Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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Hydroxyzine D8
CAS:Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Formula:C21H27ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:382.95Alimemazine D6
CAS:Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formula:C18H22N2SPurezza:98%Colore e forma:SolidPeso molecolare:304.481-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS:MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formula:C6H9ClN2O2Colore e forma:SolidPeso molecolare:176.601Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Formula:C10H16N8S2Purezza:98%Colore e forma:SolidPeso molecolare:312.42Acrivastine D7
CAS:Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.Formula:C22H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:355.48Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formula:C32H39NO4Purezza:98%Colore e forma:SolidPeso molecolare:507.69Emedastine Difumarate
CAS:Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formula:C25H34N4O9Colore e forma:SolidPeso molecolare:534.56Diphenylpyraline
CAS:Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.Formula:C19H23NOColore e forma:SolidPeso molecolare:281.39Gizzerosine
CAS:Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.Formula:C11H20N4O2Colore e forma:SolidPeso molecolare:240.3WZ4141
CAS:WZ4141 is an intermediate in compound synthesis.Formula:C16H13N3O2Purezza:98%Colore e forma:SolidPeso molecolare:279.29Doxepin D3 Hydrochloride
CAS:Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 andFormula:C19H22ClNOPurezza:98%Colore e forma:SolidPeso molecolare:318.86Cetirizine D8
CAS:Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formula:C21H25ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:396.94Cetirizine D4
CAS:Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formula:C21H25ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:392.91Clobenpropit dihydrobromide
CAS:Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)Formula:C14H19Br2ClN4SPurezza:99.86%Colore e forma:SolidPeso molecolare:470.7Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purezza:≥95%Colore e forma:White Crystalline Powder SolidPeso molecolare:265.35Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formula:C15H19N3Purezza:≥95%Colore e forma:SolidPeso molecolare:241.33Fenspiride
CAS:Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.Formula:C15H20N2O2Colore e forma:SolidPeso molecolare:260.33Emedastine
CAS:Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.Formula:C17H26N4OPurezza:97.1% - 97.76%Colore e forma:OilPeso molecolare:302.41Ref: TM-T3979
1mg37,00€5mg79,00€10mg115,00€25mg187,00€50mg279,00€100mg415,00€500mg933,00€1mL*10mM (DMSO)87,00€Fexofenadine hydrochloride
CAS:Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,Formula:C32H39NO4·HClPurezza:99.39% - ≥95%Colore e forma:SolidPeso molecolare:538.13Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formula:C17H18O9Purezza:99.03% - 99.49%Colore e forma:SolidPeso molecolare:366.32Ref: TM-TN1008
1mg96,00€2mg139,00€5mg227,00€10mg364,00€25mg600,00€50mg845,00€100mg1.121,00€1mL*10mM (DMSO)235,00€Conessine
CAS:<p>Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.</p>Formula:C24H40N2Purezza:99.65%Colore e forma:SolidPeso molecolare:356.59Chlorpheniramine
CAS:Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.Formula:C16H19ClN2Colore e forma:SolidPeso molecolare:274.79Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColore e forma:SolidPeso molecolare:228.21Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formula:C21H27ClN2O2Purezza:99.54% - ≥95%Colore e forma:Oil SolidPeso molecolare:374.9Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purezza:>99.99%Colore e forma:SolidPeso molecolare:362.3SCH-37370
CAS:SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Formula:C21H21ClN2OPurezza:99.07%Colore e forma:SolidPeso molecolare:352.86Ref: TM-T19686
1mg48,00€5mg89,00€10mg115,00€25mg195,00€50mg290,00€100mg393,00€200mg520,00€1mL*10mM (DMSO)90,00€H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurezza:98.81%Colore e forma:SolidPeso molecolare:316.79GSK189254A
CAS:GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Formula:C21H25N3O2Purezza:98.71% - 99.858%Colore e forma:SolidPeso molecolare:351.44Ref: TM-TQ0066
1mg52,00€5mg88,00€10mg120,00€25mg216,00€50mg350,00€100mg505,00€200mg727,00€1mL*10mM (DMSO)67,00€S 38093
CAS:S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formula:C17H24N2O2Purezza:99.95%Colore e forma:SolidPeso molecolare:288.38Ref: TM-T4099
2mg38,00€5mg52,00€10mg80,00€25mg131,00€50mg210,00€100mg334,00€200mg467,00€1mL*10mM (DMSO)52,00€Bilastine
CAS:Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration ofFormula:C28H37N3O3Purezza:99.86% - >99.99%Colore e forma:SolidPeso molecolare:463.61Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Colore e forma:SolidPeso molecolare:314.852Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:356.44Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurezza:99.78%Colore e forma:SolidPeso molecolare:331.86Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFormula:C21H28N2O2Purezza:99.53%Colore e forma:White Or Similar To White PowderPeso molecolare:340.46Clobenpropit 2HBr
CAS:Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formula:C14H17ClN4SColore e forma:SolidPeso molecolare:308.83Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purezza:99.13% - 99.81%Colore e forma:SolidPeso molecolare:311.63Osthole
CAS:Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Formula:C15H16O3Purezza:99.93% - 99.96%Colore e forma:Fine White PowderPeso molecolare:244.29HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purezza:99.51%Colore e forma:SolidPeso molecolare:614.57Triprolidine
CAS:Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formula:C19H22N2Colore e forma:SolidPeso molecolare:278.39Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purezza:98.25%Colore e forma:SolidPeso molecolare:233.182-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purezza:99.42%Colore e forma:SolidPeso molecolare:195.09Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Formula:C8H12N2Purezza:99.87% - 99.87%Colore e forma:Yellowish Liquid Liquid LiquidPeso molecolare:136.19Dioxopromethazine
CAS:Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formula:C17H20N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:316.42Buclizine
CAS:Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Formula:C28H33ClN2Colore e forma:SolidPeso molecolare:433.03Desloratadine
CAS:Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.Formula:C19H19ClN2Purezza:99.79% - >99.99%Colore e forma:SolidPeso molecolare:310.82C-Type Natriuretic Peptide (CNP) (1-22), human
CAS:C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Formula:C93H157N27O28S3Purezza:>99.99%Colore e forma:SolidPeso molecolare:2197.6Ref: TM-TP1187
1mg119,00€5mg414,00€10mg658,00€25mg945,00€50mg1.264,00€100mg1.700,00€200mg2.270,00€500µg88,00€Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formula:C32H39NO4Purezza:99.35%Colore e forma:White To Off-White SolidPeso molecolare:501.66Tiaramide hydrochloride
CAS:Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formula:C15H19Cl2N3O3SPurezza:98.48%Colore e forma:SolidPeso molecolare:392.3Ref: TM-T28972
1mg70,00€5mg137,00€10mg187,00€25mg315,00€50mg472,00€100mg658,00€200mg930,00€1mL*10mM (DMSO)144,00€JNJ-5207852 dihydrochloride
CAS:JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFormula:C20H34Cl2N2OPurezza:99.51%Colore e forma:SolidPeso molecolare:389.4
