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Cellule staminali

Cellule staminali

Gli inibitori delle cellule staminali sono composti che mirano specificamente alle cellule staminali e alle loro vie di segnalazione, influenzando la loro capacità di autorinnovarsi e differenziarsi. Questi inibitori sono cruciali nella ricerca focalizzata sul controllo del comportamento delle cellule staminali, sulla comprensione dei processi di sviluppo e sullo sviluppo di terapie per malattie come il cancro, dove si ritiene che le cellule staminali svolgano un ruolo chiave. Presso CymitQuimica, offriamo una varietà di inibitori delle cellule staminali per supportare la tua ricerca in medicina rigenerativa, biologia dello sviluppo e oncologia.

Trovati 463 prodotti di "Cellule staminali"

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  • BDP5290

    CAS:
    BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.)
    Formula:C17H18ClN7O
    Purezza:97.22%
    Colore e forma:Solid
    Peso molecolare:371.82
  • Teplinovivint

    CAS:
    Teplinovivint is a potent inhibitor of the Wnt/β-catenin signaling pathway, demonstrating anti-inflammatory properties with potential utility in tendinopathy
    Formula:C25H26N6O2
    Purezza:97.21%
    Colore e forma:Solid
    Peso molecolare:442.51
  • GSK429286A

    CAS:
    <p>GSK429286A (RHO-15) is a specific inhibitor of ROCK1/2 (IC50: 14/63 nM).</p>
    Formula:C21H16F4N4O2
    Purezza:97.68% - 98.49%
    Colore e forma:Solid
    Peso molecolare:432.37
  • LY3200882

    CAS:
    LY3200882 is a highly selective inhibitor of TGF-β receptor type 1 (TGFβRI).
    Formula:C24H29N5O3
    Purezza:99.46% - 99.63%
    Colore e forma:Solid
    Peso molecolare:435.52
  • AZD1080

    CAS:
    AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor.
    Formula:C19H18N4O2
    Purezza:97.72% - 99.75%
    Colore e forma:Solid
    Peso molecolare:334.37
  • PF-670462

    CAS:
    PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.
    Formula:C19H22Cl2FN5
    Purezza:99.42% - 99.72%
    Colore e forma:Solid
    Peso molecolare:410.32
  • 2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide

    CAS:
    2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide (GDC046), a potent lead analog, has good kinase selectivity and physicochemical properties.
    Formula:C16H13Cl2N3O2
    Purezza:98.77%
    Colore e forma:Solid
    Peso molecolare:350.2
  • Fosciclopirox

    CAS:
    Fosciclopirox (CPX-POM), the phosphoryloxymethyl ester of CPX (Ciclopirox Prodrug, CPX-POM), selectively delivers the active metabolite, CPX, to the entire
    Formula:C13H20NO6P
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:317.27
  • XMU-MP-1

    CAS:
    XMU-MP-1 is a reversible and selective MST1/2 kinase inhibitor, IC50 values for MST1 and MST2 are 71.1 nM and 38.1 nM, respectively. High-Quality, Low-Cost!
    Formula:C17H16N6O3S2
    Purezza:99.68% - 99.86%
    Colore e forma:Solid
    Peso molecolare:416.48
  • SH-4-54

    CAS:
    SH-4-54 is a most potent, small molecule, nonphosphorylated STAT3 inhibitor.
    Formula:C29H27F5N2O5S
    Purezza:98% - 99.12%
    Colore e forma:Solid
    Peso molecolare:610.59
  • ROCK-IN-2

    CAS:
    ROCK-IN-2 (Azaindole 1) is a selective and ATP-competitive ROCK inhibitor with IC50 of 0.6 and 1.1 nM for human ROCK-1 and ROCK-2.
    Formula:C18H13ClF2N6O
    Purezza:97.29%
    Colore e forma:Solid
    Peso molecolare:402.79
  • GS87

    CAS:
    GS87 is a highly specific inhibitor of GSK3 (glycogen synthase kinase 3) that induces extensive differentiation of AML cells.
    Formula:C16H11N5O2S
    Purezza:98.86%
    Colore e forma:Solid
    Peso molecolare:337.36
  • Tegatrabetan

    CAS:
    Tegatrabetan (BC2059) is a small molecule inhibitor of the Wnt/beta-catenin pathway with potential antineoplastic activity.
    Formula:C28H36N4O6S2
    Purezza:98.01% - 99.18%
    Colore e forma:Solid
    Peso molecolare:588.74
  • SAR407899

    CAS:
    SAR407899 is Rho kinase inhibitor potently inhibits endothelin-1-induced constriction of renal resistance arteries.
    Formula:C14H16N2O2
    Purezza:99.42%
    Colore e forma:Solid
    Peso molecolare:244.29
  • IWP-O1

    CAS:
    IWP-O1 is a highly potent Porcupine (Porcn) inhibitor (EC50: 80 pM), effectively suppresses the phosphorylation of Dvl2/3 and LRP6 in HeLa cells.
    Formula:C26H20N6O
    Purezza:99.12%
    Colore e forma:Solid
    Peso molecolare:432.48
  • Hydroxyfasudil Hydrochloride

    CAS:
    Hydroxyfasudil Hydrochloride (HA 1100 hydrochloride) is a ROCK1/2 inhibitor (IC50s: 0.73/0.72 μM).
    Formula:C14H18ClN3O3S
    Purezza:98.05%
    Colore e forma:Solid
    Peso molecolare:343.83
  • IQ 1

    CAS:
    <p>IQ 1 has multiple roles, such as maintaining the multifunctionality of mouse ESCs, decreasing Wnt-stimulated phosphorylation, blocking PP2A/Nkd interactions.</p>
    Formula:C21H22N4O2
    Purezza:98.57% - ≥95%
    Colore e forma:Solid
    Peso molecolare:362.42
  • BIO-013077-01

    CAS:
    BIO-013077-01 is a potent TGFbeta family type I receptors antagonist.
    Formula:C17H13N5
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:287.32
  • FM-381

    CAS:
    FM381, a JAK3 inhibitor with 127 pM IC50, is 410-3600x more selective over JAK1/2/TYK2.
    Formula:C24H24N6O2
    Purezza:98.44%
    Colore e forma:Solid
    Peso molecolare:428.49
  • Galunisertib

    CAS:
    Galunisertib (LY2157299) is a selective TGF-β receptor type I (TGF-βRI) inhibitor. Galunisertib has antitumor activity. Cost-effective and quality-assured.
    Formula:C22H19N5O
    Purezza:97.09% - 99.98%
    Colore e forma:Solid
    Peso molecolare:369.42