
Recettore del glucagone
I recettori del glucagone sono GPCR che mediano gli effetti del glucagone, un ormone coinvolto nella regolazione dell'omeostasi del glucosio promuovendo la degradazione del glicogeno e il rilascio di glucosio dal fegato. Questi recettori sono fondamentali nella gestione dei livelli di zucchero nel sangue e sono di particolare interesse nello studio del diabete e dei disturbi metabolici. Gli antagonisti dei recettori del glucagone sono studiati come potenziali trattamenti per l'iperglicemia nel diabete di tipo 2. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori del glucagone di alta qualità per supportare la tua ricerca in endocrinologia, diabete e regolazione metabolica.
Trovati 195 prodotti di "Recettore del glucagone"
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Glucagon receptor antagonists-2
CAS:Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.Formula:C22H30FNO2Purezza:98%Colore e forma:SolidPeso molecolare:359.48BAY-27-9955
CAS:BAY-27-9955 is a glucagon receptor antagonist.Formula:C23H31FOColore e forma:SolidPeso molecolare:342.49GCGR antagonist 2
CAS:Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.Formula:C28H26N4O2Colore e forma:SolidPeso molecolare:450.53MS012
CAS:MS012 is a Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase (Kd = 46 ± 15 nM).Formula:C22H35N5O2Colore e forma:SolidPeso molecolare:401.55L-168049
CAS:L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.Formula:C24H20BrClN2OPurezza:>99.99%Colore e forma:SolidPeso molecolare:467.79Ref: TM-T22893
1mg52,00€5mg111,00€10mg180,00€25mg378,00€50mg560,00€100mg800,00€500mg1.644,00€1mL*10mM (DMSO)123,00€NNC 92-1687
CAS:NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.Formula:C15H12N2O3SPurezza:98.70% - 99.96%Colore e forma:SolidPeso molecolare:300.33MK3577
CAS:MK3577 is a glucagon receptor antagonist.Formula:C30H30ClFN2O3Colore e forma:SolidPeso molecolare:521.02Antitumor agent-101
CAS:Antitumor agent-101 is a selective, covalent inhibitor targeting lysine methyltransferases G9a/GLP, demonstrating IC50 values of 8.5 nM for G9a and 5.5 nM forFormula:C26H38N6O3Purezza:98%Colore e forma:SolidPeso molecolare:482.62MK 0893
CAS:MK 0893 is a potent and selective Glucagon Receptor (GR) antagonist competitive, reversible cAMP activity, which attenuates blood glucose elevation.Formula:C32H27Cl2N3O4Purezza:98.79%Colore e forma:SolidPeso molecolare:588.48GLP-1R agonist 3
CAS:GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used to study diabetes and obesity.Formula:C31H28FN5O4Purezza:97.19%Colore e forma:SolidPeso molecolare:553.58GLP-1R agonist 10
CAS:GLP-1R agonist 10 is a GLP-1 agonist (EC50: 0.051 nM).Formula:C29H29ClFN5O4Colore e forma:SolidPeso molecolare:566.02GLP-1R agonist 9
CAS:GLP-1R agonist 9 acts as a GLP-1R agonist, demonstrating efficacy with EC50 values of 1.1 nM and 11 nM against CHO GLP-1R Clone H6 and Clone C6, respectively.Formula:C32H30ClF2N3O5Colore e forma:SolidPeso molecolare:610.05GLP-1R agonist 17
CAS:GLP-1R agonist 17 excels in stimulating GLP-1 receptors, useful for cardiovascular metabolic disease research.Formula:C28H26ClFN4O4SColore e forma:SolidPeso molecolare:569.05Glucagon receptor antagonists-3
CAS:Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.Formula:C22H30FNO2Purezza:98%Colore e forma:SolidPeso molecolare:359.48GLP-1 receptor agonist 3
CAS:GLP-1 receptor agonist 3 is a GLP-1 receptor agonist,Example 4A-1, has EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively.Formula:C31H30FN5O4Purezza:98%Colore e forma:SolidPeso molecolare:555.6LGD-6972 sodium
CAS:LGD-6972 sodium is a glucagon receptor antagonist.Formula:C43H46N2NaO5SPurezza:98%Colore e forma:SolidPeso molecolare:725.9GLP-1R agonist 12
CAS:GLP-1R agonist 12 (Compound 123) 是一种 GLP-1R 激动剂,能够用于研究糖尿病。Formula:C34H36N6O4Colore e forma:SolidPeso molecolare:592.69Adomeglivant
CAS:Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.Formula:C32H36F3NO4Purezza:99.91%Colore e forma:SolidPeso molecolare:555.63Ref: TM-T14130
1mg38,00€5mg80,00€10mg120,00€25mg188,00€50mg354,00€100mg588,00€200mg868,00€1mL*10mM (DMSO)87,00€Lotiglipron
CAS:<p>Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.</p>Formula:C31H31ClN4O5Purezza:98.3%Colore e forma:SolidPeso molecolare:575.05LGD-6972
CAS:<p>LGD-6972 is an antagonist of glucagon receptor.</p>Formula:C43H46N2O5SPurezza:98.8% - 99.62%Colore e forma:SolidPeso molecolare:702.9
