Src
Gli inibitori di Src sono composti che prendono di mira le chinasi della famiglia Src, coinvolte in vari processi cellulari, tra cui crescita, differenziazione e angiogenesi. Le chinasi Src svolgono un ruolo critico nelle vie di segnalazione che promuovono la formazione di nuovi vasi sanguigni nei tumori. Inibendo Src, è possibile interrompere queste vie, riducendo così l'angiogenesi e la crescita tumorale. Gli inibitori di Src sono ampiamente utilizzati nella ricerca sul cancro e nello sviluppo terapeutico. Presso CymitQuimica, offriamo una selezione completa di inibitori di Src di alta qualità per supportare la tua ricerca in oncologia, segnalazione cellulare e angiogenesi.
Trovati 82 prodotti di "Src"
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MNS
CAS:MNS is a tyrosine kinases inhibitor, inhibits Syk, Src, p97 with IC50 of 2.5 μM, 29.3 μM and 1.7 μM, respectively.Formula:C9H7NO4Purezza:98.53%Colore e forma:Yellow PowderPeso molecolare:193.16lavendustin C
CAS:lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.Formula:C14H13NO5Purezza:98.06%Colore e forma:Yellow To Tan PowderPeso molecolare:275.26Ref: TM-T4185
1mg42,00€2mg55,00€5mg93,00€10mg152,00€25mg330,00€50mg492,00€100mg707,00€1mL*10mM (DMSO)90,00€PP1
CAS:PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is 5 nM/ 6 nM, respectively.Formula:C16H19N5Purezza:99% - 99.88%Colore e forma:Off-White To Grey SolidPeso molecolare:281.36Ref: TM-T6196
1mg40,00€2mg52,00€5mg88,00€10mg118,00€25mg202,00€50mg283,00€100mg444,00€500mg998,00€1mL*10mM (DMSO)94,00€WH-4-023
CAS:WH-4-023 (Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor. It also potently inhibits SIK.Formula:C32H36N6O4Purezza:98% - 99.75%Colore e forma:SolidPeso molecolare:568.67Ref: TM-T1811
2mg51,00€5mg74,00€10mg99,00€25mg162,00€50mg197,00€100mg350,00€1mL*10mM (DMSO)Prezzo su richiesta1-NM-PP1
CAS:1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.Formula:C20H21N5Purezza:98% - 98.93%Colore e forma:White Cyrstalline SolidPeso molecolare:331.41Ref: TM-T2153
1mg48,00€2mg63,00€5mg84,00€10mg132,00€25mg271,00€50mg505,00€100mg668,00€1mL*10mM (DMSO)90,00€Masitinib mesylate
CAS:Masitinib mesylate (AB-1010 mesylate) is a selective and orally bioavailable c-Kit inhibitor (IC50 of 200 nM,540/800 nM,510 nM for human recombinant c-Kit;Formula:C29H34N6O4S2Purezza:97.67% - 98.44%Colore e forma:SolidPeso molecolare:594.75KX1-004
CAS:KX1-004, a potential protective drug for NIHL, is an effective small molecule inhibitor of Src-PTK.Formula:C16H13FN2O2Purezza:99.39% - ≥95%Colore e forma:SolidPeso molecolare:284.29Ref: TM-T1812
1mg43,00€2mg56,00€5mg93,00€10mg152,00€25mg268,00€50mg442,00€100mg622,00€500mg1.305,00€1mL*10mM (DMSO)92,00€squarunkinA
CAS:squarunkinA is a novel modulator of the UNC119-Cargo Interaction, potently and selectively inhibiting the binding of a myristoylated peptide representing the N-Formula:C25H32F3N5O4Purezza:99.29%Colore e forma:SolidPeso molecolare:523.55PP121
CAS:PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.Formula:C17H17N7Purezza:98.45% - 99.93%Colore e forma:SolidPeso molecolare:319.36Scutellarein
CAS:Scutellarein (6-Hydroxyapigenin) reduces inflammatory responses by inhibiting Src kinase activity.Formula:C15H10O6Purezza:98.02% - 99.63%Colore e forma:SolidPeso molecolare:286.24Ref: TM-T3319
2mg38,00€5mg52,00€10mg75,00€25mg109,00€50mg159,00€100mg227,00€200mg338,00€1mL*10mM (DMSO)59,00€1-Naphthyl PP1 hydrochloride
CAS:1-Naphthyl PP1 hydrochloride (1-NA-PP 1 hydrochloride) is a selective inhibitor of src family kinases v-SrcFormula:C19H20ClN5Purezza:98.63%Colore e forma:SolidPeso molecolare:353.85Periplocin
CAS:Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.Formula:C36H56O13Purezza:99.66% - 99.74%Colore e forma:SolidPeso molecolare:696.82Ref: TM-T5S1982
1mg35,00€5mg77,00€10mg106,00€25mg170,00€50mg253,00€100mg375,00€500mg892,00€1mL*10mM (DMSO)107,00€Tetramethylcurcumin
CAS:Tetramethylcurcumin is a novel curcumin analog, is an effective inhibitors of STAT3 phosphorylation, DNA binding activity, and transactivation in vitro.it alsoFormula:C25H28O6Purezza:97.69% - 99.94%Colore e forma:SolidPeso molecolare:424.49Bafetinib
CAS:Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.Formula:C30H31F3N8OPurezza:94.16% - 99.68%Colore e forma:SolidPeso molecolare:576.62Ref: TM-T6311
1mg34,00€2mg49,00€5mg74,00€10mg98,00€25mg150,00€50mg178,00€100mg333,00€200mg432,00€1mL*10mM (DMSO)95,00€7-Hydroxy-4H-chromen-4-one
CAS:7-Hydroxy-4H-chromen-4-one (7-hydroxy-4-benzopyrone) is a Src kinase inhibitor (IC50 of <300 μM).Formula:C9H6O3Purezza:97.65%Colore e forma:SolidPeso molecolare:162.14XL228
CAS:XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).Formula:C22H31N9OPurezza:99.07%Colore e forma:SolidPeso molecolare:437.54Ref: TM-T17267
1mg52,00€2mg73,00€5mg94,00€10mg141,00€25mg244,00€50mg371,00€100mg552,00€1mL*10mM (DMSO)104,00€Tirbanibulin
CAS:Tirbanibulin (KX2-391) is a highly selective Src kinase inhibitor that has demonstrated efficacy in pre-Clinicalal animal models of a variety of cancers.Formula:C26H29N3O3Purezza:99.43% - 99.67%Colore e forma:SolidPeso molecolare:431.53Ref: TM-T6345
1mg35,00€5mg64,00€10mg77,00€25mg150,00€50mg266,00€100mg447,00€200mg640,00€1mL*10mM (DMSO)66,00€ENMD-2076
CAS:ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.Formula:C21H25N7Purezza:97.63% - ≥95%Colore e forma:SolidPeso molecolare:375.47PD-089828
CAS:PD 089828 inhibits FGFR1, PDGFRβ, EGFR (IC50s: 0.15-5.47 μM), and c-Src (IC50: 0.18 μM).Formula:C18H18Cl2N6OPurezza:97.39%Colore e forma:SolidPeso molecolare:405.28PD173955
CAS:PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR andFormula:C21H16Cl2N4OSPurezza:98.52% - 98.99%Colore e forma:SolidPeso molecolare:443.35Ref: TM-T3063
2mg35,00€5mg50,00€10mg92,00€25mg166,00€50mg248,00€100mg371,00€200mg530,00€1mL*10mM (DMSO)94,00€AMG-47a
CAS:AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.Formula:C29H28F3N5O2Purezza:98%Colore e forma:SolidPeso molecolare:535.56OXSI-2
CAS:OXSI-2 (Syk Inhibitor) is an inhibitor of Syk with an EC50 of 313 nM and an IC50 of 14 nM.Formula:C18H15N3O3SPurezza:98%Colore e forma:Dark Orange SolidPeso molecolare:353.39TC-S 7003
CAS:TC-S 7003 (Lck Inhibitor) is a Lck inhibitor with anti-inflammatory activity that inhibits T-cell proliferation and can be used to study arthritis.Formula:C31H30N8OPurezza:99.74%Colore e forma:SolidPeso molecolare:530.62A 419259 trihydrochloride
CAS:A 419259 trihydrochloride (RK 20449 trihydrochloride) is an Src family kinases inhibitor (IC50s: 9 nM, 3 nM and 3 nM for Src, Lck and Lyn).Formula:C29H37Cl3N6OPurezza:99.75% - 99.96%Colore e forma:SolidPeso molecolare:592BT424
CAS:BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation and renal fibrosis in the UUO model [1].Formula:C22H15BCl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:421.08TL02-59
CAS:TL02-59: Fgr inhibitor (IC50=0.03nM), also targets Lyn (0.1nM), Hck (160nM), halts acute myelogenous leukemia growth.Formula:C32H34F3N5O4Purezza:98.77%Colore e forma:SolidPeso molecolare:609.64Ref: TM-T13186
1mg49,00€2mg62,00€5mg93,00€10mg133,00€25mg260,00€50mg401,00€100mg557,00€200mg790,00€1mL*10mM (DMSO)111,00€KB SRC 4
CAS:KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits the growth of cancer cells.CAS 번호13460-73-83-4Formula:C32H23ClN8Purezza:98.83% - 99.34%Colore e forma:SolidPeso molecolare:555.03Ref: TM-T11745
1mg73,00€5mg167,00€10mg238,00€25mg504,00€50mgPrezzo su richiesta1mL*10mM (DMSO)188,00€TG 100572 Hydrochloride
CAS:TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.
Formula:C26H27Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:512.43CH6953755
CAS:CH6953755: oral YES1 kinase inhibitor, IC50 1.8 nM, potent, selective, anticancer, halts cell proliferation.Formula:C26H22F2N6O4SPurezza:98.87%Colore e forma:SolidPeso molecolare:552.55Ref: TM-T10784
1mg55,00€5mg116,00€10mg177,00€25mg348,00€50mg557,00€100mg893,00€1mL*10mM (DMSO)141,00€Src Inhibitor 3
CAS:Src Inhibitor 3 blocks c-Src kinase (IC50 <3 nM CSK HTRF, <4 nM Caliper), boosting T cell growth from receptor signals.Formula:C34H32ClFN8O4Purezza:98.35%Colore e forma:SolidPeso molecolare:671.12Ref: TM-T13000
1mg96,00€5mg177,00€10mg304,00€25mg480,00€50mg665,00€100mgPrezzo su richiesta1mL*10mM (DMSO)264,00€CGP062464
CAS:CGP062464 is an inhibitor of the tyrosine kinase c-Src, with an IC50 of less than 50 nM. It is utilized in research related to osteoporosis and tumor-induced hypercalcemia.Formula:C18H14N4Colore e forma:SolidPeso molecolare:286.331N-Deshydroxyethyl Dasatinib-C3-NH2
CAS:N-Deshydroxyethyl Dasatinib-C3-NH2 is a target protein ligand-linker conjugate, comprising an LCK ligand and a PROTAC linker, designed to recruit E3 ligase. It is utilized in the synthesis of [PROTACSJ11646].Formula:C23H29ClN8OSColore e forma:SolidPeso molecolare:501.05
