Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurezza:99.77% - >99.99%Colore e forma:White To Slightly Yellowish Crystalline SolidPeso molecolare:341.88Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formula:C21H27Cl3N2O3Purezza:99.4% - 99.97%Colore e forma:SolidPeso molecolare:461.81Mepyramine maleate
CAS:Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Formula:C21H27N3O5Purezza:99.51% - 99.7%Colore e forma:White Crystalline PowderPeso molecolare:401.47Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurezza:99.85%Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecolare:320.88Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Formula:C13H16N4Purezza:98.34% - 99.73%Colore e forma:SolidPeso molecolare:228.29Amitriptyline hydrochloride
CAS:Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFormula:C20H24ClNPurezza:97% - 99.94%Colore e forma:Crystals White To Off-White PowderPeso molecolare:313.86Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formula:C19H19NSPurezza:97.50%Colore e forma:SolidPeso molecolare:293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€Loratadine
CAS:<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Formula:C22H23ClN2O2Purezza:99.71% - 99.98%Colore e forma:White PowderPeso molecolare:382.88Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formula:C16H20N2·C4H4O4Purezza:99.85%Colore e forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecolare:356.42Chlorpheniramine maleate
CAS:Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Formula:C20H23ClN2O4Purezza:99.64% - 99.98%Colore e forma:Odorless White Crystalline Solid Or White Powder With A Bitter TastePeso molecolare:390.87KSK67
CAS:KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with KiFormula:C22H27N3O2Purezza:99.94%Colore e forma:SoildPeso molecolare:365.47Betahistine mesylate
CAS:<p>Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.</p>Formula:C8H12N2·2(CH4O3S)Purezza:98% - 99.85%Colore e forma:CoaPeso molecolare:328.4Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonistFormula:C7H13N3O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:171.2Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Formula:C21H31N3O3Purezza:99.59%Colore e forma:SolidPeso molecolare:373.49Ref: TM-T9770
1mg111,00€2mg166,00€5mg274,00€10mg439,00€25mg725,00€50mg1.017,00€100mg1.359,00€500mg2.745,00€1mL*10mM (DMSO)283,00€Methapyrilene hydrochloride
CAS:Methapyrilene hydrochloride is a biochemical.Formula:C14H20ClN3SColore e forma:Liquid Solution) 5 5 (Ntp 1992)Peso molecolare:297.85Tecastemizole
CAS:Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formula:C19H21FN4Purezza:99.70%Colore e forma:SolidPeso molecolare:324.4Ref: TM-T26253
1mg57,00€5mg125,00€10mg177,00€25mg304,00€50mg437,00€100mg615,00€500mg1.225,00€1mL*10mM (DMSO)138,00€KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Formula:C26H28N4O3Purezza:97.51%Colore e forma:SoildPeso molecolare:444.53Cetirizine D8 dihydrochloride
CAS:Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.Formula:C21H26Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:433.4Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formula:C20H25N5O3SPurezza:99.32%Colore e forma:SolidPeso molecolare:415.51Histamine H4 receptor antagonist-1
CAS:Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.Formula:C30H38N8O2Colore e forma:SolidPeso molecolare:542.68Sufotidine
CAS:Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.Formula:C20H31N5O3SPurezza:99.03% - 99.92%Colore e forma:SolidPeso molecolare:421.56Thioperamide maleate
CAS:Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formula:C19H28N4O4SPurezza:98.48%Colore e forma:SolidPeso molecolare:408.52Conessine hydrobromide
CAS:Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Formula:C24H41BrN2Colore e forma:SolidPeso molecolare:437.51Diphenhydramine hydrochloride
CAS:<p>DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.</p>Formula:C17H22ClNOPurezza:99.84%Colore e forma:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Peso molecolare:291.82Dalcotidine
CAS:<p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>Formula:C18H29N3O2Purezza:99.11%Colore e forma:SolidPeso molecolare:319.44Sigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFormula:C26H27N3OPurezza:98%Colore e forma:SolidPeso molecolare:397.51Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Colore e forma:Odour SolidOxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.Formula:C20H23N5O5SPurezza:97.34%Colore e forma:SoildPeso molecolare:445.49Bodilisant
CAS:Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.Formula:C27H34BF2N3OColore e forma:SolidPeso molecolare:465.4Nizatidine
CAS:Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Formula:C12H21N5O2S2Purezza:99.43%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:331.46Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Formula:C21H25ClN2O3Colore e forma:SolidPeso molecolare:388.89Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurezza:99.77% - 99.86%Colore e forma:SoildPeso molecolare:296.37Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formula:C21H27Cl3N2O3Colore e forma:SolidPeso molecolare:461.81H4R antagonist 3
CAS:H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFormula:C19H21ClN4SPurezza:98%Colore e forma:SolidPeso molecolare:372.924-Methylhistamine
CAS:4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer andFormula:C6H11N3Purezza:98%Colore e forma:SolidPeso molecolare:125.17Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Colore e forma:SolidPeso molecolare:341.091Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Formula:C19H21N3O2Colore e forma:SolidPeso molecolare:323.39Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Colore e forma:Odour SolidDexchlorpheniramine free base
CAS:Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Formula:C16H19ClN2Purezza:98%Colore e forma:Oily Liquid SolidPeso molecolare:274.79JNJ-10181457 (hydrochloride)
CAS:JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFormula:C20H30Cl2N2OColore e forma:SolidPeso molecolare:385.37Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formula:C10H20ClNO4Purezza:90% - 99.77%Colore e forma:SolidPeso molecolare:253.72(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H25Cl2N3OPurezza:98%Colore e forma:SolidPeso molecolare:418.363-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Formula:C19H19ClN2OColore e forma:SolidPeso molecolare:326.82(+)-Dropropizine
CAS:(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.Formula:C13H20N2O2Purezza:>99.99%Colore e forma:White Or Off White Crystalline PowderPeso molecolare:236.31Cetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Formula:C30H28Cl2N2Colore e forma:SolidPeso molecolare:487.46Cetirizine methyl ester
CAS:Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Formula:C22H27ClN2O3Colore e forma:SolidPeso molecolare:402.91AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Formula:C27H19F3N4O4SColore e forma:SolidPeso molecolare:552.52Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Formula:C19H21N5O3SPurezza:99.67%Colore e forma:SolidPeso molecolare:399.47Ref: TM-T68122
1mg378,00€5mg895,00€10mg1.216,00€25mg1.786,00€50mg2.442,00€100mg3.287,00€500mg6.603,00€Alimemazine D6
CAS:Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formula:C18H22N2SPurezza:98%Colore e forma:SolidPeso molecolare:304.48Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formula:C17H22N3O4PPurezza:98%Colore e forma:CoaPeso molecolare:363.35
