Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 729 prodotti di "Recettore adrenergico"
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RS100329 hydrochloride
CAS:RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.Formula:C20H26ClF3N4O3Purezza:99.95%Colore e forma:SolidPeso molecolare:462.89Ref: TM-T23253
1mg35,00€5mg64,00€10mg104,00€25mg220,00€50mg328,00€100mg469,00€500mgPrezzo su richiestaL-796568 free base
CAS:L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).Formula:C31H27F3N4O3S2Colore e forma:SolidPeso molecolare:624.7LK 204-545
CAS:LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.Formula:C25H32N4O6Colore e forma:SolidPeso molecolare:484.54NGD9002
CAS:NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.Formula:C20H31N5OPurezza:98%Colore e forma:SolidPeso molecolare:357.49Vatinoxan hydrochloride
CAS:Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.Formula:C20H27ClN4O4SPurezza:98%Colore e forma:SolidPeso molecolare:454.97Domesticine, (-)-
CAS:Domesticine, (-)- is an antagonist of alpha-1D-adrenoceptor.Formula:C19H19NO4Purezza:98%Colore e forma:SolidPeso molecolare:325.36GW-597901
CAS:GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.Formula:C25H38N2O6SColore e forma:SolidPeso molecolare:494.64Epinephrine HCl
CAS:Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.Formula:C9H14ClNO3Purezza:99.48%Colore e forma:SolidPeso molecolare:219.67KUC-7322
CAS:Ritobegron is used as a selective β3-adrenoceptor agonist and the prodrug of the active compound, KUC-7322.Formula:C21H27NO5Colore e forma:SolidPeso molecolare:373.44Vemtoberant
CAS:Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.Formula:C29H37N3O8S2Colore e forma:SolidPeso molecolare:619.75Abediterol
CAS:Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.Formula:C25H30F2N2O4Colore e forma:SolidPeso molecolare:460.51BMS-194449
CAS:BMS-194449 is a full beta 3 agonist.Formula:C24H24F4N2O6SColore e forma:SolidPeso molecolare:544.52β3-AR agonist 1
CAS:β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/Formula:C22H28N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:444.55L-796568 dihydrochloride
CAS:L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.Formula:C31H29Cl2F3N4O3S2Colore e forma:SolidPeso molecolare:697.62Ritodrine
CAS:Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].Formula:C17H21NO3Colore e forma:SolidPeso molecolare:287.35Binedaline
CAS:Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formula:C19H23N3Purezza:98%Colore e forma:SolidPeso molecolare:293.41Dibenamine hydrochloride
CAS:<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Formula:C16H19Cl2NPurezza:96.43%Colore e forma:Oily Liquid SolidPeso molecolare:296.23Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurezza:99.73%Colore e forma:SolidPeso molecolare:555.65Pronetalol
CAS:Pronethalol ((±)-Pronethalol), a non-selective β-adrenergic antagonist, effectively inhibits Sox2 expression and offers protection against Digitalis-induced ventricular arrhythmias. Additionally, it can reverse such arrhythmias and limit the development of cerebral arteriovenous malformations (AVMs) [1] [2].Formula:C15H19NOColore e forma:SolidPeso molecolare:229.32SDZ-NVI-085
CAS:SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.Formula:C15H21NO2SColore e forma:SolidPeso molecolare:279.4Indacaterol acetate
CAS:Indacaterol acetate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C26H32N2O5Colore e forma:SolidPeso molecolare:452.54Ro-70-0004
CAS:Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.Formula:C20H24F4N4O3Colore e forma:SolidPeso molecolare:444.42Phentolamine Analogue 1
CAS:Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formula:C17H19N3OPurezza:99.96%Colore e forma:SolidPeso molecolare:281.35Ref: TM-T12444
1mg86,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)172,00€Bunazosin Hydrochloride
CAS:Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.Formula:C19H28ClN5O3Purezza:99.12%Colore e forma:SolidPeso molecolare:409.91N-5984
CAS:<p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>Formula:C20H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:391.854-hydroxy Nebivolol hydrochloride
CAS:4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.Formula:C22H25F2NO5HClColore e forma:SolidPeso molecolare:457.9(-)-Isoproterenol hydrochloride
CAS:(-)-Isoproterenol hydrochloride is used as a β-adrenergic receptor agonist in the treatment of bradycardia and as a bronchodilator.Formula:C11H17NO3·CIHColore e forma:SolidPeso molecolare:247.72BI-167107
CAS:BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).Formula:C21H26N2O4Colore e forma:SolidPeso molecolare:370.44AGN 192836
CAS:AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).Formula:C12H13N3O2Colore e forma:SolidPeso molecolare:231.25β3-AR agonist 2
CAS:β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Formula:C27H38N4O7SPurezza:98%Colore e forma:SolidPeso molecolare:562.68Bufuralol (hydrochloride)
CAS:Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.Formula:C16H24ClNO2Colore e forma:SolidPeso molecolare:297.82Todralazine hydrochloride
CAS:Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Formula:C11H13ClN4O2Purezza:99.91%Colore e forma:SolidPeso molecolare:268.7Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formula:C20H33N3O4·HClColore e forma:White Crystalline SolidPeso molecolare:415.96Bufuralol
CAS:Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Formula:C16H23NO2Purezza:98.26%Colore e forma:SolidPeso molecolare:261.36Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formula:C30H30ClN5O4SColore e forma:SolidPeso molecolare:592.11N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Formula:C20H23Cl2NO5Colore e forma:SolidPeso molecolare:428.31Indacaterol xinafoate
CAS:Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C35H36N2O6Colore e forma:SolidPeso molecolare:580.67Prenalterol hydrochloride
CAS:Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Formula:C12H20ClNO3Colore e forma:SolidPeso molecolare:261.75Deriglidole
CAS:Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Formula:C16H21N3Purezza:98.12% - 99.03%Colore e forma:SolidPeso molecolare:255.36OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purezza:99.79%Colore e forma:SolidPeso molecolare:421.58Ref: TM-T13804
1mg187,00€5mg455,00€10mg620,00€25mg940,00€50mg1.264,00€100mg1.663,00€200mg2.252,00€1mL*10mM (DMSO)567,00€CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purezza:99.40% - 99.58%Colore e forma:SolidPeso molecolare:494.46Ref: TM-T30846
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€α1 adrenoceptor-MO-1
CAS:α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Formula:C20H24ClN5OPurezza:99.20% - 99.29%Colore e forma:SolidPeso molecolare:385.89Ref: TM-T10003
1mg198,00€5mg393,00€10mg542,00€25mg785,00€50mg1.074,00€100mg1.454,00€200mg1.967,00€1mL*10mM (DMSO)467,00€Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Formula:C18H22ClNO4Purezza:99.82%Colore e forma:SolidPeso molecolare:351.83(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formula:C12H19NO3Purezza:99.73%Colore e forma:SolidPeso molecolare:225.280990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormula:C21H21N5Purezza:98.99%Colore e forma:SolidPeso molecolare:343.42Ref: TM-T13983
1mg202,00€5mg512,00€10mg740,00€25mg1.121,00€50mg1.539,00€100mg2.072,00€1mL*10mM (DMSO)535,00€Bometolol Hydrochloride
CAS:Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.Formula:C25H33ClN2O7Purezza:98%Colore e forma:SolidPeso molecolare:508.99Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Formula:C23H30N6O4Purezza:98%Colore e forma:SolidPeso molecolare:454.52Vibegron
CAS:Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Formula:C26H28N4O3Colore e forma:SolidPeso molecolare:444.53(±)-Penbutolol
CAS:(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.Formula:C18H29NO2Colore e forma:SolidPeso molecolare:291.43Sulfinalol hydrochloride
CAS:Sulfinalol hydrochloride is an orally active β-adrenoceptor (β-adrenoceptor) antagonist that exhibits direct vasodilatory activity. It is also classified as an antihypertensive agent.Formula:C20H28ClNO4SColore e forma:SolidPeso molecolare:413.96
