
Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 389 prodotti per "Recettore dell'istamina".
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2-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purezza:99.42%Colore e forma:SolidPeso molecolare:195.09cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formula:C16H14O2Purezza:98.15%Colore e forma:SolidPeso molecolare:238.2812Ref: TM-T8586
1mg58,00€1mL*10mM (DMSO)105,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€SCH-37370
CAS:SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Formula:C21H21ClN2OPurezza:99.07%Colore e forma:White SolidPeso molecolare:352.86Ref: TM-T19686
1mg46,00€5mg85,00€1mL*10mM (DMSO)86,00€10mg109,00€25mg185,00€50mg275,00€100mg371,00€200mg494,00€Acitazanolast
CAS:Acitazanolast (WP-871) is an anti-allergic drug candidate.Formula:C9H7N5O3Purezza:98.25%Colore e forma:SolidPeso molecolare:233.18Hydroxyzine
CAS:Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formula:C21H27ClN2O2Purezza:98.7% - ≥95%Colore e forma:SolidPeso molecolare:374.9Fenspiride
CAS:Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.Formula:C15H20N2O2Colore e forma:SolidPeso molecolare:260.33Tribenoside
CAS:Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formula:C29H34O6Purezza:≥98%Colore e forma:Yellow OilPeso molecolare:478.58Lodoxamide
CAS:Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formula:C11H6ClN3O6Purezza:99.13% - 99.96%Colore e forma:SolidPeso molecolare:311.63Bilastine
CAS:Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration ofFormula:C28H37N3O3Purezza:99.86% - >99.99%Colore e forma:White SolidPeso molecolare:463.61Conessine
CAS:Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.Formula:C24H40N2Purezza:99.65% - 99.93%Colore e forma:SolidPeso molecolare:356.59H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurezza:98.81%Colore e forma:SolidPeso molecolare:316.79C-Type Natriuretic Peptide (CNP) (1-22), human
CAS:C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Formula:C93H157N27O28S3Purezza:>99.99%Colore e forma:White SolidPeso molecolare:2197.6Ref: TM-TP1187
500µg84,00€1mg113,00€5mg391,00€10mg623,00€25mg895,00€50mg1.198,00€100mg1.611,00€200mg2.152,00€Tiaramide hydrochloride
CAS:Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formula:C15H19Cl2N3O3SPurezza:98.48%Colore e forma:SolidPeso molecolare:392.3Ref: TM-T28972
1mg66,00€5mg130,00€1mL*10mM (DMSO)137,00€10mg177,00€25mg299,00€50mg447,00€100mg623,00€200mg882,00€Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColore e forma:SolidPeso molecolare:228.21HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purezza:99.51%Colore e forma:SolidPeso molecolare:614.57Bepotastine Besilate
CAS:Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).Formula:C21H25ClN2O3·C6H6O3SPurezza:99.83% - 99.9%Colore e forma:Brown Viscous LiquidPeso molecolare:547.06Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurezza:99.79%Colore e forma:SolidPeso molecolare:234.19Clobenpropit 2HBr
CAS:Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formula:C14H17ClN4SColore e forma:SolidPeso molecolare:308.83VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Formula:C15H19N5Purezza:99.44% - 99.57%Colore e forma:SolidPeso molecolare:269.34Buclizine
CAS:Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Formula:C28H33ClN2Colore e forma:SolidPeso molecolare:433.03
