
AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 617 prodotti di "AChR"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cevimeline
CAS:Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.Formula:C10H17NOSColore e forma:Off-White SolidPeso molecolare:199.31Dexetimide
CAS:Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.Formula:C23H26N2O2Colore e forma:SolidPeso molecolare:362.46Varenicline Hydrochloride
CAS:Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).Formula:C13H14ClN3Purezza:99.854%Colore e forma:SolidPeso molecolare:247.72Cevimeline hydrochloride
CAS:Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.Formula:C10H18ClOSColore e forma:SolidPeso molecolare:235.77Glycerophosphoinositol choline
CAS:Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.Formula:C14H32NO12PColore e forma:SolidPeso molecolare:437.38(±)-Darifenacin
CAS:(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.Formula:C28H30N2O2Colore e forma:SolidPeso molecolare:426.55VU0467485
CAS:VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.Formula:C17H17FN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:360.41Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurezza:98.9%Colore e forma:SolidPeso molecolare:213.7Pirmenol hydrochloride
CAS:Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μMFormula:C22H31ClN2OColore e forma:SolidPeso molecolare:374.95Tebanicline dihydrochloride
CAS:Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.Formula:C9H13Cl3N2OColore e forma:SolidPeso molecolare:271.57SSR180711 hydrochloride
CAS:SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Formula:C14H18BrClN2O2Purezza:99.22%Colore e forma:SolidPeso molecolare:361.66(S)-(+)-Dimethindene maleate
CAS:(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFormula:C24H28N2O4Purezza:99.94%Colore e forma:SolidPeso molecolare:408.49NBTGR
CAS:NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).Formula:C17H18N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:434.43Sabcomeline hydrochloride
CAS:Sabcomeline is a selective M1 receptor partial agonist.Formula:C10H16ClN3OColore e forma:SolidPeso molecolare:229.71Biperiden
CAS:Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.Formula:C21H29NOPurezza:99.65%Colore e forma:Crystals SolidPeso molecolare:311.46Ispronicline
CAS:Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitiveFormula:C14H22N2OPurezza:97.70% - 99.16%Colore e forma:SolidPeso molecolare:234.34DL-Cystine
CAS:DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .Formula:C6H12N2O4S2Colore e forma:SolidPeso molecolare:240.3ABT-107
CAS:ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.Formula:C19H20N4OColore e forma:SolidPeso molecolare:320.396NS3861 fumarate
CAS:NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.Formula:C16H18BrNO4SColore e forma:SolidPeso molecolare:400.29NSC 23766
CAS:NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Formula:C24H35N7Purezza:99.49%Colore e forma:SolidPeso molecolare:421.58Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Formula:C40H42ClN5O7Purezza:97.94% - 98.4%Colore e forma:SolidPeso molecolare:740.24Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Formula:C14H30N2O4·2Cl·2H2OPurezza:99.87%Colore e forma:White SolidPeso molecolare:397.34Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Formula:C9H12Cl2N2OPurezza:91.74% - 98.78%Colore e forma:SolidPeso molecolare:235.11VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purezza:97.56%Colore e forma:SolidPeso molecolare:316.15KH7
CAS:KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Formula:C17H15BrN4O2SPurezza:98.43%Colore e forma:SolidPeso molecolare:419.3Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formula:C17H17N5O6SPurezza:99.69% - 99.74%Colore e forma:Off-White SolidPeso molecolare:419.41VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Formula:C18H28ClN3O3Purezza:99% - 99.97%Colore e forma:SolidPeso molecolare:369.89Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Formula:C21H26ClNO2Purezza:99.5%Colore e forma:SolidPeso molecolare:359.89VU0152100
CAS:<p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>Formula:C18H19N3O2SPurezza:99.56%Colore e forma:SolidPeso molecolare:341.43NS9283
CAS:<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Formula:C14H8N4OPurezza:99.12%Colore e forma:SolidPeso molecolare:248.24ML380
CAS:<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Formula:C23H25F3N4O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:494.53α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formula:C69H107N23O24S4Purezza:94.82% - 97.79%Colore e forma:SolidPeso molecolare:1770.99Isopropamide Iodide
CAS:<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Formula:C23H33IN2OPurezza:99.67%Colore e forma:SolidPeso molecolare:480.43Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurezza:99.76% - >99.99%Colore e forma:White SolidPeso molecolare:203.75Nitenpyram
CAS:<p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>Formula:C11H15ClN4O2Purezza:99.03%Colore e forma:Light-Yellow CrystalPeso molecolare:270.72Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Formula:C6H8ClN5O2SPurezza:99.71% - 99.87%Colore e forma:Solid PowderPeso molecolare:249.68VU0467154
CAS:VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Formula:C17H15F3N4O3S2Purezza:99.51% - 99.53%Colore e forma:SolidPeso molecolare:444.45Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formula:C19H29N5O3·2(C2H4O2)Purezza:99.60%Colore e forma:SolidPeso molecolare:495.58Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurezza:99.20%Colore e forma:SolidPeso molecolare:320.84Mc-Val-Ala-PAB
CAS:<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Formula:C25H34N4O6Purezza:98.34% - 99.24%Colore e forma:SolidPeso molecolare:486.56PSEM 89S TFA
CAS:<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Formula:C18H23F3N2O5Purezza:99.9%Colore e forma:SolidPeso molecolare:404.38Solifenacin hydrochloride
CAS:Solifenacin Hcl is a muscarinic receptor antagonist.Formula:C23H27ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:398.93Oxyphencyclimine Hydrochloride
CAS:<p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>Formula:C20H29ClN2O3Purezza:99.55%Colore e forma:SolidPeso molecolare:380.91Mecamylamine
CAS:<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Formula:C11H21NColore e forma:SolidPeso molecolare:167.29Sofpironium bromide
CAS:<p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>Formula:C22H32BrNO5Purezza:98.85%Colore e forma:SolidPeso molecolare:470.4Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formula:C10H21NPurezza:98.18% - 99.28%Colore e forma:Colorless - Light Yellow Clear LiquidPeso molecolare:155.28Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purezza:99.89%Colore e forma:White Crystalline PowderPeso molecolare:202.21Propiverine
CAS:Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.Formula:C23H29NO3Colore e forma:SolidPeso molecolare:367.48NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Formula:C14H9Cl2F3N2O2Purezza:99.11%Colore e forma:SolidPeso molecolare:365.13Varenicline Tartrate
CAS:<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Formula:C13H13N3·C4H6O6Purezza:98.23% - 98.32%Colore e forma:Tan SolidPeso molecolare:361.35Oxyphenonium bromide
CAS:<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Formula:C21H34BrNO3Purezza:98.96%Colore e forma:SolidPeso molecolare:428.404Dronedarone
CAS:<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Formula:C31H44N2O5SPurezza:98.85% - 99.58%Colore e forma:SolidPeso molecolare:556.76EB-3D
CAS:EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Formula:C30H36Br2N4O2Purezza:99.48%Colore e forma:SolidPeso molecolare:644.4Propantheline
CAS:Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Formula:C23H30NO3Colore e forma:SolidPeso molecolare:368.49MC-Val-Cit-PABC-PNP
CAS:MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.Formula:C35H43N7O11Purezza:97.2% - 98.055%Colore e forma:SolidPeso molecolare:737.76Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Formula:C16H19N3O5Purezza:99.76%Colore e forma:SolidPeso molecolare:333.34Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Formula:C10H22ClNColore e forma:SolidPeso molecolare:191.74Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Formula:C12H16N2O4Purezza:98%Colore e forma:SolidPeso molecolare:207.23VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurezza:98.46%Colore e forma:SolidPeso molecolare:355.41Adiphenine
CAS:Adiphenine is an inhibitor of nicotinic receptors.Formula:C20H25NO2Colore e forma:SolidPeso molecolare:311.42Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Formula:C19H23N3O3Purezza:99.96%Colore e forma:SolidPeso molecolare:341.4Aclidinium bromide
CAS:<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Formula:C26H30NO4S2·BrPurezza:99.53% - 99.69%Colore e forma:SolidPeso molecolare:564.55Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H17ClN2OS·HClPurezza:98.34% - 99.85%Colore e forma:SolidPeso molecolare:357.3suvn-911
CAS:suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.Formula:C11H14Cl2N2OPurezza:98.88%Colore e forma:SolidPeso molecolare:261.15JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Formula:C19H20ClFN4Purezza:99.72%Colore e forma:SolidPeso molecolare:358.84Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Formula:C29H34BrNO2Purezza:98.4% - 99.89%Colore e forma:SolidPeso molecolare:508.49VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Formula:C16H9ClF3NO2Purezza:100%Colore e forma:SolidPeso molecolare:339.7(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Formula:C13H17NO2Colore e forma:SolidPeso molecolare:219.284Oxyphencyclimine
CAS:Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.Formula:C20H28N2O3Colore e forma:SolidPeso molecolare:344.45mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Formula:C23H26ClIN2O2Purezza:99.87%Colore e forma:SolidPeso molecolare:524.82Benzetimide hydrochloride
CAS:Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Formula:C23H27ClN2O2Purezza:99.32%Colore e forma:Off-White PowderPeso molecolare:398.93Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formula:C44H48ClN5O11Colore e forma:SolidPeso molecolare:858.34Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formula:C23H26N2O2Purezza:99.87%Colore e forma:SolidPeso molecolare:362.46Pirmenol
CAS:Pirmenol is a new antiarrhythmic drugFormula:C22H30N2OPurezza:97.24%Colore e forma:SolidPeso molecolare:338.49LY2119620
CAS:LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Formula:C19H24ClN5O3SPurezza:99.7%Colore e forma:SolidPeso molecolare:437.94Cyclodrine hydrochloride
CAS:Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study ofFormula:C19H30ClNO3Purezza:98.59%Colore e forma:SolidPeso molecolare:355.9Ilmetropium iodide
CAS:Ilmetropium iodide is a bronchodilator.Formula:C20H30INO3Purezza:98.45%Colore e forma:SolidPeso molecolare:459.36Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Formula:C28H30N2O2Purezza:99.78%Colore e forma:SolidPeso molecolare:426.55BNC210
CAS:BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.Formula:C17H23N3O3Purezza:97.05% - >99.99%Colore e forma:SolidPeso molecolare:317.38Brompheniramine
CAS:Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formula:C16H19BrN2Colore e forma:SolidPeso molecolare:319.24Harman hydrochloride
CAS:Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.Formula:C12H11ClN2Purezza:99.35%Colore e forma:SolidPeso molecolare:218.68Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Formula:C16H20N2O2Purezza:98.63%Colore e forma:SolidPeso molecolare:272.34Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Formula:C24H40O10S2Purezza:98%Colore e forma:SolidPeso molecolare:552.7W-84 dibromide
CAS:<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Formula:C32H44Br2N4O4Purezza:95.56%Colore e forma:SolidPeso molecolare:708.52Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formula:C18H27ClN2O4Purezza:99.74%Colore e forma:SolidPeso molecolare:370.87CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Formula:C19H15Cl2N3O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:388.25SEN12333
CAS:<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Formula:C20H25N3O2Purezza:99.02%Colore e forma:SolidPeso molecolare:339.43Glycopyrrolate
CAS:Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Formula:C19H28BrNO3Purezza:99.41% - 99.64%Colore e forma:SolidPeso molecolare:398.339-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purezza:99.35% - 99.37%Colore e forma:SolidPeso molecolare:163.184BP-TQS
CAS:4BP-TQS is an allosteric agonist of α7 nAChRs.Formula:C18H17BrN2O2SPurezza:99.96%Colore e forma:SolidPeso molecolare:405.31PNU-282987 S enantiomer free base
CAS:PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Formula:C14H17ClN2OPurezza:99.74%Colore e forma:SolidPeso molecolare:264.75BQCA
CAS:<p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>Formula:C18H15NO4Purezza:97.22%Colore e forma:SolidPeso molecolare:309.32TBPB
CAS:<p>TBPB is an allosteric M1 mAChR agonist.</p>Formula:C25H32N4OPurezza:97.87% - 99.9%Colore e forma:SolidPeso molecolare:404.55Piperidolate
CAS:Piperidolate inhibits intestinal cramp induced by acetylcholineFormula:C21H25NO2Purezza:98.45%Colore e forma:SolidPeso molecolare:323.43Dicyclomine
CAS:Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.Formula:C19H35NO2Colore e forma:SolidPeso molecolare:309.49A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Formula:C17H21ClN4Purezza:99.83%Colore e forma:SolidPeso molecolare:316.83DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Formula:C19H23Cl2N3Purezza:99.91%Colore e forma:SolidPeso molecolare:364.31Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purezza:98.12%Colore e forma:SolidPeso molecolare:597.75Ethyl (triphenylphosphoranylidene) acetate
CAS:<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Formula:C22H21O2PPurezza:97.985%Colore e forma:White Or Slight Yellow PowderPeso molecolare:348.37Fesoterodine
CAS:Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.Formula:C26H37NO3Purezza:97.1%Colore e forma:SolidPeso molecolare:411.58
