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AChR

AChR

Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.

Trovati 619 prodotti di "AChR"

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  • Cynandione A
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    Cynandione A

    CAS:
    Cynandione A is an acetophenone derived from Cynanchum wilfordii with anti-inflammatory activity.
    Formula:C16H14O6
    Purezza:99.62%
    Colore e forma:Solid
    Peso molecolare:302.28

    Ref: TM-T70277

  • Timepidium bromide
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    Timepidium bromide

    CAS:
    Timepidium bromide is an agent of anticholinergic.
    Formula:C17H22BrNOS2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:400.4

    Ref: TM-T12825

  • UFP-512
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    UFP-512

    CAS:
    UFP-512 is a selective delta-opioid (DOP) receptor agonist.
    Formula:C31H33N5O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:555.62

    Ref: TM-T29046

  • BMS-933043
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    BMS-933043

    CAS:
    BMS-933043: α7 nAChR partial agonist, binds rat (Ki=3.3 nM) & human (Ki=8.1 nM), agonist with EC50=23.4 nM (calcium assay), 0.14-0.29 μM (electrophysiology).
    Formula:C16H19N7O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:325.37

    Ref: TM-T26865

  • ABT-418 hydrochloride
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    ABT-418 hydrochloride

    CAS:
    ABT-418 HCl enhances cognition and reduces anxiety as a selective nAChRs agonist, researched for Alzheimer's.
    Formula:C9H15ClN2O
    Colore e forma:Solid
    Peso molecolare:202.68

    Ref: TM-T10224

  • Zamifenacin fumarate
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    Zamifenacin fumarate

    CAS:
    Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.
    Formula:C31H33NO7
    Purezza:99.88%
    Colore e forma:Solid
    Peso molecolare:531.6

    Ref: TM-T13385

  • AR420626
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    AR420626

    CAS:
    AR420626: selective FA3R agonist, guards against SALS, effects blocked by BHB, a FA3R antagonist.
    Formula:C21H18Cl2N2O3
    Purezza:98.62%
    Colore e forma:Solid
    Peso molecolare:417.29

    Ref: TM-T26647

  • VU 0255035
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    VU 0255035

    CAS:
    <p>VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.</p>
    Formula:C18H20N6O3S2
    Purezza:98.09% - 98.1%
    Colore e forma:Solid
    Peso molecolare:432.52

    Ref: TM-T23508

  • Tiotropium Bromide hydrate
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    Tiotropium Bromide hydrate

    CAS:
    Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.
    Formula:C19H24BrNO5S2
    Purezza:98.44% - 99.41%
    Colore e forma:Solid
    Peso molecolare:490.43

    Ref: TM-T6707

  • Homatropine hydrochloride
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    Homatropine hydrochloride

    CAS:
    Homatropine hydrochloride is an orally active anticholinergic agent that induces rapid pupil dilation with cycloplegic effects and possesses antitussive
    Formula:C16H22ClNO3
    Colore e forma:Solid
    Peso molecolare:311.8

    Ref: TM-T80637

  • mAChR antagonist 1
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    mAChR antagonist 1

    CAS:
    Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes,
    Formula:C19H22N2O2
    Colore e forma:Solid
    Peso molecolare:310.39

    Ref: TM-T81888

  • Tematropium
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    Tematropium

    CAS:
    Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.
    Formula:C21H31NO8S
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:457.54

    Ref: TM-T10732

  • Logo CymitQuimica
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    nAChR antagonist 1

    CAS:
    Compound B15, a potent α7 nAChR antagonist, IC50 = 3.3 μM, promising for research on schizophrenia, Alzheimer's, and inflammation.
    Formula:C19H22N4O2
    Colore e forma:Solid
    Peso molecolare:338.4

    Ref: TM-T61064

  • UB 165
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    UB 165

    CAS:
    Subtype-selective nicotinic agonist
    Formula:C13H15ClN2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:234.72

    Ref: TM-T23485

  • (+)-Cevimeline hydrochloride hemihydrate
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    (+)-Cevimeline hydrochloride hemihydrate

    (+)-Cevimeline HCl hemihydrate is a muscarinic agonist for dry mouth in Sjogren's with rapid absorption, differing metabolism in species.
    Formula:C10H19ClNO1·5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:244.78

    Ref: TM-T13460

  • 1,9-Dideoxyforskolin
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    1,9-Dideoxyforskolin

    CAS:
    The compound is an inactive analog of forskolin(an adenylyl cyclase activator).
    Formula:C22H34O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:378.5

    Ref: TM-T22467

  • LY593093
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    LY593093

    CAS:
    LY593093 is a selective partial orthosteric agonist of M1 muscarinic acetylcholine receptor.
    Formula:C32H30FN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:507.6

    Ref: TM-T27961

  • VU6007496
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    VU6007496

    CAS:
    <p>VU6007496 is a highly selective and CNS-penetrating M1 positive allosteric modulator (PAM) that exhibits good pharmacokinetics (PK).</p>
    Formula:C25H27N5O2
    Colore e forma:Solid
    Peso molecolare:429.51

    Ref: TM-T200762

  • TDI-11861
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    TDI-11861

    CAS:
    TDI-11861 is a second-gen sAC (ADCY10) inhibitor with an IC50 of 5.5 nM and slow dissociation.
    Formula:C22H25ClF2N6O3
    Colore e forma:Solid
    Peso molecolare:494.92

    Ref: TM-T73297

  • TAAR1 agonist 2
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    TAAR1 agonist 2

    CAS:
    TAAR1 agonist 2 (compound 30), a full agonist at trace amine-associated receptor 1 (TAAR1) (pEC50=7.5), also displays agonistic properties at H1 receptors and activates various muscarinic acetylcholine receptors, including the M2 receptor (pEC50=5). This compound is utilized in researching neuropsychiatric diseases.
    Formula:C9H11NO
    Colore e forma:Solid
    Peso molecolare:149.19

    Ref: TM-T200140