Proteasi serina
Gli inibitori delle serin proteasi sono composti che inibiscono le serin proteasi, un gruppo di enzimi caratterizzati da un residuo di serina nel loro sito attivo. Queste proteasi sono coinvolte in numerosi processi fisiologici, tra cui la digestione, la risposta immunitaria, la coagulazione del sangue e l'infiammazione. Gli inibitori delle serin proteasi sono importanti per studiare le malattie in cui questi enzimi sono disregolati, come le malattie cardiovascolari, il cancro e le condizioni infiammatorie. Presso CymitQuimica, offriamo inibitori delle serin proteasi per supportare la tua ricerca in enzimologia, meccanismi delle malattie e interventi terapeutici.
Trovati 56 prodotti per "Proteasi serina".
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Nonacog alfa
CAS:Nonacog alfa (BAX326), a recombinant human factor IX, is utilized in the study of hemophilia B [1].Colore e forma:LiquidMeOSuc-AAPF-CMK
CAS:MeOSuc-AAPF-CMK (MeOSuc-Ala-Ala-Pro-Phe-CH2Cl) is a potent inhibitor of the enzyme proteinase K [1].Formula:C26H35ClN4O7Colore e forma:SolidPeso molecolare:551.03Suc-AAP-Abu-pNA
CAS:Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,Formula:C25H34N6O9Colore e forma:SolidPeso molecolare:562.57C1 Esterase Inhibitor (Human)
C1 Esterase Inhibitor (Human) is a glycoprotein derived from human plasma and acts as a serine protease inhibitor. It inactivates enzymes like C1r, C1s, and mannose-binding lectin-associated serine proteases (MASP) through covalent binding. This compound possesses anti-inflammatory properties and is utilized to prevent angioedema attacks associated with hereditary angioedema.Colore e forma:Odour LiquidChymotrypsinogen
CAS:Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .Colore e forma:SolidPKR-IN-C51
CAS:PKR-IN-C51 is ATP-competitive protein kinase R (PKR) inhibitor that inhibits intracellular PKR activation and autophosphorylation. Ser/Thr kinase.Formula:C23H21N5Purezza:98.94%Colore e forma:Yellow SolidPeso molecolare:367.45Ref: TM-T24647
2mg82,00€5mg120,00€1mL*10mM (DMSO)133,00€10mg192,00€25mg356,00€50mg530,00€100mg755,00€2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urineFormula:C13H16O3Purezza:99.53% - 99.81%Colore e forma:SolidPeso molecolare:220.26Ref: TM-T8802
1mg82,00€1mL*10mM (DMSO)146,00€5mg168,00€10mg244,00€25mg404,00€50mg567,00€100mg767,00€500mg1.521,00€WNK463
CAS:WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).Formula:C21H24F3N7O2Purezza:>99.99% - ≥95%Colore e forma:SolidPeso molecolare:463.46Benzamidine hydrochloride
CAS:Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.Formula:C7H9ClN2Purezza:99.64% - 99.97%Colore e forma:SolidPeso molecolare:156.612-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
CAS:2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.Formula:C14H7BrClNO2Purezza:97.36%Colore e forma:SolidPeso molecolare:336.57ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Formula:C22H19N3O2SPurezza:99.12% - 99.87%Colore e forma:SolidPeso molecolare:389.47Ref: TM-T3423
1mg34,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg92,00€25mg178,00€50mg295,00€100mg474,00€500mg1.035,00€WNK-IN-11
CAS:WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)Formula:C21H21Cl2N5OSPurezza:98.32%Colore e forma:SolidPeso molecolare:462.4Ref: TM-T5456
1mg87,00€5mg172,00€1mL*10mM (DMSO)188,00€10mg280,00€25mg474,00€50mg683,00€100mg964,00€500mg1.918,00€KKI-5 acetate(97145-43-2 free base)
KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.Formula:C37H59N11O11Purezza:99.74%Colore e forma:White SolidPeso molecolare:833.95Cetraxate hydrochloride
CAS:Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.Formula:C17H24ClNO4Purezza:99.75%Colore e forma:SolidPeso molecolare:341.83Alvelestat
CAS:Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.Formula:C25H22F3N5O4SPurezza:98% - >99.99%Colore e forma:White SolidPeso molecolare:545.53Ref: TM-T3107
1mg34,00€2mg43,00€5mg56,00€1mL*10mM (DMSO)74,00€10mg84,00€25mg148,00€50mg219,00€100mg349,00€500mg830,00€Lanadelumab
CAS:Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.Purezza:95% - 97.4% (SDS-PAGE); 99.2% (SEC-HPLC)Colore e forma:Transparent LiquidPeso molecolare:145.70 kDaAnti-Matriptase Antibody
Anti-Matriptase Antibody is a human antibody expressed in CHO cells.Purezza:95.8% (SDS-PAGE); 99.2% (SEC-HPLC) - 95.8% (SDS-PAGE); 99.2% (SEC-HPLC)Colore e forma:Transparent LiquidPeso molecolare:144.27 kDaGalegenimab
CAS:Galegenimab (RG 6147) is an Fab targeting HtrA1, capable of blocking proteolytic cleavage of biglycan (an HtrA1 substrate), suitable for AMD research.Purezza:95% - 95.8% (SDS-PAGE); 99.7% (SEC-HPLC)Colore e forma:Transparent LiquidPeso molecolare:46.87 kDaMEGA-9
CAS:MEGA-9 (Nonanoyl-N-Methylglucamide) solubilizes membrane protein and can be used as a nonionic detergent.Formula:C16H33NO6Purezza:99.9%Colore e forma:White SolidPeso molecolare:335.44ZM223 hydrochloride (2031177-48-5 free base)
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.Formula:C23H18ClF3N4O2S2Purezza:98%Colore e forma:SolidPeso molecolare:538.99
