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DPP-4

DPP-4

Gli inibitori di DPP-4 sono composti che inibiscono la Dipeptidil Peptidasi-4, un enzima coinvolto nell'inattivazione degli ormoni incretinici, che regolano il metabolismo del glucosio. Inibendo la DPP-4, questi composti aiutano a prolungare l'azione degli ormoni incretinici, migliorando la secrezione di insulina e riducendo i livelli di glucosio nel sangue. Gli inibitori di DPP-4 sono ampiamente utilizzati nel trattamento del diabete di tipo 2 e nella ricerca sui disturbi metabolici. Presso CymitQuimica, offriamo inibitori di DPP-4 per supportare la tua ricerca in endocrinologia, gestione del diabete e malattie metaboliche.

Trovati 20 prodotti di "DPP-4"

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  • 3-Pyridylacetic acid hydrochloride

    CAS:
    <p>3-Pyridylacetic acid HCl (3-PAA) is a strong acid, reactive with amines/alcohols/acids, and an organic catalyst.</p>
    Formula:C7H8ClNO2
    Purezza:99.31% - 99.95%
    Colore e forma:White To Beige Crystalline Powder
    Peso molecolare:173.6
  • Retagliptin Phosphate

    CAS:
    <p>Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.</p>
    Formula:C19H21F6N4O7P
    Purezza:98.70%
    Colore e forma:Solid
    Peso molecolare:562.36
  • Begelomab

    CAS:
    Begelomab (SAND-26) is a mouse-derived monoclonal antibody targeting DPP-4/CD26. Begelomab can be used to study severe refractory inflammatory myopathies.
    Purezza:97.8% (SDS-PAGE); 98.3% (SEC-HPLC) - 97.8% (SDS-PAGE); 98.3% (SEC-HPLC)
    Colore e forma:Liquid
  • Saxagliptin hydrate

    CAS:
    Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).
    Formula:C18H25N3O2·H2O
    Purezza:99.52%
    Colore e forma:Solid
    Peso molecolare:333.43
  • Denagliptin

    CAS:
    Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study of
    Formula:C20H18F3N3O
    Purezza:99.12%
    Colore e forma:Solid
    Peso molecolare:373.37
  • DPP-IV-IN-2

    CAS:
    DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).
    Formula:C18H26N4O5
    Purezza:99.08%
    Colore e forma:Solid
    Peso molecolare:378.42
  • DPP4/CD26 Protein, Mouse, Recombinant (hFc)


    DPP4/CD26 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.
    Purezza:99% - > 95 % as determined by SDS-PAGE.
    Colore e forma:Lyophilized Powder
    Peso molecolare:112.9 kDa (predicted)
  • DPP4/CD26 Protein, Mouse, Recombinant (His)


    DPP4/CD26 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.
    Colore e forma:Lyophilized Powder
    Peso molecolare:85.9 kDa (predicted)
  • Alogliptin Benzoate

    CAS:
    Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.
    Formula:C25H27N5O4
    Purezza:99.94% - >99.99%
    Colore e forma:White Powder
    Peso molecolare:461.51
  • Diprotin A

    CAS:
    Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.
    Formula:C17H31N3O4
    Purezza:99.29%
    Colore e forma:White Powder
    Peso molecolare:341.45
  • Saxagliptin

    CAS:
    <p>Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.</p>
    Formula:C18H25N3O2
    Purezza:99.17% - 99.95%
    Colore e forma:Solid
    Peso molecolare:315.41
  • Alogliptin

    CAS:
    Alogliptin (SYR-322)(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of <10 nM, exhibits greater than 10, 000-fold selectivity over DPP-8 and DPP-9
    Formula:C18H21N5O2
    Purezza:99.63%
    Colore e forma:Solid
    Peso molecolare:339.39
  • Anagliptin

    CAS:
    Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.
    Formula:C19H25N7O2
    Purezza:97.59% - 99.98%
    Colore e forma:Solid
    Peso molecolare:383.45
  • Picolamine

    CAS:
    <p>Picolamine acts as a potential inhibitor of DPP-4.</p>
    Formula:C6H8N2
    Purezza:98.3%
    Colore e forma:Light Yellow Liquid
    Peso molecolare:108.14
  • Teneligliptin

    CAS:
    <p>Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.</p>
    Formula:C22H30N6OS
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:426.58
  • Cofrogliptin

    CAS:
    Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).
    Formula:C18H19F5N4O3S
    Colore e forma:Solid
    Peso molecolare:466.43
  • Gosogliptin

    CAS:
    Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.
    Formula:C17H24F2N6O
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:366.41
  • P32/98 hemifumarate

    CAS:
    P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.
    Formula:C22H40N4O6S2
    Purezza:99.46%
    Colore e forma:Solid
    Peso molecolare:520.71
  • Imigliptin

    CAS:
    Imigliptin Dihydrochloride, a selective dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type II diabetes.
    Formula:C21H24N6O
    Purezza:99.12%
    Colore e forma:Solid
    Peso molecolare:376.46
  • TS-021

    CAS:
    TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.
    Formula:C17H24FN3O5S
    Purezza:>99.99% - >99.99%
    Colore e forma:Solid
    Peso molecolare:401.45