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Recettore degli oppioidi

Recettore degli oppioidi

I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.

Trovati 326 prodotti di "Recettore degli oppioidi"

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  • Trimebutine maleate

    CAS:
    <p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>
    Formula:C26H33NO9
    Purezza:99.76% - 99.98%
    Colore e forma:White Solid
    Peso molecolare:503.55

    Ref: TM-T1197

    1g
    34,00€
  • ZT 52656A hydrochloride

    CAS:
    ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
    Formula:C19H26ClF3N2O
    Purezza:98.78%
    Colore e forma:Solid
    Peso molecolare:390.87

    Ref: TM-T13414

    1mg
    540,00€
    5mg
    1.198,00€
    10mg
    1.786,00€
    25mg
    3.030,00€
    50mg
    3.924,00€
    1mL*10mM (DMSO)
    1.026,00€
  • Matrine

    CAS:
    Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
    Formula:C15H24N2O
    Purezza:99.77% - >99.99%
    Colore e forma:Solid
    Peso molecolare:248.36

    Ref: TM-T2870

    25mg
    43,00€
    50mg
    58,00€
    100mg
    81,00€
    200mg
    117,00€
    500mg
    250,00€
    1mL*10mM (DMSO)
    49,00€
  • CP 866087

    CAS:
    CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
    Formula:C24H30N2O3S
    Purezza:99.22% - 99.74%
    Colore e forma:Solid
    Peso molecolare:426.57

    Ref: TM-T31081L

    1mg
    185,00€
    5mg
    459,00€
    10mg
    657,00€
    25mg
    1.026,00€
    50mg
    1.415,00€
  • Naltrexone hydrochloride

    CAS:
    <p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>
    Formula:C20H24ClNO4
    Purezza:98.72% - 99.65%
    Colore e forma:White Crystalline Powder
    Peso molecolare:377.862

    Ref: TM-T0963

    1g
    163,00€
    25mg
    35,00€
    50mg
    44,00€
    100mg
    55,00€
    500mg
    111,00€
  • Apitegromab

    CAS:
    Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including
    Purezza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)
    Colore e forma:Liquid

    Ref: TM-T77445

    1mg
    160,00€
    5mg
    472,00€
    10mg
    755,00€
    25mg
    1.121,00€
    50mg
    1.501,00€
  • Moguisteine

    CAS:
    Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.
    Formula:C16H21NO5S
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:339.41

    Ref: TM-T1169

    50mg
    34,00€
    1mL*10mM (DMSO)
    34,00€
  • BTRX-335140

    CAS:
    <p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>
    Formula:C25H32FN5O2
    Purezza:98% - 99.89%
    Colore e forma:Solid
    Peso molecolare:453.55

    Ref: TM-T14835

    1mg
    105,00€
    2mg
    155,00€
    5mg
    250,00€
    10mg
    406,00€
    25mg
    840,00€
    50mg
    1.378,00€
    100mg
    1.882,00€
    200mg
    2.632,00€
  • Meptazinol hydrochloride

    CAS:
    Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
    Formula:C15H23NO·HCl
    Purezza:99.75%
    Colore e forma:White Solid
    Peso molecolare:269.81

    Ref: TM-T0201

    5mg
    48,00€
    10mg
    55,00€
    25mg
    87,00€
    50mg
    116,00€
    100mg
    168,00€
    200mg
    227,00€
    1mL*10mM (DMSO)
    55,00€
  • Alvimopan

    CAS:
    <p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>
    Formula:C25H32N2O4
    Purezza:99.47% - 99.78%
    Colore e forma:Solid
    Peso molecolare:424.53

    Ref: TM-T1242

    1mg
    48,00€
    5mg
    88,00€
    10mg
    135,00€
    25mg
    245,00€
    50mg
    378,00€
    100mg
    560,00€
    200mg
    797,00€
  • Loperamide hydrochloride

    CAS:
    Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
    Formula:C29H34Cl2N2O2
    Purezza:99.91% - >99.99%
    Colore e forma:Crystals Practically Insoluble In Water
    Peso molecolare:513.50

    Ref: TM-T0209

    1g
    107,00€
    50mg
    44,00€
    100mg
    55,00€
    500mg
    85,00€
    1mL*10mM (DMSO)
    55,00€
  • Sinomenine hydrochloride

    CAS:
    Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
    Formula:C19H24ClNO4
    Purezza:99.43%
    Colore e forma:Solid
    Peso molecolare:365.85

    Ref: TM-T2921

    1g
    70,00€
    200mg
    34,00€
    500mg
    52,00€
  • Samidorphan HCl

    CAS:
    <p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>
    Formula:C21H27ClN2O4
    Purezza:96.79% - 97.85%
    Colore e forma:Soild
    Peso molecolare:406.9

    Ref: TM-T67888L

    1mg
    164,00€
    5mg
    393,00€
    10mg
    582,00€
    25mg
    930,00€
    50mg
    1.254,00€
    100mg
    1.691,00€
  • LY2940094

    CAS:
    LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
    Formula:C22H23ClF2N4O2S
    Purezza:99.4%
    Colore e forma:Solid
    Peso molecolare:480.96

    Ref: TM-T15799

    1mg
    81,00€
    2mg
    106,00€
    5mg
    163,00€
    10mg
    274,00€
    25mg
    542,00€
    50mg
    778,00€
    100mg
    1.074,00€
    1mL*10mM (DMSO)
    180,00€
  • DPDPE

    CAS:
    DPDPE is selective δ-opioid receptor agonist peptide.
    Formula:C30H39N5O7S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:645.79

    Ref: TM-TP2036

    1mg
    545,00€
  • ICI 174,864

    CAS:
    <p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>
    Formula:C38H53N5O7
    Purezza:98%
    Colore e forma:White Solid
    Peso molecolare:691.87

    Ref: TM-TP2013

    1mg
    677,00€
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Colore e forma:Odour Solid

    Ref: TM-L2610

    1mg
    Prezzo su richiesta
  • Biphalin TFA

    CAS:
    <p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>
    Formula:C46H56N10O10·xC2HF3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:909.00 (free base)

    Ref: TM-T80074

    5mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • [DPro10] Dynorphin A (1-11)acetate,porcine


    [DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.
    Formula:C65H107N21O15
    Purezza:99.59%
    Colore e forma:Soild
    Peso molecolare:1422.7

    Ref: TM-T76341L

    2mg
    38,00€
    5mg
    59,00€
    10mg
    87,00€
    25mg
    131,00€
    50mg
    190,00€
    100mg
    279,00€
    200mg
    394,00€
  • β-Endorphin, equine TFA


    β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3
    Formula:C156H249F3N42O46S
    Colore e forma:Solid
    Peso molecolare:3537.96

    Ref: TM-T76027

    5mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta