C19H23N3Purezza:98%Colore e forma:SolidPeso molecolare:293.41Bunazosin Hydrochloride
CAS:Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.Formula:C19H28ClN5O3Purezza:99.12%Colore e forma:SolidPeso molecolare:409.91Vatinoxan hydrochloride
CAS:Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.Formula:C20H27ClN4O4SPurezza:98%Colore e forma:SolidPeso molecolare:454.97L-796568 free base
CAS:L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).Formula:C31H27F3N4O3S2Colore e forma:SolidPeso molecolare:624.7LK 204-545
CAS:LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.Formula:C25H32N4O6Colore e forma:SolidPeso molecolare:484.54Vemtoberant
CAS:Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.Formula:C29H37N3O8S2Colore e forma:SolidPeso molecolare:619.75NGD9002
CAS:NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.Formula:C20H31N5OPurezza:98%Colore e forma:SolidPeso molecolare:357.49KUC-7322
CAS:Ritobegron is used as a selective β3-adrenoceptor agonist and the prodrug of the active compound, KUC-7322.Formula:C21H27NO5Colore e forma:SolidPeso molecolare:373.44Epinephrine HCl
CAS:Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.Formula:C9H14ClNO3Purezza:99.48%Colore e forma:SolidPeso molecolare:219.67N-5984
CAS:<p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>Formula:C20H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:391.854-hydroxy Nebivolol hydrochloride
CAS:4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.Formula:C22H25F2NO5HClColore e forma:SolidPeso molecolare:457.9Todralazine hydrochloride
CAS:Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Formula:C11H13ClN4O2Purezza:99.91%Colore e forma:SolidPeso molecolare:268.7(-)-Isoproterenol hydrochloride
CAS:(-)-Isoproterenol hydrochloride is used as a β-adrenergic receptor agonist in the treatment of bradycardia and as a bronchodilator.Formula:C11H17NO3·CIHColore e forma:SolidPeso molecolare:247.72BI-167107
CAS:BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).Formula:C21H26N2O4Colore e forma:SolidPeso molecolare:370.44Indacaterol acetate
CAS:Indacaterol acetate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C26H32N2O5Colore e forma:SolidPeso molecolare:452.54RS 17053 hydrochloride
CAS:RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.Formula:C24H30Cl2N2O2Purezza:99.27%Colore e forma:SolidPeso molecolare:449.41Bufuralol
CAS:Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Formula:C16H23NO2Purezza:98.26%Colore e forma:SolidPeso molecolare:261.36Prenalterol hydrochloride
CAS:Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Formula:C12H20ClNO3Colore e forma:SolidPeso molecolare:261.75Domesticine, (-)-
CAS:Domesticine, (-)- is an antagonist of alpha-1D-adrenoceptor.Formula:C19H19NO4Purezza:98%Colore e forma:SolidPeso molecolare:325.36GW-597901
CAS:GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.Formula:C25H38N2O6SColore e forma:SolidPeso molecolare:494.64Indacaterol xinafoate
CAS:Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C35H36N2O6Colore e forma:SolidPeso molecolare:580.67AGN 192836
CAS:AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).Formula:C12H13N3O2Colore e forma:SolidPeso molecolare:231.25Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formula:C20H33N3O4·HClColore e forma:White Crystalline SolidPeso molecolare:415.96BU-E 75
CAS:BU-E 75 is an agonist of the histamine H2.Formula:C21H24F2N6Colore e forma:SolidPeso molecolare:398.45Dibenamine hydrochloride
CAS:<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Formula:C16H19Cl2NPurezza:96.43%Colore e forma:Oily Liquid SolidPeso molecolare:296.23OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purezza:99.79%Colore e forma:SolidPeso molecolare:421.58Ref: TM-T13804
1mg187,00€5mg455,00€10mg620,00€25mg940,00€50mg1.264,00€100mg1.663,00€200mg2.252,00€1mL*10mM (DMSO)567,00€α1 adrenoceptor-MO-1
CAS:α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Formula:C20H24ClN5OPurezza:99.20% - 99.29%Colore e forma:SolidPeso molecolare:385.89Ref: TM-T10003
1mg198,00€5mg393,00€10mg542,00€25mg785,00€50mg1.074,00€100mg1.454,00€200mg1.967,00€1mL*10mM (DMSO)467,00€Deriglidole
CAS:Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Formula:C16H21N3Purezza:98.12% - 99.03%Colore e forma:SolidPeso molecolare:255.360990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormula:C21H21N5Purezza:98.99%Colore e forma:SolidPeso molecolare:343.42Ref: TM-T13983
1mg202,00€5mg512,00€10mg740,00€25mg1.121,00€50mg1.539,00€100mg2.072,00€1mL*10mM (DMSO)535,00€(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formula:C12H19NO3Purezza:99.73%Colore e forma:SolidPeso molecolare:225.28Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Formula:C18H22ClNO4Purezza:99.82%Colore e forma:SolidPeso molecolare:351.83CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purezza:99.40% - 99.58%Colore e forma:SolidPeso molecolare:494.46Ref: TM-T30846
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Meluadrine
CAS:Meluadrine, a potent agonist of the β2 adrenergic receptor, is one of the metabolites of Tulobuterol [1].Formula:C12H18ClNO2Peso molecolare:243.732,3-MDMA hydrochloride
CAS:2,3-MDMA hydrochloride is an inhibitor of the noradrenalin transporter and serotonin transporter, with IC50 values of 6.2 μM and 82 μM, respectively.Formula:C11H16ClNO2Peso molecolare:229.703Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Formula:C23H30N6O4Purezza:98%Colore e forma:SolidPeso molecolare:454.52Butopamine hydrochloride
CAS:Butopamine hydrochloride is an orally active inotropic compound that is more effective at increasing heart rate compared to Dobutamine.Formula:C18H24ClNO3Colore e forma:SolidPeso molecolare:337.84Ersentilide
CAS:Ersentilide, a benzamide derivative, functions as both a β1-adrenergic receptor antagonist and an Ikr blocker. It has demonstrated efficacy in animal models of cardiac arrhythmias.Formula:C21H26N4O5SColore e forma:SolidPeso molecolare:446.52Nipradolol
CAS:Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.Formula:C15H22N2O6Colore e forma:SolidPeso molecolare:326.35Org-6906
CAS:DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.Formula:C13H16ClNPurezza:98%Colore e forma:SolidPeso molecolare:221.73BRL-37344
CAS:<p>BRL-37344 is a selective β3-adrenergic receptor agonist. It significantly reduces the body weight of obese mice.</p>Formula:C19H22ClNO4Colore e forma:SolidPeso molecolare:363.84Carazolol hydrochloride
CAS:Carazolol (BM 51052) hydrochloride is a potent antagonist of β1/β2-adrenoceptors and also serves as a powerful and selective agonist of β3-adrenoceptors. It is utilized in research focusing on hypertension.Formula:C18H23ClN2O2Peso molecolare:334.84SAR-150640
CAS:SAR-150640, a selective β3-adrenergic receptor agonist, prevents an increase in MMP activity and production observed after LPS stimulation or in cases of chorioamnionitis.Formula:C25H35ClN2O7SColore e forma:SolidPeso molecolare:543.07L-654284
CAS:L-654284 is an α2-adrenergic receptor antagonist characterized by its notable selectivity. It competes with 3H-clonidine and 3H-rauwolscine for binding in vitro, exhibiting Ki values of 0.8 nM and 1.1 nM, respectively. L-654284 effectively blocks the pre-ejaculatory effects of clonidine in isolated rat vas deferens, with a pA2 value of 9.1. The compound demonstrates significant selectivity for α2 over α1 adrenergic receptors, with a Ki value of 110 nM against 3H-prazosin binding. In vivo, L-654284 significantly increases the turnover of norepinephrine in the rat cerebral cortex, indicating its activity in blocking α2-adrenergic receptors within the central nervous system.Formula:C18H24N2O4SColore e forma:SolidPeso molecolare:364.46AA 497 (Free Base)
CAS:AA 497, a beta-2 agonist, causes relaxation and suppresses Ca spike frequency.Formula:C14H21NO3Purezza:98%Colore e forma:SolidPeso molecolare:251.32(±)-Penbutolol
CAS:(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.Formula:C18H29NO2Colore e forma:SolidPeso molecolare:291.43Sulfinalol hydrochloride
CAS:Sulfinalol hydrochloride is an orally active β-adrenoceptor (β-adrenoceptor) antagonist that exhibits direct vasodilatory activity. It is also classified as an antihypertensive agent.Formula:C20H28ClNO4SColore e forma:SolidPeso molecolare:413.96LK 11
CAS:LK-11, an alkaloid derivative, inhibits the passive uptake of norepinephrine (NA) by synaptic vesicles in the thalamus, similarly to cocaine.Formula:C15H26N2O3Colore e forma:SolidPeso molecolare:282.38Aclidinium
CAS:Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, exhibiting bronchodilator properties. It effectively reduces lung hyperinflation, enhances lung function, and prolongs exercise endurance time. This compound is commonly utilized in studies focusing on chronic obstructive pulmonary disease (COPD).Formula:C26H30NO4S2Colore e forma:SolidPeso molecolare:484.65TAAR1 agonist 3
CAS:TAAR1 agonist 3 is a potent agonist of Trace Amine-Associated Receptor 1 (TAAR1) with a pEC50 value of 7.6. Additionally, it acts as a full agonist at the α2AR with a pEC50 of 6. TAAR1 agonist 3 is utilized in the research of neuropsychiatric disorders.Formula:C10H13NOColore e forma:SolidPeso molecolare:163.22(Rac)-Nebivolol
CAS:(Rac)-Nebivolol, a racemic β1-adrenergic blocker (IC50=0.8 nM), has vasodilatory properties and mitigates ethanol-induced cardiac harm.Formula:C22H25F2NO4Colore e forma:SolidPeso molecolare:405.43RU 52583
CAS:RU 52583 is an alpha 2-adrenergic receptor antagonist.Formula:C18H20N2Purezza:98%Colore e forma:SolidPeso molecolare:264.36Anti-MRSA agent 19
CAS:Anti-MRSA agent 19 (Compound 1) is an antibiotic that exhibits activity against Staphylococcus aureus. It is active against 40 clinical isolates from the CDC, representing diverse bacterial species with various resistance factors, including resistance to vancomycin, aminoglycoside/tetracycline, and oxazolidinone (median MIC=4 μg/mL).Formula:C15H10Cl3NO4Colore e forma:SolidPeso molecolare:374.6Vibegron
CAS:Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Formula:C26H28N4O3Colore e forma:SolidPeso molecolare:444.53Bometolol Hydrochloride
CAS:Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.Formula:C25H33ClN2O7Purezza:98%Colore e forma:SolidPeso molecolare:508.99Mafoprazine
CAS:Mafoprazine, a phenylpiperazine derivative, exhibits varying affinities for neuronal receptors, primarily exerting its antipsychotic effects through blocking D2 receptors and enhancing α-adrenergic activity. It also increases the activity of dopamine metabolites.Formula:C22H28FN3O3Colore e forma:SolidPeso molecolare:401.47Metrazoline
CAS:<p>Metrazoline (o-Methyl-tracizoline) acts as a ligand for adrenergic receptors (low affinity) and imidazoline I2 receptors.</p>Formula:C14H16N2O4Colore e forma:SolidPeso molecolare:276.288(S)-Bucindolol
CAS:(S)-Bucindolol is an enantiomer of bucindolol, specifically a β1-adrenergic receptor antagonist. It is primarily utilized in research related to heart failure.Formula:C22H25N3O2Colore e forma:SolidPeso molecolare:363.45PF-9404C
CAS:PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.Formula:C16H25N3O9Purezza:98%Colore e forma:SolidPeso molecolare:403.38HOKU-81
CAS:HOKU-81is a new bronchodilator and is one of the metabolites of tulobuterol.Formula:C12H18ClNO2Colore e forma:SolidPeso molecolare:243.73Picumeterol
CAS:Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth muscle relaxation. Picumeterol is a pure R enantiomer that can be used to improve lung function and reduce airway hyperreactivity in patients with asthma.Formula:C21H29Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:426.38N-methyl-2-AI (hydrochloride)
CAS:N-methyl-2-AI (hydrochloride) is a useful organic compound for research related to life sciences. The catalog number is T66396 and the CAS number is 10408-85-2.Formula:C10H14ClNColore e forma:SolidPeso molecolare:183.684-Hydroxyatomoxetine
CAS:4-Hydroxyatomoxetine, an active metabolite of Atomoxetine, is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.Formula:C17H21NO2Purezza:98%Colore e forma:SolidPeso molecolare:271.351-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol
CAS:1-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol is a useful organic compound for research related to life sciences. The catalog number is T65156 and the CAS number is 24155-42-8.Formula:C11H10Cl2N2OColore e forma:SolidPeso molecolare:257.114-Hydroxypropranolol hydrochloride
CAS:4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors (pA2s: 8.24 and 8.26).Formula:C16H22ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:311.8SKF 89748
CAS:SKF 89748 is an agonists of alpha 1-adrenoceptor.Formula:C12H17NOSPurezza:98%Colore e forma:SolidPeso molecolare:223.33SB251023
CAS:SB251023 is an agonist of β3-adrenoceptor.Formula:C28H34NO6PColore e forma:SolidPeso molecolare:511.55
