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Recettore del glucagone

Recettore del glucagone

I recettori del glucagone sono GPCR che mediano gli effetti del glucagone, un ormone coinvolto nella regolazione dell'omeostasi del glucosio promuovendo la degradazione del glicogeno e il rilascio di glucosio dal fegato. Questi recettori sono fondamentali nella gestione dei livelli di zucchero nel sangue e sono di particolare interesse nello studio del diabete e dei disturbi metabolici. Gli antagonisti dei recettori del glucagone sono studiati come potenziali trattamenti per l'iperglicemia nel diabete di tipo 2. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori del glucagone di alta qualità per supportare la tua ricerca in endocrinologia, diabete e regolazione metabolica.

Trovati 195 prodotti di "Recettore del glucagone"

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  • Avexitide acetate

    CAS:
    Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
    Formula:C155H246N40O53S
    Purezza:96.64% - 98.65%
    Colore e forma:Solid
    Peso molecolare:3549.91
  • PF-06882961

    CAS:
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C31H30FN5O4
    Purezza:97.19% - 99.56%
    Colore e forma:Solid
    Peso molecolare:555.6
  • Volagidemab

    CAS:
    <p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>
    Purezza:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)
    Colore e forma:Liquid
  • Retatrutide

    CAS:
    <p>Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.</p>
    Formula:C221H342N46O68
    Purezza:98.31%
    Colore e forma:Solid
    Peso molecolare:4732.09
  • Tirzepatide monosodium salt


    Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.
    Formula:C225H347N48O68Na
    Purezza:99.69%
    Colore e forma:Soild
    Peso molecolare:4835.51
  • Crotedumab

    CAS:
    Crotedumab (REGN1193) is a humanized antibody targeting GCGR, which reduces fasting blood glucose and improves glucose tolerance, used in diabetes research.
    Purezza:>95%
    Colore e forma:Liquid
  • Glucagon (1-29), bovine, human, porcine hydrochloride

    CAS:
    Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.
    Formula:C153H225N43O49S·ClH
    Purezza:95.65% - 98.03%
    Colore e forma:Solid
    Peso molecolare:3519.21
  • Orforglipron

    CAS:
    Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1
    Formula:C48H48F2N10O5
    Purezza:99.47% - 99.8%
    Colore e forma:Solid
    Peso molecolare:882.96
  • Retatrutide sodium salt


    Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.
    Purezza:99.97%
    Colore e forma:Soild
  • GLP-1R agonist 34

    CAS:
    GLP-1R agonist 34 (Compound 1) is an orally active small molecule agonist of the glucagon-like peptide-1 receptor (GLP-1R). It enhances insulin secretion, suppresses glucagon release, and slows gastric emptying, thereby effectively reducing blood glucose levels. GLP-1R agonist 34 holds potential for research into metabolic disorders such as type 2 diabetes, obesity, and non-alcoholic steatohepatitis (NASH).
    Formula:C50H50F2N10O5
    Colore e forma:Solid
    Peso molecolare:908.99
  • GLP-1R Agonist DMB

    CAS:
    GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
    Formula:C13H15Cl2N3O2S
    Purezza:99.52%
    Colore e forma:Solid
    Peso molecolare:348.25
  • GLP-1R Antagonist 1

    CAS:
    <p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>
    Formula:C16H11ClF6N4O2
    Purezza:99.84%
    Colore e forma:Solid
    Peso molecolare:440.73
  • HAEGTFTSD

    CAS:
    HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.
    Formula:C40H57N11O17
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:963.94
  • Tirzepatide

    CAS:
    Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.
    Formula:C225H348N48O68
    Purezza:99.52% - 99.99%
    Colore e forma:Solid
    Peso molecolare:4813.45
  • HAEGT

    CAS:
    <p>HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.</p>
    Formula:C20H31N7O9
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:513.5
  • Glucagon receptor antagonists-1

    CAS:
    Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.
    Formula:C29H34FNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:447.58
  • V-0219 hydrochloride


    <p>V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.</p>
    Formula:C20H26ClF3N4O2
    Purezza:99.97%
    Colore e forma:Soild
    Peso molecolare:446.89
  • GLP-1 moiety from Dulaglutide


    GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist.
    Formula:C149H221N37O49
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3314.62
  • HAEGTFTSD acetate(926018-45-3 free base)


    HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from
    Formula:C42H61N11O19
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1024.01
  • GLP-1 receptor agonist 13


    Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].
    Formula:C25H23ClF2N6O
    Colore e forma:Solid
    Peso molecolare:496.94
  • Albiglutide Fragment

    CAS:
    <p>Albiglutide fragment is a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).</p>
    Formula:C148H224N40O45
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3283.6
  • 6α-Methylprednisolone 21-hemisuccinate sodium salt

    CAS:
    6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone), a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
    Formula:C26H33NaO8
    Purezza:99.65%
    Colore e forma:Lyophilized Powder
    Peso molecolare:496.53
  • Cinnamtannin A2

    CAS:
    <p>Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.</p>
    Formula:C60H50O24
    Colore e forma:Solid
    Peso molecolare:1155.02
  • Tirzepatide hydrochloride


    Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.
    Formula:C225H349N48O68Cl
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4849.91
  • Survodutide TFA


    Survodutide TFA (BI 456906 TFA) is a GCGR/GLP-1R dual agonist, a peptide compound used in obesity research.
    Formula:C192H289N47O61·xC2HF3OC2
    Purezza:99.29% - 99.96%
    Colore e forma:Solid
    Peso molecolare:4231.62 (free base)
  • Secretin (28-54), human TFA


    <p>Secretin (28-54), human TFA is a 27-amino acid peptide that works on the human Secretin receptor.</p>
    Formula:C132H221N44F3O42
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3153.48
  • VU0453379

    CAS:
    VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).
    Formula:C26H34N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:434.57
  • GLP-1 receptor agonist 4

    CAS:
    GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.
    Formula:C51H44Cl2N4O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:879.82
  • Glucagon (19-29), human

    CAS:
    Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.
    Formula:C61H89N15O18S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1352.53
  • Glucagon-like peptide 1 (1-37), human

    CAS:
    Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.
    Formula:C186H275N51O59
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4169.48
  • Secretin (28-54), human

    CAS:
    Secretin (28-54), human, is a 27-amino acid residue peptide with a C-terminal amidation, acting on human secretin receptors.
    Formula:C130H220N44O40
    Purezza:98%
    Colore e forma:Powder
    Peso molecolare:3039.46
  • Albenatide

    CAS:
    <p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>
    Formula:C26H47N7O9S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:633.76
  • HAEGTFTSDVS

    CAS:
    HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.
    Formula:C48H71N13O20
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1150.18
  • Pal-Glu(OSu)-OH

    CAS:
    <p>Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.</p>
    Formula:C25H42N2O7
    Colore e forma:Solid
    Peso molecolare:482.618
  • TT-OAD2

    CAS:
    <p>TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.</p>
    Formula:C50H49Cl4N3O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:929.75
  • GLP-2(1-33)(human)

    CAS:
    GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.
    Formula:C165H254N44O55S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3766.19
  • HAEGTFT

    CAS:
    HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.
    Formula:C33H47N9O12
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:761.78
  • SDV-Exendin-3/4


    SDV-Exendin-3/4 is a 32-amino acid peptide.
    Formula:NA
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3443.87
  • Acmopatide

    CAS:
    Acmopatide (Compound E-153) is a dual agonist of GIP and GLP-1 receptors and can be utilized in diabetes research.
    Colore e forma:Solid
  • GTFTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS


    GTFTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS is an Exendin-4 peptide derivative.
    Peso molecolare:3850.31
  • Glucagon Receptor Antagonist Inactive Control

    CAS:
    Glucagon Receptor Antagonist Inactive Control is a Glucagon receptor antagonist that can be used in related research in the field of life sciences.
    Formula:C21H23BrN2OS
    Colore e forma:Solid
    Peso molecolare:431.39
  • TE-8105


    TE-8105 is a GLP-1 receptor agonist that demonstrates prolonged and enhanced efficacy in models of diabetes, obesity, and non-alcoholic steatohepatitis (NASH).
    Colore e forma:Odour Solid
  • Zovaglutide

    CAS:
    Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.
    Colore e forma:Solid
  • [Gly8]-GLP-1(7-37) acetate


    [Gly8]-GLP-1(7-37) acetate is a derivative of GLP-1, where glycine at position 8 is replaced with alanine. [Gly8]-GLP-1(7-37) acetate is also a peptide fragment of the GLP-1 receptor (GLP-1R) agonist, Dulaglutide.
    Colore e forma:Odour Solid
  • WB4-24

    CAS:
    WB4-24 is a GLP-1 receptor agonist that enhances the release of β-endorphin in microglia. It exhibits antiallodynic, anti-inflammatory, and analgesic effects in mouse models of inflammation induced by formalin, carrageenan, and CFA.
    Formula:C52H48N4O14S2
    Colore e forma:Solid
    Peso molecolare:1017.09
  • Berobenatide

    CAS:
    Berobenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist.
    Colore e forma:Solid
  • Peptide C105Y TFA


    Peptide C105Y TFA is a cell-penetrating peptide synthesized based on the amino acid sequence of residues 359-374 of α1-antitrypsin. It enhances the gene expression of DNA nanoparticles.
    Formula:C97H148N20O23S·xC2HF3O2
  • GLP-1R agonist 20


    GLP-1R agonist 20 (Compound I-132) is an agonist of the glucagon-like peptide-1 receptor (GLP-1 receptor), with an EC50 value of 0.0162 nM.
    Formula:C31H30Cl2F2N4O5
    Peso molecolare:646.15613
  • SPN009


    SPN009 (Sequence 3) is a GLP-1 receptor (GLP-1 Receptor) agonist, with an EC50 of 2.84 nM, and improves type 2 diabetes in DB/DB mouse models.
    Formula:C191H299N45O59
    Peso molecolare:4167.17798
  • Anti-GLP-1R Antibody


    Anti-GLP-1R Antibody is an anti-GLP-1R antibody that can be used for immunohistochemistry of paraffin sections.
    Purezza:98.3% (SDS-PAGE); 97.2% (SEC-HPLC) - 98.3% (SDS-PAGE); 97.2% (SEC-HPLC)
    Colore e forma:Odour Liquid
  • Secretin, canine TFA


    Secretin, canine TFA, is an endocrine hormone that stimulates the secretion of pancreatic fluid rich in bicarbonate. Additionally, Secretin, canine TFA, can regulate the primary cell functions and paracellular permeability of gastric monolayer cells through an Src kinase-dependent pathway.
    Colore e forma:Odour Solid
  • Sorbinicate

    CAS:
    <p>Sorbinicate is an antihypercholesterolaemic and vasodilating nicotinic acid ester.</p>
    Formula:C42H32N6O12
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:812.74
  • Semaglutide, FITC labeled


    Semaglutide (FITC-labeled Semaglutide) is a long-acting analog of human glucagon-like peptide-1, functioning as an agonist of the GLP-1 receptor. It shows potential for research related to type 2 diabetes.
    Formula:C209H304N46O63S
    Peso molecolare:4498.17191
  • GIP/GLP-1 dual receptor agonist-1 sodium


    GIP/GLP-1 dual receptor agonist-1 (Compound 4) (sodium) functions as a GIP/GLP-1 receptor agonist. This compound is applicable for research into metabolic disorders and liver diseases, including non-alcoholic steatohepatitis (NASH) and non-alcoholic fatty liver disease (NAFLD).
    Colore e forma:Odour Solid
  • GLP-1(7-36), amide acetate

    CAS:
    GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.
    Formula:C151H230N40O47
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:3357.68
  • Apraglutide

    CAS:
    Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.
    Formula:C172H263N43O52
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3765.25
  • Dulaglutide

    CAS:
    <p>Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).</p>
    Colore e forma:Solid
  • Taspoglutide

    CAS:
    Taspoglutide is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist(EC50 value of 0.06 nM),and for treatment of type 2 diabetes
    Formula:C152H232N40O45
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3339.763
  • LSN3160440

    CAS:
    LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.
    Formula:C27H27Cl2N3O
    Colore e forma:Solid
    Peso molecolare:480.43
  • Des His1, Glu8 Exendin-4


    Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose and is used in the study of diabetes and obesity.
    Formula:C179H277N47O59S
    Purezza:99.92%
    Colore e forma:Solid
    Peso molecolare:4063.46
  • Secretin, porcine

    CAS:
    Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.
    Formula:C130H220N44O41·xC2H4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:N/A
  • TT-OAD2 free base

    CAS:
    TT-OAD2 free base, a non-peptide GLP-1 receptor agonist, can treat diabetes; has an EC50 of 5 nM.
    Formula:C50H47Cl2N3O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:856.83
  • {Val1}-Exendin-3/4


    {Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.
    Formula:NA
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3241.7
  • GLP-1R agonist 14

    CAS:
    GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].
    Formula:C45H42F2N10O5
    Colore e forma:Solid
    Peso molecolare:840.88
  • GIP/GLP-1 dual receptor agonist-1

    CAS:
    Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.
    Colore e forma:Solid
  • HAEGTFTSDVS acetate


    HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.
    Formula:C50H75N13O22
    Purezza:97.47%
    Colore e forma:Solid
    Peso molecolare:1210.2
  • GLP-1R agonist 29


    <p>GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.</p>
    Colore e forma:Odour Solid
  • Exendin-3/4 (59-86)


    Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.
    Formula:NA
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3055.49
  • GLP-1(7-37)

    CAS:
    GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.
    Formula:C151H228N40O47
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3355.67
  • Mazdutide acetate(2259884-03-0 free base)


    Mazdutide acetate is a potent (GLP-1R and GCGR agonist that stimulates insulin secretion from mouse pancreatic islets , which can be used to study obesity.
    Purezza:98.41%
    Colore e forma:Odour Solid
  • Bay 55-9837

    CAS:
    Selective VPAC2 agonist; EC50: 0.4 nM (VPAC2), 100 nM (VPAC1), >1000 nM (PAC1). Enhances insulin secretion, reduces HIV-1 replication.
    Formula:C167H270N52O46
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3742.29
  • Semaglutide TFA


    Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels and reduces cardiovascular risk in diabetic patients
    Formula:C189H290F3N45O61
    Purezza:99.69%
    Colore e forma:Solid
    Peso molecolare:4225.6482
  • Survodutide

    CAS:
    Survodutide (BI 456906) is a dual agonist of glucagon and glucagon-like peptide 1 (GLP-1) receptor (GLP Receptor) that reduces body weight in HbA1c16 diabetes.
    Formula:C192H289N47O61
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:4229.0957
  • VU0453379 hydrochloride


    VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.
    Formula:C26H35ClN4O2
    Colore e forma:Solid
    Peso molecolare:471.03
  • 3-Deoxyglucosone

    CAS:
    3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with protein
    Formula:C6H10O5
    Purezza:95%
    Colore e forma:Solid
    Peso molecolare:162.14
  • Ribupatide

    CAS:
    Ribupatide is a dual agonist of gastric inhibitory polypeptide (GIP) and glucagon-like peptide 1 (GLP-1) receptors and can be utilized in antidiabetic research.
    Colore e forma:Solid
  • Albiglutide fragment TFA


    Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as a
    Formula:C148H224N40O45·xC2HF3O2
    Colore e forma:Solid
  • Vensemaglutide

    CAS:
    Vensemaglutide is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in research related to diabetes or other metabolic disorders.
    Formula:C214H337N49O67
    Peso molecolare:4668.25
  • (R)-V-0219 hydrochloride


    (R)-V-0219 hydrochloride: Oral GLP-1R PAM, enantiomer of V-0219, triggers Ca2+ flux in hGLP-1R HEK cells.
    Formula:C20H26ClF3N4O2
    Colore e forma:Solid
    Peso molecolare:446.89
  • GLP-1R agonist 26

    CAS:
    Compound 1, also known as GLP-1R agonist 26, is an agonist of the glucagon-like peptide-1 receptor (GLP-1R) with an EC50 of <10 nM.
    Formula:C32H29FN6O4S
    Peso molecolare:612.67
  • Maridebart

    CAS:
    Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].
    Colore e forma:Liquid
  • Oxyntomodulin

    CAS:
    GLP-1 analog modulates appetite, boosts metabolism, and curbs gastric acid. Increases cAMP, mildly stimulates glucagon receptor.
    Formula:C192H295N59O60S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4421.86
  • GLP-1 receptor agonist 8

    CAS:
    GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.
    Formula:C34H36ClFN6O4
    Colore e forma:Solid
    Peso molecolare:647.14
  • [Des-His1,Glu9]-Glucagon amide

    CAS:
    Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.
    Formula:C148H221N41O47S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3358.68
  • GLP-1R agonist 27


    <p>GLP-1R agonist 27 (compound 21) is a potent and orally active GLP-1R agonist. It enhances the accumulation of cyclic adenosine monophosphate (cAMP), reduces blood glucose levels, and decreases food intake. GLP-1R agonist 27 shows potential for research in obesity and type 2 diabetes mellitus (T2DM).</p>
    Formula:C32H33N5O4Se
    Colore e forma:Solid
    Peso molecolare:630.6
  • Liraglutide acetate

    CAS:
    Liraglutide acetate is the acetate salt form of Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in the study of type 2 diabetes.
    Formula:C172H265N43O51·xC2H4O2
    Peso molecolare:3751.20 (free base)
  • (S)-V-0219 hydrochloride


    (S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.
    Formula:C20H26ClF3N4O2
    Colore e forma:Solid
    Peso molecolare:446.89
  • GLP-1R agonist 15

    CAS:
    GLP-1R agonist 15 (Compound 101) is a GLP-1 receptor agonist [1] .
    Formula:C46H47FN8O7S
    Colore e forma:Solid
    Peso molecolare:874.98
  • Gulgafafusp alfa

    CAS:
    Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].
    Colore e forma:Liquid
  • PHI-27 (porcine)

    CAS:
    PHI-27 (porcine) is a porcine-derived peptide consisting of 27 amino acids, utilized in the identification of peptide hormones and other bioactive peptides [1].
    Formula:C136H216N36O40
    Peso molecolare:2995.39
  • DD202-114

    CAS:
    DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.
    Formula:C33H35FN4O5
    Peso molecolare:586.65
  • Glucagon-like peptide 1 (1-37), human TFA


    Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.
    Formula:C188H276N51F3O61
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4283.5
  • (Asp28)-Glucagon (1-29) (human, rat, porcine)

    CAS:
    "(Asp28)-Glucagon (1-29) (human, rat, porcine)" is an analog of glucagon with an aspartic acid (Asp) substitution at position 28, notably enhancing its aqueous
    Formula:C153H224N42O50S
    Peso molecolare:3483.73
  • GLP-1R agonist 16

    CAS:
    Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].
    Formula:C50H58FN10O6P
    Colore e forma:Solid
    Peso molecolare:945.03
  • GLP-1R agonist 4

    CAS:
    GLP-1R agonist 4, potentially for diabetes research, is a potent GLP-1R stimulator linked to hypoglycemia.
    Formula:C32H30ClF2N3O5
    Colore e forma:Solid
    Peso molecolare:610.05
  • SAR441255


    SAR441255 is a potent unimolecular peptide that acts as a GLP-1/GIP/GCG receptor triagonist, demonstrating balanced activation across all three target receptors
    Colore e forma:Odour Solid
  • FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS


    FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS is an Exendin-4 peptide derivative.
    Colore e forma:Solid
    Peso molecolare:3692.15
  • Dapiglutide

    CAS:
    Dapiglutide (ZP7570) is a long-acting GLP-1R & GLP-2R dual agonist for SBS research.
    Colore e forma:Solid
  • GRPP (human)

    CAS:
    GRPP (human), a 30-amino-acid peptide derived from Gcg, modestly elevates plasma insulin levels while reducing plasma glucagon concentrations.
    Formula:C136H215N41O58S
    Colore e forma:Solid
    Peso molecolare:3384.47
  • GLP-1(28-36)amide TFA


    GLP-1(28-36)amide TFA, a nonapeptide cleavage product of GLP-1, shows antioxidant properties with anti-diabetic and cardioprotective effects.
    Formula:C56H86F3N15O11
    Colore e forma:Solid
    Peso molecolare:1202.37
  • GLP-1(9-36)amide TFA


    GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.
    Formula:C142H215F3N36O45
    Colore e forma:Solid
    Peso molecolare:3203.43
  • Pegapamodutide

    CAS:
    Pegapamodutide (LY-2944876) is a dual glucagon-GLP-1 receptor agonist utilized in research concerning type 2 diabetes and obesity [1].
  • Utreglutide

    CAS:
    Utreglutide is a potent glucagon-like peptide 1 (GLP-1) receptor agonit [1] .
    Formula:C191H298N46O58
    Colore e forma:Solid
    Peso molecolare:4166.67
  • Bay 55-9837 TFA


    Bay 55-9837 TFA is a VPAC2 agonist with a 0.65 nM Kd, potential for type 2 diabetes research.
    Formula:C150H240F3ClN44O44
    Colore e forma:Solid
    Peso molecolare:3456.22
  • Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide


    Biotin-labeled GLP-1-(7-36) amide; a gut peptide that enhances insulin release.
    Formula:C165H252N44O48S
    Colore e forma:Solid
    Peso molecolare:3652.1
  • Tirzepatide TFA


    Tirzepatide TFA, a GIP and GLP-1 agonist, targets type 2 diabetes treatment.
    Formula:C227H349F3N48O70
    Colore e forma:Solid
    Peso molecolare:4927.47
  • GLP-1R agonist 19

    CAS:
    GLP-1R agonist 19 (M3190) is a potent, selective GLP-1 receptor agonist that demonstrates excellent plasma and liver microsomal stability, along with low hERG toxicity [1].
    Formula:C94H136FN21O25
    Colore e forma:Solid
    Peso molecolare:1979.21
  • Exendin-4 (3-39)

    CAS:
    <p>Exendin-4 (3-39) is a truncated peptide missing first 2 amino acids of Exendin-4, a potent GLP-1r agonist used in diabetes and HPA axis research.</p>
    Formula:C176H272N46O58S
    Colore e forma:Solid
    Peso molecolare:3992.44
  • VIP(6-28)(human, rat, porcine, bovine)

    CAS:
    VIP(6-28) blocks VIP-induced cAMP signaling in humans, rats, pigs, and cows.
    Formula:C126H207N37O34S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2816.28
  • Orforglipron hemicalcium hydrate

    CAS:
    Orforglipron hemicalcium hydrate (LY3502970 hemicalcium hydrate; GLP-1 receptor agonist 1 hemicalcium hydrate) represents the hemicalcium hydrate form of the calcium salt of Orforglipron, an orally active agonist targeting the Glucagon-like peptide-1 receptor (GLP-1R). This compound has demonstrated efficacy in mitigating type 2 diabetes [1].
    Formula:C48H48F2N10O5Ca·H2O
    Colore e forma:Solid
    Peso molecolare:921.02
  • Secretin (33-59), rat TFA


    Secretin (33-59), rat (TFA), a 27-aa peptide, stimulates the secretin receptor, increasing pancreas secretion of bicarbonate, enzymes, and K+.
    Formula:C131H217F3N42O44
    Colore e forma:Solid
    Peso molecolare:3141.37
  • Ecnoglutide

    CAS:
    Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .
    Formula:C194H304N48O61
    Colore e forma:Solid
    Peso molecolare:4284.76
  • Pemvidutide TFA


    Pemvidutide (TFA), a GLP-1R/GCGR dual agonist, effectively reduces body weight, liver fat, and serum lipid levels, and is utilized in research on non-alcoholic
    Formula:C182H275N39O54·xC2HF3O2
    Colore e forma:Solid
    Peso molecolare:3873.35 (free base)
  • GLP-1 receptor agonist 9 citrate


    <p>GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.</p>
    Formula:C38H39ClFN3O12
    Purezza:98.76%
    Colore e forma:Solid
    Peso molecolare:784.18
  • GLP-1 (9-36) amide

    CAS:
    GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
    Formula:C140H214N36O43
    Purezza:97%
    Colore e forma:Solid
    Peso molecolare:3089.41
  • (S, R)-LSN 3318839

    CAS:
    (S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
    Formula:C26H23Cl2N3O2
    Purezza:99.41%
    Colore e forma:Soild
    Peso molecolare:480.39
  • GLP-1R/GIPR agonist-1


    GLP-1R/GIPR agonist-1 is a dual receptor agonist for GLP-1 (glucagon-like peptide-1) and GIP (glucose-dependent insulinotropic polypeptide). It mimics the action of endogenous hormones GLP-1 and GIP, enhancing insulin secretion while suppressing glucagon release, thus lowering blood sugar. This compound is used in research related to metabolic disorders such as diabetes, obesity, and non-alcoholic steatohepatitis (NASH).
    Formula:C220H342N55O69
    Peso molecolare:4858.49434
  • Glucagon (1-29), bovine, human, porcine

    CAS:
    Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.
    Formula:C153H225N43O49S
    Purezza:99.56% - 99.56%
    Colore e forma:Solid
    Peso molecolare:3482.75
  • SCO-267

    CAS:
    SCO-267 is a full agonist of GPR40/FFAR1, stimulating insulin secretion and GLP-1 release in diabetic rats, improving glucose tolerance,type 2 diabetes.
    Formula:C36H46N4O5
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:614.77
  • GLP-1 receptor agonist 2

    CAS:
    GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C30H31ClFN5O4
    Colore e forma:Solid
    Peso molecolare:580.05
  • GLP-1 receptor agonist 7

    CAS:
    GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.
    Formula:C31H30ClFN4O5
    Colore e forma:Solid
    Peso molecolare:593.05
  • GLP-1R modulator C16

    CAS:
    GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
    Formula:C21H26ClFN2O3
    Purezza:99.6% - >99.99%
    Colore e forma:Solid
    Peso molecolare:408.89
  • V-0219

    CAS:
    V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
    Formula:C20H25F3N4O2
    Purezza:99.91%
    Colore e forma:Soild
    Peso molecolare:410.43
  • GLP-1R modulator C5

    CAS:
    GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.
    Formula:C24H21NO3
    Purezza:99.59%
    Colore e forma:Solid
    Peso molecolare:371.43
  • Anti-GCGR Antibody (7J909)


    Anti-GCGR Antibody (7J909) is an antibody targeting GCGR. Anti-GCGR Antibody (7J909) can be used in ELISA.
    Colore e forma:Odour Liquid
  • Tirzepatide Acetate(2023788-19-2 free base)


    Tirzepatide (LY3298176) Acetate (2023788-19-2 free base) is a new molecule that can control blood glucose levels.Cost-effective and quality-assured.
    Formula:C227H352N48O70
    Purezza:97.3% - 98.05%
    Colore e forma:Solid
    Peso molecolare:4873.5
  • PF-06882961 Tris

    CAS:
    PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C35H41FN6O7
    Purezza:98.74% - 99.79%
    Colore e forma:Solid
    Peso molecolare:676.7
  • GRA Ex-25

    CAS:
    <p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>
    Formula:C29H36F3N3O5
    Purezza:98.2% - 98.88%
    Colore e forma:Solid
    Peso molecolare:563.61
  • Shanzhiside methyl ester

    CAS:
    Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.
    Formula:C17H26O11
    Purezza:98.998% - 99.32%
    Colore e forma:Solid
    Peso molecolare:406.38
  • Lixisenatide acetate (320367-13-3 free base)

    CAS:
    <p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>
    Formula:C215H347N61O65S·6C2H4O2
    Purezza:98% - 99.9%
    Colore e forma:Solid
    Peso molecolare:5218.88
  • BETP

    CAS:
    BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
    Formula:C20H17F3N2O2S
    Purezza:98.51%
    Colore e forma:Solid
    Peso molecolare:406.42
  • HAEGTFTSDVSSYLE


    <p>HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.</p>
    Formula:C71H103N17O28
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:1642.71
  • GLP-1(7-36), amide

    CAS:
    GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.
    Formula:C149H226N40O45
    Purezza:99.85%
    Colore e forma:White Powder
    Peso molecolare:3297.63
  • Exendin-4

    CAS:
    <p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>
    Formula:C184H282N50O60S
    Purezza:97.71% - 99.78%
    Colore e forma:Solid
    Peso molecolare:4186.57
  • Semaglutide

    CAS:
    Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
    Formula:C187H291N45O59
    Purezza:96.92% - 99.78%
    Colore e forma:Solid
    Peso molecolare:4114
  • Liraglutide

    CAS:
    Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.
    Formula:C172H265N43O51
    Purezza:97.65% - 99.04%
    Colore e forma:Solid
    Peso molecolare:3751.25
  • Oxyntomodulin acetate


    Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
    Purezza:99.24%
    Colore e forma:Liquid
    Peso molecolare:N/A
  • Bay 55-9837 acetate


    Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
    Purezza:98.27%
    Colore e forma:Liquid
    Peso molecolare:N/A
  • Secretin (33-59), rat

    CAS:
    <p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>
    Formula:C129H216N42O42
    Purezza:98.12%
    Colore e forma:Solid
    Peso molecolare:3027.35
  • Glucagon (19-29), human acetate


    Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
    Formula:C63H93N15O20S
    Purezza:98.11%
    Colore e forma:Solid
    Peso molecolare:1412.57
  • HAEGTFT acetate(926018-95-3 free base)


    HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
    Formula:C35H51N9O14
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:821.84
  • Exendin-4 acetate

    CAS:
    <p>Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).</p>
    Formula:C186H286N50O62S
    Purezza:98.48% - 99.78%
    Colore e forma:Solid
    Peso molecolare:4247
  • Albiglutide TFA (782500-75-8 free base)


    <p>Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).</p>
    Formula:C150H225F3N40O47
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:3397.63
  • Teduglutide acetate


    <p>Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy.</p>
    Formula:C166H256N44O56S
    Purezza:97.39%
    Colore e forma:Soild
    Peso molecolare:3812.13
  • ML-SI3

    CAS:
    CCG-143140 is a GLP-1 receptor inverse agonists.
    Formula:C23H31N3O3S
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:429.58
  • Exenatide

    CAS:
    Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.
    Formula:C186H286N50O62S
    Purezza:99.42%
    Colore e forma:Solid
    Peso molecolare:4247
  • Glucagon-like peptide 1 (1-37), human acetate


    Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
    Purezza:98%
    Colore e forma:Liquid
    Peso molecolare:N/A
  • Cotadutide acetate


    Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.
    Formula:C169H256N42O57
    Purezza:98.28%
    Colore e forma:Solid
    Peso molecolare:3788.14
  • GLP-1(7-37) acetate(106612-94-6 free base)

    CAS:
    Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
    Formula:C151H228N40O47
    Purezza:98.89%
    Colore e forma:Solid
    Peso molecolare:3355.67
  • Avexitide

    CAS:
    Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
    Formula:C149H234N40O47S
    Purezza:98% - 99.65%
    Colore e forma:Solid
    Peso molecolare:3369.76
  • GLP-1 receptor agonist 9

    CAS:
    <p>1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.</p>
    Formula:C32H31ClFN3O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:592.06
  • PF-06291874

    CAS:
    PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
    Formula:C26H28F3N3O4
    Purezza:99.12% - 99.27%
    Colore e forma:Solid
    Peso molecolare:503.51
  • NNC-0640

    CAS:
    NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
    Formula:C29H31N7O4S
    Purezza:97.04%
    Colore e forma:Solid
    Peso molecolare:573.67
  • GLP-1 Receptor modulator 1

    CAS:
    GLP-1 Receptormodulator 1 (Compound 7) is an effective positive allosteric modulator of the GLP-1 receptor. It is utilized in the research of obesity and type 2 diabetes.
    Formula:C18H21NOS
    Peso molecolare:299.43
  • GLP-1R agonist 1

    CAS:
    GLP-1R agonist 1, an imidazole derivative and potent GLP-1R activator, may aid diabetes research.
    Formula:C32H29ClFN3O5
    Colore e forma:Solid
    Peso molecolare:590.04
  • (S)-V-0219


    (S)-V-0219: oral, GLP-1R PAM, boosts calcium in hGLP-1R HEK cells, lowers glucose, curbs hunger in mice.
    Formula:C20H25F3N4O2
    Colore e forma:Solid
    Peso molecolare:410.43
  • PF-06412154 HCl

    CAS:
    PF-06412154 HCl is a glucagon receptor antagonist.
    Formula:C24H28ClN3O3
    Colore e forma:Solid
    Peso molecolare:441.96
  • Glucagon receptor antagonists-5

    CAS:
    Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.
    Formula:C30H29ClF3N3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:572.02
  • Efpeglenatide

    CAS:
    Efpeglenatide is a long-acting GLP-1 receptor agonist that improves insulin sensitivity, lowers blood glucose, delays weight gain, and supports metabolic disease research.
    Purezza:100% - 100%
    Colore e forma:Solid
  • (R)-V-0219


    (R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.
    Formula:C20H25F3N4O2
    Colore e forma:Solid
    Peso molecolare:410.43
  • Glucagon receptor antagonists-2

    CAS:
    Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.
    Formula:C22H30FNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:359.48
  • BAY-27-9955

    CAS:
    BAY-27-9955 is a glucagon receptor antagonist.
    Formula:C23H31FO
    Colore e forma:Solid
    Peso molecolare:342.49
  • GCGR antagonist 2

    CAS:
    Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.
    Formula:C28H26N4O2
    Colore e forma:Solid
    Peso molecolare:450.53
  • MS012

    CAS:
    MS012 is a Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase (Kd = 46 ± 15 nM).
    Formula:C22H35N5O2
    Colore e forma:Solid
    Peso molecolare:401.55
  • L-168049

    CAS:
    L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.
    Formula:C24H20BrClN2O
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:467.79
  • NNC 92-1687

    CAS:
    NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.
    Formula:C15H12N2O3S
    Purezza:98.70% - 99.96%
    Colore e forma:Solid
    Peso molecolare:300.33
  • MK3577

    CAS:
    MK3577 is a glucagon receptor antagonist.
    Formula:C30H30ClFN2O3
    Colore e forma:Solid
    Peso molecolare:521.02
  • Antitumor agent-101

    CAS:
    Antitumor agent-101 is a selective, covalent inhibitor targeting lysine methyltransferases G9a/GLP, demonstrating IC50 values of 8.5 nM for G9a and 5.5 nM for
    Formula:C26H38N6O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:482.62
  • MK 0893

    CAS:
    MK 0893 is a potent and selective Glucagon Receptor (GR) antagonist competitive, reversible cAMP activity, which attenuates blood glucose elevation.
    Formula:C32H27Cl2N3O4
    Purezza:98.79%
    Colore e forma:Solid
    Peso molecolare:588.48
  • GLP-1R agonist 3

    CAS:
    GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used to study diabetes and obesity.
    Formula:C31H28FN5O4
    Purezza:97.19%
    Colore e forma:Solid
    Peso molecolare:553.58
  • GLP-1R agonist 10

    CAS:
    GLP-1R agonist 10 is a GLP-1 agonist (EC50: 0.051 nM).
    Formula:C29H29ClFN5O4
    Colore e forma:Solid
    Peso molecolare:566.02
  • GLP-1R agonist 9

    CAS:
    GLP-1R agonist 9 acts as a GLP-1R agonist, demonstrating efficacy with EC50 values of 1.1 nM and 11 nM against CHO GLP-1R Clone H6 and Clone C6, respectively.
    Formula:C32H30ClF2N3O5
    Colore e forma:Solid
    Peso molecolare:610.05
  • GLP-1R agonist 17

    CAS:
    GLP-1R agonist 17 excels in stimulating GLP-1 receptors, useful for cardiovascular metabolic disease research.
    Formula:C28H26ClFN4O4S
    Colore e forma:Solid
    Peso molecolare:569.05
  • Glucagon receptor antagonists-3

    CAS:
    Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.
    Formula:C22H30FNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:359.48
  • GLP-1 receptor agonist 3

    CAS:
    GLP-1 receptor agonist 3 is a GLP-1 receptor agonist,Example 4A-1, has EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively.
    Formula:C31H30FN5O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:555.6
  • LGD-6972 sodium

    CAS:
    LGD-6972 sodium is a glucagon receptor antagonist.
    Formula:C43H46N2NaO5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:725.9
  • GLP-1R agonist 12

    CAS:
    GLP-1R agonist 12 (Compound 123) 是一种 GLP-1R 激动剂,能够用于研究糖尿病。
    Formula:C34H36N6O4
    Colore e forma:Solid
    Peso molecolare:592.69
  • Adomeglivant

    CAS:
    Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
    Formula:C32H36F3NO4
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:555.63
  • Lotiglipron

    CAS:
    <p>Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.</p>
    Formula:C31H31ClN4O5
    Purezza:98.3%
    Colore e forma:Solid
    Peso molecolare:575.05
  • LGD-6972

    CAS:
    <p>LGD-6972 is an antagonist of glucagon receptor.</p>
    Formula:C43H46N2O5S
    Purezza:98.8% - 99.62%
    Colore e forma:Solid
    Peso molecolare:702.9
  • GLP-1R agonist 8

    CAS:
    GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 < 2 nM).
    Formula:C33H32N4O5
    Colore e forma:Solid
    Peso molecolare:564.63
  • GLP-1 receptor agonist 15

    CAS:
    GLP-1 receptor agonist 15 (Example 4) is a GLP receptor agonist with an EC50 of 0.74 nM. It exhibits an IC50 of 10.1 μM against the hERG potassium ion channel. This compound is applicable for research in the diabetes field.
    Formula:C32H31ClFN3O5
    Colore e forma:Solid
    Peso molecolare:592.057
  • LXT34

    CAS:
    LXT34 (Example 2) is a GPR120 agonist with anti-inflammatory properties. This compound enhances GLP-1 formation in the gastrointestinal tract and improves insulin resistance in macrophages and pancreatic cells. LXT34 is applicable in studies related to inflammatory conditions, such as type 2 diabetes, obesity, and non-alcoholic fatty liver disease.
    Formula:C18H21NO3S
    Colore e forma:Solid
    Peso molecolare:331.43
  • GLP-1 receptor agonist 11

    CAS:
    GLP-1 Receptor Agonist 11 (compound 3) acts as an effective agonist for the GLP Receptor, finding use in research related to conditions like diabetes and non-alc. fatty liver disease [1].
    Formula:C31H31ClFN3O4
    Colore e forma:Solid
    Peso molecolare:564.05
  • GLP-1R modulator-1

    CAS:
    GLP-1R modulator-1 (Compound 384) is a potent and orally active selective agonist of the glucagon-like peptide-1 receptor (GLP-1R). It activates G protein-coupled signaling, leading to increased intracellular cAMP levels, enhanced insulin secretion, delayed gastric emptying, and reduced appetite. GLP-1R modulator-1 holds potential for research in type 2 diabetes, obesity, and non-alcoholic steatohepatitis (NASH).
    Formula:C41H38ClFN6O4
    Colore e forma:Solid
    Peso molecolare:733.23
  • DS79932728

    CAS:
    DS79932728 is an orally active inhibitor of G9a and GLP, with IC50 values of 12.6 nM and 75.7 nM, respectively. It induces the production of γ-globin, thereby increasing fetal hemoglobin (HbF) levels. In cynomolgus monkey models, DS79932728 enhances the proportion of F-reticulocytes (F-rets) and shows good oral absorption characteristics.
    Formula:C19H25N3O
    Colore e forma:Solid
    Peso molecolare:311.421
  • GLP-1R agonist 33

    CAS:
    GLP-1R agonist 33 (Compound 224) is a GLP-1 receptor agonist with potential applications in research related to diabetes, obesity, and non-alcoholic fatty liver disease (NAFLD).
    Formula:C30H27FN6O4
    Colore e forma:Solid
    Peso molecolare:554.57
  • PF-06372222

    CAS:
    <p>PF-06372222: a small-molecule that modulates GCGR and antagonizes GLP-1R, affecting insulin and glucagon.</p>
    Formula:C26H28F3N5O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:515.53
  • GLP-1 receptor agonist 12

    CAS:
    Compound 20A, known as GLP-1 receptor agonist 12, acts as an agonist of the GLP receptor. It is utilized in researching diseases like diabetes [1].
    Formula:C31H31FN6O4
    Peso molecolare:570.61
  • DA-302168S

    CAS:
    <p>DA-302168S is an orally active, selective GLP-1R agonist with an EC50 value of 1.32 nM. It promotes insulin secretion and has a hypoglycemic effect. Additionally, DA-302168S reduces food intake. It primarily activates GLP-1R in humans and monkeys, with minimal effect on GLP-1R in rats, mice, and dogs. DA-302168S can be used for research in type 2 diabetes and obesity.</p>
    Formula:C33H24ClF2N3O5
    Colore e forma:Solid
    Peso molecolare:616.011
  • SCH-900822

    CAS:
    SCH-900822 is a potent and selective glucagon receptor antagonist.
    Formula:C34H43Cl2N7O2
    Colore e forma:Solid
    Peso molecolare:652.66
  • GLP-1 receptor agonist 16

    CAS:
    GLP-1 receptoragonist 16 (Example 53) is a GLP-1 agonist applicable for research in diabetes, obesity, or diseases related to non-alcoholic steatohepatitis.
    Formula:C33H31ClFN3O4
    Colore e forma:Solid
    Peso molecolare:588.068
  • GLP-1 receptor agonist 10

    CAS:
    GLP-1 Receptor Agonist 10 (Compound 42), an agonist of the GLP receptor, reduces glucose excursions and inhibits food intake in mice. It is useful for research into type 2 diabetes (T2DM) and obesity [1].
    Formula:C30H28F4N6O5
    Peso molecolare:628.57
  • LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purezza:99.21%
    Colore e forma:Solid
    Peso molecolare:480.39
  • Anti-GLP1R Antibody


    <p>Anti-GLP1R Antibody is a human antibody expressed in CHO cells, targeting GLP1R. For isotype controls, refer to Human IgG1 kappa, Isotype Control.</p>
    Colore e forma:Odour Liquid

    Ref: TM-T9901A-804

    1mg
    Fuori produzione
    5mg
    Fuori produzione
    Prodotto fuori produzione