Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 445 prodotti di "Recettore della dopamina"
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Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFormula:C21H22CL2N4OSPurezza:97.97% - 99.82%Colore e forma:SolidPeso molecolare:449.4Tetrahydropalmatine
CAS:Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epilepticFormula:C21H25NO4Purezza:99.59% - 99.95%Colore e forma:SolidPeso molecolare:355.43Spiperone
CAS:Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formula:C23H26FN3O2Purezza:99.34% - 99.91%Colore e forma:SolidPeso molecolare:395.47Talquetamab
CAS:Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment of multiple myeloma.Colore e forma:LiquidPeso molecolare:144.59 kDaQuetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purezza:99.32% - >99.99%Colore e forma:White Crystalline SolidPeso molecolare:883.09Oxidopamine hydrobromide
CAS:Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Formula:C8H12BrNO3Purezza:98.22% - 99.88%Colore e forma:Beige To Brown Fine Crystalline PowderPeso molecolare:250.09Paliperidone
CAS:Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Formula:C23H27FN4O3Purezza:95% - 99.08%Colore e forma:Off White To Light Orange Coloured SolidPeso molecolare:426.48BP 897 hydrochloride
CAS:BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.Formula:C26H32ClN3O2Purezza:99.42%Colore e forma:SolidPeso molecolare:454Haloperidol
CAS:Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Formula:C21H23ClFNO2Purezza:98.69% - 98.97%Colore e forma:Crystals SolidPeso molecolare:375.86ONC206
CAS:ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations andFormula:C23H22F2N4OPurezza:99.38% - 99.81%Colore e forma:SolidPeso molecolare:408.44Benserazide hydrochloride
CAS:Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.Formula:C10H15N3O5·HClPurezza:98.63% - 99.74%Colore e forma:White Crystalline SolidPeso molecolare:293.7Vanicoside E
CAS:Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formula:C53H52O22Colore e forma:SolidPeso molecolare:1040.97D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Colore e forma:Odour SolidDETQ
CAS:DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.Formula:C22H25Cl2NO3Colore e forma:SolidPeso molecolare:422.34Neuromedin N
CAS:Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Formula:C38H63N7O8Purezza:98%Colore e forma:SolidPeso molecolare:745.95Fenoldopam
CAS:Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).Formula:C16H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:305.76Losulazine
CAS:Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.Formula:C27H22F4N4O3SPurezza:98.83%Colore e forma:SolidPeso molecolare:558.55Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Colore e forma:Odour Solid[18F]-Labeled L-dopa precursor
CAS:[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formula:C35H36N2O7Colore e forma:SolidPeso molecolare:596.67MLS1082
CAS:MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formula:C24H23N3O2Purezza:99.53%Colore e forma:SolidPeso molecolare:385.46ABT 724 trihydrochloride
CAS:ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formula:C17H22Cl3N5Purezza:99.91%Colore e forma:SolidPeso molecolare:402.75Ref: TM-T22019
5mg40,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)44,00€(Iso)-WAY-260022
CAS:(Iso)-WAY-260022 ((Iso)-NRI-022) is a stereoisomer of WAY-260022, a norepinephrine reuptake inhibitor and selective inhibitor of 5-hydroxytryptamine and dopamine transport proteins.Formula:C21H31F3N2O2Purezza:97.68% - 99.36%Colore e forma:SoildPeso molecolare:400.48Onzigolide
CAS:Onzigolide (BIM-23A760) is a dual agonist for D2R and SSTR2 with strong dopamine and somatostatin properties.Formula:C86H116N16O12S4Colore e forma:SolidPeso molecolare:1694.21Octodrine
CAS:Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.Formula:C8H19NPurezza:99.98%Colore e forma:Clear Colorless To Light Yellow LiquidPeso molecolare:129.24D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nMFormula:C22H27Cl2N3OPurezza:98%Colore e forma:SolidPeso molecolare:420.38D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Formula:C27H37NO5Purezza:98%Colore e forma:SolidPeso molecolare:455.59Clomipramine D3
CAS:Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formula:C19H23ClN2Purezza:98%Colore e forma:SolidPeso molecolare:317.87A 31472
CAS:A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H22ClNColore e forma:SolidPeso molecolare:335.87N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS:N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Formula:C10H16ClNColore e forma:SolidPeso molecolare:185.69S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Formula:C29H29N3O2Purezza:98%Colore e forma:SolidPeso molecolare:451.56MOR agonist-3
MOR agonist-3 (Compound 84) is a dual D3R/MOR antagonist with K i values of 382 nM and 55.2 nM, respectively.Colore e forma:Odour SolidAmisulpride hydrochloride
CAS:Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Formula:C17H28ClN3O4SColore e forma:SolidPeso molecolare:405.94Dopamine D2 receptor agonist-2
CAS:Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
Formula:C25H31Cl2N5OSPurezza:98.93%Colore e forma:SoildPeso molecolare:520.527-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Formula:C16H22INOColore e forma:SolidPeso molecolare:371.262A 77636 hydrochloride
CAS:A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).Formula:C20H28ClNO3Purezza:99.57%Colore e forma:SolidPeso molecolare:365.89ADTN hydrobromide
CAS:ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).Formula:C10H14BrNO2Colore e forma:SolidPeso molecolare:260.13MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:680.71LE 300
CAS:LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formula:C20H22N2Purezza:97.91% - 98.79%Colore e forma:SolidPeso molecolare:290.4PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formula:C22H30N2O3SColore e forma:SolidPeso molecolare:402.55Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78Cabergoline
CAS:Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.
Formula:C26H37N5O2Purezza:97.69% - 99.86%Colore e forma:White Crystalline SolidPeso molecolare:451.6O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Formula:C14H16Cl2O2Colore e forma:SolidPeso molecolare:287.18Haloperidol D4
CAS:Haloperidol D4 is deuterium-labeled haloperidol.Formula:C21H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:379.89ADTN
CAS:ADTN is an agonist of the dopamine receptor.Formula:C10H13NO2Purezza:98%Colore e forma:SolidPeso molecolare:179.22(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Formula:C159H252N40O58Purezza:98%Colore e forma:SolidPeso molecolare:3651.95Fluphenazine free base
CAS:Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Formula:C22H26F3N3OSColore e forma:SolidPeso molecolare:437.52Quinelorane
CAS:Quinelorane is dextrorotary isomer.Formula:C14H22N4Colore e forma:SolidPeso molecolare:246.35N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formula:C15H22ClNO2Purezza:98.85% - 99.54%Colore e forma:SolidPeso molecolare:283.79Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Formula:C22H26ClNO4SColore e forma:SolidPeso molecolare:435.96
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