Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 326 prodotti di "Recettore degli oppioidi"
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BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Formula:C29H39N5O7Purezza:>99.99%Colore e forma:SolidPeso molecolare:569.65Ref: TM-TP1905
2mg42,00€5mg62,00€10mg87,00€25mg154,00€50mg274,00€100mg487,00€200mg692,00€1mL*10mM (DMSO)78,00€DAMGO TFA (78123-71-4(Free base))
DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.Formula:C28H36F3N5O8Purezza:98.67% - 99.76%Colore e forma:SolidPeso molecolare:627.6Asimadoline hydrochloride
CAS:Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.Formula:C27H31ClN2O2Purezza:98.94% - 99.32%Colore e forma:SolidPeso molecolare:451.01Ref: TM-T4691
1mg35,00€5mg73,00€10mg111,00€25mg227,00€50mg338,00€100mg500,00€500mg1.074,00€1mL*10mM (DMSO)81,00€Endomorphin 1
CAS:Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).Formula:C34H38N6O5Purezza:95.92%Colore e forma:Solid (Solid Powder )Peso molecolare:610.7Salvinorin A
CAS:Salvinorin A is a non-nitrogenous κ-opioid selective agonist.Formula:C23H28O8Purezza:99.06%Colore e forma:SolidPeso molecolare:432.46Ref: TM-T23306
1mg274,00€5mg663,00€10mg947,00€25mg1.415,00€50mg1.890,00€100mg2.547,00€1mL*10mM (DMSO)735,00€GRT2932Q
CAS:GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].Formula:C25H26ClN3OColore e forma:SolidPeso molecolare:419.95σ1 Receptor/μ Opioid receptor modulator 1
CAS:σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).Formula:C24H31FN2O2Colore e forma:SolidPeso molecolare:398.51ML 190
CAS:ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.Formula:C27H32N6O3Purezza:99.88%Colore e forma:SolidPeso molecolare:488.58Ref: TM-T22995
1mg72,00€5mg156,00€10mg235,00€25mg502,00€50mg805,00€100mg1.083,00€1mL*10mM (DMSO)169,00€ADL-5859 HCl
CAS:ADL-5859 is a delta-opioid receptor agonist.Formula:C24H28N2O3Purezza:98%Colore e forma:SolidPeso molecolare:392.49Enadoline (Free Base)
CAS:Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.Formula:C24H32N2O3Colore e forma:SolidPeso molecolare:396.52SR8993
CAS:SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.Formula:C25H37FN4Purezza:98%Colore e forma:SolidPeso molecolare:412.59BMS-986124
CAS:BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.Formula:C16H15BrClNO3S2Colore e forma:SolidPeso molecolare:448.78BW 373U86
CAS:BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [Formula:C27H37N3O2Colore e forma:SolidPeso molecolare:435.6GSK1521498
CAS:GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H23F2N4O4PPurezza:98%Colore e forma:SolidPeso molecolare:500.43DDD028
CAS:DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.Formula:C20H20N2Purezza:98%Colore e forma:SolidPeso molecolare:288.39TIPP
CAS:TIPP is an agent of delta opioid antagonist.Formula:C37H38N4O6Purezza:98%Colore e forma:SolidPeso molecolare:634.72SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Formula:C28H31NOPurezza:99.54%Colore e forma:SolidPeso molecolare:397.55Ici 174865
CAS:Ici 174865 is a delta opioid receptor antagonist agent.Formula:C38H53N5O7Colore e forma:SolidPeso molecolare:691.86Dup 747
CAS:Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.Formula:C24H28Cl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:447.4LY2048978
CAS:LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.Formula:C19H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:312.41μ opioid receptor agonist 2
CAS:μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.Formula:C25H34N4OColore e forma:SolidPeso molecolare:406.56Anrikefon
CAS:Anrikefon (HSK21542) is a kappa opioid receptor agonist with analgesic effect .Formula:C39H57N7O5Peso molecolare:703.91AT-076
CAS:AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.Formula:C26H35N3O3Colore e forma:SolidPeso molecolare:437.57GSK1521498 free base (hydrochloride)
CAS:GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H21ClF2N4Purezza:98%Colore e forma:SolidPeso molecolare:438.9AZD7268
CAS:AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.Formula:C29H30N4O2SColore e forma:SolidPeso molecolare:498.64ML138
CAS:ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.Formula:C19H14Cl2N4OSColore e forma:SolidPeso molecolare:417.31CP-866087
CAS:CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H28N2O2Purezza:99.56% - >99.99%Colore e forma:SoildPeso molecolare:376.49Opioid receptor modulator 1
CAS:Opioid receptor modulator 1 is a modulator of opioid receptor.Formula:C18H23NO2Purezza:98%Colore e forma:SolidPeso molecolare:285.38CR-665 Acetate
CAS:CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.Formula:C38H53N9O6Colore e forma:SolidPeso molecolare:731.899JTC-801 free base
CAS:JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).Formula:C26H25N3O2Purezza:98%Colore e forma:SolidPeso molecolare:411.5Loperamide oxide
CAS:Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.Formula:C29H33ClN2O3Colore e forma:SolidPeso molecolare:493.04ORL1 antagonist 1
CAS:ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).Formula:C20H22ClN5Purezza:98.92%Colore e forma:SolidPeso molecolare:367.88Ref: TM-T12320
1mg52,00€5mg111,00€10mg163,00€25mg235,00€50mg333,00€100mg447,00€200mg592,00€1mL*10mM (DMSO)114,00€Diallyl G
CAS:Diallyl G is a delta-opioid receptor antagonist agent.Formula:C38H53N5O8Colore e forma:SolidPeso molecolare:707.86Axomadol
CAS:Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.Formula:C16H25NO3Purezza:98%Colore e forma:SolidPeso molecolare:279.37LY 164929
CAS:LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.Formula:C28H41N5O4Colore e forma:SolidPeso molecolare:511.66Azoenkephalin
CAS:Azoenkephalin is the azo bridge between tyrosine & phenylalanine of enkephalin molecule.Formula:C28H35N7O7Colore e forma:SolidPeso molecolare:581.62Viminol
CAS:Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.Formula:C21H31ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:362.94ICI 154,129
CAS:Selective δ opioid antagonistFormula:C34H46N4O6SPurezza:98%Colore e forma:SolidPeso molecolare:638.82GSK1521498 free base
CAS:<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Formula:C24H20F2N4Purezza:99.85%Colore e forma:SolidPeso molecolare:402.44Ref: TM-T11478L
1mg125,00€5mg297,00€10mg545,00€25mg1.063,00€50mg1.617,00€100mg2.451,00€1mL*10mM (DMSO)328,00€LY2444296
CAS:LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).Formula:C24H22F2N2O2Purezza:99.18%Colore e forma:SolidPeso molecolare:408.44PF-4455242 HCl
CAS:PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.Formula:C21H29ClN2O2SPurezza:99.59%Colore e forma:SolidPeso molecolare:408.99LY 281217
CAS:LY 281217, an organic opioid agonist, can produce analgesic effects in mice.Formula:C32H42N4O6Purezza:98%Colore e forma:SolidPeso molecolare:578.7Endomorphin 1 acetate
CAS:Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.Formula:C36H42N6O7Purezza:99.74%Colore e forma:SolidPeso molecolare:670.75Norbinaltorphimine
CAS:nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.Formula:C40H43N3O6Colore e forma:SolidPeso molecolare:661.79DIPPA hydrochloride
CAS:κ receptor antagonistFormula:C22H24Cl3N3OSPurezza:98%Colore e forma:SolidPeso molecolare:484.87ICI 199,441 hydrochloride
CAS:ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.Formula:C21H25Cl3N2OPurezza:99.57%Colore e forma:SolidPeso molecolare:427.8Ref: TM-T22849
2mg34,00€5mg50,00€10mg80,00€25mg145,00€50mg226,00€100mg331,00€200mg465,00€1mL*10mM (DMSO)62,00€Bevenopran
CAS:Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.Formula:C20H26N4O4Purezza:98.69% - 98.9%Colore e forma:SolidPeso molecolare:386.44Ref: TM-T14551
1mg65,00€5mg137,00€10mg197,00€25mg316,00€50mg430,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)150,00€JNJ-20788560
CAS:<p>JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).</p>Formula:C25H28N2O2Purezza:98.02%Colore e forma:SolidPeso molecolare:388.5ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Formula:C25H32N2O3Purezza:98.58%Colore e forma:SolidPeso molecolare:408.53Ref: TM-T23002
5mg47,00€10mg67,00€25mg118,00€50mg185,00€100mg266,00€200mg379,00€1mL*10mM (DMSO)34,00€SCH-486757
CAS:SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.Formula:C24H23Cl2N3OPurezza:99.53% - >99.99%Colore e forma:SolidPeso molecolare:440.37Trimebutine CTB salt
CAS:Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.Formula:C29H36N2O8S2Purezza:99.85% - >99.99%Colore e forma:SolidPeso molecolare:604.74IPAG
CAS:IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.Formula:C17H22IN3Purezza:99.65%Colore e forma:SolidPeso molecolare:395.28AT-121
CAS:AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).Formula:C24H38N4O3SPurezza:98.49% - 99.97%Colore e forma:SolidPeso molecolare:462.65Ref: TM-T37610
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€ADL-5747
CAS:ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletalFormula:C24H28N2O3Purezza:98.94% - 99.74%Colore e forma:SolidPeso molecolare:392.49ICI 204,448
CAS:ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.Formula:C23H27Cl3N2O4Purezza:>99.99%Colore e forma:SolidPeso molecolare:501.83NNC 63-0532
CAS:NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.Formula:C27H29N3O3Purezza:99.53%Colore e forma:SolidPeso molecolare:443.54GR 89696 fumarate
CAS:GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.Formula:C23H29Cl2N3O7Purezza:99.84%Colore e forma:SolidPeso molecolare:530.4N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFormula:C33H33ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:541.08Mu opioid receptor antagonist 7
CAS:Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (Formula:C22H27ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:386.91Deltakephalin
CAS:Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.Formula:C34H48N6O10Purezza:98%Colore e forma:SolidPeso molecolare:700.78μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purezza:98%Colore e forma:SolidPeso molecolare:352.47Trap-101 hydrochloride
CAS:nociceptin/orphanin FQ (NOP) receptor antagonistFormula:C24H36ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:434.02μ opioid receptor agonist 1
CAS:μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that canFormula:C26H38N4OColore e forma:SolidPeso molecolare:422.61FK 33-824
CAS:FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.Formula:C29H41N5O7SPurezza:98%Colore e forma:SolidPeso molecolare:603.73DPI-3290
CAS:DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potentFormula:C30H34FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:487.61ADL-08-0011
CAS:ADL-08-0011 is an metabolite of alvimopan.Formula:C23H29NO3Colore e forma:SolidPeso molecolare:367.49MR2034
CAS:MR2034 is an agonist of kappa-Opioid receptor. MR2034 stimulates hypothalamic-pituitary-adrenal axis.Formula:C19H27NO2Colore e forma:SolidPeso molecolare:301.42SNC 162
CAS:SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.Formula:C27H37N3OPurezza:98%Colore e forma:SolidPeso molecolare:419.6Naloxonazine
CAS:Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.Formula:C38H42N4O6Colore e forma:SolidPeso molecolare:650.76Frakefamide
CAS:Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.Formula:C30H34FN5O5Purezza:98%Colore e forma:SolidPeso molecolare:563.62ADL 08-0011 HCl
CAS:ADL 08-0011, a μ-opioid antagonist with Ki 0.25 nM, is derived from alvimopan by gut microbes and counteracts loperamide effects in rats.Formula:C23H30ClNO3Colore e forma:SolidPeso molecolare:403.947ICI 204448
CAS:ICI 204448 is a potent and peripherally selective κ-opioid agonist.Formula:C23H26Cl2N2O4Colore e forma:SolidPeso molecolare:465.37Ro 48-6791
CAS:Ro 48-6791, a GABA receptor agonist, is used potentially for anesthesia.Formula:C21H25FN6O2Colore e forma:SolidPeso molecolare:412.46Naloxonazine dihydrochloride
CAS:μ1 receptor antagonistFormula:C38H43ClN4O6Purezza:98%Colore e forma:SolidPeso molecolare:687.22CYT-1010
CAS:CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.Formula:C35H40N6O5Purezza:98%Colore e forma:SolidPeso molecolare:624.73Salvinorin A Carbamate
CAS:Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.Formula:C22H27NO8Colore e forma:SolidPeso molecolare:433.457R-84760 hydrochloride
CAS:R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.Formula:C19H25Cl3N2OSColore e forma:SolidPeso molecolare:435.84Icalcaprant
CAS:Icalcaprant is a kappa-opioid receptor antagonist [1].Formula:C23H26N4O3Purezza:98%Colore e forma:SolidPeso molecolare:406.48Prodilidine hydrochloride
CAS:Prodilidine hydrochloride is an opioid analgesic.Formula:C15H22ClNO2Colore e forma:SolidPeso molecolare:283.79BNTX maleate
CAS:δ1 opioid receptor antagonistFormula:C31H31NO8Purezza:98%Colore e forma:SolidPeso molecolare:545.58Sunobinop
CAS:Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.Formula:C26H33N3O3Colore e forma:SolidPeso molecolare:435.56CCG258747
CAS:CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.Formula:C28H27FN4O4Colore e forma:SolidPeso molecolare:502.54GNTI dihydrochloride
CAS:κ opioid receptor antagonistFormula:C27H30ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:508.01Mu opioid receptor antagonist 2
Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.Formula:C25H28N2O4SColore e forma:SolidPeso molecolare:452.57BW 443C
CAS:BW 443C is a selective agonist of mu-opioid receptor.Formula:C33H46N10O10Colore e forma:SolidPeso molecolare:742.791MTI013
MTI013 is a selective inhibitor of SARS-CoV-2 nsp14 Mtase (IC50: 2.98 µM) and an antiviral agent (IC50: 10.33 µM in HCoV-229E infected Huh7 cells). Additionally, MTI013 demonstrates synergistic antiviral effects when used in conjunction with the RdRp inhibitor SHEN26.Formula:C24H26N6O4SColore e forma:SolidPeso molecolare:494.57σ1 Receptor/μ Opioid receptor modulator 2
CAS:Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.Formula:C23H31N3OPeso molecolare:365.51Daeatal
CAS:Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.Formula:C56H93N19O10Purezza:98%Colore e forma:SolidPeso molecolare:1192.46SB-612111
CAS:SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Formula:C24H29Cl2NOColore e forma:SolidPeso molecolare:418.40SB-612111 hydrochloride
SB-612111 is a potent ORL-1 antagonist, with high affinity (Ki: 0.33 nM) and µ-receptor activity (Ki: 57.6 nM), blocking Nociceptin-induced pain.Formula:C24H30Cl3NOColore e forma:SolidPeso molecolare:454.86RX 809055AX
CAS:RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.Formula:C29H29ClN2O4Colore e forma:SolidPeso molecolare:505SC13
CAS:SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.Formula:C26H30N2O5Colore e forma:SolidPeso molecolare:450.53BU09059
CAS:BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).Formula:C28H37N3O5Purezza:98%Colore e forma:SolidPeso molecolare:495.61Mu opioid receptor antagonist 3
Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.Formula:C25H28N2O4SColore e forma:SolidPeso molecolare:452.576β-Naltrexol
CAS:6β-Naltrexol is a peripherally selective opioid antagonist that reduces constipation from opioids while minimizing central nervous system effects.Formula:C20H25NO4Purezza:99.933%Colore e forma:SolidPeso molecolare:343.42Mu opioid receptor antagonist 8
CAS:<p>Muopioid Receptor Antagonist 8 (368) serves as an antagonist to the μ-opioid receptor, significantly inhibiting the activation of Gi induced by met-enkephalin at the µOR.</p>Formula:C36H35N3O4SColore e forma:SolidPeso molecolare:605.75Naltrindole 5′-isothiocyanate
CAS:Naltrindole 5′-isothiocyanate (5'-NTII) is an irreversible delta opioid receptor antagonist that counters the analgesic effects induced by DSLET without altering the effects caused by DPDPE.Formula:C27H25N3O3SColore e forma:SolidPeso molecolare:471.571Norbinaltorphimine dihydrochloride
CAS:Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.Formula:C40H45Cl2N3O6Purezza:98.17% - 99.88%Colore e forma:SolidPeso molecolare:734.71Ref: TM-T12241
1mg38,00€5mg85,00€10mg120,00€25mg235,00€50mg409,00€100mg652,00€200mg908,00€1mL*10mM (DMSO)124,00€J-113397
CAS:J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).Formula:C24H37N3O2Purezza:98%Colore e forma:SolidPeso molecolare:399.57Opioid receptor antagonist 1
CAS:<p>Opioid receptor antagonist 1 (Compound 10) is an Orvinol-based antagonist of opioid receptors. It exhibits activity as an antagonist against the analgesic properties of morphine.</p>Formula:C24H29ClF3NO4Colore e forma:SolidPeso molecolare:487.94
