
AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 619 prodotti di "AChR"
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Iperoxo
CAS:Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.Formula:C10H17IN2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:324.16PHA 543613
CAS:PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.Formula:C15H17N3O2Purezza:99.43% - 99.96%Colore e forma:SolidPeso molecolare:271.31JNJ-39393406
CAS:JNJ-39393406 is an α7 nicotinic acetylcholine receptor positive allosteric modulator for the study of tobacco dependence and Alzheimer's disease.Formula:C19H18F2N6O3Purezza:98.5%Colore e forma:SolidPeso molecolare:416.38Oxotremorine M iodide
CAS:Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.Formula:C11H19IN2OPurezza:99.57%Colore e forma:SolidPeso molecolare:322.19NKY80
CAS:NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.Formula:C12H11N3O2Purezza:99.88%Colore e forma:SolidPeso molecolare:229.23LG 50643
CAS:LG 50643 is a muscarinic antagonist.Formula:C24H34INO2Purezza:98%Colore e forma:SolidPeso molecolare:495.44PTAC oxalate
CAS:muscarinic receptor ligandFormula:C14H21N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:359.46A-424274
CAS:A-424274 is a positive allosteric modulator of α4β2 neuronal nicotinic receptor.Formula:C14H15N3Purezza:98%Colore e forma:SolidPeso molecolare:225.29LY2033298
CAS:LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.Formula:C13H14ClN3O2SPurezza:98.78%Colore e forma:SolidPeso molecolare:311.793-Bromocytisine
CAS:3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).Formula:C11H13BrN2OPurezza:99.974%Colore e forma:SolidPeso molecolare:269.14Tolterodine Dimer
CAS:Tolterodine Dimer is a derivative of Tolterodine -- a muscarinic receptor antagonist that is used to treat patients with overactive bladder.Formula:C35H41NO2Colore e forma:SolidPeso molecolare:507.71APS3
CAS:APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].Formula:C18H7Cl2F6N5O5S2Colore e forma:SolidPeso molecolare:622.31Adenylyl cyclase-IN-1
CAS:Adenylyl cyclase-IN-1 is a potential adenylyl cyclase inhibitor for ocular hypotonia research [1].Formula:C9H8N2S3Colore e forma:SolidPeso molecolare:240.37ASP8302
CAS:ASP8302 is an allosteric potentiator of the muscarinic M3 receptor. It enhances urination efficiency and reduces residual urine volume in two rat models of voiding dysfunction. ASP8302 is useful for investigating diseases associated with bladder dysfunction.Formula:C26H32ClN7O3S2Colore e forma:SolidPeso molecolare:590.16ICL-CCIC-0019
CAS:ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.Formula:C26H44Br2N4Purezza:99.54%Colore e forma:SolidPeso molecolare:572.46Hydroxy Varenicline
CAS:Hydroxy varenicline, a metabolite of the nicotinic acetylcholine receptor (nAChR) agonist varenicline, functions within the biochemical pathway by interacting with nAChR sites.Formula:C13H13N3OColore e forma:SolidPeso molecolare:227.267L 687306
CAS:L 687306 is a partial agonist of muscarinic M1 receptors. It is also a highly competitive antagonist at cardiac M2 receptors and ileal M3 muscarinic receptors.Formula:C11H15N3OColore e forma:SolidPeso molecolare:205.26Muscarine tosylate
CAS:Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].Formula:C16H27NO5SColore e forma:SolidPeso molecolare:345.45N-Demethyl MK-6884
CAS:N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.Formula:C24H23N5OColore e forma:SolidPeso molecolare:397.47VU0453595
CAS:<p>VU0453595 is a M1 positive allosteric modulator (PAM).</p>Formula:C18H15FN4OPurezza:99.91%Colore e forma:SolidPeso molecolare:322.34
