
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 443 prodotti di "Recettore della dopamina"
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Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formula:C20H29FN2O3Purezza:98.97% - >99.99%Colore e forma:SolidPeso molecolare:364.45Ref: TM-T70302
1mg359,00€5mg842,00€10mg1.035,00€25mg1.663,00€50mg2.072,00€100mg2.660,00€1mL*10mM (DMSO)677,00€Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Formula:C22H26ClNPurezza:98%Colore e forma:SolidPeso molecolare:339.9Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Formula:C20H25BrN4OColore e forma:SolidPeso molecolare:417.34SKF-104557
CAS:N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.Formula:C13H18N2OColore e forma:SolidPeso molecolare:218.29A 68930 hydrochloride
CAS:A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].Formula:C16H18ClNO3Colore e forma:Off-White SolidPeso molecolare:307.77A-77636
CAS:A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Formula:C20H27NO3Purezza:98%Colore e forma:SolidPeso molecolare:329.43SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Formula:C19H22BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:376.29Tau-aggregation-IN-1
CAS:Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).Formula:C28H37N5O2SColore e forma:SolidPeso molecolare:507.69SB269652
CAS:SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.Formula:C27H30N4OPurezza:98%Colore e forma:SolidPeso molecolare:426.55DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurezza:96.7%Colore e forma:SolidPeso molecolare:228.12GBR 13069 dihydrochloride
CAS:GBR 13069 dihydrochloride is a dopamine uptake inhibitor.Formula:C28H32Cl2F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:521.47Octoclothepin maleate salt
CAS:Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.Formula:C23H25ClN2O4SColore e forma:SolidPeso molecolare:460.97RTI 336
CAS:RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.Formula:C24H26Cl2N2OPurezza:98%Colore e forma:SolidPeso molecolare:429.38SV-156
CAS:SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).Formula:C21H23BrN2O2Colore e forma:SolidPeso molecolare:415.32D4R agonist-1
CAS:D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.Formula:C19H22N4SPurezza:98.44%Colore e forma:SolidPeso molecolare:338.47SKF-75670 Hydrobromide
CAS:SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.Formula:C17H20BrNO2Colore e forma:SolidPeso molecolare:350.25FR 64822
CAS:FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Formula:C11H14N4OColore e forma:SolidPeso molecolare:218.26S-3608
CAS:S-3608 is an atypical dopamine agonist.Formula:C16H20ClN3OSColore e forma:SolidPeso molecolare:337.87UNC9995
CAS:UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).Formula:C20H21Cl2N3OSPurezza:98%Colore e forma:SolidPeso molecolare:422.37NPEC-caged-dopamine
CAS:Dopamine receptor agonistFormula:C17H18N2O6Purezza:98%Colore e forma:SolidPeso molecolare:346.33RBI-257 Maleate
CAS:RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.Formula:C25H32IN3O5Colore e forma:SolidPeso molecolare:581.44Quinelorane dihydrochloride
CAS:Dopamine D2 and D3 receptor agonistFormula:C14H23ClN4Purezza:98%Colore e forma:SolidPeso molecolare:282.81A412997
CAS:A412997 is a selective agonist of dopamine D4 receptor.Formula:C19H23N3OPurezza:98%Colore e forma:SolidPeso molecolare:309.41SKF-83822
CAS:SKF-83822 is an agonist of dopamine D1-like receptor.Formula:C20H22ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:343.85BRD5814
CAS:BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.Formula:C21H23ClF3NO2Colore e forma:SolidPeso molecolare:413.86JPC-211
CAS:JPC-211 is an agonist of dopamine-receptor.Formula:C17H27NO2Purezza:98%Colore e forma:SolidPeso molecolare:277.4SB-277011 dihydrochloride
CAS:SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.Formula:C28H32Cl2N4OPurezza:98%Colore e forma:SolidPeso molecolare:511.49(+)-UH 232 maleate
CAS:D2 antagonistFormula:C18H29NOPurezza:98%Colore e forma:SolidPeso molecolare:275.43Quinpirole Hydrochloride
CAS:Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and miceFormula:C13H22ClN3Purezza:98%Colore e forma:SolidPeso molecolare:255.792-CMDO
CAS:2-CMDO is a Dopamine D2-like receptor antagonist.Formula:C23H23ClN2O5Purezza:98%Colore e forma:SolidPeso molecolare:442.89SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Formula:C18H20ClNO2Purezza:98.68%Colore e forma:SolidPeso molecolare:317.81Dopamine D2 receptor antagonist-1
CAS:Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.Formula:C14H17N3SPurezza:99.86%Colore e forma:SolidPeso molecolare:259.37Ref: TM-T11077
1mg60,00€5mg127,00€10mg188,00€25mg354,00€50mg518,00€100mg730,00€1mL*10mM (DMSO)140,00€Indatraline hydrochloride
CAS:Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)Formula:C16H16Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:328.66JHW 007 hydrochloride
CAS:JHW 007 hydrochloride is a Dopamine uptake inhibitor.Formula:C24H30ClF2NOPurezza:98%Colore e forma:SolidPeso molecolare:421.95SKF-82958
CAS:SKF 82958 is a D1/D5 receptor full agonist.Formula:C19H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:329.82CL-216303 HCl
CAS:CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.Formula:C11H12Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:264.58SKF83822 hydrobromide
CAS:SKF83822 hydrobromide is a dopamine D1-like receptor agonist.Formula:C20H23BrClNO2Purezza:98%Colore e forma:SolidPeso molecolare:424.76Piperidine-MO-1
CAS:Piperidine-MO-1 is a dopamine receptor modulator, with an ED50 of 68 μmol/kg on increase of DOPAC in the rat striatum.Formula:C14H21ClFNO2SPurezza:99.88%Colore e forma:SolidPeso molecolare:321.84PF2562
CAS:PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Formula:C19H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:331.37Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formula:C19H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:329.82ST-198
CAS:ST-198 is a dopamine D3 receptor antagonist.Formula:C22H26N2OPurezza:98%Colore e forma:SolidPeso molecolare:334.45CGP 25454A
CAS:CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.Formula:C15H21Cl2N3O2Colore e forma:SolidPeso molecolare:346.25SKF 83959 hydrobromide
CAS:SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.Formula:C18H21BrClNO2Purezza:98%Colore e forma:SolidPeso molecolare:398.72R(+)-6-Bromo-APB HBr
CAS:R(+)-6-Bromo-APB HBr is used as a D1 Dopamine receptor agonist.Formula:C19H21Br2NO2Purezza:98%Colore e forma:SolidPeso molecolare:455.18PD-89211
CAS:PD 89211 selectively blocks dopamine D4.2 receptor >800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).Formula:C19H21ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:356.85Dopamine D4 receptor antagonist-1
CAS:Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.Formula:C18H19ClN4Colore e forma:SolidPeso molecolare:326.82Lenperone
CAS:Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic.Formula:C22H23F2NO2Colore e forma:SolidPeso molecolare:371.42BAK2-66
CAS:BAK2-66 is a selective antagonist of the dopamine D3 receptor.Formula:C23H24Cl2FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:464.36Brl 20596
CAS:Brl 20596 is a central dopamine antagonist in the class of anilide.Formula:C20H24ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:373.88Mosapramine
CAS:Mosapramine is a dopamine D2-receptor antagonist.Formula:C28H35ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:479.06R-SKF-38393A HCl
CAS:R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.Formula:C16H18ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:291.77CAD031
CAS:CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.Formula:C18H14F6N2O2Colore e forma:SolidPeso molecolare:404.31Trimopam
CAS:Trimopam is a dopamine receptor agonist of the benzazepine group.Formula:C19H23NO2Colore e forma:SolidPeso molecolare:297.39ADR-851 HCl
CAS:ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.Formula:C14H19Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:332.23PD 119819
CAS:PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.Formula:C21H25Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:438.35SKF-80723 HBr
CAS:SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.Formula:C16H16BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:334.21Fluphenazine Decanoate Dihydrochloride
CAS:Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.Formula:C32H46Cl2F3N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:664.69TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColore e forma:SolidPeso molecolare:413.68PF-592379
CAS:PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).Formula:C13H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:235.33FAUC-3019
CAS:FAUC-3019 is a partial agonist of the dopamine D(4) receptor.Formula:C22H24N2OColore e forma:SolidPeso molecolare:332.44Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Colore e forma:SolidPeso molecolare:219.33PG 01037 dihydrochloride
CAS:PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.Formula:C26H28Cl4N4OPurezza:99.89%Colore e forma:SolidPeso molecolare:554.34Ref: TM-T23143
1mg39,00€2mg52,00€5mg74,00€10mg97,00€25mg144,00€50mg207,00€100mg306,00€200mg522,00€1mL*10mM (DMSO)87,00€YQA14
CAS:YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.Formula:C23H27ClN4O3Purezza:99.52%Colore e forma:SolidPeso molecolare:442.94GBR-13069 dimethanesulfonate
CAS:GBR-13069 dimethanesulfonate is a dopamine reuptake inhibitor.Formula:C30H38F2N2O7S2Colore e forma:SolidPeso molecolare:640.76Oxypertine
CAS:Oxypertine, an indole-derived antipsychotic, treats psychoses like mania, schizophrenia, and severe anxiety, akin to chlorpromazine.Formula:C23H29N3O2Colore e forma:SolidPeso molecolare:379.5Milenperone
CAS:Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.Formula:C22H23ClFN3O2Purezza:98.09% - 99.84%Colore e forma:SolidPeso molecolare:415.89GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Formula:C28H34Cl2N2OPurezza:98.08%Colore e forma:SolidPeso molecolare:485.49CCG 203769
CAS:CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.Formula:C8H14N2O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:202.27Ref: TM-T10705
1mg88,00€5mg187,00€10mg264,00€25mg469,00€50mg657,00€100mg944,00€500mg1.882,00€1mL*10mM (DMSO)207,00€Benperidol
CAS:Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formula:C22H24FN3O2Purezza:99.91%Colore e forma:SolidPeso molecolare:381.44Ref: TM-T26360
1mg116,00€5mg276,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)279,00€U 99194 maleate
CAS:U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formula:C21H31NO6Purezza:99.45%Colore e forma:SolidPeso molecolare:393.47MLS1547
CAS:MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Formula:C19H19ClN4OPurezza:99.64%Colore e forma:SolidPeso molecolare:354.83Remoxipride hydrochloride
CAS:Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-Formula:C16H24BrClN2O3Purezza:99.88%Colore e forma:SolidPeso molecolare:407.73Molindone
CAS:<p>Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.</p>Formula:C16H24N2O2Purezza:99.37% - 99.46%Colore e forma:Off-White SolidPeso molecolare:276.37Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Formula:C14H20FNO2SPurezza:99.39%Colore e forma:SolidPeso molecolare:285.38Seridopidine
CAS:Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.Formula:C14H20FNO2SPurezza:99.77%Colore e forma:SolidPeso molecolare:285.387-Hydroxy-DPAT hydrobromide
CAS:7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formula:C16H26BrNOPurezza:99.73%Colore e forma:SolidPeso molecolare:328.29SK609 HCl
CAS:SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.Formula:C10H15Cl2NPurezza:99.02%Colore e forma:SolidPeso molecolare:220.14PF-00217830
CAS:PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.Formula:C26H30N4O2Purezza:98.72%Colore e forma:SolidPeso molecolare:430.54A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formula:C20H27F3N6OSPurezza:98.80%Colore e forma:SolidPeso molecolare:456.53Ref: TM-T10213
1mg89,00€5mg198,00€10mg279,00€25mg434,00€50mg562,00€100mg780,00€200mg1.035,00€1mL*10mM (DMSO)227,00€Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formula:C23H24FN3O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formula:C21H22ClFN4O2Purezza:96.57%Colore e forma:SolidPeso molecolare:416.88BP14979
CAS:BP14979 is D3R-selective partial agonist.Formula:C23H34N4O2Purezza:98.29% - 99.73%Colore e forma:SolidPeso molecolare:398.54NGD 94-1
CAS:NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.Formula:C18H20N6Purezza:99.61%Colore e forma:SolidPeso molecolare:320.39PD 168568 dihydrochloride
CAS:PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Formula:C22H29Cl2N3OPurezza:99.71%Colore e forma:SolidPeso molecolare:422.39Ref: TM-T12383
5mg48,00€10mg58,00€25mg117,00€50mg170,00€100mg248,00€200mg348,00€1mL*10mM (DMSO)60,00€CyPPA
CAS:<p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>Formula:C16H23N5Purezza:99.88%Colore e forma:SolidPeso molecolare:285.39Medifoxamine
CAS:Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.MedifoxamineFormula:C16H19NO2Purezza:98.88%Colore e forma:SolidPeso molecolare:257.33Ref: TM-T24444
1mg99,00€5mg235,00€10mg354,00€25mg635,00€50mg893,00€100mg1.159,00€1mL*10mM (DMSO)259,00€SB-277011
CAS:SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).Formula:C28H30N4OPurezza:99.39%Colore e forma:SolidPeso molecolare:438.56Ref: TM-T12861
1mg47,00€5mg58,00€10mg93,00€25mg158,00€50mg254,00€100mgPrezzo su richiesta1mL*10mM (DMSO)60,00€Brilaroxazine
CAS:Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Formula:C22H25Cl2N3O3Purezza:99.36%Colore e forma:SolidPeso molecolare:450.36Ref: TM-T14782
1mg105,00€5mg250,00€10mg406,00€25mg700,00€50mg1.008,00€100mg1.378,00€200mg1.833,00€1mL*10mM (DMSO)283,00€JNJ-37822681 dihydrochloride
CAS:JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的,可快速解离的多巴胺 D2受体拮抗剂,与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。Formula:C17H19Cl2F5N4Purezza:99.78%Colore e forma:SolidPeso molecolare:445.26LY3154885
CAS:LY3154885 is an orally active dopamine D1 receptor orthosteric modulator (PAM) that reduces the risk of drug-drug interactions (DDI).Formula:C23H23Cl2N3O2Colore e forma:SolidPeso molecolare:444.35CY 208-243
CAS:CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.Formula:C19H18N2Purezza:98%Colore e forma:SolidPeso molecolare:274.36PW0464
CAS:PW0464 ((Rac)-Razpipadon) is a non-catechol D1R agonist and potent omplete G protein biased ligand with an EC50 (Gs-cAMP)=5.8 nM for neurological disorders.Formula:C19H17F2N3O4Purezza:98.78%Colore e forma:SolidPeso molecolare:389.35Ref: TM-T36946
1mg169,00€5mg408,00€10mg670,00€25mg1.296,00€50mg1.941,00€100mg2.608,00€1mL*10mM (DMSO)449,00€SKF 81297 hydrobromide
CAS:SKF 81297 hydrobromide, a selective agonist of the dopamine D1-like receptor,exhibits central activity and is widely used to study the neuromodulatory effects.Formula:C16H17BrClNO2Purezza:99.52%Colore e forma:SolidPeso molecolare:370.67Dihydrexidine
CAS:Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.Formula:C17H17NO2Purezza:98%Colore e forma:SolidPeso molecolare:267.32AJ-76 hydrochloride
CAS:AJ-76 hydrochloride ((+)-AJ 76 hydrochloride) serves as a dopamine autoreceptor antagonist, exhibiting pK i values of 6.95 for hD3, 6.67 for hD4, 6.37 for hD2S, 6.21 for hD2L, and 6.07 for rD2 receptors, indicating its binding affinity strength across these receptor types.Formula:C15H24ClNOColore e forma:SolidPeso molecolare:269.81LBT 999
CAS:LBT 999 is used as a dopamine reuptake inhibitor.Formula:C20H26FNO2Colore e forma:SolidPeso molecolare:331.42Carbidine dihydrochloride
CAS:Carbidine, a gamma-carboline derivative, is an atypical antipsychotic that modulates dopamine release and tyrosine hydroxylase activity.Formula:C13H20Cl2N2Purezza:98.59%Colore e forma:SolidPeso molecolare:275.217Z1078601926
CAS:Z1078601926 is an allosteric inhibitor of the human dopamine transporter (hDAT) and exhibits a synergistic effect when combined with Nomifensine [1].Formula:C14H19FN2OColore e forma:SolidPeso molecolare:250.31ABT-670
CAS:ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.Formula:C19H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:325.4SKF 81297
CAS:SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].Formula:C16H16ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:289.76
