Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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GT-2331
CAS:GT-2331 is a histamine H3 receptor antagonist.Formula:C14H20N2Colore e forma:SolidPeso molecolare:216.32APD-916
CAS:APD-916, an H3 receptor antagonist, exhibits favorable pharmacokinetic properties. Oral administration of APD-916 has been demonstrated to enhance wakefulness in various animal models.Formula:C23H31NO3SColore e forma:SolidPeso molecolare:401.56Embramine hydrochloride
CAS:Embramine hydrochloride is a monoethanolamine derivative utilized for its antihistaminic and anticholinergic properties [1].Formula:C18H23BrClNOColore e forma:SolidPeso molecolare:384.74JNJ-28583867
CAS:JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.Formula:C24H32N2O2SColore e forma:SolidPeso molecolare:412.59GSK-1004723
CAS:GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.Formula:C39H49ClN4O2Colore e forma:SolidPeso molecolare:641.28Cipralisant
CAS:Cipralisant: H3 receptor antagonist (in vivo), agonist (in vitro, pKi 9.9), Ki 0.47 nM in rats, may treat ADHD.Formula:C14H20N2Purezza:98%Colore e forma:SolidPeso molecolare:216.32Hydroxydione
CAS:Hydroxydione, a neuroactive steroid with general anesthetic properties, is utilized in anesthesia-related research [1] [2].Formula:C21H32O3Colore e forma:SolidPeso molecolare:332.48Cipralisant maleate
CAS:Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.Formula:C18H24N2O4Colore e forma:SolidPeso molecolare:332.39H3 receptor antagonist 1
CAS:H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.Formula:C20H28F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:350.45Levocabastine
CAS:Levocarbastine: 2nd-gen H1 antagonist, treats allergic conjunctivitis, selective NTS2 neurotensin inhibitor.Formula:C26H29FN2O2Colore e forma:SolidPeso molecolare:420.52H4R antagonist 2
CAS:H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoidFormula:C13H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:259.31ST-1006
CAS:ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.Formula:C16H20Cl2N6Purezza:99.96% - 99.98%Colore e forma:SolidPeso molecolare:367.28Ref: TM-T34709
1mg90,00€5mg198,00€10mg316,00€25mg513,00€50mg633,00€100mg785,00€200mg1.045,00€1mL*10mM (DMSO)Prezzo su richiestaEnerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purezza:99.7%Colore e forma:SoildPeso molecolare:398.50Ref: TM-T67828
1mg52,00€2mg71,00€5mg107,00€10mg170,00€25mg359,00€50mg462,00€100mg645,00€200mg873,00€1mL*10mM (DMSO)117,00€H3R antagonist 1
CAS:H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).Formula:C19H23N3O3Colore e forma:SolidPeso molecolare:341.4Tixanox sodium
CAS:Tixanox sodium effectively blocks histamine release in the lungs triggered by anti-IgE. It has also been demonstrated that when administered orally, Tixanox sodium can successfully counteract exercise-induced asthma.Formula:C15H9NaO5SColore e forma:SolidPeso molecolare:324.28H3R antagonist 5
CAS:H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.Formula:C23H32N2O4Colore e forma:SolidPeso molecolare:400.511CI-624
CAS:CI-624 reduces the secretion and output of hydrogen ions, sodium ions, potassium ions, and pepsin. This compound may be utilized in research focusing on cancer and autoimmune diseases.Formula:C8H8N2SColore e forma:SolidPeso molecolare:164.228H1R ligand-1
CAS:<p>H1R ligand-1 (Compound fragment 1) is a high-affinity ligand for the human histamine H1 receptor (H1R). It can serve as a scaffold for synthesizing a series of derivatives to investigate H1R binding kinetics.</p>Formula:C19H23NOColore e forma:SolidPeso molecolare:281.392Sitamaquine hydrochloride
CAS:Sitamaquine hydrochloride (WR 6026) is an orally active 8-aminoquinoline analog with antileishmanial activity. This compound inhibits mitochondrial complex II (succinate dehydrogenase) and is characterized by its lipophilic weak base properties. It rapidly accumulates in the acidic compartments of Leishmania parasites, predominantly localizing within the acidocalcisomes.Formula:C21H35Cl2N3OColore e forma:SolidPeso molecolare:416.43Arpromidine
CAS:Arpromidine (BU-E-50) acts as an agonist for the histamine H2 receptor and an antagonist for the histamine H1 receptor. It demonstrates positive inotropic effects with a lower risk of inducing arrhythmias. Arpromidine can be utilized in studies related to congestive heart failure.Formula:C21H25FN6Colore e forma:SolidPeso molecolare:380.462
