
Recettore del glucagone
I recettori del glucagone sono GPCR che mediano gli effetti del glucagone, un ormone coinvolto nella regolazione dell'omeostasi del glucosio promuovendo la degradazione del glicogeno e il rilascio di glucosio dal fegato. Questi recettori sono fondamentali nella gestione dei livelli di zucchero nel sangue e sono di particolare interesse nello studio del diabete e dei disturbi metabolici. Gli antagonisti dei recettori del glucagone sono studiati come potenziali trattamenti per l'iperglicemia nel diabete di tipo 2. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori del glucagone di alta qualità per supportare la tua ricerca in endocrinologia, diabete e regolazione metabolica.
Trovati 197 prodotti per "Recettore del glucagone".
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Retatrutide
CAS:Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.Formula:C221H342N46O68Purezza:98.31%Colore e forma:White SolidPeso molecolare:4732.09Volagidemab
CAS:Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.Purezza:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)Colore e forma:Transparent LiquidPeso molecolare:147 kDaAvexitide acetate
CAS:Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.Formula:C155H246N40O53SPurezza:96.64% - 98.65%Colore e forma:SolidPeso molecolare:3549.91Retatrutide sodium salt
Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.Purezza:99.86% - 99.97%Colore e forma:White SolidGlucagon (1-29), bovine, human, porcine hydrochloride
CAS:Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.Formula:C153H225N43O49S·ClHPurezza:95.65% - 98.50%Colore e forma:SolidPeso molecolare:3519.21Ref: TM-T15389L
1mg66,00€5mg173,00€10mg260,00€25mg449,00€50mg657,00€100mg887,00€200mg1.198,00€250mg1.368,00€PF-06882961
CAS:PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C31H30FN5O4Purezza:97.19% - 99.56%Colore e forma:SolidPeso molecolare:555.6Tirzepatide monosodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.Formula:C225H347N48O68NaPurezza:99.69%Colore e forma:SolidPeso molecolare:4835.51Ref: TM-TP1111L1
1mg236,00€5mg620,00€10mg1.018,00€25mg1.521,00€50mg2.088,00€100mg2.817,00€1g7.042,00€Crotedumab
CAS:Crotedumab (REGN1193) is a humanized antibody targeting GCGR, which reduces fasting blood glucose and improves glucose tolerance, used in diabetes research.Purezza:>95%Colore e forma:LiquidPeso molecolare:146.82 kDaOrforglipron
CAS:Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1Formula:C48H48F2N10O5Purezza:99.47% - 99.89%Colore e forma:White SolidPeso molecolare:882.96Tirzepatide hydrochloride
Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.Formula:C225H349N48O68ClPurezza:98%Colore e forma:SolidPeso molecolare:4849.91HAEGT
CAS:HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.Formula:C20H31N7O9Purezza:98%Colore e forma:SolidPeso molecolare:513.5GLP-1 receptor agonist 13
Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].Formula:C25H23ClF2N6OColore e forma:SolidPeso molecolare:496.94Albiglutide Fragment
CAS:Albiglutide fragment is a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).Formula:C148H224N40O45Purezza:98%Colore e forma:SolidPeso molecolare:3283.6GLP-1 (9-36) amide
CAS:GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.Formula:C140H214N36O43Purezza:97%Colore e forma:SolidPeso molecolare:3089.41Secretin (28-54), human TFA
Secretin (28-54), human TFA is a 27-amino acid peptide that works on the human Secretin receptor.Formula:C132H221N44F3O42Purezza:98%Colore e forma:SolidPeso molecolare:3153.48VU0453379
CAS:VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).Formula:C26H34N4O2Purezza:98%Colore e forma:SolidPeso molecolare:434.57GLP-1R Antagonist 1
CAS:GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).Formula:C16H11ClF6N4O2Purezza:99.84%Colore e forma:White SolidPeso molecolare:440.73Tirzepatide
CAS:Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.Formula:C225H348N48O68Purezza:99.52% - 99.99%Colore e forma:White SolidPeso molecolare:4813.45V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.Formula:C20H26ClF3N4O2Purezza:99.97%Colore e forma:SoildPeso molecolare:446.89Ref: TM-T60047L
1mg35,00€5mg79,00€1mL*10mM (DMSO)86,00€10mg122,00€25mg224,00€50mg333,00€100mg474,00€200mg637,00€HAEGTFTSD
CAS:HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.Formula:C40H57N11O17Purezza:98%Colore e forma:SolidPeso molecolare:963.94

