Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 736 prodotti per "Recettore adrenergico".
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PNMT-IN-1
PNMT-IN-1 (inhibitor 4) is a selective second generation inhibitor [1] of phenylethanolamine N-methyltransferase (PNMT), exhibiting a Ki value of 1.2 nM and anColore e forma:Odour SolidPafenolol
CAS:Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.Formula:C18H31N3O3Purezza:98.33%Colore e forma:White SolidPeso molecolare:337.46Carvedilol
CAS:Carvedilol (SKF 105517) Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. The S enantiomer of carvedilol nonselectively binds to and blocks beta-adrenergic receptors, thereby exerting negative inotropic and chronotropic effects, and leading to a reduction in cardiac output. In addition, both enantiomers of carvedilol bind to and block alpha 1-adrenergic receptors, thereby causing vasodilation and reducing peripheral vascular resistance.Formula:C24H26N2O4Purezza:99.73% - 99.97%Colore e forma:Colourless Crystalline PowderPeso molecolare:406.47CTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formula:C97H131F3I2N20O25S2Colore e forma:SolidPeso molecolare:2352.13(+)-ORM-10921
CAS:(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.Formula:C18H23NO2Purezza:99.23%Colore e forma:SolidPeso molecolare:285.38β2AR agonist 4
β2AR agonist 4 (compound A19) is an effective selective agonist for the β2-adrenoceptor (β2-Adrenoceptor), exhibiting an EC50 of 3.7 pM. In a rat model with COPD, β2AR agonist 4 reduces the elevation of inflammatory factors and leukocytes, thereby improving lung function.Formula:C19H23ClN2O5Peso molecolare:394.12955ACTH (1-14)
CAS:ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.Formula:C77H109N21O20SPurezza:98%Colore e forma:SolidPeso molecolare:1680.88CTP-347
CAS:CTP-347, a deuterated version of paroxetine, is potentially the best non-hormonal drug in its class for the treatment of hot flashes.Formula:C19H20FNO3Colore e forma:SolidPeso molecolare:331.38LM-189 free base
LM-189 free base is a G protein α subunit I (Gαi)-biased agonist and acts as a Gαi-biased ligand for the β2-adrenergic receptor (β2AR). It stabilizes a particular conformation in TM6 and enhances the dynamics of ICL2. LM-189 free base is useful for the development of Gαi-biased β2AR agonists.Colore e forma:Odour SolidNafetolol
CAS:Nafetolol (K 5407) is a biochemical reagent that can be used to synthesize other compounds.Formula:C19H29NO3Purezza:98.91%Colore e forma:SolidPeso molecolare:319.44Tizanidine
CAS:Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.Formula:C9H8ClN5SPurezza:99.11%Colore e forma:Yellow SolidPeso molecolare:253.71Azepexole hydrochloride
CAS:Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaestheticFormula:C9H16ClN3OPurezza:99.88% - 99.89%Colore e forma:Orange SolidPeso molecolare:217.7Ref: TM-T21787L
25mgPrezzo su richiesta50mgPrezzo su richiesta5mg34,00€1mL*10mM (DMSO)39,00€10mg50,00€AdTx1
Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.Formula:C310H481N87O100S8Purezza:98%Colore e forma:SolidPeso molecolare:7283.22ARC 239 dihydrochloride
CAS:ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).Formula:C24H31Cl2N3O3Purezza:99.72%Colore e forma:White SolidPeso molecolare:480.43O-Desmethyl Mebeverine alcohol hydrochloride
CAS:O-Desmethyl Mebeverine alcohol HCl, a metabolite of Mebeverine, is a strong α1 inhibitor, relaxing the GI tract.Formula:C15H26ClNO2Colore e forma:SolidPeso molecolare:287.83SU 4029 dihydrochloride
CAS:SU 4029 dihydrochloride is a bioactive chemical.Formula:C9H21Cl2N3OColore e forma:SolidPeso molecolare:258.19Formoterol O-β-D-Glucuronide
CAS:Formoterol O-β-D-glucuronide is a metabolite of formoterol .Formula:C25H32N2O10Colore e forma:SolidPeso molecolare:520.535Ivabradine-D3 hydrochloride
CAS:Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.Formula:C27H37ClN2O5Purezza:98%Colore e forma:SolidPeso molecolare:508.07Acrinor
CAS:Acrinor is a adrenergic beta receptor agonist.Formula:C35H46Cl2N10O8Purezza:98%Colore e forma:SolidPeso molecolare:805.72YM 09538
CAS:YM 09538 is a biochemical.Formula:C18H25ClN2O5SColore e forma:SolidPeso molecolare:416.92Mabuterol free base
CAS:Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.Formula:C13H18ClF3N2OPurezza:98%Colore e forma:SolidPeso molecolare:310.74allo-Yohimbine
CAS:allo-Yohimbine is a biochemical.Formula:C21H26N2O3Colore e forma:SolidPeso molecolare:354.44Deterenol hydrochloride
CAS:Deterenol hydrochloride, with CAS No. 23239-36-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Deterenol hydrochloride provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C11H18ClNO2Peso molecolare:231.72Dabelotine, (R)-
CAS:Dabelotine, (R)- is the R-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formula:C15H22N2O2Colore e forma:SolidPeso molecolare:262.35Phenylethanolamine A
CAS:Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.Formula:C19H24N2O4Colore e forma:SolidPeso molecolare:344.405-hydroxy Propranolol
CAS:5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.Formula:C16H21NO3Colore e forma:SolidPeso molecolare:275.348Benzoquinamide hydrochloride
CAS:Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemeticFormula:C22H33ClN2O5Purezza:97.13% - 99.56%Colore e forma:White SolidPeso molecolare:440.96Phenoxybenzamine
CAS:Phenoxybenzamine blocks α-1 receptors, potentially reducing neuroinflammation post brain trauma.Formula:C18H22ClNOPurezza:98%Colore e forma:SolidPeso molecolare:303.83Nolomirole
CAS:Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.Formula:C19H27NO4Colore e forma:SolidPeso molecolare:333.42AG-825
CAS:AG-825（Tyrphostin C15） is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (TyrphostinFormula:C19H15N3O3S2Purezza:99.52%Colore e forma:SolidPeso molecolare:397.47Ref: TM-T14138
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg105,00€25mg222,00€50mg371,00€100mg597,00€500mg1.234,00€Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formula:C25H26O13Colore e forma:SolidPeso molecolare:534.475-Bromoimidazo[1,2-A]Pyrazine
CAS:5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.Formula:C6H4BrN3Purezza:99.92%Colore e forma:SolidPeso molecolare:198.02Corynanthine
CAS:Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.Formula:C21H26N2O3Purezza:98%Colore e forma:SolidPeso molecolare:354.44LM-189
LM-189 is a G protein α subunit I (Gαi)-biased agonist and serves as a Gαi-biased ligand for the β2-adrenergic receptor (β2AR). It stabilizes a specific conformation in TM6 and enhances the dynamics of ICL2. LM-189 is useful for developing Gαi-biased β2AR agonists.Ethylnorepinephrine hydrochloride
CAS:Ethylnorepinephrine hydrochloride is a unique bronchodilator.Formula:C10H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:233.69Dabelotine, (S)-
CAS:Dabelotine, (S)- is the S-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formula:C15H22N2O2Colore e forma:SolidPeso molecolare:262.35(±)5(6)-EET
CAS:5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.473Metaterol
CAS:Metaterol is a bioactive chemical.Formula:C11H17NO2Colore e forma:SolidPeso molecolare:195.2582Amitraz
CAS:Prodotto controllatoAmitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.Formula:C19H23N3Purezza:99.88%Colore e forma:SolidPeso molecolare:293.41Prazobind
CAS:Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.Formula:C23H27N5O3Colore e forma:SolidPeso molecolare:421.501D-Epinephrine
CAS:D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.Formula:C9H13NO3Colore e forma:SolidPeso molecolare:183.2O-Desmethyl Mebeverine alcohol
CAS:Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.Formula:C15H25NO2Purezza:98%Colore e forma:SolidPeso molecolare:251.36(R)-(+)-Atenolol
CAS:(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.Formula:C14H22N2O3Purezza:98.72%Colore e forma:SolidPeso molecolare:266.34SB-206606
CAS:SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.Formula:C19H22ClNO4Colore e forma:SolidPeso molecolare:363.83Oxaprotiline hydrochloride
CAS:Oxaprotiline hydrochloride is an antidepressant.Formula:C20H24ClNOPurezza:98%Colore e forma:SolidPeso molecolare:329.86Desglymidodrine
CAS:Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.Formula:C10H15NO3Purezza:99.56%Colore e forma:SolidPeso molecolare:197.23Piribedil-D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purezza:98%Colore e forma:SolidPeso molecolare:306.39Clencyclohexerol-D10
CAS:Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.Formula:C14H20Cl2N2O2Colore e forma:White SolidPeso molecolare:329.29Xylometazoline hydrochloride (Standard)
CAS:Xylometazoline hydrochloride (Standard) is the standard substance of Xylometazoline hydrochloride, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.Formula:C16H24N2·HClPeso molecolare:280.844-Hydroxyatomoxetine-D3
CAS:4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.Formula:C17H21NO2Purezza:98%Colore e forma:SolidPeso molecolare:274.37
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