CaMK
Gli inibitori della Protein-Chinasi Dipendente dal Calcio/Calmodulina (CaMK) sono composti specializzati che inibiscono l'attività della CaMK, una chinasi critica coinvolta in una varietà di processi cellulari, in particolare nel sistema nervoso. La CaMK è essenziale per tradurre i segnali di calcio in varie risposte cellulari, tra cui la plasticità sinaptica, la formazione della memoria e l'espressione genica. La disregolazione dell'attività della CaMK è associata a numerosi disturbi neurologici, rendendo questi inibitori strumenti preziosi per lo studio della segnalazione sinaptica, dell'apprendimento e della memoria. Presso CymitQuimica, offriamo inibitori della CaMK di alta qualità per supportare la tua ricerca sulla plasticità sinaptica, la funzione cognitiva e la neurofarmacologia.
Trovati 66 prodotti per "CaMK".
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Calmodulin Binding Peptide 1
CAS:Calmodulin Binding Peptide 1, a high-affinity MLCK-derived inhibitor, blocks IP3-induced Ca2+ release.Formula:C231H373N69O70S2Purezza:98%Colore e forma:SolidPeso molecolare:5301.1CAMKIV Protein, Human, Recombinant (GST)
CAMKIV Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag.Colore e forma:Lyophilized PowderPeso molecolare:79 kDa (predicted); 100 kDa (reducing conditions)A-484954
CAS:A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.Formula:C13H15N5O3Purezza:97.47% - 99.86%Colore e forma:SolidPeso molecolare:289.29Ref: TM-TQ0137
1mg40,00€2mg52,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg137,00€25mg289,00€50mg515,00€100mg733,00€KN-92 hydrochloride
CAS:KN-92 hydrochloride is an inactive derivative of KN-93.Formula:C24H26Cl2N2O3SPurezza:99.68%Colore e forma:White SolidPeso molecolare:493.45KN-92
CAS:KN-92 is an inactive analog of the CaM kinase II inhibitor KN 93.Formula:C24H25ClN2O3SColore e forma:SolidPeso molecolare:456.98KN-93
CAS:KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.Formula:C26H29ClN2O4SPurezza:99.56% - 99.95%Colore e forma:White SolidPeso molecolare:501.04Ref: TM-T2697
1mg54,00€2mg74,00€5mg107,00€1mL*10mM (DMSO)120,00€10mg146,00€25mg289,00€50mg358,00€100mg523,00€Trifluoperazine
CAS:Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formula:C21H24F3N3SPurezza:98.3% - 99.98%Colore e forma:SolidPeso molecolare:407.5NH125
CAS:NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.Formula:C27H45IN2Purezza:98.60%Colore e forma:SolidPeso molecolare:524.56Ref: TM-T6605
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg113,00€25mg250,00€50mg430,00€100mg620,00€KN-62
CAS:KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.Formula:C38H35N5O6S2Purezza:99.80% - >99.99%Colore e forma:SolidPeso molecolare:721.84Ref: TM-T2694
1mg34,00€2mg49,00€5mg71,00€10mg105,00€1mL*10mM (DMSO)105,00€25mg207,00€50mg404,00€100mg592,00€CaMKII-IN-1
CAS:CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM).Formula:C29H30ClN5O2SPurezza:99.69%Colore e forma:SolidPeso molecolare:548.1Ref: TM-T14860
1mg50,00€2mg71,00€5mg113,00€1mL*10mM (DMSO)137,00€10mg166,00€25mg334,00€50mg520,00€100mg750,00€lavendustin C
CAS:lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.Formula:C14H13NO5Purezza:98.06%Colore e forma:SolidPeso molecolare:275.26Ref: TM-T4185
1mg42,00€2mg55,00€1mL*10mM (DMSO)90,00€5mg93,00€10mg152,00€25mg330,00€50mg492,00€100mg707,00€STO-609
CAS:STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.Formula:C19H10N2O3Purezza:97.14% - 99.35%Colore e forma:SolidPeso molecolare:314.29Ref: TM-T3546
1mg39,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg120,00€25mg250,00€50mg400,00€100mg620,00€200mg873,00€CaMKP Inhibitor
CAS:CaMKP Inhibitor can inhibit CaMKP.Formula:C10H8NNaO7S2Purezza:99.91% - 99.98%Colore e forma:SolidPeso molecolare:341.28Ref: TM-T2159
1mg39,00€5mg82,00€1mL*10mM (DMSO)102,00€10mg120,00€25mg227,00€50mg334,00€100mg460,00€500mg1.035,00€Stains-All
CAS:Stains-All is a cationic dye of carbocyanine.Formula:C30H27BrN2S2Purezza:98.85% - 99.71%Colore e forma:Black SolidPeso molecolare:559.58CALP2 acetate(261969-04-4 free base)
CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.Formula:C68H104N14O13SPurezza:99.91%Colore e forma:White SolidPeso molecolare:1357.7Syntide 2 acetate(108334-68-5 free base)
Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).Formula:C70H126N20O20Purezza:99.87%Colore e forma:Purple LiquidPeso molecolare:1567.85Autocamtide-2-related inhibitory peptide TFA salt
Autocamtide-2-related inhibitory peptide TFA salt(CaM kinase II inhibitor TFA salt) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.Formula:C66H117F3N22O21Purezza:>99.99%Colore e forma:SolidPeso molecolare:1611.77Autocamtide-2-related inhibitory peptide
CAS:Autocamtide-2-related inhibitory peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.Formula:C64H116N22O19Purezza:>99.99%Colore e forma:SolidPeso molecolare:1497.74Autocamtide 2 TFA(129198-88-5 free base)
Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.Formula:C67H119F3N22O22Purezza:99.86%Colore e forma:SolidPeso molecolare:1641.79GSK3i XIII
CAS:GSK3i XIII (GSK3 inhibitor XIII) is a GSK-3 ATP-binding site inhibitor.Formula:C18H19N5Purezza:98.87%Colore e forma:SolidPeso molecolare:305.38Ref: TM-T24111
1mg63,00€5mg114,00€1mL*10mM (DMSO)128,00€10mg172,00€25mg279,00€50mg406,00€100mg572,00€
