Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formula:C21H21D8Cl3N2O2Colore e forma:SolidPeso molecolare:455.88Methaphenilene hydrochloride
CAS:Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Formula:C15H21ClN2SPurezza:99.84%Colore e forma:SolidPeso molecolare:296.86Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formula:C18H17D3N2Colore e forma:SolidPeso molecolare:267.38Proxyfan Oxalate
CAS:Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Formula:C15H18N2O5Colore e forma:SolidPeso molecolare:306.31Amthamine
CAS:Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Formula:C6H11N3SColore e forma:SoildPeso molecolare:157.24Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Formula:C16H18N2O2Purezza:98.00%Colore e forma:SolidPeso molecolare:270.33Roxatidine acetate
CAS:Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Formula:C19H28N2O4Purezza:98%Colore e forma:White Or Off-White PowderPeso molecolare:348.44Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormula:C19H28ClN5O12Purezza:98.8%Colore e forma:SolidPeso molecolare:553.91VUF 8430 dihydrobromide
CAS:histamine H4 receptor full agonistFormula:C4H12BrN5SPurezza:98%Colore e forma:SolidPeso molecolare:242.14BMH-7
CAS:BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.Formula:C20H21N5OPurezza:99.71%Colore e forma:SolidPeso molecolare:347.41Tei 6472
CAS:Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Formula:C32H39N3O5Purezza:98%Colore e forma:SolidPeso molecolare:545.67Nα-Methylhistamine dihydrochloride
CAS:Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.Formula:C6H13Cl2N3Purezza:98%Colore e forma:SolidPeso molecolare:198.094Amthamine dihydrobromide
CAS:H2 agonistFormula:C6H13Br2N3SPurezza:98%Colore e forma:SolidPeso molecolare:319.06Carcainium chloride
CAS:Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.Formula:C18H22ClN3O2Purezza:99.89%Colore e forma:SolidPeso molecolare:347.84Bavisant dihydrochloride
CAS:Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.Formula:C19H29Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:402.36DA 4643
CAS:DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.Formula:C12H16Cl2N6SPurezza:98%Colore e forma:SolidPeso molecolare:347.26Mequitamium iodide
CAS:Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.Formula:C21H25IN2SColore e forma:SolidPeso molecolare:464.41Impentamine dihydrobromide
CAS:Impentamine dihydrobromide is a histamine H3 receptor antagonist.Formula:C8H17Br2N3Purezza:98%Colore e forma:SolidPeso molecolare:315.05Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Formula:C19H21ClN2OSColore e forma:SolidPeso molecolare:360.9AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purezza:98%Colore e forma:SolidPeso molecolare:504.53AHR-14310C
CAS:AHR-14310C is a long-acting and nonsedating H1-antihistamine.Formula:C24H28F2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:430.49NNC-38-1049
CAS:NNC-38-1049 is a novel selective antagonist of histamine H3.Formula:C19H25ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:348.87Aplysamine-1
CAS:Aplysamine-1 is an antagonist of histamine H3 receptor.Formula:C15H24Br2N2OPurezza:98%Colore e forma:SolidPeso molecolare:408.17Embramine
CAS:Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.Formula:C18H22BrNOPurezza:98%Colore e forma:SolidPeso molecolare:348.28Linadryl hydrochloride
CAS:Linadryl hydrochloride may have antihistamine activity.Formula:C19H24ClNO2Colore e forma:SolidPeso molecolare:333.85Ramixotidine
CAS:Ramixotidine is a competitive antagonist of histamine H2-receptor.Formula:C16H21N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:335.42GT 2016
CAS:GT 2016 is a H3 receptor antagonist.Formula:C19H31N3OPurezza:98%Colore e forma:SolidPeso molecolare:317.47Niperotidine
CAS:Niperotidine is an antagonist of histamine H2-receptor.Formula:C20H26N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:434.51Dacemazine hydrochloride
CAS:Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.Formula:C16H17ClN2OSPurezza:98%Colore e forma:SolidPeso molecolare:320.84JNJ-39220675
CAS:JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.Formula:C21H24FN3O2Purezza:98.13% - 99.89%Colore e forma:SolidPeso molecolare:369.43Adriforant hydrochloride
CAS:Adriforant hydrochloride is an antagonist of histamine H4 receptor.Formula:C13H25Cl3N6Purezza:98%Colore e forma:SolidPeso molecolare:371.74ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurezza:97.45%Colore e forma:SolidPeso molecolare:306.29Setastine HCl
CAS:Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.Formula:C22H29Cl2NOColore e forma:SolidPeso molecolare:394.38Seliforant
CAS:Seliforant is a histamine H4 receptor antagonist.Formula:C12H21N5Purezza:98%Colore e forma:SolidPeso molecolare:235.33A 987306
CAS:A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.Formula:C18H25N5OColore e forma:SolidPeso molecolare:327.42Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Formula:C15H20BrIN4SPurezza:98%Colore e forma:SolidPeso molecolare:495.22PF-03654746 Tosylate
CAS:PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.Formula:C25H32F2N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:494.6Hetramine
CAS:Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.Formula:C15H20N4Purezza:98%Colore e forma:SolidPeso molecolare:256.35Fenethazine
CAS:Fenethazine is an effective antihistamine used as an antiallergic drug.Formula:C16H18N2SColore e forma:SolidPeso molecolare:270.39HSR-609
CAS:HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.Formula:C21H21FN2O3Purezza:98%Colore e forma:SolidPeso molecolare:368.4Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Formula:C13H22N6Purezza:99.84%Colore e forma:SolidPeso molecolare:262.35FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:418.55ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Formula:C24H28ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:397.94H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Formula:C11H11BrN8Colore e forma:SolidPeso molecolare:335.16(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formula:C23H32N6O3SPurezza:99.54%Colore e forma:SolidPeso molecolare:472.6Ref: TM-T10000
1mg148,00€5mg284,00€10mg411,00€25mg645,00€50mg867,00€100mg1.121,00€1mL*10mM (DMSO)369,00€Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Formula:C22H24ClN3OPurezza:99.35%Colore e forma:White Crystal PowderPeso molecolare:381.90Zaltidine
CAS:Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.Formula:C8H10N6SPurezza:98%Colore e forma:SolidPeso molecolare:222.27JNJ-10191584
CAS:JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammationFormula:C13H15ClN4OColore e forma:SolidPeso molecolare:278.74Alimemazine
CAS:Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.Formula:C18H22N2SPurezza:98%Colore e forma:Crystals SolidPeso molecolare:298.45Aminopotentidine
CAS:H2 antagonistFormula:C26H35N7O2Purezza:98%Colore e forma:SolidPeso molecolare:477.6Zolantidine dimaleate
CAS:H2 receptor antagonistFormula:C26H31N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:497.61BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Formula:C12H19N5O2S2Purezza:98%Colore e forma:SolidPeso molecolare:329.44ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Formula:C22H22N2OPurezza:99.94%Colore e forma:SolidPeso molecolare:330.42Ref: TM-T14087
1mg47,00€5mg87,00€10mg140,00€25mg285,00€50mg432,00€100mg628,00€200mg879,00€1mL*10mM (DMSO)96,00€(R)-Mequitazine
CAS:(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.Formula:C20H22N2SColore e forma:SolidPeso molecolare:322.47A-304121
CAS:A-304121 is a histamine H(3) receptor.Formula:C20H29N3O3Colore e forma:SolidPeso molecolare:359.46OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Formula:C19H30ClN3SColore e forma:SolidPeso molecolare:367.98JNJ 10181457 dihydrochloride
CAS:JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.Formula:C20H28N2OPurezza:98%Colore e forma:SolidPeso molecolare:312.45Mianserin
CAS:Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.Formula:C18H20N2Purezza:99.85%Colore e forma:SolidPeso molecolare:264.36Wy 49051
CAS:Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).Formula:C28H33N5O3Purezza:99.89%Colore e forma:SolidPeso molecolare:487.59Ref: TM-T13352
1mg104,00€5mg198,00€10mg288,00€25mg452,00€50mg607,00€100mg785,00€200mg1.045,00€1mL*10mM (DMSO)264,00€ROS 234
CAS:ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.Formula:C13H15N5Colore e forma:SolidPeso molecolare:241.29Mizolastine dihydrochloride
CAS:Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).Formula:C24H27Cl2FN6OPurezza:98%Colore e forma:SolidPeso molecolare:505.42Phenyltoloxamine
CAS:Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).Formula:C17H21NOColore e forma:SolidPeso molecolare:255.35GSK334429
CAS:GSK334429 is an antagonist of histamine H3 receptor.Formula:C20H29F3N4OColore e forma:SolidPeso molecolare:398.47Sequifenadine
CAS:Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].Formula:C22H27NOColore e forma:SolidPeso molecolare:321.46A-940894
CAS:A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.Formula:C17H21N5Colore e forma:SolidPeso molecolare:295.38Immepip
CAS:Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.Formula:C9H15N3Colore e forma:SolidPeso molecolare:165.24Repirinast
CAS:Repirinast is a mediator release inhibitor. It is used to treat asthma.Formula:C20H21NO5Colore e forma:SolidPeso molecolare:355.38N-Acetylhistamine
CAS:N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.Formula:C7H11N3OPurezza:99.51%Colore e forma:SolidPeso molecolare:153.18Izuforant
CAS:Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).Formula:C12H12BrN7Colore e forma:SolidPeso molecolare:334.17A-943931
CAS:A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.Formula:C17H21N5Purezza:99.79%Colore e forma:SolidPeso molecolare:295.38Pitolisant oxalate
CAS:Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formula:C19H28ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:385.88PF-03654746
CAS:PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.Formula:C18H24F2N2OPurezza:98.85% - 99.57%Colore e forma:SolidPeso molecolare:322.39AZD5213
CAS:AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.Formula:C19H25N3O2Colore e forma:SolidPeso molecolare:327.42Pirolate
CAS:Pirolate is a receptor of histamine H1.Formula:C16H15N3O5Purezza:98%Colore e forma:SolidPeso molecolare:329.31Bepotastine tosylate
CAS:Bepotastine tosylate: Oral 2nd-gen H1 antagonist, inhibits histamine effects on NGF; treats conjunctivitis, urticaria.Formula:C28H33ClN2O6SColore e forma:SolidPeso molecolare:561.09VUF-10497
CAS:VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).Formula:C18H20ClN5SPurezza:98%Colore e forma:SolidPeso molecolare:373.9Phenindamine
CAS:Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].Formula:C19H19NColore e forma:SolidPeso molecolare:261.36Acreozast
CAS:Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.Formula:C15H14ClN3O6Colore e forma:SolidPeso molecolare:367.74CP19
CAS:CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].Formula:C26H30N2O5Colore e forma:SolidPeso molecolare:450.53Phenindamine Tartrate
CAS:Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.Formula:C23H25NO6Colore e forma:SolidPeso molecolare:411.454INCB38579
CAS:INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.Formula:C25H34N6OColore e forma:SolidPeso molecolare:434.58GSK 189254 HCl
CAS:GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.Formula:C21H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.9Nebidrazine
CAS:Nebidrazine is an alpha-adrenoceptor agonist.Formula:C9H8Cl2N6Colore e forma:SolidPeso molecolare:271.11Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purezza:98%Colore e forma:SolidPeso molecolare:392.54Loratadine N-oxide
CAS:Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.Formula:C22H23ClN2O3Colore e forma:SolidPeso molecolare:398.88MK-0249
CAS:<p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>Formula:C23H24F3N3O2Purezza:99.90%Colore e forma:SolidPeso molecolare:431.45A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColore e forma:SolidPeso molecolare:349.47SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Formula:C23H28Cl2F2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:489.38Thioperamide
CAS:histamine H3 and H4 antagonist/inverse agonistFormula:C15H24N4SPurezza:98%Colore e forma:White SolidPeso molecolare:292.44VUF 5681 dihydrobromide
CAS:histamine H3 receptor silent antagonistFormula:C11H21Br2N3Purezza:98%Colore e forma:SolidPeso molecolare:355.11VUF 8430
CAS:VUF 8430 is a selective agonist for the H4 receptor.Formula:C4H11N5SPurezza:98%Colore e forma:SolidPeso molecolare:161.23UK-9040
CAS:UK-9040 inhibits gastric secretory.Formula:C23H31NSPurezza:98%Colore e forma:SolidPeso molecolare:353.56(R)-(-)-α-Methylhistamine dihydrobromide
CAS:(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).Formula:C6H13Br2N3Purezza:98%Colore e forma:SolidPeso molecolare:287Carbinoxamine
CAS:Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.Formula:C16H19ClN2OPurezza:98%Colore e forma:LiquidPeso molecolare:290.79PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.Formula:C19H26F2N2O3Purezza:99.44%Colore e forma:SoildPeso molecolare:368.42Carcinine
CAS:Carcinine ditrifluoroacetate is a H3 receptor antagonist.Formula:C8H14N4OPurezza:98%Colore e forma:SolidPeso molecolare:182.22JNJ-28610244
CAS:JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.Formula:C16H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:271.36Setastine
CAS:Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.Formula:C22H28ClNOColore e forma:SolidPeso molecolare:357.92Rocastine
CAS:Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.Formula:C13H19N3OSPurezza:98.26%Colore e forma:SolidPeso molecolare:265.37H3 receptor-MO-1
CAS:H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.Formula:C20H27N3O2Purezza:99.11%Colore e forma:SolidPeso molecolare:341.45Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFormula:C31H37N5O3Purezza:96.68%Colore e forma:SolidPeso molecolare:527.66CP-66948
CAS:CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.Formula:C13H20N6SPurezza:99.14%Colore e forma:SolidPeso molecolare:292.4PF-03654764
CAS:PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.Formula:C20H28F2N2OPurezza:>99.99%Colore e forma:SolidPeso molecolare:350.45Lavoltidine
CAS:Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.Formula:C19H29N5O2Purezza:98.30% - 98.36%Colore e forma:SolidPeso molecolare:359.47H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Formula:C19H24ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:377.86Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Formula:C20H25ClN2OSColore e forma:SolidPeso molecolare:376.94Vapitadine dihydrochloride
CAS:Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.Formula:C17H22Cl2N4OPurezza:98.28% - 99.30%Colore e forma:SolidPeso molecolare:369.29JNJ 10191584 maleate
CAS:JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).Formula:C17H19ClN4O5Purezza:99.37%Colore e forma:SolidPeso molecolare:394.81Azatadine
CAS:Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).Formula:C20H22N2Purezza:98%Colore e forma:SolidPeso molecolare:290.4Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Formula:C14H23N7SPurezza:98%Colore e forma:SolidPeso molecolare:321.44VUF14862
CAS:VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C26H32N4O2Colore e forma:SolidPeso molecolare:432.56Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Colore e forma:SolidPeso molecolare:431.91UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Formula:C17H22N6SColore e forma:SolidPeso molecolare:342.46Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Formula:C12H9N3O2Colore e forma:SolidPeso molecolare:227.22BL 6341A
CAS:BL 6341A is related to Tumor data and H2-antagonists or anti-histaminsFormula:C9H14N8OS3Colore e forma:SolidPeso molecolare:346.46(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H24ClN3OColore e forma:SolidPeso molecolare:381.9Aceprometazine
CAS:Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].Formula:C19H22N2OSColore e forma:SolidPeso molecolare:326.46Noberastine maleate
CAS:Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.Formula:C25H29N5O9Colore e forma:SolidPeso molecolare:543.53ROS 234 dioxalate
CAS:ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)Formula:C17H19N5O8Purezza:98%Colore e forma:SolidPeso molecolare:421.37Fenspiride-d5
CAS:Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.Formula:C15H15D5N2O2Colore e forma:SolidPeso molecolare:265.36GSK-239512
CAS:GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.Formula:C23H27N3O2Purezza:99.62% - 99.74%Colore e forma:SolidPeso molecolare:377.48S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFormula:C6H11NO2SPurezza:98%Colore e forma:SolidPeso molecolare:161.22Dacemazine
CAS:Dacemazine is used to treat depression.Formula:C16H16N2OSColore e forma:SolidPeso molecolare:284.38VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C25H32N4O2Colore e forma:SolidPeso molecolare:420.55Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Formula:C19H17NO7Purezza:95% - 97.34%Colore e forma:SolidPeso molecolare:371.34Dothiepin HCl
CAS:Dothiepin HCl: TCA, SNRI, with antihistamine, antiadrenergic, anticholinergic, and sodium block properties.Formula:C19H22ClNSColore e forma:SolidPeso molecolare:331.9FR-A 19
CAS:FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.Formula:C25H34Cl3F2N5Colore e forma:SolidPeso molecolare:548.93KY 234
CAS:KY 234 is a thromboxane synthetase antagonist.Formula:C33H35N5O2Colore e forma:SolidPeso molecolare:533.676(S)-Azelastine
CAS:(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.Formula:C22H24ClN3OColore e forma:SolidPeso molecolare:381.9VUF 8328
CAS:VUF 8328 is an agonist of histamine H(3) receptor.Formula:C7H12N4SPurezza:98%Colore e forma:SolidPeso molecolare:184.26ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFormula:C24H27NO2Purezza:99.83% - 99.98%Colore e forma:SolidPeso molecolare:361.48Immethridine dihydrobromide
CAS:Immethridine dihydrobromide is a histamine H3 receptor agonist.Formula:C9H11Br2N3Purezza:97.61% - 98.14%Colore e forma:SolidPeso molecolare:321.01Proxyfan
CAS:Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Formula:C13H16N2OPurezza:99.68%Colore e forma:SolidPeso molecolare:216.28DF-1111301
CAS:DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.Formula:C15H25Cl2N3OPurezza:99.17%Colore e forma:SolidPeso molecolare:334.29Noberastine
CAS:Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.Formula:C17H21N5OPurezza:99.72% - >99.99%Colore e forma:SolidPeso molecolare:311.38KP136
CAS:KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).Formula:C16H18N4O3Purezza:98.3% - 98.61%Colore e forma:SolidPeso molecolare:314.34JZP-361
CAS:JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.Formula:C22H20ClN5OPurezza:99.82%Colore e forma:SolidPeso molecolare:405.88Pitolisant
CAS:Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formula:C17H26ClNOPurezza:99.84%Colore e forma:SolidPeso molecolare:295.85Ref: TM-T60636
5mg48,00€10mg70,00€25mg120,00€50mg188,00€100mg311,00€500mg747,00€1mL*10mM (DMSO)52,00€KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formula:C25H26N4OPurezza:99.60%Colore e forma:SolidPeso molecolare:398.5Impromidine hydrochloride
CAS:Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.Formula:C14H26Cl3N7SPurezza:99.82%Colore e forma:SolidPeso molecolare:430.83NP10679
CAS:NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.Formula:C23H26F3N3O3Purezza:99.43%Colore e forma:SolidPeso molecolare:449.47Clemastine
CAS:Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Formula:C21H26ClNOPurezza:99.21%Colore e forma:SolidPeso molecolare:343.89Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Formula:C19H27N3O2Purezza:99.21% - 99.65%Colore e forma:SolidPeso molecolare:329.44Ref: TM-TQ0046
1mg43,00€5mg96,00€10mg134,00€25mg221,00€50mg325,00€100mg465,00€500mgPrezzo su richiesta1mL*10mM (DMSO)94,00€Linetastine
CAS:Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.Formula:C35H40N2O6Purezza:99.99%Colore e forma:SolidPeso molecolare:584.7D18024
CAS:<p>D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.</p>Formula:C29H31ClFN3OPurezza:99.86%Colore e forma:SolidPeso molecolare:492.03Enerisant hydrochloride
CAS:Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteinsFormula:C22H31ClN4O3Purezza:99.95%Colore e forma:SolidPeso molecolare:434.96Abt-288
CAS:ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.Formula:C23H24N4OPurezza:98.17% - 98.49%Colore e forma:SolidPeso molecolare:372.46KSK68
CAS:KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.Formula:C23H28N2O2Purezza:99.11%Colore e forma:SolidPeso molecolare:364.48Efletirizine
CAS:Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.Formula:C21H24F2N2O3Purezza:99.39%Colore e forma:SolidPeso molecolare:390.42Antihistamine-1
CAS:Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。Formula:C23H24FN5Purezza:99.69%Colore e forma:SolidPeso molecolare:389.47Ref: TM-T10335
5mg58,00€10mg92,00€25mg177,00€50mg334,00€100mgPrezzo su richiesta1mL*10mM (DMSO)64,00€Eclazolast
CAS:<p>Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.</p>Formula:C12H12ClNO4Purezza:98.36% - 98.58%Colore e forma:SolidPeso molecolare:269.68Irdabisant
CAS:Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.Formula:C18H23N3O2Purezza:99.96%Colore e forma:SolidPeso molecolare:313.39UCB-35440
CAS:UCB-35440, a 5-lipoxygenase inhibitor and a histamine H1 receptor antagonist, is used potentially for the treatment of dermatitis.Formula:C31H34ClN5O4Colore e forma:SolidPeso molecolare:576.09Meclizine N-oxide
CAS:Meclizine N-oxide, a metabolite of the histamine H1 receptor antagonist meclizine (1), also acts as a degradation product and potential impurity in commercial meclizine preparations (2).Formula:C25H27ClN2OColore e forma:SolidPeso molecolare:407Levocabastine hydrochloride
CAS:Levocabastine HCl is an agent with antihistaminic activity.Formula:C26H30ClFN2O2Colore e forma:SolidPeso molecolare:456.98Quinotolast sodium
CAS:Quinotolast sodium inhibits histamine, LTC4 and PGD2 release in a concentration-dependent manner in the concentration range of 1-100 μg/mL.Formula:C17H12N6NaO3Purezza:98%Colore e forma:SolidPeso molecolare:371.312A-349821
CAS:A-349821 is an H3 receptor agonist radioligand.Formula:C28H35F3N2O5Colore e forma:SolidPeso molecolare:536.59CI-949
CAS:CI-949 inhibits LTC4/D4, histamine, TXB2 release (IC50: 0.5, 11.4, 0.1 μM).Formula:C20H20N6O3Purezza:98%Colore e forma:SolidPeso molecolare:392.41Ebrotidine
CAS:Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a potent antisecretory activity and evidenced gastroprotection.Formula:C14H17BrN6O2S3Purezza:97.519%Colore e forma:SolidPeso molecolare:477.42Minocromil
CAS:Minocromil is a new agent of Anti-asthmatic.Formula:C18H16N2O6Purezza:98%Colore e forma:SolidPeso molecolare:356.33GT-2331
CAS:GT-2331 is a histamine H3 receptor antagonist.Formula:C14H20N2Colore e forma:SolidPeso molecolare:216.32APD-916
CAS:APD-916, an H3 receptor antagonist, exhibits favorable pharmacokinetic properties. Oral administration of APD-916 has been demonstrated to enhance wakefulness in various animal models.Formula:C23H31NO3SColore e forma:SolidPeso molecolare:401.56Embramine hydrochloride
CAS:Embramine hydrochloride is a monoethanolamine derivative utilized for its antihistaminic and anticholinergic properties [1].Formula:C18H23BrClNOColore e forma:SolidPeso molecolare:384.74JNJ-28583867
CAS:JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.Formula:C24H32N2O2SColore e forma:SolidPeso molecolare:412.59GSK-1004723
CAS:GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.Formula:C39H49ClN4O2Colore e forma:SolidPeso molecolare:641.28Cipralisant
CAS:Cipralisant: H3 receptor antagonist (in vivo), agonist (in vitro, pKi 9.9), Ki 0.47 nM in rats, may treat ADHD.Formula:C14H20N2Purezza:98%Colore e forma:SolidPeso molecolare:216.32Hydroxydione
CAS:Hydroxydione, a neuroactive steroid with general anesthetic properties, is utilized in anesthesia-related research [1] [2].Formula:C21H32O3Colore e forma:SolidPeso molecolare:332.48Cipralisant maleate
CAS:Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.Formula:C18H24N2O4Colore e forma:SolidPeso molecolare:332.39H3 receptor antagonist 1
CAS:H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.Formula:C20H28F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:350.45Levocabastine
CAS:Levocarbastine: 2nd-gen H1 antagonist, treats allergic conjunctivitis, selective NTS2 neurotensin inhibitor.Formula:C26H29FN2O2Colore e forma:SolidPeso molecolare:420.52H4R antagonist 2
CAS:H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoidFormula:C13H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:259.31ST-1006
CAS:ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.Formula:C16H20Cl2N6Purezza:99.96% - 99.98%Colore e forma:SolidPeso molecolare:367.28Ref: TM-T34709
1mg90,00€5mg198,00€10mg316,00€25mg513,00€50mg633,00€100mg785,00€200mg1.045,00€1mL*10mM (DMSO)Prezzo su richiestaEnerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purezza:99.7%Colore e forma:SoildPeso molecolare:398.50Ref: TM-T67828
1mg52,00€2mg71,00€5mg107,00€10mg170,00€25mg359,00€50mg462,00€100mg645,00€200mg873,00€1mL*10mM (DMSO)117,00€H3R antagonist 1
CAS:H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).Formula:C19H23N3O3Colore e forma:SolidPeso molecolare:341.4Tixanox sodium
CAS:Tixanox sodium effectively blocks histamine release in the lungs triggered by anti-IgE. It has also been demonstrated that when administered orally, Tixanox sodium can successfully counteract exercise-induced asthma.Formula:C15H9NaO5SColore e forma:SolidPeso molecolare:324.28H3R antagonist 5
CAS:H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.Formula:C23H32N2O4Colore e forma:SolidPeso molecolare:400.511CI-624
CAS:CI-624 reduces the secretion and output of hydrogen ions, sodium ions, potassium ions, and pepsin. This compound may be utilized in research focusing on cancer and autoimmune diseases.Formula:C8H8N2SColore e forma:SolidPeso molecolare:164.228H1R ligand-1
CAS:<p>H1R ligand-1 (Compound fragment 1) is a high-affinity ligand for the human histamine H1 receptor (H1R). It can serve as a scaffold for synthesizing a series of derivatives to investigate H1R binding kinetics.</p>Formula:C19H23NOColore e forma:SolidPeso molecolare:281.392Sitamaquine hydrochloride
CAS:Sitamaquine hydrochloride (WR 6026) is an orally active 8-aminoquinoline analog with antileishmanial activity. This compound inhibits mitochondrial complex II (succinate dehydrogenase) and is characterized by its lipophilic weak base properties. It rapidly accumulates in the acidic compartments of Leishmania parasites, predominantly localizing within the acidocalcisomes.Formula:C21H35Cl2N3OColore e forma:SolidPeso molecolare:416.43Arpromidine
CAS:Arpromidine (BU-E-50) acts as an agonist for the histamine H2 receptor and an antagonist for the histamine H1 receptor. It demonstrates positive inotropic effects with a lower risk of inducing arrhythmias. Arpromidine can be utilized in studies related to congestive heart failure.Formula:C21H25FN6Colore e forma:SolidPeso molecolare:380.462Nedocromil sodium
CAS:Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Formula:C19H17NNaO7Purezza:98%Colore e forma:SolidPeso molecolare:394.335Histamine H3 antagonist-1
CAS:<p>Compound 10o, a histamine H3 antagonist-1, functions as both a histamine H3 antagonist and a serotonin reuptake inhibitor, making it useful for research in depression [1].</p>Formula:C24H28F3N3O2Colore e forma:SolidPeso molecolare:447.49ONO-8809
CAS:ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.Formula:C30H46BrNO4SPurezza:98%Colore e forma:SolidPeso molecolare:596.66(R)-(-)-α-Methylhistamine dihydrochloride
CAS:R(-)-alpha-Methylhistamine 2HCl is an effective and selective agonist of the H3 histamine receptor.Formula:C6H13Cl2N3Colore e forma:SolidPeso molecolare:198.09Imetit dihydrobromide
CAS:Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM).Formula:C6H12Br2N4SPurezza:98%Colore e forma:SolidPeso molecolare:332.06
