
PAI-1
Il Plasminogen Activator Inhibitor-1 (PAI-1) è un inibitore delle serin proteasi che regola la fibrinolisi inibendo l'attivatore tissutale del plasminogeno (tPA) e l'urochinasi (uPA). Livelli elevati di PAI-1 sono associati a un aumento del rischio di trombosi, malattie cardiovascolari e sindrome metabolica. Gli inibitori di PAI-1 sono oggetto di ricerca per il loro potenziale nel trattamento di queste condizioni. Presso CymitQuimica, offriamo inibitori di PAI-1 per supportare la tua ricerca in ematologia, salute cardiovascolare e malattie metaboliche.
Trovati 30 prodotti per "PAI-1".
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UK-371804 HCl
CAS:UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-Formula:C14H17Cl2N5O4SPurezza:98%Colore e forma:SolidPeso molecolare:422.29Diaplasinin
CAS:Diaplasinin (PAI-749) is a potent inhibitor of plasminogen activator inhibitor-1 (PAI-1) with antithrombotic activity, used in cardiovascular disease research.Formula:C32H31N5OPurezza:99.02%Colore e forma:Yellow SolidPeso molecolare:501.62Ref: TM-T25915
1mg57,00€5mg120,00€1mL*10mM (DMSO)133,00€10mg178,00€25mg409,00€50mg708,00€100mg1.153,00€p-Aminobenzamidine dihydrochloride
CAS:4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase typeFormula:C7H11Cl2N3Purezza:99.00% - 99.56%Colore e forma:SolidPeso molecolare:208.088SK-216
CAS:SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.Formula:C29H29NNa2O6Purezza:98.29%Colore e forma:SolidPeso molecolare:533.52AZ3976
CAS:AZ3976 is an inhibitor of PAI-1 with an IC50 of 16 μM in a plasma clot lysis assay. AZ3976 displays profibrinolytic activities.Formula:C15H19N5O3Purezza:98.14%Colore e forma:White SolidPeso molecolare:317.34Aleplasinin
CAS:Aleplasinin (PAZ 417) is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and a key negative regulator of the fibrinolyticFormula:C28H27NO3Purezza:99.21%Colore e forma:SolidPeso molecolare:425.52Ref: TM-T29856
1mg54,00€5mg114,00€1mL*10mM (DMSO)126,00€10mg178,00€25mg409,00€50mg620,00€100mg982,00€200mg1.314,00€PPACK
CAS:PPACK: synthetic peptide, irreversibly inhibits thrombin (Ki = 0.24 nM), prevents platelet activation.Formula:C21H31ClN6O3Purezza:98%Colore e forma:SolidPeso molecolare:450.96ZK824190
CAS:ZK824190: oral uPA inhibitor, IC50 - uPA 237 nM, tPA 1600 nM, Plasmin 1850 nM.Formula:C22H20F2N2O4Purezza:98.84%Colore e forma:White SolidPeso molecolare:414.4Ref: TM-T13408
1mg152,00€5mg306,00€1mL*10mM (DMSO)318,00€10mg442,00€25mg675,00€50mg900,00€100mg1.224,00€GGACK
CAS:GGACK (H-Glu-Gly-Arg-CMK) is an irreversible substrate-like inhibitor of the serine protease urokinase-type plasminogen activator (uPA).Formula:C14H25ClN6O5Colore e forma:SolidPeso molecolare:392.84BT-114143
CAS:BT-114143 is a plasminogen activator inhibitor with an IC50 of 8.42 μM. It is applicable in research related to hemorrhagic diseases caused by excessive fibrinolysis, including traumatic bleeding, severe menorrhagia, postpartum hemorrhage, and complications of hemophilia.Formula:C8H11N2O3PColore e forma:SolidPeso molecolare:214.158
