
Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Formula:C21H25ClN2O3Colore e forma:SolidPeso molecolare:388.89Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurezza:99.77% - 99.86%Colore e forma:SoildPeso molecolare:296.37Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formula:C21H27Cl3N2O3Colore e forma:SolidPeso molecolare:461.81H4R antagonist 3
CAS:H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFormula:C19H21ClN4SPurezza:98%Colore e forma:SolidPeso molecolare:372.924-Methylhistamine
CAS:<p>4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and</p>Formula:C6H11N3Purezza:98%Colore e forma:SolidPeso molecolare:125.17Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Colore e forma:SolidPeso molecolare:341.091Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Formula:C19H21N3O2Colore e forma:SolidPeso molecolare:323.39Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Colore e forma:Odour SolidDexchlorpheniramine free base
CAS:Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Formula:C16H19ClN2Purezza:98%Colore e forma:Oily Liquid SolidPeso molecolare:274.79JNJ-10181457 (hydrochloride)
CAS:JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFormula:C20H30Cl2N2OColore e forma:SolidPeso molecolare:385.37Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formula:C10H20ClNO4Purezza:90% - 99.77%Colore e forma:SolidPeso molecolare:253.72(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H25Cl2N3OPurezza:98%Colore e forma:SolidPeso molecolare:418.363-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Formula:C19H19ClN2OColore e forma:SolidPeso molecolare:326.82(+)-Dropropizine
CAS:(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.Formula:C13H20N2O2Purezza:>99.99%Colore e forma:White Or Off White Crystalline PowderPeso molecolare:236.31Cetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Formula:C30H28Cl2N2Colore e forma:SolidPeso molecolare:487.46Cetirizine methyl ester
CAS:Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Formula:C22H27ClN2O3Colore e forma:SolidPeso molecolare:402.91AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Formula:C27H19F3N4O4SColore e forma:SolidPeso molecolare:552.52Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Formula:C19H21N5O3SPurezza:99.67%Colore e forma:SolidPeso molecolare:399.47Alimemazine D6
CAS:Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formula:C18H22N2SPurezza:98%Colore e forma:SolidPeso molecolare:304.48Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formula:C17H22N3O4PPurezza:98%Colore e forma:CoaPeso molecolare:363.35
