
Recettore della bradichinina
I recettori della bradichinina sono GPCR che mediano gli effetti della bradichinina, un peptide coinvolto nelle risposte infiammatorie, nella percezione del dolore e nella regolazione della pressione sanguigna. Esistono due principali tipi di recettori della bradichinina, B1 e B2, ognuno dei quali svolge ruoli distinti nei processi fisiopatologici. Gli antagonisti dei recettori della bradichinina sono utilizzati nel trattamento di condizioni come l'angioedema ereditario, il dolore cronico e l'ipertensione. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori della bradichinina di alta qualità per supportare la tua ricerca in infiammazione, gestione del dolore e biologia cardiovascolare.
Trovati 60 prodotti di "Recettore della bradichinina"
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Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Formula:C34H36Cl2N6O5S·2ClHPurezza:99.17% - 99.58%Colore e forma:SoildPeso molecolare:784.58Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Formula:C36H49Cl3N6O6SColore e forma:SolidPeso molecolare:800.23Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Formula:C61H94N18O13SColore e forma:SolidPeso molecolare:1319.58Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Formula:C59H89N19O13SPurezza:98%Colore e forma:White SolidPeso molecolare:1304.52[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.Formula:C50H75N15O10Purezza:98%Colore e forma:SolidPeso molecolare:1046.23Bombinakinin M
CAS:Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.Formula:C100H159N31O24Purezza:98%Colore e forma:SolidPeso molecolare:2179.55Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].Formula:C47H75N13O11Purezza:98%Colore e forma:SolidPeso molecolare:998.18(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Formula:C52H77N15O14Purezza:99.46%Colore e forma:SolidPeso molecolare:1136.26Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Formula:C47H66N12O11Purezza:98%Colore e forma:SolidPeso molecolare:975.11B-Raf IN 14
CAS:B-Raf IN 14 is a BRAF inhibitor.Formula:C15H14BrN5O3SPurezza:98.38%Colore e forma:SolidPeso molecolare:424.27[Des-Arg9]-Bradykinin acetate
CAS:[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.Formula:C46H65N11O12Purezza:99.05%Colore e forma:SolidPeso molecolare:964.07Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formula:C49H75N15O12SPurezza:98%Colore e forma:SolidPeso molecolare:1098.29[Des-Arg10]-HOE I40 TFA
<p>[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.</p>Formula:C53H77N15O12S·xC2HF3O2Colore e forma:SolidDes-Arg9-[Leu8]-Bradykinin acetate
CAS:Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].Formula:C43H67N11O12Purezza:98%Colore e forma:SolidPeso molecolare:930.06Bombinakinin M acetate
<p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>Formula:C102H163N31O26Purezza:99.80%Colore e forma:SolidPeso molecolare:2239.58NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.Formula:C62H91N19O15Purezza:97.72%Colore e forma:SolidPeso molecolare:1342.5Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFormula:C87H142N34O29S2Peso molecolare:2192.4Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Formula:C36H50Cl4N6O6SColore e forma:SolidPeso molecolare:836.7Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFormula:C56H85N17O12Purezza:98%Colore e forma:SolidPeso molecolare:1188.38Zoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Formula:C12H11NO3SPurezza:99.62%Colore e forma:SolidPeso molecolare:249.29NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Formula:C60H87N19O13Purezza:98%Colore e forma:SolidPeso molecolare:1282.48FR190997
CAS:FR190997 is an agonist of bradykinin B2 receptor.Formula:C37H33Cl2N5O5Colore e forma:SolidPeso molecolare:698.59FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Formula:C30H28BrCl2N5O4Purezza:98%Colore e forma:SolidPeso molecolare:673.38Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Formula:C16H28N6O4Purezza:98%Colore e forma:SolidPeso molecolare:368.43L 366811
CAS:L 366811 is a potent oxytocin antagonist.Formula:C43H56N8O6Colore e forma:SolidPeso molecolare:780.95JMV-1645
CAS:JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.Formula:C49H69N13O12SPurezza:98%Colore e forma:SolidPeso molecolare:1064.23MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Formula:C60H90N20O11SPurezza:98%Colore e forma:SolidPeso molecolare:1299.56Lys-[Des-Arg9]Bradykinin TFA
CAS:<p>Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.</p>Formula:C54H75F6N13O15Colore e forma:SolidPeso molecolare:1260.24Bradykinin (1-7)
CAS:Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formula:C35H52N10O9Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:756.85Bradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Formula:C30H45N9O8Purezza:98%Colore e forma:SolidPeso molecolare:659.73Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Formula:C50H73N13O11Purezza:98%Colore e forma:SolidPeso molecolare:1032.21Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Formula:C50H73N15O11Colore e forma:SolidPeso molecolare:1060.228Lys-[Hyp3]-Bradykinin
CAS:Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Formula:C56H85N17O13Colore e forma:SolidPeso molecolare:1204.38[Des-Arg9]-Bradykinin
CAS:<p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>Formula:C44H61N11O10Purezza:98%Colore e forma:SolidPeso molecolare:904.02Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formula:C27H40N8O6Colore e forma:SolidPeso molecolare:572.66Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormula:C49H70N12O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1035.15Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Formula:C61H93N19O15SPurezza:99.68% - 99.90%Colore e forma:SolidPeso molecolare:1364.575-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formula:C4H6N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:130.1Bradykinin
CAS:Bradykinin is an inflammatory mediator.Formula:C50H73N15O11Purezza:99.68%Colore e forma:SolidPeso molecolare:1060.21Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purezza:99.89%Colore e forma:SolidPeso molecolare:239.27ELN-441958
CAS:ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.Formula:C29H29ClN4O2Purezza:99.88%Colore e forma:SolidPeso molecolare:501.02SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Formula:C42H53ClN4O7SPurezza:98.59% - 99.16%Colore e forma:SolidPeso molecolare:793.41Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formula:C52H77N15O13Purezza:>99.99%Colore e forma:SolidPeso molecolare:1120.26Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formula:C54H75F6N13O15Purezza:97.35%Colore e forma:SolidPeso molecolare:1260.24[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1018.05Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purezza:>99.99%Colore e forma:SolidPeso molecolare:904.02R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Formula:C59H82F3N13O14Purezza:>99.99%Colore e forma:SolidPeso molecolare:1254.36Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purezza:99.86%Colore e forma:SolidPeso molecolare:1248.43Lys-[Des-Arg9]Bradykinin acetate
<p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and</p>Formula:C52H77N13O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1092.27Fulimetibant
CAS:Fulimetibant is a bradykinin receptor antagonist.Formula:C25H21F4N3O3Colore e forma:SolidPeso molecolare:487.45Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Formula:C34H36Cl2N6O5SPurezza:98%Colore e forma:SolidPeso molecolare:711.66NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Formula:C59H95N19O14Colore e forma:SolidPeso molecolare:1294.5BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purezza:98%Colore e forma:SolidPeso molecolare:698.55B 4148
CAS:B 4148 is a bradykinin inhibitor.Formula:C62H95N19O14S2Colore e forma:SolidPeso molecolare:1394.67Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormula:C25H34N4O5SPurezza:99.62% - 99.67%Colore e forma:SolidPeso molecolare:502.63MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formula:C22H19ClF4N2O4Purezza:99.88%Colore e forma:SolidPeso molecolare:486.84NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Formula:C36H45N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:659.84BI-113823
CAS:BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.Formula:C26H44N4O5SColore e forma:SolidPeso molecolare:524.716Fasitibant
CAS:<p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>Formula:C36H49Cl2N6O6SColore e forma:SolidPeso molecolare:764.78FK-3657
CAS:FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.Formula:C30H27Cl2N5O4Colore e forma:SolidPeso molecolare:592.47

