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Autofagia

Autofagia

Gli inibitori dell'autofagia mirano al processo cellulare di autofagia, che comporta la degradazione e il riciclo dei componenti cellulari attraverso i lisosomi. L'autofagia è un meccanismo critico per mantenere l'omeostasi cellulare, ma la sua disfunzione è implicata in varie malattie, tra cui il cancro, la neurodegenerazione e le infezioni. Gli inibitori dell'autofagia possono bloccare questo processo, rendendoli strumenti preziosi per studiare il ruolo dell'autofagia nelle malattie e sviluppare strategie terapeutiche. Presso CymitQuimica, offriamo inibitori dell'autofagia per supportare la tua ricerca in biologia cellulare, oncologia e malattie neurodegenerative.

Trovati 1483 prodotti di "Autofagia"

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  • ZX-29

    CAS:
    ZX-29: Strong ALK inhibitor; IC50 - ALK 2.1 nM, L1196M 1.3 nM, G1202R 3.9 nM; triggers autophagy; anti-cancer.
    Formula:C23H28ClN7O3S
    Purezza:98.32%
    Colore e forma:Solid
    Peso molecolare:518.03
  • Trimetazidine dihydrochloride

    CAS:
    Trimetazidine, an anti-ischemic agent, enhances myocardial glucose use, inhibits fat metabolism, and helps with angina.
    Formula:C14H24Cl2N2O3
    Purezza:99.58%
    Colore e forma:Crystalline Solid
    Peso molecolare:339.258
  • LG-100064

    CAS:
    LG-100064 is an agonist of retinoid-X-receptor (RXR)(EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ and RXRγ)
    Formula:C23H26O3
    Purezza:98.65%
    Colore e forma:Solid
    Peso molecolare:350.45
  • Felodipine

    CAS:
    Felodipine (CGH-869) is a longlasting 1, 4-dihydropyridine calcium channel repressor.
    Formula:C18H19Cl2NO4
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:384.25
  • Sulfadoxine

    CAS:
    Sulfadoxine (Sulphadoxine) is a broad-spectrum sulfanilamide and a synthetic analog of para-aminobenzoic acid (PABA) with bacteriostatic and antimalarial
    Formula:C12H14N4O4S
    Purezza:99.67%
    Colore e forma:White Or White Crystalline Powder
    Peso molecolare:310.33
  • Sulindac

    CAS:
    Sulindac (Sulindac sulfoxide) is a sulfinylindene derivative prodrug with potential antineoplastic activity.
    Formula:C20H17FO3S
    Purezza:99.09% - 99.15%
    Colore e forma:Yellow Solid
    Peso molecolare:356.41
  • Doxorubicin hydrochloride

    CAS:
    Doxorubicin hydrochloride (Adriamycin) belongs to the anthracycline class of antibiotics and is an inhibitor of human DNA topoisomerase I/II (IC50=0.8/2.67 μM).
    Formula:C27H29NO11·HCl
    Purezza:98% - 99.52%
    Colore e forma:Orange-Red At Neutral Phs And Violet Blue Over Ph 9 (Ntp 1992)
    Peso molecolare:579.99
  • Oxidopamine hydrochloride

    CAS:
    Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.
    Formula:C8H12ClNO3
    Purezza:98.34% - 99.85%
    Colore e forma:Physical Description Beige Solid (Ntp 1992)
    Peso molecolare:205.64
  • Oxidopamine hydrobromide

    CAS:
    Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.
    Formula:C8H12BrNO3
    Purezza:98.22% - 99.88%
    Colore e forma:Beige To Brown Fine Crystalline Powder
    Peso molecolare:250.09
  • Carvedilol phosphate hemihydrate

    CAS:
    Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent.
    Formula:C24H26N2O4·5H2O·H3O4P
    Purezza:99.24% - 99.98%
    Colore e forma:Solid
    Peso molecolare:513.49
  • Erlotinib hydrochloride

    CAS:
    <p>Erlotinib hydrochloride (NSC 718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of non-small cell lung cancer.</p>
    Formula:C22H23N3O4·HCl
    Purezza:99.78% - 99.85%
    Colore e forma:White Or Off-White Powder
    Peso molecolare:429.9
  • Ezetimibe

    CAS:
    <p>Ezetimibe (SCH 58235) is a Dietary Cholesterol Absorption Inhibitor. The physiologic effect of ezetimibe is by means of Decreased Cholesterol Absorption.</p>
    Formula:C24H21F2NO3
    Purezza:97.28% - 99.77%
    Colore e forma:Solid
    Peso molecolare:409.43
  • Pyrazinamide

    CAS:
    Pyrazinamide (Pyrazinecarboxamide), an antimycobacterial, is utilized therapeutically as an antitubercular agent, which is a synthetic pyrazinoic acid amide
    Formula:C5H5N3O
    Purezza:99.71% - 99.9%
    Colore e forma:Crystals Physical Description White Powder Sublimes From 318°F (Ntp 1992)
    Peso molecolare:123.11
  • Baicalin

    CAS:
    Baicalin (Baicalein 7-O-β-D-glucuronide) is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV
    Formula:C21H18O11
    Purezza:90.08% - 99.32%
    Colore e forma:Yellow Powder
    Peso molecolare:446.36
  • 9-ING-41

    CAS:
    9-ING-41 is a glycogen synthase kinase-3 inhibitor.
    Formula:C22H13FN2O5
    Purezza:99.32%
    Colore e forma:Solid
    Peso molecolare:404.35
  • Amiodarone hydrochloride

    CAS:
    Amiodarone HCl: Antianginal, class III antiarrhythmic. Lengthens heart muscle action, slows heart rate, reduces vascular resistance.
    Formula:C25H29I2NO3·HCl
    Purezza:99.82% - ≥95%
    Colore e forma:White To Cream Crystalline Powder
    Peso molecolare:681.78
  • Itraconazole

    CAS:
    Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes required for ERGOSTEROL synthesis.
    Formula:C35H38Cl2N8O4
    Purezza:98% - 99.90%
    Colore e forma:Off-White Crystalline Solid
    Peso molecolare:705.63
  • Lomustine

    CAS:
    Lomustine (NSC-79037) is an alkylating agent of value against both hematologic malignancies and solid tumors.
    Formula:C9H16ClN3O2
    Purezza:98.36% - 99.44%
    Colore e forma:Solid Solid
    Peso molecolare:233.7
  • Taurine

    CAS:
    <p>Taurine (2-Aminoethanesulfonic acid) is an organic acid widely distributed in animal tissues and is one of the constituents of bile acids. Cost-effective and quality-assured.</p>
    Formula:C2H7NO3S
    Purezza:99.81% - 99.87%
    Colore e forma:White Crystalline Powder
    Peso molecolare:125.15
  • Naproxen

    CAS:
    Naproxen ((S)-Naproxen) is a propionic acid derivative and a non-steroidal anti-inflammatory drug (NSAID) with anti-inflammatory, antipyretic and analgesic
    Formula:C14H14O3
    Purezza:99.6% - 99.89%
    Colore e forma:Crystals From Acetone-Hexane Solid
    Peso molecolare:230.26