
Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 728 prodotti di "Recettore adrenergico"
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AG-825
CAS:AG-825(Tyrphostin C15) is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (TyrphostinFormula:C19H15N3O3S2Purezza:99.52%Colore e forma:Yellow SolidPeso molecolare:397.47Formoterol O-β-D-Glucuronide
CAS:Formoterol O-β-D-glucuronide is a metabolite of formoterol .Formula:C25H32N2O10Colore e forma:SolidPeso molecolare:520.535Amitraz
CAS:<p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>Formula:C19H23N3Purezza:99.88%Colore e forma:White/Pale Yellow Crystalline SolidPeso molecolare:293.41CTP-347
CAS:CTP-347, a deuterated version of paroxetine, is potentially the best non-hormonal drug in its class for the treatment of hot flashes.Formula:C19H20FNO3Peso molecolare:331.38ARC 239 dihydrochloride
CAS:<p>ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).</p>Formula:C24H31Cl2N3O3Purezza:99.72%Colore e forma:SolidPeso molecolare:480.43Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Formula:C10H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:233.69S(-)-Bisoprolol fumarate
CAS:S(-)-Bisoprolol fumarate is a selective β1-blocker for hypertension and heart research.Formula:C18H31NO4·xC4H4O4Colore e forma:SolidPeso molecolare:441.521(±)5(6)-EET
CAS:5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.473(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Formula:C14H22N2O3Purezza:98.72%Colore e forma:SolidPeso molecolare:266.34Prazobind
CAS:Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.Formula:C23H27N5O3Colore e forma:SolidPeso molecolare:421.501L-770644 dihydrochloride
CAS:L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Formula:C30H38ClN7O4SColore e forma:SolidPeso molecolare:628.19Corynanthine
CAS:Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.Formula:C21H26N2O3Purezza:98%Colore e forma:SolidPeso molecolare:354.44Carvedilol
CAS:<p>Carvedilol (SKF 105517) Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. The S enantiomer of carvedilol nonselectively binds to and blocks beta-adrenergic receptors, thereby exerting negative inotropic and chronotropic effects, and leading to a reduction in cardiac output. In addition, both enantiomers of carvedilol bind to and block alpha 1-adrenergic receptors, thereby causing vasodilation and reducing peripheral vascular resistance.</p>Formula:C24H26N2O4Purezza:99.73% - 99.97%Colore e forma:Colourless Crystalline PowderPeso molecolare:406.47YS-49 monohydrate
YS-49, a PI3K/Akt activator, curbs RhoA/PTEN; inhibits VSMC growth by inducing HO-1; an isoquinoline alkaloid that stimulates cardiac β-adrenoceptors.Formula:C20H22BrNO3Colore e forma:SolidPeso molecolare:404.3Metaraminol
CAS:Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.Formula:C9H13NO2Colore e forma:SolidPeso molecolare:167.21Phenylethanolamine A
CAS:Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.Formula:C19H24N2O4Colore e forma:SolidPeso molecolare:344.40Abediterol napadisylate
CAS:Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formula:C60H68F4N4O14S2Purezza:98%Colore e forma:SolidPeso molecolare:1209.32Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].Purezza:98%Colore e forma:Odour SolidUpidosin
CAS:<p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>Formula:C31H33N3O4Purezza:99.66%Colore e forma:SolidPeso molecolare:511.61(+)-ORM-10921
CAS:(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.Formula:C18H23NO2Purezza:99.23%Colore e forma:SoildPeso molecolare:285.38

