AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 617 prodotti di "AChR"
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Ethybenztropine HCl
CAS:Ethybenztropine HCl is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.Formula:C22H28ClNOColore e forma:SolidPeso molecolare:357.92Esoxybutynin Chloride
CAS:(S)-oxybutynin, with antimuscarinic effects, is being developed for urinary incontinence.Formula:C22H32ClNO3Colore e forma:SolidPeso molecolare:393.95AR-R 17779 hydrochloride
CAS:AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.Formula:C9H15ClN2O2Colore e forma:SolidPeso molecolare:218.68Elucaine
CAS:Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.Formula:C19H23NO2Purezza:98%Colore e forma:SolidPeso molecolare:297.39(R,R)-Glycopyrrolate
CAS:(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.Formula:C19H28BrNO3Purezza:98%Colore e forma:SolidPeso molecolare:398.34SIB 1508Y maleate
CAS:neuronal nicotinic ACh receptor agonistFormula:C16H18N2O4Purezza:98%Colore e forma:SolidPeso molecolare:302.33LRE1
CAS:<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Formula:C12H13ClN4SPurezza:>99.99%Colore e forma:SolidPeso molecolare:280.78Terodiline
CAS:Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.Formula:C20H27NPurezza:98.20% - 99.59%Colore e forma:SolidPeso molecolare:281.44Methacholine bromide
CAS:<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Formula:C8H18BrNO2Colore e forma:SolidPeso molecolare:240.141Nuvenzepine
CAS:Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.Formula:C19H20N4O2Purezza:98%Colore e forma:SolidPeso molecolare:336.39DA 4626
CAS:DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.Formula:C14H18N4Purezza:98%Colore e forma:SolidPeso molecolare:242.32PQCA
CAS:<p>PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.</p>Formula:C22H20N4O3Purezza:99.88%Colore e forma:SolidPeso molecolare:388.42Telenzepine
CAS:Telenzepine is a potent and selective M1 antimuscarinic.Formula:C19H22N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:370.47AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Formula:C20H29FN2O2Colore e forma:SolidPeso molecolare:348.45Neramexane Mesylate
CAS:<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Formula:C12H27NO3SPurezza:98%Colore e forma:SolidPeso molecolare:265.41ML381
CAS:ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.Formula:C21H21N3O4Colore e forma:SolidPeso molecolare:379.41ML169
CAS:ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).Formula:C21H17BrFN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:506.34Zamifenacin
CAS:Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.Formula:C27H29NO3Purezza:98%Colore e forma:SolidPeso molecolare:415.52BNC375
CAS:BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).Formula:C19H23ClN2O3SPurezza:98%Colore e forma:SolidPeso molecolare:394.92(R,R)-Reboxetine mesylate
CAS:(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.Formula:C20H27NO6SColore e forma:SolidPeso molecolare:409.5M1 ligand 1
CAS:Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.Formula:C20H21NO2Colore e forma:SolidPeso molecolare:307.39Benzatropine
CAS:Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.Formula:C21H25NOPurezza:98%Colore e forma:SolidPeso molecolare:307.43Penehyclidine hydrochloride
CAS:<p>Penehyclidine hydrochloride: M1/M3 antagonist, activates NF-κB, anti-inflammatory, anticholinergic.</p>Formula:C20H30ClNO2Purezza:99.79%Colore e forma:SolidPeso molecolare:351.91Muscarine iodide
CAS:Muscarinic acetylcholine receptor agonistFormula:C9H20INO2Purezza:98%Colore e forma:SolidPeso molecolare:301.17Tridihexethyl chloride
CAS:Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.Formula:C21H36ClNOColore e forma:SolidPeso molecolare:353.97TC 2559 difumarate
CAS:partial agonist of α4β2 nicotinic acetylcholine receptorFormula:C12H18N2OC4H404Purezza:98%Colore e forma:SolidPeso molecolare:380.39TC299423
CAS:TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.Formula:C11H15N3Colore e forma:SolidPeso molecolare:189.26SM-21 maleate
CAS:Increases release of acetylcholine,σ2 antagonistFormula:C22H28ClNO7Purezza:98%Colore e forma:SolidPeso molecolare:453.91Sulfoxaflor
CAS:Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.Formula:C10H10F3N3OSPurezza:99.56%Colore e forma:SolidPeso molecolare:277.27TC 1698 dihydrochloride
CAS:nicotinic α7 receptor agonistFormula:C13H18N2Purezza:98%Colore e forma:SolidPeso molecolare:202.3Beperidium iodide
CAS:Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).Formula:C23H34IN3O3Colore e forma:SolidPeso molecolare:527.44WIN 62,577
CAS:WIN 62,577 is a allosteric antagonist of mAChR.Formula:C29H31N3OPurezza:98%Colore e forma:SolidPeso molecolare:437.58SIB-1553A hydrochloride
CAS:SIB-1553A hydrochloride is a nicotinic acetylcholine receptor agonist and a selective neuronal nAChR ligandFormula:C13H20ClNOSPurezza:99.56% - 99.73%Colore e forma:SolidPeso molecolare:273.82Benzamide Derivative 1
CAS:Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.Formula:C22H34ClN3O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:423.98Alvameline
CAS:Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.Formula:C9H15N5Purezza:98%Colore e forma:SolidPeso molecolare:193.25Muscarine chloride
CAS:Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.Formula:C9H20ClNO2Colore e forma:SolidPeso molecolare:209.71Quifenadine
CAS:Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.Formula:C20H23NOPurezza:98%Colore e forma:SolidPeso molecolare:293.4DAU 5884 hydrochloride
CAS:muscarinic M3 receptor antagonistFormula:C17H22ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:351.83Nelonicline
CAS:Nelonicline is a selective agonist of neuronal nicotinic receptors.Formula:C17H19N3OSPurezza:98%Colore e forma:SolidPeso molecolare:313.42Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurezza:99.67%Colore e forma:White Crystalline PowderPeso molecolare:322.83PF-03635659
CAS:PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.Formula:C28H32N2O3Purezza:98.39% - 99.85%Colore e forma:SolidPeso molecolare:444.57NKY80
CAS:NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.Formula:C12H11N3O2Purezza:99.88%Colore e forma:SolidPeso molecolare:229.23rel-(1R,2R)-Vesamicol Hydrochloride
CAS:rel-(1R,2R)-Vesamicol Hydrochloride is a acetylcholine transport inhibitor.Formula:C17H26ClNOPurezza:99.88%Colore e forma:SolidPeso molecolare:295.85Desformylflustrabromine hydrochloride
CAS:Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.Formula:C17H12INO5Purezza:99.79%Colore e forma:SolidPeso molecolare:437.19Temiverine hydrochloride
CAS:Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.Formula:C24H36ClNO3Purezza:99.26% - 99.43%Colore e forma:SolidPeso molecolare:422ASM-024
CAS:ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.Formula:C15H25N2Purezza:99.74%Colore e forma:SolidPeso molecolare:233.37Posatirelin
CAS:Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.Formula:C17H28N4O4Purezza:99.43% - 99.95%Colore e forma:SolidPeso molecolare:352.43Oxotremorine M iodide
CAS:Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.Formula:C11H19IN2OPurezza:99.57%Colore e forma:SolidPeso molecolare:322.19JNJ-39393406
CAS:JNJ-39393406 is an α7 nicotinic acetylcholine receptor positive allosteric modulator for the study of tobacco dependence and Alzheimer's disease.Formula:C19H18F2N6O3Purezza:98.5%Colore e forma:SolidPeso molecolare:416.38Xanomeline
CAS:<p>Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.</p>Formula:C14H23N3OSPurezza:99.61%Colore e forma:SolidPeso molecolare:281.42NB001
CAS:NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.Formula:C12H20N6OPurezza:99.69%Colore e forma:Off-White To Pale Pink SolidPeso molecolare:264.33AQW051
CAS:AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.Formula:C19H22N2OPurezza:99.94%Colore e forma:SolidPeso molecolare:294.39Aceclidine
CAS:Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocularFormula:C9H15NO2Purezza:>99.99%Colore e forma:SolidPeso molecolare:169.22Tribendimidine
CAS:<p>Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.</p>Formula:C28H32N6Purezza:≥98%Colore e forma:SolidPeso molecolare:452.59McN-A 343
CAS:<p>McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.</p>Formula:C14H18Cl2N2O2Purezza:99.65%Colore e forma:SolidPeso molecolare:317.21Xanomeline oxalate
CAS:Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.Formula:C16H25N3O5SPurezza:99.1%Colore e forma:SolidPeso molecolare:371.45SCH-900271
CAS:SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.Formula:C14H16N2O4Purezza:98.82% - 99.93%Colore e forma:SolidPeso molecolare:276.29Iperoxo
CAS:Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.Formula:C10H17IN2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:324.16Otenzepad
CAS:Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Formula:C24H31N5O2Purezza:99.79%Colore e forma:SolidPeso molecolare:421.54PHA 543613
CAS:PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.Formula:C15H17N3O2Purezza:99.43% - 99.96%Colore e forma:SolidPeso molecolare:271.31GSK233705
CAS:GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.Formula:C24H29BrN2Purezza:99.87% - 99.98%Colore e forma:SolidPeso molecolare:425.4Dimethindene
CAS:Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.Formula:C20H24N2Purezza:98.3% - 98.99%Colore e forma:SolidPeso molecolare:292.42CP-810123
CAS:CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.Formula:C14H18N4OPurezza:98.63% - 99.60%Colore e forma:SolidPeso molecolare:258.32BMS-933043
CAS:BMS-933043: α7 nAChR partial agonist, binds rat (Ki=3.3 nM) & human (Ki=8.1 nM), agonist with EC50=23.4 nM (calcium assay), 0.14-0.29 μM (electrophysiology).Formula:C16H19N7OPurezza:98%Colore e forma:SolidPeso molecolare:325.37L 687306
CAS:L 687306 is a partial agonist of muscarinic M1 receptors. It is also a highly competitive antagonist at cardiac M2 receptors and ileal M3 muscarinic receptors.Formula:C11H15N3OColore e forma:SolidPeso molecolare:205.26ABT-418 hydrochloride
CAS:ABT-418 HCl enhances cognition and reduces anxiety as a selective nAChRs agonist, researched for Alzheimer's.Formula:C9H15ClN2OColore e forma:SolidPeso molecolare:202.68N-Demethyl MK-6884
CAS:N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.Formula:C24H23N5OColore e forma:SolidPeso molecolare:397.47APS3
CAS:APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].Formula:C18H7Cl2F6N5O5S2Colore e forma:SolidPeso molecolare:622.31LY2033298
CAS:LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.Formula:C13H14ClN3O2SPurezza:98.78%Colore e forma:SolidPeso molecolare:311.79ICL-CCIC-0019
CAS:<p>ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.</p>Formula:C26H44Br2N4Purezza:99.54%Colore e forma:SolidPeso molecolare:572.463-Bromocytisine
CAS:3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).Formula:C11H13BrN2OPurezza:99.974%Colore e forma:SolidPeso molecolare:269.14Adenylyl cyclase-IN-1
CAS:Adenylyl cyclase-IN-1 is a potential adenylyl cyclase inhibitor for ocular hypotonia research [1].Formula:C9H8N2S3Colore e forma:SolidPeso molecolare:240.37Zamifenacin fumarate
CAS:Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.Formula:C31H33NO7Purezza:99.88%Colore e forma:SolidPeso molecolare:531.6Homatropine hydrochloride
CAS:Homatropine hydrochloride is an orally active anticholinergic agent that induces rapid pupil dilation with cycloplegic effects and possesses antitussiveFormula:C16H22ClNO3Colore e forma:SolidPeso molecolare:311.8Tiotropium Bromide hydrate
CAS:Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.Formula:C19H24BrNO5S2Purezza:98.44% - 99.41%Colore e forma:SolidPeso molecolare:490.43mAChR antagonist 1
CAS:Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes,Formula:C19H22N2O2Colore e forma:SolidPeso molecolare:310.39Tolterodine Dimer
CAS:Tolterodine Dimer is a derivative of Tolterodine -- a muscarinic receptor antagonist that is used to treat patients with overactive bladder.Formula:C35H41NO2Colore e forma:SolidPeso molecolare:507.71Timepidium bromide
CAS:Timepidium bromide is an agent of anticholinergic.Formula:C17H22BrNOS2Purezza:98%Colore e forma:SolidPeso molecolare:400.4AR420626
CAS:AR420626: selective FA3R agonist, guards against SALS, effects blocked by BHB, a FA3R antagonist.Formula:C21H18Cl2N2O3Purezza:98.62%Colore e forma:SolidPeso molecolare:417.29LG 50643
CAS:LG 50643 is a muscarinic antagonist.Formula:C24H34INO2Purezza:98%Colore e forma:SolidPeso molecolare:495.44ASP8302
CAS:ASP8302 is an allosteric potentiator of the muscarinic M3 receptor. It enhances urination efficiency and reduces residual urine volume in two rat models of voiding dysfunction. ASP8302 is useful for investigating diseases associated with bladder dysfunction.Formula:C26H32ClN7O3S2Colore e forma:SolidPeso molecolare:590.16Muscarine tosylate
CAS:Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].Formula:C16H27NO5SColore e forma:SolidPeso molecolare:345.45Hydroxy Varenicline
CAS:Hydroxy varenicline, a metabolite of the nicotinic acetylcholine receptor (nAChR) agonist varenicline, functions within the biochemical pathway by interacting with nAChR sites.Formula:C13H13N3OColore e forma:SolidPeso molecolare:227.267VU 0255035
CAS:<p>VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.</p>Formula:C18H20N6O3S2Purezza:98.09% - 98.1%Colore e forma:SolidPeso molecolare:432.52Cynandione A
CAS:Cynandione A is an acetophenone derived from Cynanchum wilfordii with anti-inflammatory activity.Formula:C16H14O6Purezza:99.62%Colore e forma:SolidPeso molecolare:302.28PTAC oxalate
CAS:muscarinic receptor ligandFormula:C14H21N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:359.46VU0453595
CAS:<p>VU0453595 is a M1 positive allosteric modulator (PAM).</p>Formula:C18H15FN4OPurezza:99.91%Colore e forma:SolidPeso molecolare:322.34UFP-512
CAS:UFP-512 is a selective delta-opioid (DOP) receptor agonist.Formula:C31H33N5O5Purezza:98%Colore e forma:SolidPeso molecolare:555.62A-424274
CAS:A-424274 is a positive allosteric modulator of α4β2 neuronal nicotinic receptor.Formula:C14H15N3Purezza:98%Colore e forma:SolidPeso molecolare:225.29Tematropium
CAS:Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.Formula:C21H31NO8SPurezza:99.89%Colore e forma:SolidPeso molecolare:457.54(+)-Sparteine sulfate pentahydrate
(+)-sparteine (sulfate pentahydrate) is a ganglion blocker that competitively blocks nicotinic acetylcholine receptors in neurons.Formula:C15H38N2O9SColore e forma:SolidPeso molecolare:422.54WIN 62577
CAS:WIN 62577 is a species-selective tachykinin NK1 receptor antagonist and also serves as an allosteric enhancer with micromolar potency at M3 receptors. Additionally, WIN 62577 demonstrates potent antiviral activity against SARS-CoV-2.Formula:C29H31N3OColore e forma:SolidPeso molecolare:437.576(S)-Albuterol
CAS:<p>(S)-Albuterol functions as a muscarinic receptor and phospholipase C activator, enhancing the intracellular free calcium concentration in airway smooth muscle cells.</p>Formula:C13H21NO3Colore e forma:SolidPeso molecolare:239.311nAChR antagonist 1
CAS:Compound B15, a potent α7 nAChR antagonist, IC50 = 3.3 μM, promising for research on schizophrenia, Alzheimer's, and inflammation.Formula:C19H22N4O2Colore e forma:SolidPeso molecolare:338.4Dihydro-β-erythroidine hydrobromide
CAS:Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H22BrNO3Purezza:98%Colore e forma:White SolidPeso molecolare:356.26p-F-HHSiD hydrochloride
CAS:p-F-HHSiD (p-Fluorohexahydrosiladifenidol) hydrochloride is a selective M3mAChR antagonist. It is capable of inhibiting acetylcholine-mediated vasodilation in human umbilical vein endothelial cells (HUVEC).Formula:C20H33ClFNOSiPeso molecolare:386.019VU6007496
CAS:<p>VU6007496 is a highly selective and CNS-penetrating M1 positive allosteric modulator (PAM) that exhibits good pharmacokinetics (PK).</p>Formula:C25H27N5O2Colore e forma:SolidPeso molecolare:429.51TAAR1 agonist 2
CAS:TAAR1 agonist 2 (compound 30), a full agonist at trace amine-associated receptor 1 (TAAR1) (pEC50=7.5), also displays agonistic properties at H1 receptors and activates various muscarinic acetylcholine receptors, including the M2 receptor (pEC50=5). This compound is utilized in researching neuropsychiatric diseases.Formula:C9H11NOColore e forma:SolidPeso molecolare:149.19VU6016235
CAS:VU6016235 is a structurally unique, orally available, and highly selective tricyclic M4 muscarinic acetylcholine receptor positive allosteric modulator.Formula:C21H22N4OSColore e forma:SolidPeso molecolare:378.49TDI-11861
CAS:TDI-11861 is a second-gen sAC (ADCY10) inhibitor with an IC50 of 5.5 nM and slow dissociation.Formula:C22H25ClF2N6O3Colore e forma:SolidPeso molecolare:494.92
