
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 443 prodotti di "Recettore della dopamina"
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SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Formula:C10H14ClNColore e forma:SolidPeso molecolare:183.68Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Colore e forma:SolidPeso molecolare:491.49Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formula:C32H44F3N3O2SPurezza:98.14%Colore e forma:SolidPeso molecolare:591.77Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formula:C17H18Cl3NOPurezza:98.86% - 99.93%Colore e forma:SolidPeso molecolare:358.69Aplindore
CAS:Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formula:C18H18N2O3Colore e forma:SolidPeso molecolare:310.35FAUC 213
CAS:<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Formula:C18H19ClN4Purezza:99.84%Colore e forma:SolidPeso molecolare:326.82Metoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Colore e forma:SolidPeso molecolare:372.72Sonepiprazole mesylate
CAS:Sonepiprazole mesylate is a selective D4 antagonistFormula:C22H31N3O6S2Colore e forma:SolidPeso molecolare:497.63FAUC 346
CAS:FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formula:C24H29N3O2SPurezza:99.46%Colore e forma:SolidPeso molecolare:423.57Ref: TM-T9081
2mg35,00€5mg49,00€10mg81,00€25mg145,00€50mg235,00€100mg379,00€200mg517,00€1mL*10mM (DMSO)55,00€Vanoxerine dihydrochloride
CAS:Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)Formula:C28H34Cl2F2N2OPurezza:98.16% - 98.35%Colore e forma:White SolidPeso molecolare:523.49Pramipexole dihydrochloride hydrate
CAS:Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formula:C10H17N3S·2HCl·H2OPurezza:99.68%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:302.26Ref: TM-T6951
10mg47,00€25mg74,00€50mg119,00€100mg170,00€200mg255,00€500mg430,00€1mL*10mM (DMSO)47,00€Sultopride hydrochloride
CAS:Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formula:C17H27ClN2O4SPurezza:≥95%Colore e forma:White Or Yellowish PowderPeso molecolare:390.93Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurezza:99.78%Colore e forma:SolidPeso molecolare:331.86J-147
CAS:J-147, a curcumin derivative, is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging.Formula:C18H17F3N2O2Purezza:99.61% - >99.99%Colore e forma:SolidPeso molecolare:350.33Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormula:C40H67N7O10Purezza:99.95%Colore e forma:SolidPeso molecolare:805.9D-tetrahydropalmatine
CAS:D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.Formula:C21H25NO4Purezza:99.34%Colore e forma:SolidPeso molecolare:355.43Ref: TM-T4S0779
2mg44,00€5mg64,00€10mg97,00€25mg182,00€50mg273,00€100mg393,00€200mg558,00€1mL*10mM (DMSO)65,00€Pergolide
CAS:Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormula:C19H26N2SPurezza:99.95%Colore e forma:SolidPeso molecolare:314.49Ref: TM-T21340
2mg38,00€5mg57,00€10mg80,00€25mg116,00€50mg167,00€100mg250,00€200mg370,00€1mL*10mM (DMSO)64,00€Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formula:C19H16F3N3O3Purezza:99.33% - 99.8%Colore e forma:SolidPeso molecolare:391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Trimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formula:C21H29ClN2O5Purezza:99.52%Colore e forma:SolidPeso molecolare:424.92Bromocriptine mesylate
CAS:Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)Formula:C33H44BrN5O8SPurezza:99.85% - 99.96%Colore e forma:White SolidPeso molecolare:750.7PD-168077 maleate
CAS:PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formula:C24H26N4O5Purezza:99.13%Colore e forma:SolidPeso molecolare:450.49Ref: TM-T5047
2mg35,00€5mg52,00€10mg80,00€25mg150,00€50mg245,00€100mg364,00€200mg517,00€1mL*10mM (DMSO)58,00€Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formula:C17H25N3O5SPurezza:99.65%Colore e forma:SolidPeso molecolare:383.46Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formula:C18H19ClN4OPurezza:98.65% - 99.94%Colore e forma:SolidPeso molecolare:342.82Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formula:C23H31ClN4O2SPurezza:99.37%Colore e forma:White SolidPeso molecolare:463SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurezza:98% - 99.83%Colore e forma:SolidPeso molecolare:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€A-381393
CAS:A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Formula:C20H24N4Purezza:99.00%Colore e forma:SolidPeso molecolare:320.43Ref: TM-T5397
1mg40,00€5mg80,00€10mg117,00€25mg210,00€50mg304,00€100mg437,00€200mg615,00€1mL*10mM (DMSO)88,00€Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formula:C24H23ClF3NPurezza:99.99%Colore e forma:SolidPeso molecolare:417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurezza:99.78% - >99.99%Colore e forma:SolidPeso molecolare:463.87Pridopidine
CAS:Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formula:C15H23NO2SPurezza:95.2% - 99.89%Colore e forma:SolidPeso molecolare:281.41lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurezza:95.83% - 99.95%Colore e forma:SolidPeso molecolare:565.7Ropinirole hydrochloride
CAS:Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Formula:C16H24N2O·HClPurezza:99.87% - 99.98%Colore e forma:Off-White SolidPeso molecolare:296.84(-)-Isocorypalmine
CAS:(-)-Isocorypalmine ((S)-Tetrahydrocolumbamine), a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.Formula:C20H23NO4Purezza:98.18% - 99.97%Colore e forma:SolidPeso molecolare:341.4Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formula:C11H16ClNO4Purezza:95.00%Colore e forma:SolidPeso molecolare:261.7Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purezza:99.33%Colore e forma:SolidPeso molecolare:354.27MPTP hydrochloride
CAS:MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.Formula:C12H16ClNPurezza:96.35% - >99.99%Colore e forma:SolidPeso molecolare:209.72Ref: TM-T4081
5mg35,00€10mg50,00€25mg85,00€50mg138,00€100mg187,00€200mg298,00€500mg472,00€1mL*10mM (DMSO)52,00€Phenelzine
CAS:Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formula:C8H12N2Purezza:98%Colore e forma:LiquidPeso molecolare:136.19Ref: TM-T9540
5mgPrezzo su richiesta10mgPrezzo su richiesta25mgPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiesta200mgPrezzo su richiesta500mgPrezzo su richiestaZatebradine
CAS:Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formula:C26H36N2O5Purezza:98%Colore e forma:SolidPeso molecolare:456.57Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formula:C10H17N3SPurezza:99.78%Colore e forma:SolidPeso molecolare:211.33Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purezza:99.41% - >99.99%Colore e forma:SolidPeso molecolare:517.66Protein deglycase DJ-1 against-1
CAS:Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formula:C24H23N3O4Purezza:97.23%Colore e forma:SolidPeso molecolare:417.46(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS:(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H14D5Cl2N3SColore e forma:SolidPeso molecolare:289.28L-745870
CAS:L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formula:C18H19ClN4Purezza:98%Colore e forma:SolidPeso molecolare:326.82Ropinirole
CAS:Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Formula:C16H24N2OPurezza:99.68%Colore e forma:SolidPeso molecolare:260.38Dopamine D4 receptor ligand 2
CAS:Compound 17, a dopamine D4 receptor ligand, exhibits high potency and selectivity with IC 50 values of 0.057 nM for D4, and >1000, 220, and 270 nM for D2, 5-HT1A, and α1 receptors, respectively [1].Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88Vanoxerine
CAS:Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).Formula:C28H32F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:450.56Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.27Lergotrile mesylate
CAS:Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.Formula:C18H22ClN3O3SColore e forma:SolidPeso molecolare:395.9Bromperidol decanoate
CAS:Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.Formula:C31H41BrFNO3Colore e forma:SolidPeso molecolare:574.56LY 171859
CAS:LY 171859 is an agonist of D2-receptor.Formula:C17H14O5Purezza:98%Colore e forma:SolidPeso molecolare:298.29Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Formula:C22H25NO6Purezza:98%Colore e forma:SolidPeso molecolare:399.44Clothixamide
CAS:Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.Formula:C24H28ClN3OSPurezza:95.51%Colore e forma:SolidPeso molecolare:442.02CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purezza:98%Colore e forma:SolidPeso molecolare:231.33'-Fluorobenzylspiperone maleate
CAS:<p>ligand for the D2 receptor</p>Formula:C34H35F2N3O6Purezza:98%Colore e forma:SolidPeso molecolare:619.66NGB 2904 hydrochloride
CAS:dopamine D3 receptor antagonistFormula:C28H30Cl3N3OPurezza:98%Colore e forma:SolidPeso molecolare:530.92Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Formula:C25H31NOPurezza:98%Colore e forma:SolidPeso molecolare:361.52PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Formula:C11H17N3SPurezza:98%Colore e forma:SolidPeso molecolare:223.34U-101958 Maleate
CAS:U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.Formula:C25H33N3O5Purezza:98%Colore e forma:SolidPeso molecolare:455.55Roxindole hydrochloride
CAS:Dopamine D2 autoreceptor agonistFormula:C23H27ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:382.93Sch 24518
CAS:Sc h24518 is an antagonist of D1 receptor.Formula:C16H17BrClNOPurezza:98%Colore e forma:SolidPeso molecolare:354.67Sultopride
CAS:Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.Formula:C17H26N2O4SColore e forma:SolidPeso molecolare:354.46GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Colore e forma:SolidPeso molecolare:530.665Lergotrile
CAS:Lergotrile is used as an enzyme Inhibitor (Prolactin).Formula:C17H18ClN3Purezza:98%Colore e forma:SolidPeso molecolare:299.8CJB-090 2HCl
CAS:CJB-090 2HCl is a partial agonist of the dopamine D3 receptor.Formula:C26H30Cl4N4OColore e forma:SolidPeso molecolare:556.35Oxiperomide
CAS:Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.Formula:C20H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:337.42Gyki 32887
CAS:Gyki 32887 is a dopamine agonist.Formula:C23H28N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:516.57Amitifadine free base
CAS:Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.Formula:C11H11Cl2NColore e forma:SolidPeso molecolare:228.12A 69024
CAS:A 69024 is a highly selective antagonist of dopamine D-1 receptor.Formula:C20H24BrNO4Purezza:98%Colore e forma:SolidPeso molecolare:422.31Seproxetine HCl
CAS:Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.Formula:C16H17ClF3NOPurezza:98%Colore e forma:SolidPeso molecolare:331.76A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurezza:98%Colore e forma:SolidPeso molecolare:337.89Clopenthixol
CAS:Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.Formula:C22H25ClN2OSColore e forma:SolidPeso molecolare:400.96SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:403.86U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColore e forma:SolidPeso molecolare:325.45PF-06256142
CAS:PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).Formula:C21H16N4O2Purezza:98%Colore e forma:SolidPeso molecolare:356.38Remoxipride
CAS:Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.Formula:C16H23BrN2O3Purezza:98%Colore e forma:SolidPeso molecolare:371.27A68930
CAS:A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.Formula:C16H17NO3Colore e forma:SolidPeso molecolare:271.31Zelandopam free base
CAS:Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.Formula:C15H15NO4Colore e forma:SolidPeso molecolare:273.28PD168,077
CAS:PD168,077 is an agonist of dopamine D4 receptor. It has a facilitatory effect on memory consolidation.Formula:C20H22N4OPurezza:98%Colore e forma:SolidPeso molecolare:334.41Savoxepin mesylate
CAS:Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.Formula:C26H30N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:466.59Nafadotride
CAS:Nafadotride is a dopamine D3 receptor antagonist.Formula:C22H27N3O2Colore e forma:SolidPeso molecolare:365.47WAY-260022
CAS:WAY-260022 is the norepinephrine transporter inhibitor.Formula:C21H31F3N2O2Purezza:97.61% - 99.41%Colore e forma:SolidPeso molecolare:400.48(R)-PF-06256142
CAS:(R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.Formula:C21H16N4O2Colore e forma:SolidPeso molecolare:356.38L 741742 hydrochloride
CAS:L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.Formula:C23H26Cl2N2OPurezza:99.9%Colore e forma:SolidPeso molecolare:417.37SV293
CAS:SV293 is a selective antagonist of D2 dopamine receptor.Formula:C22H26N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:382.52Org-10490
CAS:Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.Formula:C17H19NOPurezza:98%Colore e forma:SolidPeso molecolare:253.34ST-836
CAS:ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H34N4OSPurezza:98%Colore e forma:SolidPeso molecolare:414.61GBR 12783
CAS:GBR 12783 enhances memory, boosts rat hippocampal acetylcholine, and is a potent dopamine uptake inhibitor with IC50s of 1.8/1.2 nM in rats/mice.Formula:C28H32N2OPurezza:98%Colore e forma:SolidPeso molecolare:412.57Foscarbidopa
CAS:Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.Formula:C10H15N2O7PPurezza:96.17% - 97.27%Colore e forma:SolidPeso molecolare:306.21Talipexole
CAS:Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.Formula:C10H15N3SPurezza:98%Colore e forma:SolidPeso molecolare:209.31UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Formula:C23H28Cl2N4O2Purezza:98.78% - 98.78%Colore e forma:SolidPeso molecolare:463.4Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formula:C13H18N2Purezza:98%Colore e forma:SolidPeso molecolare:202.3PD 120697
CAS:PD 120697 is a dopamine antagonist with central dopamine agonist properties.Formula:C11H15N3SPurezza:98%Colore e forma:SolidPeso molecolare:221.32Acetophenazine
CAS:Acetophenazine is an anxiolytic compound that is used in the study of depression.Formula:C23H29N3O2SPurezza:99.30%Colore e forma:SoildPeso molecolare:411.56L-750,667 Trihydrochloride
CAS:L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.Formula:C18H22Cl3IN4Purezza:99.63%Colore e forma:SolidPeso molecolare:527.66Tesofensine
CAS:Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.Formula:C17H23Cl2NOPurezza:98%Colore e forma:SolidPeso molecolare:328.286-Chloromelatonin
CAS:6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.Formula:C13H15ClN2O2Purezza:97.26% - 99.25%Colore e forma:SolidPeso molecolare:266.72Ref: TM-T22530
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€CP-226269
CAS:<p>CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.</p>Formula:C18H19FN4Purezza:99.08%Colore e forma:SolidPeso molecolare:310.37(-)-GSK598809
CAS:(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.Formula:C22H23F4N5OSPurezza:98%Colore e forma:SolidPeso molecolare:481.51Lenperone HCl
CAS:Lenperone HCl is a dopamine antagonist and an antipsychotic agent.Formula:C22H24ClF2NO2Purezza:98%Colore e forma:SolidPeso molecolare:407.88Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formula:C20H29FN2O3Purezza:98.97% - >99.99%Colore e forma:SolidPeso molecolare:364.45Ref: TM-T70302
1mg359,00€5mg842,00€10mg1.035,00€25mg1.663,00€50mg2.072,00€100mg2.660,00€1mL*10mM (DMSO)677,00€Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Formula:C22H26ClNPurezza:98%Colore e forma:SolidPeso molecolare:339.9Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Formula:C20H25BrN4OColore e forma:SolidPeso molecolare:417.34SKF-104557
CAS:N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.Formula:C13H18N2OColore e forma:SolidPeso molecolare:218.29A 68930 hydrochloride
CAS:A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].Formula:C16H18ClNO3Colore e forma:Off-White SolidPeso molecolare:307.77A-77636
CAS:A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Formula:C20H27NO3Purezza:98%Colore e forma:SolidPeso molecolare:329.43SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Formula:C19H22BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:376.29Tau-aggregation-IN-1
CAS:Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).Formula:C28H37N5O2SColore e forma:SolidPeso molecolare:507.69SB269652
CAS:SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.Formula:C27H30N4OPurezza:98%Colore e forma:SolidPeso molecolare:426.55DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurezza:96.7%Colore e forma:SolidPeso molecolare:228.12GBR 13069 dihydrochloride
CAS:GBR 13069 dihydrochloride is a dopamine uptake inhibitor.Formula:C28H32Cl2F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:521.47Octoclothepin maleate salt
CAS:Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.Formula:C23H25ClN2O4SColore e forma:SolidPeso molecolare:460.97RTI 336
CAS:RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.Formula:C24H26Cl2N2OPurezza:98%Colore e forma:SolidPeso molecolare:429.38SV-156
CAS:SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).Formula:C21H23BrN2O2Colore e forma:SolidPeso molecolare:415.32D4R agonist-1
CAS:D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.Formula:C19H22N4SPurezza:98.44%Colore e forma:SolidPeso molecolare:338.47SKF-75670 Hydrobromide
CAS:SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.Formula:C17H20BrNO2Colore e forma:SolidPeso molecolare:350.25FR 64822
CAS:FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Formula:C11H14N4OColore e forma:SolidPeso molecolare:218.26S-3608
CAS:S-3608 is an atypical dopamine agonist.Formula:C16H20ClN3OSColore e forma:SolidPeso molecolare:337.87UNC9995
CAS:UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).Formula:C20H21Cl2N3OSPurezza:98%Colore e forma:SolidPeso molecolare:422.37NPEC-caged-dopamine
CAS:Dopamine receptor agonistFormula:C17H18N2O6Purezza:98%Colore e forma:SolidPeso molecolare:346.33RBI-257 Maleate
CAS:RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.Formula:C25H32IN3O5Colore e forma:SolidPeso molecolare:581.44Quinelorane dihydrochloride
CAS:Dopamine D2 and D3 receptor agonistFormula:C14H23ClN4Purezza:98%Colore e forma:SolidPeso molecolare:282.81A412997
CAS:A412997 is a selective agonist of dopamine D4 receptor.Formula:C19H23N3OPurezza:98%Colore e forma:SolidPeso molecolare:309.41SKF-83822
CAS:SKF-83822 is an agonist of dopamine D1-like receptor.Formula:C20H22ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:343.85BRD5814
CAS:BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.Formula:C21H23ClF3NO2Colore e forma:SolidPeso molecolare:413.86JPC-211
CAS:JPC-211 is an agonist of dopamine-receptor.Formula:C17H27NO2Purezza:98%Colore e forma:SolidPeso molecolare:277.4SB-277011 dihydrochloride
CAS:SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.Formula:C28H32Cl2N4OPurezza:98%Colore e forma:SolidPeso molecolare:511.49(+)-UH 232 maleate
CAS:D2 antagonistFormula:C18H29NOPurezza:98%Colore e forma:SolidPeso molecolare:275.43Quinpirole Hydrochloride
CAS:Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and miceFormula:C13H22ClN3Purezza:98%Colore e forma:SolidPeso molecolare:255.792-CMDO
CAS:2-CMDO is a Dopamine D2-like receptor antagonist.Formula:C23H23ClN2O5Purezza:98%Colore e forma:SolidPeso molecolare:442.89SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Formula:C18H20ClNO2Purezza:98.68%Colore e forma:SolidPeso molecolare:317.81Dopamine D2 receptor antagonist-1
CAS:Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.Formula:C14H17N3SPurezza:99.86%Colore e forma:SolidPeso molecolare:259.37Ref: TM-T11077
1mg60,00€5mg127,00€10mg188,00€25mg354,00€50mg518,00€100mg730,00€1mL*10mM (DMSO)140,00€Indatraline hydrochloride
CAS:Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)Formula:C16H16Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:328.66JHW 007 hydrochloride
CAS:JHW 007 hydrochloride is a Dopamine uptake inhibitor.Formula:C24H30ClF2NOPurezza:98%Colore e forma:SolidPeso molecolare:421.95SKF-82958
CAS:SKF 82958 is a D1/D5 receptor full agonist.Formula:C19H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:329.82CL-216303 HCl
CAS:CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.Formula:C11H12Cl3NPurezza:98%Colore e forma:SolidPeso molecolare:264.58SKF83822 hydrobromide
CAS:SKF83822 hydrobromide is a dopamine D1-like receptor agonist.Formula:C20H23BrClNO2Purezza:98%Colore e forma:SolidPeso molecolare:424.76Piperidine-MO-1
CAS:Piperidine-MO-1 is a dopamine receptor modulator, with an ED50 of 68 μmol/kg on increase of DOPAC in the rat striatum.Formula:C14H21ClFNO2SPurezza:99.88%Colore e forma:SolidPeso molecolare:321.84PF2562
CAS:PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Formula:C19H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:331.37Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formula:C19H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:329.82ST-198
CAS:ST-198 is a dopamine D3 receptor antagonist.Formula:C22H26N2OPurezza:98%Colore e forma:SolidPeso molecolare:334.45CGP 25454A
CAS:CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.Formula:C15H21Cl2N3O2Colore e forma:SolidPeso molecolare:346.25SKF 83959 hydrobromide
CAS:SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.Formula:C18H21BrClNO2Purezza:98%Colore e forma:SolidPeso molecolare:398.72R(+)-6-Bromo-APB HBr
CAS:R(+)-6-Bromo-APB HBr is used as a D1 Dopamine receptor agonist.Formula:C19H21Br2NO2Purezza:98%Colore e forma:SolidPeso molecolare:455.18PD-89211
CAS:PD 89211 selectively blocks dopamine D4.2 receptor >800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).Formula:C19H21ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:356.85Dopamine D4 receptor antagonist-1
CAS:Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.Formula:C18H19ClN4Colore e forma:SolidPeso molecolare:326.82Lenperone
CAS:Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic.Formula:C22H23F2NO2Colore e forma:SolidPeso molecolare:371.42BAK2-66
CAS:BAK2-66 is a selective antagonist of the dopamine D3 receptor.Formula:C23H24Cl2FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:464.36Brl 20596
CAS:Brl 20596 is a central dopamine antagonist in the class of anilide.Formula:C20H24ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:373.88Mosapramine
CAS:Mosapramine is a dopamine D2-receptor antagonist.Formula:C28H35ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:479.06R-SKF-38393A HCl
CAS:R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.Formula:C16H18ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:291.77CAD031
CAS:CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.Formula:C18H14F6N2O2Colore e forma:SolidPeso molecolare:404.31Trimopam
CAS:Trimopam is a dopamine receptor agonist of the benzazepine group.Formula:C19H23NO2Colore e forma:SolidPeso molecolare:297.39ADR-851 HCl
CAS:ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.Formula:C14H19Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:332.23PD 119819
CAS:PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.Formula:C21H25Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:438.35SKF-80723 HBr
CAS:SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.Formula:C16H16BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:334.21Fluphenazine Decanoate Dihydrochloride
CAS:Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.Formula:C32H46Cl2F3N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:664.69TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColore e forma:SolidPeso molecolare:413.68PF-592379
CAS:PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).Formula:C13H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:235.33FAUC-3019
CAS:FAUC-3019 is a partial agonist of the dopamine D(4) receptor.Formula:C22H24N2OColore e forma:SolidPeso molecolare:332.44Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Colore e forma:SolidPeso molecolare:219.33PG 01037 dihydrochloride
CAS:PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.Formula:C26H28Cl4N4OPurezza:99.89%Colore e forma:SolidPeso molecolare:554.34Ref: TM-T23143
1mg39,00€2mg52,00€5mg74,00€10mg97,00€25mg144,00€50mg207,00€100mg306,00€200mg522,00€1mL*10mM (DMSO)87,00€YQA14
CAS:YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.Formula:C23H27ClN4O3Purezza:99.52%Colore e forma:SolidPeso molecolare:442.94GBR-13069 dimethanesulfonate
CAS:GBR-13069 dimethanesulfonate is a dopamine reuptake inhibitor.Formula:C30H38F2N2O7S2Colore e forma:SolidPeso molecolare:640.76Oxypertine
CAS:Oxypertine, an indole-derived antipsychotic, treats psychoses like mania, schizophrenia, and severe anxiety, akin to chlorpromazine.Formula:C23H29N3O2Colore e forma:SolidPeso molecolare:379.5Milenperone
CAS:Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.Formula:C22H23ClFN3O2Purezza:98.09% - 99.84%Colore e forma:SolidPeso molecolare:415.89GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Formula:C28H34Cl2N2OPurezza:98.08%Colore e forma:SolidPeso molecolare:485.49CCG 203769
CAS:CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.Formula:C8H14N2O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:202.27Ref: TM-T10705
1mg88,00€5mg187,00€10mg264,00€25mg469,00€50mg657,00€100mg944,00€500mg1.882,00€1mL*10mM (DMSO)207,00€Benperidol
CAS:Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formula:C22H24FN3O2Purezza:99.91%Colore e forma:SolidPeso molecolare:381.44Ref: TM-T26360
1mg116,00€5mg276,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€1mL*10mM (DMSO)279,00€U 99194 maleate
CAS:U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formula:C21H31NO6Purezza:99.45%Colore e forma:SolidPeso molecolare:393.47MLS1547
CAS:MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Formula:C19H19ClN4OPurezza:99.64%Colore e forma:SolidPeso molecolare:354.83Remoxipride hydrochloride
CAS:Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-Formula:C16H24BrClN2O3Purezza:99.88%Colore e forma:SolidPeso molecolare:407.73Molindone
CAS:<p>Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.</p>Formula:C16H24N2O2Purezza:99.37% - 99.46%Colore e forma:Off-White SolidPeso molecolare:276.37Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Formula:C14H20FNO2SPurezza:99.39%Colore e forma:SolidPeso molecolare:285.38Seridopidine
CAS:Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.Formula:C14H20FNO2SPurezza:99.77%Colore e forma:SolidPeso molecolare:285.387-Hydroxy-DPAT hydrobromide
CAS:7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formula:C16H26BrNOPurezza:99.73%Colore e forma:SolidPeso molecolare:328.29SK609 HCl
CAS:SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.Formula:C10H15Cl2NPurezza:99.02%Colore e forma:SolidPeso molecolare:220.14PF-00217830
CAS:PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.Formula:C26H30N4O2Purezza:98.72%Colore e forma:SolidPeso molecolare:430.54A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formula:C20H27F3N6OSPurezza:98.80%Colore e forma:SolidPeso molecolare:456.53Ref: TM-T10213
1mg89,00€5mg198,00€10mg279,00€25mg434,00€50mg562,00€100mg780,00€200mg1.035,00€1mL*10mM (DMSO)227,00€Fananserin
CAS:Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formula:C23H24FN3O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:425.52Ref: TM-T15270
2mg42,00€5mg56,00€10mg81,00€25mg116,00€50mg170,00€100mg250,00€200mg369,00€1mL*10mM (DMSO)62,00€Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formula:C21H22ClFN4O2Purezza:96.57%Colore e forma:SolidPeso molecolare:416.88BP14979
CAS:BP14979 is D3R-selective partial agonist.Formula:C23H34N4O2Purezza:98.29% - 99.73%Colore e forma:SolidPeso molecolare:398.54NGD 94-1
CAS:NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.Formula:C18H20N6Purezza:99.61%Colore e forma:SolidPeso molecolare:320.39PD 168568 dihydrochloride
CAS:PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Formula:C22H29Cl2N3OPurezza:99.71%Colore e forma:SolidPeso molecolare:422.39Ref: TM-T12383
5mg48,00€10mg58,00€25mg117,00€50mg170,00€100mg248,00€200mg348,00€1mL*10mM (DMSO)60,00€CyPPA
CAS:<p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>Formula:C16H23N5Purezza:99.88%Colore e forma:SolidPeso molecolare:285.39Medifoxamine
CAS:Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.MedifoxamineFormula:C16H19NO2Purezza:98.88%Colore e forma:SolidPeso molecolare:257.33Ref: TM-T24444
1mg99,00€5mg235,00€10mg354,00€25mg635,00€50mg893,00€100mg1.159,00€1mL*10mM (DMSO)259,00€SB-277011
CAS:SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).Formula:C28H30N4OPurezza:99.39%Colore e forma:SolidPeso molecolare:438.56Ref: TM-T12861
1mg47,00€5mg58,00€10mg93,00€25mg158,00€50mg254,00€100mgPrezzo su richiesta1mL*10mM (DMSO)60,00€Brilaroxazine
CAS:Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Formula:C22H25Cl2N3O3Purezza:99.36%Colore e forma:SolidPeso molecolare:450.36Ref: TM-T14782
1mg105,00€5mg250,00€10mg406,00€25mg700,00€50mg1.008,00€100mg1.378,00€200mg1.833,00€1mL*10mM (DMSO)283,00€JNJ-37822681 dihydrochloride
CAS:JNJ-37822681 dihydrochloride 是特异性的、有中枢活性的,可快速解离的多巴胺 D2受体拮抗剂,与多巴胺 D2L 受体结合的亲和力适中 (Ki=158 nM)。JNJ-37822681 dihydrochloride 在精神分裂症和躁郁症领域有研究价值。Formula:C17H19Cl2F5N4Purezza:99.78%Colore e forma:SolidPeso molecolare:445.26LY3154885
CAS:LY3154885 is an orally active dopamine D1 receptor orthosteric modulator (PAM) that reduces the risk of drug-drug interactions (DDI).Formula:C23H23Cl2N3O2Colore e forma:SolidPeso molecolare:444.35CY 208-243
CAS:CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.Formula:C19H18N2Purezza:98%Colore e forma:SolidPeso molecolare:274.36PW0464
CAS:PW0464 ((Rac)-Razpipadon) is a non-catechol D1R agonist and potent omplete G protein biased ligand with an EC50 (Gs-cAMP)=5.8 nM for neurological disorders.Formula:C19H17F2N3O4Purezza:98.78%Colore e forma:SolidPeso molecolare:389.35Ref: TM-T36946
1mg169,00€5mg408,00€10mg670,00€25mg1.296,00€50mg1.941,00€100mg2.608,00€1mL*10mM (DMSO)449,00€SKF 81297 hydrobromide
CAS:SKF 81297 hydrobromide, a selective agonist of the dopamine D1-like receptor,exhibits central activity and is widely used to study the neuromodulatory effects.Formula:C16H17BrClNO2Purezza:99.52%Colore e forma:SolidPeso molecolare:370.67Dihydrexidine
CAS:Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.Formula:C17H17NO2Purezza:98%Colore e forma:SolidPeso molecolare:267.32AJ-76 hydrochloride
CAS:AJ-76 hydrochloride ((+)-AJ 76 hydrochloride) serves as a dopamine autoreceptor antagonist, exhibiting pK i values of 6.95 for hD3, 6.67 for hD4, 6.37 for hD2S, 6.21 for hD2L, and 6.07 for rD2 receptors, indicating its binding affinity strength across these receptor types.Formula:C15H24ClNOColore e forma:SolidPeso molecolare:269.81LBT 999
CAS:LBT 999 is used as a dopamine reuptake inhibitor.Formula:C20H26FNO2Colore e forma:SolidPeso molecolare:331.42Carbidine dihydrochloride
CAS:Carbidine, a gamma-carboline derivative, is an atypical antipsychotic that modulates dopamine release and tyrosine hydroxylase activity.Formula:C13H20Cl2N2Purezza:98.59%Colore e forma:SolidPeso molecolare:275.217Z1078601926
CAS:Z1078601926 is an allosteric inhibitor of the human dopamine transporter (hDAT) and exhibits a synergistic effect when combined with Nomifensine [1].Formula:C14H19FN2OColore e forma:SolidPeso molecolare:250.31ABT-670
CAS:ABT-670 is a selective agonist of dopamine D4 receptor. For human D4, ferret D4, and rat D4, the EC50 values are 89 nM, 160 nM, and 93 nM , respectively.Formula:C19H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:325.4SKF 81297
CAS:SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].Formula:C16H16ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:289.76
