Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 326 prodotti di "Recettore degli oppioidi"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
DPDPE TFA (88373-73-3 free base)
CAS:DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.Formula:C32H40F3N5O9S2Purezza:99.39%Colore e forma:SolidPeso molecolare:759.81Gluten Exorphin C
CAS:Gluten exorphin C is an opioid peptide derived from wheat gluten.Formula:C29H45N5O8Purezza:99.39%Colore e forma:SolidPeso molecolare:591.7Naloxegol oxalate
CAS:Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.Formula:C36H55NO15Purezza:99.67% - >99.99%Colore e forma:SolidPeso molecolare:741.83Nalmefene hydrochloride
CAS:Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.Formula:C21H26ClNO3Purezza:98% - 99.85%Colore e forma:SolidPeso molecolare:375.89ADL-5859
CAS:ADL-5859 HCl is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFormula:C24H28N2O3·HClPurezza:98.78% - 99.11%Colore e forma:SolidPeso molecolare:428.95Ref: TM-T6175
1mg52,00€2mg70,00€5mg96,00€10mg170,00€25mg338,00€50mg520,00€100mg748,00€500mg1.549,00€1mL*10mM (DMSO)114,00€Alvimopan monohydrate
CAS:Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.Formula:C25H34N2O5Purezza:98%Colore e forma:SolidPeso molecolare:442.55MCOPPB
CAS:MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.Formula:C26H40N4Colore e forma:SolidPeso molecolare:408.62GR 89696 free base
CAS:GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.Formula:C19H25Cl2N3O3Colore e forma:SolidPeso molecolare:414.33EST73502 hydrochloride
CAS:EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.Formula:C19H27ClF2N2O2Colore e forma:SolidPeso molecolare:388.88LY2940094 tartrate
CAS:LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.Formula:C26H29ClF2N4O8SColore e forma:SolidPeso molecolare:631.04MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Formula:C26H43Cl3N4Purezza:99.89% - 99.91%Colore e forma:SolidPeso molecolare:518.01Ref: TM-T2071
2mg34,00€5mg50,00€10mg87,00€25mg163,00€50mg255,00€100mg375,00€200mg535,00€1mL*10mM (DMSO)58,00€Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purezza:>99.99%Colore e forma:SolidPeso molecolare:768.86Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formula:C27H35N5O7SPurezza:≥95%Colore e forma:White Lyophilised SolidPeso molecolare:573.66Endomorphin 2
CAS:EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.Formula:C32H37N5O5Purezza:99.64%Colore e forma:SolidPeso molecolare:571.67EST73502 HCl
CAS:EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Formula:C19H27ClF2N2O2Purezza:99.96%Colore e forma:SolidPeso molecolare:388.88Ref: TM-T39284
1mg92,00€5mg180,00€10mg258,00€25mg424,00€50mg598,00€100mg792,00€200mg1.074,00€1mL*10mM (DMSO)197,00€JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Formula:C26H25N3O2·HClPurezza:99.27% - 99.59%Colore e forma:SolidPeso molecolare:447.96BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purezza:98.42%Colore e forma:SolidPeso molecolare:448.78Ref: TM-T26869
1mg48,00€5mg96,00€10mg160,00€25mg311,00€50mg472,00€100mg658,00€200mg929,00€1mL*10mM (DMSO)96,00€Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formula:C19H23NO4Purezza:99.02% - 99.73%Colore e forma:White PowderPeso molecolare:329.39ADL-5747 (HCl)
CAS:ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.Formula:C24H29ClN2O3Colore e forma:SolidPeso molecolare:428.95PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formula:C19H27N3O2SPurezza:99.93% - >99.99%Colore e forma:SolidPeso molecolare:361.5BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Formula:C31H34O4Purezza:99.09%Colore e forma:SolidPeso molecolare:470.6GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purezza:99.75%Colore e forma:SolidPeso molecolare:530.4Ref: TM-T9459
1mg87,00€2mg143,00€5mg188,00€10mg283,00€25mg509,00€50mg727,00€100mg1.017,00€1mL*10mM (DMSO)250,00€LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purezza:97.77%Colore e forma:SolidPeso molecolare:407.89Ref: TM-TQ0091
1mg52,00€2mg74,00€5mg116,00€10mg180,00€25mg298,00€50mgPrezzo su richiesta1mL*10mM (DMSO)127,00€DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Formula:C26H35N5O6Purezza:98.83% - 99.92%Colore e forma:SolidPeso molecolare:513.59Ref: TM-T4351
1mg50,00€2mg60,00€5mg87,00€10mg140,00€25mg283,00€50mg423,00€100mg623,00€1mL*10mM (DMSO)88,00€Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C50H72N15O15SPurezza:>99.99%Colore e forma:SolidPeso molecolare:1326.26Ref: TM-T7567L
1mg48,00€5mg125,00€10mg180,00€25mg325,00€50mg467,00€100mg645,00€200mg868,00€1mL*10mM (DMSO)187,00€[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Formula:C29H39N5O7Purezza:98.06%Colore e forma:SolidPeso molecolare:569.65Difelikefalin acetate
CAS:Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.Formula:C38H57N7O8Purezza:99.55%Colore e forma:SolidPeso molecolare:739.9BAM 22P acetate
BAM 22P acetate is a potent opioid agonist.Formula:C132H188N38O33S2Purezza:99.87%Colore e forma:SoildPeso molecolare:2899.27Ref: TM-TP1211L
1mg105,00€5mg398,00€10mg595,00€25mg1.064,00€50mg1.434,00€100mg1.948,00€200mg2.622,00€Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.Formula:C101H159N31O25Purezza:99.69%Colore e forma:SolidPeso molecolare:2207.58(D-Ser2)-Leu-Enkephalin-Thr
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.Formula:C33H46N6O10Purezza:94.17%Colore e forma:SoildPeso molecolare:686.75Porcine dynorphin A(1-13) acetate
Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.Formula:C77H130N24O17Purezza:99.14%Colore e forma:SolidPeso molecolare:1664Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Formula:C76H119N21O19Purezza:99.72%Colore e forma:SolidPeso molecolare:1630.89CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Formula:C53H70F3N13O13S2Purezza:99.62%Colore e forma:SolidPeso molecolare:1218.33Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Formula:C63H101F3N22O17Purezza:97.64%Colore e forma:SolidPeso molecolare:1495.61Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.Formula:C46H74N14O11Purezza:99.84%Colore e forma:SolidPeso molecolare:999.17[Met5]-Enkephalin, amide TFA
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.Formula:C29H37F3N6O8SPurezza:99.81%Colore e forma:SolidPeso molecolare:686.7Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formula:C31H40F3N5O9Purezza:98.79%Colore e forma:SolidPeso molecolare:683.67Ref: TM-T20435L
1mg86,00€2mg111,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formula:C51H79N15O16Purezza:95.54%Colore e forma:SolidPeso molecolare:1158.26N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formula:C30H39N5O8Purezza:>99.99%Colore e forma:SolidPeso molecolare:597.66b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Formula:C25H31N3O7Purezza:98.99%Colore e forma:SolidPeso molecolare:485.53Ref: TM-T21660L
5mg44,00€10mg60,00€25mg93,00€50mg138,00€100mg202,00€200mg301,00€1mL*10mM (DMSO)58,00€Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Formula:C51H73N15O11Purezza:98.59%Colore e forma:SolidPeso molecolare:1072.22Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Formula:C51H68N12O13Purezza:99.66%Colore e forma:SolidPeso molecolare:1057.16Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.Formula:C59H95N19O14Purezza:99.88%Colore e forma:SolidPeso molecolare:1294.53[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.Formula:C30H42N6O8Purezza:99.36%Colore e forma:SolidPeso molecolare:614.69Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.Formula:C31H41N7O9Purezza:98.92%Colore e forma:SoildPeso molecolare:655.7Ref: TM-T23076L
1mg309,00€2mg462,00€5mg697,00€10mg1.054,00€25mg1.549,00€50mg2.110,00€100mg2.840,00€1mL*10mM (DMSO)947,00€AR-M 1000390 hydrochloride
CAS:ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.Formula:C23H29ClN2OPurezza:98.66%Colore e forma:SolidPeso molecolare:384.94Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purezza:99.45% - 99.78%Colore e forma:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecolare:361.39BRL 52537 hydrochloride
CAS:BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Formula:C18H25Cl3N2OPurezza:99.04%Colore e forma:SolidPeso molecolare:391.76Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formula:C26H27FN2O2Purezza:99.9% - 99.97%Colore e forma:SolidPeso molecolare:418.5Ref: TM-TQ0082
1mg40,00€2mg52,00€5mg88,00€10mg126,00€25mg259,00€50mg406,00€100mg607,00€1mL*10mM (DMSO)87,00€BMS986188
CAS:BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.Formula:C30H31BrO4Purezza:98.76%Colore e forma:SolidPeso molecolare:535.47
![[D-Ala2]leucine-enkephalin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1367.webp&w=3840&q=75)
![[Met5]-Enkephalin, amide TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1254.webp&w=3840&q=75)
![[Leu5]-Enkephalin, amide acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1113L.webp&w=3840&q=75)
