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AChR

AChR

Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.

Trovati 617 prodotti di "AChR"

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  • Cevimeline

    CAS:
    Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.
    Formula:C10H17NOS
    Colore e forma:Off-White Solid
    Peso molecolare:199.31
  • Dexetimide

    CAS:
    Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.
    Formula:C23H26N2O2
    Colore e forma:Solid
    Peso molecolare:362.46
  • Varenicline Hydrochloride

    CAS:
    Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).
    Formula:C13H14ClN3
    Purezza:99.854%
    Colore e forma:Solid
    Peso molecolare:247.72
  • Cevimeline hydrochloride

    CAS:
    Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.
    Formula:C10H18ClOS
    Colore e forma:Solid
    Peso molecolare:235.77
  • Glycerophosphoinositol choline

    CAS:
    Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.
    Formula:C14H32NO12P
    Colore e forma:Solid
    Peso molecolare:437.38
  • (±)-Darifenacin

    CAS:
    (±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.
    Formula:C28H30N2O2
    Colore e forma:Solid
    Peso molecolare:426.55
  • VU0467485

    CAS:
    VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.
    Formula:C17H17FN4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:360.41
  • Clorprenaline

    CAS:
    Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.
    Formula:C11H16ClNO
    Purezza:98.9%
    Colore e forma:Solid
    Peso molecolare:213.7
  • Pirmenol hydrochloride

    CAS:
    Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM
    Formula:C22H31ClN2O
    Colore e forma:Solid
    Peso molecolare:374.95
  • Tebanicline dihydrochloride

    CAS:
    Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.
    Formula:C9H13Cl3N2O
    Colore e forma:Solid
    Peso molecolare:271.57
  • SSR180711 hydrochloride

    CAS:
    SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.
    Formula:C14H18BrClN2O2
    Purezza:99.22%
    Colore e forma:Solid
    Peso molecolare:361.66
  • (S)-(+)-Dimethindene maleate

    CAS:
    (S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors
    Formula:C24H28N2O4
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:408.49
  • NBTGR

    CAS:
    NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
    Formula:C17H18N6O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:434.43
  • Sabcomeline hydrochloride

    CAS:
    Sabcomeline is a selective M1 receptor partial agonist.
    Formula:C10H16ClN3O
    Colore e forma:Solid
    Peso molecolare:229.71
  • Biperiden

    CAS:
    Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.
    Formula:C21H29NO
    Purezza:99.65%
    Colore e forma:Crystals Solid
    Peso molecolare:311.46
  • Ispronicline

    CAS:
    Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitive
    Formula:C14H22N2O
    Purezza:97.70% - 99.16%
    Colore e forma:Solid
    Peso molecolare:234.34
  • DL-Cystine

    CAS:
    DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .
    Formula:C6H12N2O4S2
    Colore e forma:Solid
    Peso molecolare:240.3
  • ABT-107

    CAS:
    ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.
    Formula:C19H20N4O
    Colore e forma:Solid
    Peso molecolare:320.396
  • NS3861 fumarate

    CAS:
    NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.
    Formula:C16H18BrNO4S
    Colore e forma:Solid
    Peso molecolare:400.29
  • NSC 23766

    CAS:
    NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.
    Formula:C24H35N7
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:421.58
  • Batefenterol

    CAS:
    <p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>
    Formula:C40H42ClN5O7
    Purezza:97.94% - 98.4%
    Colore e forma:Solid
    Peso molecolare:740.24
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Formula:C14H30N2O4·2Cl·2H2O
    Purezza:99.87%
    Colore e forma:White Solid
    Peso molecolare:397.34
  • Tebanicline hydrochloride

    CAS:
    Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.
    Formula:C9H12Cl2N2O
    Purezza:91.74% - 98.78%
    Colore e forma:Solid
    Peso molecolare:235.11
  • VU0119498

    CAS:
    VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.
    Formula:C15H10BrNO2
    Purezza:97.56%
    Colore e forma:Solid
    Peso molecolare:316.15
  • KH7

    CAS:
    KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.
    Formula:C17H15BrN4O2S
    Purezza:98.43%
    Colore e forma:Solid
    Peso molecolare:419.3
  • Nitrobenzylthioinosine

    CAS:
    <p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>
    Formula:C17H17N5O6S
    Purezza:99.69% - 99.74%
    Colore e forma:Off-White Solid
    Peso molecolare:419.41
  • VU0357017 hydrochloride

    CAS:
    VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.
    Formula:C18H28ClN3O3
    Purezza:99% - 99.97%
    Colore e forma:Solid
    Peso molecolare:369.89
  • Piperidolate hydrochloride

    CAS:
    Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.
    Formula:C21H26ClNO2
    Purezza:99.5%
    Colore e forma:Solid
    Peso molecolare:359.89
  • VU0152100

    CAS:
    <p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>
    Formula:C18H19N3O2S
    Purezza:99.56%
    Colore e forma:Solid
    Peso molecolare:341.43
  • NS9283

    CAS:
    <p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>
    Formula:C14H8N4O
    Purezza:99.12%
    Colore e forma:Solid
    Peso molecolare:248.24
  • ML380

    CAS:
    <p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>
    Formula:C23H25F3N4O3S
    Purezza:99.69%
    Colore e forma:Solid
    Peso molecolare:494.53
  • α-Conotoxin MII acetate


    α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.
    Formula:C69H107N23O24S4
    Purezza:94.82% - 97.79%
    Colore e forma:Solid
    Peso molecolare:1770.99
  • Isopropamide Iodide

    CAS:
    <p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>
    Formula:C23H33IN2O
    Purezza:99.67%
    Colore e forma:Solid
    Peso molecolare:480.43
  • Mecamylamine hydrochloride

    CAS:
    Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.
    Formula:C11H22ClN
    Purezza:99.76% - >99.99%
    Colore e forma:White Solid
    Peso molecolare:203.75
  • Nitenpyram

    CAS:
    <p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>
    Formula:C11H15ClN4O2
    Purezza:99.03%
    Colore e forma:Light-Yellow Crystal
    Peso molecolare:270.72
  • Clothianidin

    CAS:
    Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.
    Formula:C6H8ClN5O2S
    Purezza:99.71% - 99.87%
    Colore e forma:Solid Powder
    Peso molecolare:249.68
  • VU0467154

    CAS:
    VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.
    Formula:C17H15F3N4O3S2
    Purezza:99.51% - 99.53%
    Colore e forma:Solid
    Peso molecolare:444.45
  • Syn-Ake acetate

    CAS:
    Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.
    Formula:C19H29N5O3·2(C2H4O2)
    Purezza:99.60%
    Colore e forma:Solid
    Peso molecolare:495.58
  • Encenicline

    CAS:
    Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.
    Formula:C16H17ClN2OS
    Purezza:99.20%
    Colore e forma:Solid
    Peso molecolare:320.84
  • Mc-​Val-​Ala-​PAB

    CAS:
    <p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>
    Formula:C25H34N4O6
    Purezza:98.34% - 99.24%
    Colore e forma:Solid
    Peso molecolare:486.56
  • PSEM 89S TFA

    CAS:
    <p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>
    Formula:C18H23F3N2O5
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:404.38
  • Solifenacin hydrochloride

    CAS:
    Solifenacin Hcl is a muscarinic receptor antagonist.
    Formula:C23H27ClN2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:398.93
  • Oxyphencyclimine Hydrochloride

    CAS:
    <p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>
    Formula:C20H29ClN2O3
    Purezza:99.55%
    Colore e forma:Solid
    Peso molecolare:380.91
  • Mecamylamine

    CAS:
    <p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>
    Formula:C11H21N
    Colore e forma:Solid
    Peso molecolare:167.29
  • Sofpironium bromide

    CAS:
    <p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>
    Formula:C22H32BrNO5
    Purezza:98.85%
    Colore e forma:Solid
    Peso molecolare:470.4
  • Pempidine

    CAS:
    Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.
    Formula:C10H21N
    Purezza:98.18% - 99.28%
    Colore e forma:Colorless - Light Yellow Clear Liquid
    Peso molecolare:155.28
  • Dinotefuran

    CAS:
    Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.
    Formula:C7H14N4O3
    Purezza:99.89%
    Colore e forma:White Crystalline Powder
    Peso molecolare:202.21
  • Propiverine

    CAS:
    Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.
    Formula:C23H29NO3
    Colore e forma:Solid
    Peso molecolare:367.48
  • NS 1738

    CAS:
    NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)
    Formula:C14H9Cl2F3N2O2
    Purezza:99.11%
    Colore e forma:Solid
    Peso molecolare:365.13
  • Varenicline Tartrate

    CAS:
    <p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>
    Formula:C13H13N3·C4H6O6
    Purezza:98.23% - 98.32%
    Colore e forma:Tan Solid
    Peso molecolare:361.35
  • Oxyphenonium bromide

    CAS:
    <p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>
    Formula:C21H34BrNO3
    Purezza:98.96%
    Colore e forma:Solid
    Peso molecolare:428.404
  • Dronedarone

    CAS:
    <p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>
    Formula:C31H44N2O5S
    Purezza:98.85% - 99.58%
    Colore e forma:Solid
    Peso molecolare:556.76
  • EB-3D

    CAS:
    EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.
    Formula:C30H36Br2N4O2
    Purezza:99.48%
    Colore e forma:Solid
    Peso molecolare:644.4
  • Propantheline

    CAS:
    Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.
    Formula:C23H30NO3
    Colore e forma:Solid
    Peso molecolare:368.49
  • MC-Val-Cit-PABC-PNP

    CAS:
    MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.
    Formula:C35H43N7O11
    Purezza:97.2% - 98.055%
    Colore e forma:Solid
    Peso molecolare:737.76
  • Bestim

    CAS:
    Bestim is an immunomodulatory dipeptide that is synthetic.
    Formula:C16H19N3O5
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:333.34
  • Pempidine HCl

    CAS:
    Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.
    Formula:C10H22ClN
    Colore e forma:Solid
    Peso molecolare:191.74
  • Rivanicline hemioxalate


    <p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>
    Formula:C12H16N2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:207.23
  • VU0152099

    CAS:
    VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
    Formula:C18H17N3O3S
    Purezza:98.46%
    Colore e forma:Solid
    Peso molecolare:355.41
  • Adiphenine

    CAS:
    Adiphenine is an inhibitor of nicotinic receptors.
    Formula:C20H25NO2
    Colore e forma:Solid
    Peso molecolare:311.42
  • Coluracetam

    CAS:
    Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.
    Formula:C19H23N3O3
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:341.4
  • Aclidinium bromide

    CAS:
    <p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>
    Formula:C26H30NO4S2·Br
    Purezza:99.53% - 99.69%
    Colore e forma:Solid
    Peso molecolare:564.55
  • Encenicline hydrochloride

    CAS:
    Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).
    Formula:C16H17ClN2OS·HCl
    Purezza:98.34% - 99.85%
    Colore e forma:Solid
    Peso molecolare:357.3
  • suvn-911

    CAS:
    suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.
    Formula:C11H14Cl2N2O
    Purezza:98.88%
    Colore e forma:Solid
    Peso molecolare:261.15
  • JHU37152

    CAS:
    JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.
    Formula:C19H20ClFN4
    Purezza:99.72%
    Colore e forma:Solid
    Peso molecolare:358.84
  • Umeclidinium bromide

    CAS:
    Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.
    Formula:C29H34BrNO2
    Purezza:98.4% - 99.89%
    Colore e forma:Solid
    Peso molecolare:508.49
  • VU0238441

    CAS:
    VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.
    Formula:C16H9ClF3NO2
    Purezza:100%
    Colore e forma:Solid
    Peso molecolare:339.7
  • (S)-UFR2709

    CAS:
    (S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.
    Formula:C13H17NO2
    Colore e forma:Solid
    Peso molecolare:219.284
  • Oxyphencyclimine

    CAS:
    Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.
    Formula:C20H28N2O3
    Colore e forma:Solid
    Peso molecolare:344.45
  • mAChR-IN-1 hydrochloride

    CAS:
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
    Formula:C23H26ClIN2O2
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:524.82
  • Benzetimide hydrochloride

    CAS:
    Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.
    Formula:C23H27ClN2O2
    Purezza:99.32%
    Colore e forma:Off-White Powder
    Peso molecolare:398.93
  • Batefenterol Succinate

    CAS:
    Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.
    Formula:C44H48ClN5O11
    Colore e forma:Solid
    Peso molecolare:858.34
  • Solifenacin

    CAS:
    Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,
    Formula:C23H26N2O2
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:362.46
  • Pirmenol

    CAS:
    Pirmenol is a new antiarrhythmic drug
    Formula:C22H30N2O
    Purezza:97.24%
    Colore e forma:Solid
    Peso molecolare:338.49
  • LY2119620

    CAS:
    LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
    Formula:C19H24ClN5O3S
    Purezza:99.7%
    Colore e forma:Solid
    Peso molecolare:437.94
  • Cyclodrine hydrochloride

    CAS:
    Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of
    Formula:C19H30ClNO3
    Purezza:98.59%
    Colore e forma:Solid
    Peso molecolare:355.9
  • Ilmetropium iodide

    CAS:
    Ilmetropium iodide is a bronchodilator.
    Formula:C20H30INO3
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:459.36
  • Darifenacin

    CAS:
    Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.
    Formula:C28H30N2O2
    Purezza:99.78%
    Colore e forma:Solid
    Peso molecolare:426.55
  • BNC210

    CAS:
    BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.
    Formula:C17H23N3O3
    Purezza:97.05% - >99.99%
    Colore e forma:Solid
    Peso molecolare:317.38
  • Brompheniramine

    CAS:
    Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.
    Formula:C16H19BrN2
    Colore e forma:Solid
    Peso molecolare:319.24
  • Harman hydrochloride

    CAS:
    Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.
    Formula:C12H11ClN2
    Purezza:99.35%
    Colore e forma:Solid
    Peso molecolare:218.68
  • Nor-benzetimide

    CAS:
    Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.
    Formula:C16H20N2O2
    Purezza:98.63%
    Colore e forma:Solid
    Peso molecolare:272.34
  • Ursulcholic acid

    CAS:
    Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
    Formula:C24H40O10S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:552.7
  • W-84 dibromide

    CAS:
    <p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>
    Formula:C32H44Br2N4O4
    Purezza:95.56%
    Colore e forma:Solid
    Peso molecolare:708.52
  • Nitrocaramiphen hydrochloride

    CAS:
    Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.
    Formula:C18H27ClN2O4
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:370.87
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Formula:C19H15Cl2N3O2
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:388.25
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Formula:C20H25N3O2
    Purezza:99.02%
    Colore e forma:Solid
    Peso molecolare:339.43
  • Glycopyrrolate

    CAS:
    Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.
    Formula:C19H28BrNO3
    Purezza:99.41% - 99.64%
    Colore e forma:Solid
    Peso molecolare:398.33
  • 9-Ethyladenine

    CAS:
    9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].
    Formula:C7H9N5
    Purezza:99.35% - 99.37%
    Colore e forma:Solid
    Peso molecolare:163.18
  • 4BP-TQS

    CAS:
    4BP-TQS is an allosteric agonist of α7 nAChRs.
    Formula:C18H17BrN2O2S
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:405.31
  • PNU-282987 S enantiomer free base

    CAS:
    PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
    Formula:C14H17ClN2O
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:264.75
  • BQCA

    CAS:
    <p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>
    Formula:C18H15NO4
    Purezza:97.22%
    Colore e forma:Solid
    Peso molecolare:309.32
  • TBPB

    CAS:
    <p>TBPB is an allosteric M1 mAChR agonist.</p>
    Formula:C25H32N4O
    Purezza:97.87% - 99.9%
    Colore e forma:Solid
    Peso molecolare:404.55
  • Piperidolate

    CAS:
    Piperidolate inhibits intestinal cramp induced by acetylcholine
    Formula:C21H25NO2
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:323.43
  • Dicyclomine

    CAS:
    Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.
    Formula:C19H35NO2
    Colore e forma:Solid
    Peso molecolare:309.49
  • A 582941 HCl (848591-90-2(free base))


    <p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>
    Formula:C17H21ClN4
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:316.83
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Formula:C19H23Cl2N3
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:364.31
  • Revefenacin

    CAS:
    Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.
    Formula:C35H43N5O4
    Purezza:98.12%
    Colore e forma:Solid
    Peso molecolare:597.75
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Formula:C22H21O2P
    Purezza:97.985%
    Colore e forma:White Or Slight Yellow Powder
    Peso molecolare:348.37
  • Fesoterodine

    CAS:
    Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.
    Formula:C26H37NO3
    Purezza:97.1%
    Colore e forma:Solid
    Peso molecolare:411.58