Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 443 prodotti di "Recettore della dopamina"
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SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Formula:C10H14ClNColore e forma:SolidPeso molecolare:183.68Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Colore e forma:SolidPeso molecolare:491.49Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formula:C32H44F3N3O2SPurezza:98.14%Colore e forma:SolidPeso molecolare:591.77Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formula:C17H18Cl3NOPurezza:98.86% - 99.93%Colore e forma:SolidPeso molecolare:358.69Aplindore
CAS:Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formula:C18H18N2O3Colore e forma:SolidPeso molecolare:310.35FAUC 213
CAS:<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Formula:C18H19ClN4Purezza:99.84%Colore e forma:SolidPeso molecolare:326.82Metoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Colore e forma:SolidPeso molecolare:372.72Sonepiprazole mesylate
CAS:Sonepiprazole mesylate is a selective D4 antagonistFormula:C22H31N3O6S2Colore e forma:SolidPeso molecolare:497.63FAUC 346
CAS:FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formula:C24H29N3O2SPurezza:99.46%Colore e forma:SolidPeso molecolare:423.57Ref: TM-T9081
2mg35,00€5mg49,00€10mg81,00€25mg145,00€50mg235,00€100mg379,00€200mg517,00€1mL*10mM (DMSO)55,00€Vanoxerine dihydrochloride
CAS:Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)Formula:C28H34Cl2F2N2OPurezza:98.16% - 98.35%Colore e forma:White SolidPeso molecolare:523.49Pramipexole dihydrochloride hydrate
CAS:Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formula:C10H17N3S·2HCl·H2OPurezza:99.68%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:302.26Ref: TM-T6951
10mg47,00€25mg74,00€50mg119,00€100mg170,00€200mg255,00€500mg430,00€1mL*10mM (DMSO)47,00€Sultopride hydrochloride
CAS:Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formula:C17H27ClN2O4SPurezza:≥95%Colore e forma:White Or Yellowish PowderPeso molecolare:390.93Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurezza:99.78%Colore e forma:SolidPeso molecolare:331.86J-147
CAS:J-147, a curcumin derivative, is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging.Formula:C18H17F3N2O2Purezza:99.61% - >99.99%Colore e forma:SolidPeso molecolare:350.33Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormula:C40H67N7O10Purezza:99.95%Colore e forma:SolidPeso molecolare:805.9D-tetrahydropalmatine
CAS:D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.Formula:C21H25NO4Purezza:99.34%Colore e forma:SolidPeso molecolare:355.43Ref: TM-T4S0779
2mg44,00€5mg64,00€10mg97,00€25mg182,00€50mg273,00€100mg393,00€200mg558,00€1mL*10mM (DMSO)65,00€Pergolide
CAS:Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormula:C19H26N2SPurezza:99.95%Colore e forma:SolidPeso molecolare:314.49Ref: TM-T21340
2mg38,00€5mg57,00€10mg80,00€25mg116,00€50mg167,00€100mg250,00€200mg370,00€1mL*10mM (DMSO)64,00€Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formula:C19H16F3N3O3Purezza:99.33% - 99.8%Colore e forma:SolidPeso molecolare:391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Trimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formula:C21H29ClN2O5Purezza:99.52%Colore e forma:SolidPeso molecolare:424.92Bromocriptine mesylate
CAS:Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)Formula:C33H44BrN5O8SPurezza:99.85% - 99.96%Colore e forma:White SolidPeso molecolare:750.7PD-168077 maleate
CAS:PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formula:C24H26N4O5Purezza:99.13%Colore e forma:SolidPeso molecolare:450.49Ref: TM-T5047
2mg35,00€5mg52,00€10mg80,00€25mg150,00€50mg245,00€100mg364,00€200mg517,00€1mL*10mM (DMSO)58,00€Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formula:C17H25N3O5SPurezza:99.65%Colore e forma:SolidPeso molecolare:383.46Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formula:C18H19ClN4OPurezza:98.65% - 99.94%Colore e forma:SolidPeso molecolare:342.82Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formula:C23H31ClN4O2SPurezza:99.37%Colore e forma:White SolidPeso molecolare:463SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurezza:98% - 99.83%Colore e forma:SolidPeso molecolare:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€A-381393
CAS:A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Formula:C20H24N4Purezza:99.00%Colore e forma:SolidPeso molecolare:320.43Ref: TM-T5397
1mg40,00€5mg80,00€10mg117,00€25mg210,00€50mg304,00€100mg437,00€200mg615,00€1mL*10mM (DMSO)88,00€Xaliproden hydrochloride
CAS:Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formula:C24H23ClF3NPurezza:99.99%Colore e forma:SolidPeso molecolare:417.89Ref: TM-T9272
1mg40,00€5mg85,00€10mg120,00€25mg235,00€50mg376,00€100mg540,00€200mg775,00€1mL*10mM (DMSO)96,00€Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurezza:99.78% - >99.99%Colore e forma:SolidPeso molecolare:463.87Pridopidine
CAS:Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formula:C15H23NO2SPurezza:95.2% - 99.89%Colore e forma:SolidPeso molecolare:281.41lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurezza:95.83% - 99.95%Colore e forma:SolidPeso molecolare:565.7Ropinirole hydrochloride
CAS:Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Formula:C16H24N2O·HClPurezza:99.87% - 99.98%Colore e forma:Off-White SolidPeso molecolare:296.84(-)-Isocorypalmine
CAS:(-)-Isocorypalmine ((S)-Tetrahydrocolumbamine), a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.Formula:C20H23NO4Purezza:98.18% - 99.97%Colore e forma:SolidPeso molecolare:341.4Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formula:C11H16ClNO4Purezza:95.00%Colore e forma:SolidPeso molecolare:261.7Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purezza:99.33%Colore e forma:SolidPeso molecolare:354.27MPTP hydrochloride
CAS:MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.Formula:C12H16ClNPurezza:96.35% - >99.99%Colore e forma:SolidPeso molecolare:209.72Ref: TM-T4081
5mg35,00€10mg50,00€25mg85,00€50mg138,00€100mg187,00€200mg298,00€500mg472,00€1mL*10mM (DMSO)52,00€Phenelzine
CAS:Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formula:C8H12N2Purezza:98%Colore e forma:LiquidPeso molecolare:136.19Ref: TM-T9540
5mgPrezzo su richiesta10mgPrezzo su richiesta25mgPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiesta200mgPrezzo su richiesta500mgPrezzo su richiestaZatebradine
CAS:Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formula:C26H36N2O5Purezza:98%Colore e forma:SolidPeso molecolare:456.57Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formula:C10H17N3SPurezza:99.78%Colore e forma:SolidPeso molecolare:211.33Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purezza:99.41% - >99.99%Colore e forma:SolidPeso molecolare:517.66Protein deglycase DJ-1 against-1
CAS:Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formula:C24H23N3O4Purezza:97.23%Colore e forma:SolidPeso molecolare:417.46(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS:(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H14D5Cl2N3SColore e forma:SolidPeso molecolare:289.28L-745870
CAS:L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formula:C18H19ClN4Purezza:98%Colore e forma:SolidPeso molecolare:326.82Ropinirole
CAS:Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Formula:C16H24N2OPurezza:99.68%Colore e forma:SolidPeso molecolare:260.38Dopamine D4 receptor ligand 2
CAS:Compound 17, a dopamine D4 receptor ligand, exhibits high potency and selectivity with IC 50 values of 0.057 nM for D4, and >1000, 220, and 270 nM for D2, 5-HT1A, and α1 receptors, respectively [1].Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88Vanoxerine
CAS:Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).Formula:C28H32F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:450.56Pardoprunox
CAS:Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.27Lergotrile mesylate
CAS:Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.Formula:C18H22ClN3O3SColore e forma:SolidPeso molecolare:395.9Bromperidol decanoate
CAS:Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.Formula:C31H41BrFNO3Colore e forma:SolidPeso molecolare:574.56
