
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 445 prodotti di "Recettore della dopamina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurezza:98.77% - 99.756%Colore e forma:Pale Yellow Crystals SolidPeso molecolare:315.86Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Sonepiprazole mesylate
CAS:Sonepiprazole mesylate is a selective D4 antagonistFormula:C22H31N3O6S2Colore e forma:SolidPeso molecolare:497.63Azaperone
CAS:Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Formula:C19H22FN3OPurezza:98.73%Colore e forma:White Or Off-White CrystallinePeso molecolare:327.4Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Formula:C24H25FN4O2Purezza:99.33%Colore e forma:SolidPeso molecolare:420.48Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formula:C25H27N3O2SPurezza:99.06% - 99.96%Colore e forma:SolidPeso molecolare:433.57Ref: TM-T2306
5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€1mL*10mM (DMSO)Prezzo su richiestaMetoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Colore e forma:SolidPeso molecolare:372.72FAUC 346
CAS:FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formula:C24H29N3O2SPurezza:99.46%Colore e forma:SolidPeso molecolare:423.57Ref: TM-T9081
2mg34,00€5mg50,00€10mg77,00€25mg138,00€50mg224,00€100mg359,00€200mg490,00€1mL*10mM (DMSO)52,00€Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formula:C17H18Cl3NOPurezza:98.86% - 99.93%Colore e forma:SolidPeso molecolare:358.69Fluphenazine decanoate
CAS:Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.
Formula:C32H44F3N3O2SPurezza:98.14%Colore e forma:SolidPeso molecolare:591.77Aplindore
CAS:Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formula:C18H18N2O3Colore e forma:SolidPeso molecolare:310.35Fluoroclebopride
CAS:Fluoroclebopride is a dopamine (DA) D2 receptor ligand.Formula:C20H23ClFN3O2Purezza:99.68% - 99.91%Colore e forma:SolidPeso molecolare:391.87Ref: TM-T3187
1mg34,00€5mg71,00€10mg90,00€25mg150,00€50mg222,00€100mg356,00€500mg820,00€1mL*10mM (DMSO)90,00€L-745870 trihydrochloride
CAS:L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
Formula:C18H22Cl4N4Purezza:97.52%Colore e forma:SolidPeso molecolare:436.21Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purezza:99.8% - 99.91%Colore e forma:Off-White SolidPeso molecolare:355.43Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Colore e forma:SolidPeso molecolare:491.49FAUC 213
CAS:FAUC 213 is a selective full antagonist of the dopamine D4 receptor.Formula:C18H19ClN4Purezza:99.84%Colore e forma:SolidPeso molecolare:326.82Piribedil
CAS:Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.Formula:C16H18N4O2Purezza:99.79% - 99.82%Colore e forma:SolidPeso molecolare:298.34Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68SKF38393 hydrobromide
CAS:SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Formula:C16H18BrNO2Purezza:98.99%Colore e forma:SolidPeso molecolare:336.22Rimcazole
CAS:Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Formula:C21H27N3Purezza:98%Colore e forma:SolidPeso molecolare:321.46Dasotraline
CAS:Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.Formula:C16H15Cl2NColore e forma:SolidPeso molecolare:292.2Haloperidol hydrochloride
CAS:Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.Formula:C21H24Cl2FNO2Colore e forma:SolidPeso molecolare:412.33PD 168568
CAS:PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.Formula:C22H27N3OColore e forma:SolidPeso molecolare:349.47Alizapride
CAS:Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].Formula:C16H21N5O2Colore e forma:SolidPeso molecolare:315.37OS-3-106
CAS:OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.Formula:C25H30N4O2SPurezza:99.4% - 99.57%Colore e forma:SolidPeso molecolare:450.6JNJ-37822681
CAS:JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.Formula:C17H17F5N4Purezza:99.84%Colore e forma:SolidPeso molecolare:372.34Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formula:C24H32ClNO3Purezza:99.57% - 99.77%Colore e forma:SolidPeso molecolare:417.97Tiapride
CAS:Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.Formula:C15H24N2O4SColore e forma:SolidPeso molecolare:328.43Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formula:C19H26ClNOSPurezza:99.53% - 99.56%Colore e forma:Almost White To White Crystalline PowderPeso molecolare:351.93Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formula:C20H30N2O3S2Purezza:99.70%Colore e forma:White To Off-White SolidPeso molecolare:410.59BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formula:C26H31N3O2Purezza:99.44%Colore e forma:SolidPeso molecolare:417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurezza:98.08% - 99.59%Colore e forma:SolidPeso molecolare:315.47Ref: TM-T6647
5mg50,00€10mg73,00€25mg138,00€50mg241,00€100mg358,00€200mg523,00€500mg822,00€1mL*10mM (DMSO)52,00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurezza:99.23%Colore e forma:White PowderPeso molecolare:426.57carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.
Formula:C24H31N3O2SPurezza:98.06%Colore e forma:SolidPeso molecolare:425.59Sonepiprazole hydrochloride
CAS:Sonepiprazole HCl is a a selective dopamine D4 antagonist.Formula:C21H28ClN3O3SColore e forma:SolidPeso molecolare:437.98SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Formula:C10H14ClNColore e forma:SolidPeso molecolare:183.68Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purezza:98.76% - 99.79%Colore e forma:SolidPeso molecolare:295.38Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Formula:C15H20Cl2N2O3Purezza:99.17%Colore e forma:SolidPeso molecolare:347.24Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Formula:C24H29ClFNO5Colore e forma:SolidPeso molecolare:465.95L-DOPA methyl ester (hydrochloride)
CAS:L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.
Formula:C10H14ClNO4Purezza:98.69% - 99.81%Colore e forma:White SolidPeso molecolare:247.675Tetrahydropalmatine hydrochloride
CAS:Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Formula:C21H26ClNO4Purezza:98% - 99.59%Colore e forma:SolidPeso molecolare:391.888Zuclopenthixol dihydrochloride
CAS:Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.Formula:C22H27Cl3N2OSPurezza:98%Colore e forma:SolidPeso molecolare:473.89AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Formula:C21H24ClF2NOPurezza:99.89%Colore e forma:SolidPeso molecolare:379.87Ref: TM-T39429
2mg34,00€5mg49,00€10mg75,00€25mg130,00€50mg192,00€100mg295,00€200mg442,00€1mL*10mM (DMSO)50,00€Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88L-745870 hydrochloride
CAS:L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFormula:C18H20Cl2N4Purezza:97.36%Colore e forma:SolidPeso molecolare:363.28Ref: TM-T11799
5mg40,00€10mg65,00€25mg111,00€50mg178,00€100mg259,00€200mg374,00€1mL*10mM (DMSO)34,00€Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purezza:99.83% - 99.97%Colore e forma:SolidPeso molecolare:403.52Domperidone monomaleate
CAS:Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Formula:C26H28ClN5O6Colore e forma:SolidPeso molecolare:541.98Mesdopetam
CAS:Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.Formula:C12H18FNO3SColore e forma:SolidPeso molecolare:275.34Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Colore e forma:SolidPeso molecolare:380.71Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Formula:C28H42F2N2O12S2Purezza:99.98%Colore e forma:SolidPeso molecolare:700.77
