
Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formula:C21H21D8Cl3N2O2Colore e forma:SolidPeso molecolare:455.88Methaphenilene hydrochloride
CAS:Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Formula:C15H21ClN2SPurezza:99.84%Colore e forma:SolidPeso molecolare:296.86Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formula:C18H17D3N2Colore e forma:SolidPeso molecolare:267.38Proxyfan Oxalate
CAS:Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Formula:C15H18N2O5Colore e forma:SolidPeso molecolare:306.31Amthamine
CAS:Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Formula:C6H11N3SColore e forma:SoildPeso molecolare:157.24Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Formula:C16H18N2O2Purezza:98.00%Colore e forma:SolidPeso molecolare:270.33Roxatidine acetate
CAS:Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Formula:C19H28N2O4Purezza:98%Colore e forma:White Or Off-White PowderPeso molecolare:348.44Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormula:C19H28ClN5O12Purezza:98.8%Colore e forma:SolidPeso molecolare:553.91VUF 8430 dihydrobromide
CAS:histamine H4 receptor full agonistFormula:C4H12BrN5SPurezza:98%Colore e forma:SolidPeso molecolare:242.14BMH-7
CAS:BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.Formula:C20H21N5OPurezza:99.71%Colore e forma:SolidPeso molecolare:347.41Tei 6472
CAS:Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Formula:C32H39N3O5Purezza:98%Colore e forma:SolidPeso molecolare:545.67Nα-Methylhistamine dihydrochloride
CAS:Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.Formula:C6H13Cl2N3Purezza:98%Colore e forma:SolidPeso molecolare:198.094Amthamine dihydrobromide
CAS:H2 agonistFormula:C6H13Br2N3SPurezza:98%Colore e forma:SolidPeso molecolare:319.06Carcainium chloride
CAS:Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.Formula:C18H22ClN3O2Purezza:99.89%Colore e forma:SolidPeso molecolare:347.84Bavisant dihydrochloride
CAS:Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.Formula:C19H29Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:402.36DA 4643
CAS:DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.Formula:C12H16Cl2N6SPurezza:98%Colore e forma:SolidPeso molecolare:347.26Mequitamium iodide
CAS:Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.Formula:C21H25IN2SColore e forma:SolidPeso molecolare:464.41Impentamine dihydrobromide
CAS:Impentamine dihydrobromide is a histamine H3 receptor antagonist.Formula:C8H17Br2N3Purezza:98%Colore e forma:SolidPeso molecolare:315.05Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Formula:C19H21ClN2OSColore e forma:SolidPeso molecolare:360.9AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purezza:98%Colore e forma:SolidPeso molecolare:504.53
