Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formula:C21H21D8Cl3N2O2Colore e forma:SolidPeso molecolare:455.88Methaphenilene hydrochloride
CAS:Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Formula:C15H21ClN2SPurezza:99.84%Colore e forma:SolidPeso molecolare:296.86Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formula:C18H17D3N2Colore e forma:SolidPeso molecolare:267.38Proxyfan Oxalate
CAS:Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Formula:C15H18N2O5Colore e forma:SolidPeso molecolare:306.31Amthamine
CAS:Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Formula:C6H11N3SColore e forma:SoildPeso molecolare:157.24Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Formula:C16H18N2O2Purezza:98.00%Colore e forma:SolidPeso molecolare:270.33Roxatidine acetate
CAS:Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Formula:C19H28N2O4Purezza:98%Colore e forma:White Or Off-White PowderPeso molecolare:348.44Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormula:C19H28ClN5O12Purezza:98.8%Colore e forma:SolidPeso molecolare:553.91VUF 8430 dihydrobromide
CAS:histamine H4 receptor full agonistFormula:C4H12BrN5SPurezza:98%Colore e forma:SolidPeso molecolare:242.14BMH-7
CAS:BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.Formula:C20H21N5OPurezza:99.71%Colore e forma:SolidPeso molecolare:347.41Tei 6472
CAS:Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Formula:C32H39N3O5Purezza:98%Colore e forma:SolidPeso molecolare:545.67Nα-Methylhistamine dihydrochloride
CAS:Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.Formula:C6H13Cl2N3Purezza:98%Colore e forma:SolidPeso molecolare:198.094Amthamine dihydrobromide
CAS:H2 agonistFormula:C6H13Br2N3SPurezza:98%Colore e forma:SolidPeso molecolare:319.06Carcainium chloride
CAS:Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.Formula:C18H22ClN3O2Purezza:99.89%Colore e forma:SolidPeso molecolare:347.84Bavisant dihydrochloride
CAS:Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.Formula:C19H29Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:402.36DA 4643
CAS:DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.Formula:C12H16Cl2N6SPurezza:98%Colore e forma:SolidPeso molecolare:347.26Mequitamium iodide
CAS:Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.Formula:C21H25IN2SColore e forma:SolidPeso molecolare:464.41Impentamine dihydrobromide
CAS:Impentamine dihydrobromide is a histamine H3 receptor antagonist.Formula:C8H17Br2N3Purezza:98%Colore e forma:SolidPeso molecolare:315.05Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Formula:C19H21ClN2OSColore e forma:SolidPeso molecolare:360.9AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purezza:98%Colore e forma:SolidPeso molecolare:504.53AHR-14310C
CAS:AHR-14310C is a long-acting and nonsedating H1-antihistamine.Formula:C24H28F2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:430.49NNC-38-1049
CAS:NNC-38-1049 is a novel selective antagonist of histamine H3.Formula:C19H25ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:348.87Aplysamine-1
CAS:Aplysamine-1 is an antagonist of histamine H3 receptor.Formula:C15H24Br2N2OPurezza:98%Colore e forma:SolidPeso molecolare:408.17Embramine
CAS:Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.Formula:C18H22BrNOPurezza:98%Colore e forma:SolidPeso molecolare:348.28Linadryl hydrochloride
CAS:Linadryl hydrochloride may have antihistamine activity.Formula:C19H24ClNO2Colore e forma:SolidPeso molecolare:333.85Ramixotidine
CAS:Ramixotidine is a competitive antagonist of histamine H2-receptor.Formula:C16H21N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:335.42GT 2016
CAS:GT 2016 is a H3 receptor antagonist.Formula:C19H31N3OPurezza:98%Colore e forma:SolidPeso molecolare:317.47Niperotidine
CAS:Niperotidine is an antagonist of histamine H2-receptor.Formula:C20H26N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:434.51Dacemazine hydrochloride
CAS:Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.Formula:C16H17ClN2OSPurezza:98%Colore e forma:SolidPeso molecolare:320.84JNJ-39220675
CAS:JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.Formula:C21H24FN3O2Purezza:98.13% - 99.89%Colore e forma:SolidPeso molecolare:369.43Adriforant hydrochloride
CAS:Adriforant hydrochloride is an antagonist of histamine H4 receptor.Formula:C13H25Cl3N6Purezza:98%Colore e forma:SolidPeso molecolare:371.74ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurezza:97.45%Colore e forma:SolidPeso molecolare:306.29Setastine HCl
CAS:Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.Formula:C22H29Cl2NOColore e forma:SolidPeso molecolare:394.38Seliforant
CAS:Seliforant is a histamine H4 receptor antagonist.Formula:C12H21N5Purezza:98%Colore e forma:SolidPeso molecolare:235.33A 987306
CAS:A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.Formula:C18H25N5OColore e forma:SolidPeso molecolare:327.42Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Formula:C15H20BrIN4SPurezza:98%Colore e forma:SolidPeso molecolare:495.22PF-03654746 Tosylate
CAS:PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.Formula:C25H32F2N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:494.6Hetramine
CAS:Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.Formula:C15H20N4Purezza:98%Colore e forma:SolidPeso molecolare:256.35Fenethazine
CAS:Fenethazine is an effective antihistamine used as an antiallergic drug.Formula:C16H18N2SColore e forma:SolidPeso molecolare:270.39HSR-609
CAS:HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.Formula:C21H21FN2O3Purezza:98%Colore e forma:SolidPeso molecolare:368.4Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Formula:C13H22N6Purezza:99.84%Colore e forma:SolidPeso molecolare:262.35FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:418.55ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Formula:C24H28ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:397.94H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Formula:C11H11BrN8Colore e forma:SolidPeso molecolare:335.16(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formula:C23H32N6O3SPurezza:99.54%Colore e forma:SolidPeso molecolare:472.6Ref: TM-T10000
1mg148,00€5mg284,00€10mg411,00€25mg645,00€50mg867,00€100mg1.121,00€1mL*10mM (DMSO)369,00€Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Formula:C22H24ClN3OPurezza:99.35%Colore e forma:White Crystal PowderPeso molecolare:381.90Zaltidine
CAS:Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.Formula:C8H10N6SPurezza:98%Colore e forma:SolidPeso molecolare:222.27JNJ-10191584
CAS:JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammationFormula:C13H15ClN4OColore e forma:SolidPeso molecolare:278.74Alimemazine
CAS:Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.Formula:C18H22N2SPurezza:98%Colore e forma:Crystals SolidPeso molecolare:298.45Aminopotentidine
CAS:H2 antagonistFormula:C26H35N7O2Purezza:98%Colore e forma:SolidPeso molecolare:477.6
