
Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 729 prodotti di "Recettore adrenergico"
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HEAT hydrochloride
CAS:HEAT hydrochloride is an α1-adrenoceptor antagonist.Formula:C19H22ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:331.845-Methylurapidil
CAS:5-Methylurapidil is an alpha1A-adrenoceptor antagonist.Formula:C21H31N5O3Purezza:98%Colore e forma:SolidPeso molecolare:401.5Tiamenidine
CAS:Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.Formula:C8H10ClN3SPurezza:98%Colore e forma:SolidPeso molecolare:215.7RWJ 52353
CAS:α2D adrenergic receptor agonistFormula:C11H10N2SPurezza:98%Colore e forma:SolidPeso molecolare:202.28Bucumarol (HCl)
CAS:Bucumarol is a beta-adrenergic blocking agent.Formula:C17H24ClNO4Colore e forma:SolidPeso molecolare:341.83Tiodazosin
CAS:Tiodazosin is a competitive antagonist of the postsynaptic alpha-adrenergic receptor.Formula:C18H21N7O4SPurezza:98%Colore e forma:SolidPeso molecolare:431.47A 61603
CAS:Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.Formula:C14H20BrN3O3SColore e forma:SolidPeso molecolare:390.3L 640033
CAS:L 640033 is a beta-agonist.Formula:C18H25N3OPurezza:98%Colore e forma:SolidPeso molecolare:299.41Sulfinalol
CAS:Sulfinalol is a compound that acts as an orally active β-adrenoceptor antagonist and directly induces vasodilation [1].Formula:C20H27NO4SColore e forma:SolidPeso molecolare:377.5A-123189
CAS:A-123189 is a potent, alpha1D-selective antagonist.Formula:C26H28N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:476.59(±)-Befunolol
CAS:(±)-Befunolol is a blocking agent of β-adrenoceptor.Formula:C16H21NO4Purezza:98%Colore e forma:SolidPeso molecolare:291.34(R)-Carvedilol
CAS:(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Formula:C24H26N2O4Purezza:98%Colore e forma:SolidPeso molecolare:406.47Tropodifene
CAS:Tropodifene is an inhibitor of the α-Adrenergic receptor.Formula:C25H29NO4Purezza:98%Colore e forma:SolidPeso molecolare:407.5Falintolol, (Z)-
CAS:Falintolol, (Z)-, is a novel β-adrenergic antagonist compound distinguished by the inclusion of an oxime moiety.Formula:C12H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:228.33Mezilamine
CAS:Mezilamine is an antagonist of dopamine. It also blocks presynaptic but stimulating postsynaptic alpha-adrenoceptors.Formula:C11H18ClN5SPurezza:98%Colore e forma:SolidPeso molecolare:287.81WB 4101 hydrochloride
CAS:α1A-adrenergic antagonistFormula:C19H24ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:381.85L 665871
CAS:L 665871 is used as a beta-agonist. It works as a potential swine growth promoter.Formula:C11H19N3OPurezza:98%Colore e forma:SolidPeso molecolare:209.29Amibegron hydrochloride
CAS:Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.Formula:C22H27Cl2NO4Colore e forma:SolidPeso molecolare:440.36Tetrahydrozoline nitrate
CAS:Tetrahydrozoline, an imidazoline derivative, is an α-adrenergic agonist for nasal and eye congestion studies.Formula:C13H17N3O3Colore e forma:SolidPeso molecolare:263.297Metaproterenol
CAS:Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).Formula:C11H17NO3Purezza:98%Colore e forma:SolidPeso molecolare:211.26Fenmetozole HCl
CAS:Fenmetozole HCl is an antagonist of the actions of ethanol. It attenuates the ethanol-induced reduction in cerebellar cyclic guanosine monophosphate content.Formula:C10H11Cl3N2OPurezza:98%Colore e forma:SolidPeso molecolare:281.57Ridazolol
CAS:Ridazolol is a vasodilating and cardioselective beta adrenergic blocker.Formula:C15H18Cl2N4O3Purezza:99.05%Colore e forma:SolidPeso molecolare:373.23Guanoxabenz
CAS:Guanoxabenz is an α2 adrenergic receptor agonist.Formula:C8H8Cl2N4OPurezza:98%Colore e forma:SolidPeso molecolare:247.08(S)-Carvedilol
CAS:(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Formula:C24H26N2O4Purezza:98%Colore e forma:Less Crystalline Solid Colourless Crystalline SolidPeso molecolare:406.47Detomidine
CAS:Detomidine is a nonnarcotic, synthetic α2-adrenergic agonist. Detomidine produces dose-dependent sedative and analgesic effects.Formula:C12H14N2Purezza:98%Colore e forma:White Crystalline PowderPeso molecolare:186.25SB-226552
CAS:SB-226552 is an aryloxypropanolamine selective beta3AR agonist.Formula:C25H36NO5PColore e forma:SolidPeso molecolare:461.53Undecylenoyl phenylalanine
CAS:Undecylenoyl phenylalanine (Sepiwhite msh QD) is a novel depigmenting agent, which possibly acts as an alpha-melanocyte-stimulating hormone antagonist, thus
Formula:C20H29NO3Purezza:≥98%Colore e forma:White To Pinkish Solid PowderPeso molecolare:331.45L-749372
CAS:L-749372 is the beta 3 adrenergic receptor 3-Pyridyloxypropanolamine agonist.Formula:C22H24IN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:553.41Midodrine D6 hydrochloride
CAS:Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.Formula:C12H19ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:296.78Butanserin
CAS:Butanserin is a 5-hydroxytryptamine S2-antagonist.Formula:C24H26FN3O3Purezza:98%Colore e forma:SolidPeso molecolare:423.48Methyldopa hydrochloride
CAS:L-(-)-α-Methyldopa HCl: alpha-adrenergic agonist, antihypertensive, inhibits DOPA decarboxylase.Formula:C10H14ClNO4Purezza:98%Colore e forma:SolidPeso molecolare:247.68Afurolol Hydrochloride
CAS:Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.Formula:C15H22ClNO4Purezza:98.86%Colore e forma:SolidPeso molecolare:315.79Ulimorelin
CAS:Ulimorelin, ghrelin receptor agonist (EC50: 29 nM, Ki: 16 nM), is a prokinetic and vasorelaxant via α1-adrenoceptor antagonism.Formula:C30H39FN4O4Purezza:98%Colore e forma:SolidPeso molecolare:538.65Ronactolol
CAS:Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.Formula:C20H26N2O4Colore e forma:SolidPeso molecolare:358.43Levobetaxolol
CAS:Levobetaxolol (AL-1577A/Betaxon) is a beta-blocker for ocular hypertension and glaucoma.Formula:C18H29NO3Purezza:98%Colore e forma:SolidPeso molecolare:307.43Guanfacine
CAS:Guanfacine is a selective agonist of the α2A receptor.Formula:C9H9Cl2N3OPurezza:98%Colore e forma:SolidPeso molecolare:246.09Arnolol
CAS:Arnolol, a beta blocker, slows heart rate, reduces force of beats, lowers blood pressure, and enhances blood flow.Formula:C14H23NO3Colore e forma:SolidPeso molecolare:253.34Lubabegron
CAS:Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.Formula:C29H29N3O3SColore e forma:SolidPeso molecolare:499.62Zolertine HCl
CAS:Zolertine HCl is an antagonist of alpha-Adrenoceptor.Formula:C13H19ClN6Purezza:98%Colore e forma:SolidPeso molecolare:294.78Cirazoline (free base)
CAS:Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.Formula:C13H16N2OColore e forma:SolidPeso molecolare:216.28ZD 7114 hydrochloride
CAS:β3-adrenoceptor agonistFormula:C22H31ClN2O6Purezza:98%Colore e forma:SolidPeso molecolare:454.94Protokylol
CAS:Protokylol is a β-adrenergic receptor agonist.Formula:C18H21NO5Purezza:98%Colore e forma:SolidPeso molecolare:331.36Metazosin
CAS:Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.Formula:C18H25N5O4Purezza:98%Colore e forma:SolidPeso molecolare:375.42Piribedil dihydrochloride
CAS:dopamine agonistFormula:C16H20Cl2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:371.26Todralazine
CAS:Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.Formula:C11H12N4O2Purezza:98%Colore e forma:SolidPeso molecolare:232.24BFE-55
CAS:BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptorsFormula:C14H19NO3Purezza:98%Colore e forma:SolidPeso molecolare:249.31(RS)-Butyryltimolol
CAS:(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.Formula:C17H30N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:386.51L-Alprenolol
CAS:L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.Formula:C15H23NO2Purezza:98%Colore e forma:SolidPeso molecolare:249.35Centanafadine
CAS:Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).Formula:C15H15NPurezza:98%Colore e forma:SolidPeso molecolare:209.29S(-)-Bisoprolol
CAS:S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.Formula:C18H31NO4Colore e forma:SolidPeso molecolare:325.44
