
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 443 prodotti di "Recettore della dopamina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
LY 171859
CAS:LY 171859 is an agonist of D2-receptor.Formula:C17H14O5Purezza:98%Colore e forma:SolidPeso molecolare:298.29Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Formula:C22H25NO6Purezza:98%Colore e forma:SolidPeso molecolare:399.44Clothixamide
CAS:Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.Formula:C24H28ClN3OSPurezza:95.51%Colore e forma:SolidPeso molecolare:442.02CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purezza:98%Colore e forma:SolidPeso molecolare:231.33'-Fluorobenzylspiperone maleate
CAS:<p>ligand for the D2 receptor</p>Formula:C34H35F2N3O6Purezza:98%Colore e forma:SolidPeso molecolare:619.66NGB 2904 hydrochloride
CAS:dopamine D3 receptor antagonistFormula:C28H30Cl3N3OPurezza:98%Colore e forma:SolidPeso molecolare:530.92Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Formula:C25H31NOPurezza:98%Colore e forma:SolidPeso molecolare:361.52PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Formula:C11H17N3SPurezza:98%Colore e forma:SolidPeso molecolare:223.34U-101958 Maleate
CAS:U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.Formula:C25H33N3O5Purezza:98%Colore e forma:SolidPeso molecolare:455.55Roxindole hydrochloride
CAS:Dopamine D2 autoreceptor agonistFormula:C23H27ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:382.93Sch 24518
CAS:Sc h24518 is an antagonist of D1 receptor.Formula:C16H17BrClNOPurezza:98%Colore e forma:SolidPeso molecolare:354.67Sultopride
CAS:Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.Formula:C17H26N2O4SColore e forma:SolidPeso molecolare:354.46GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Colore e forma:SolidPeso molecolare:530.665Lergotrile
CAS:Lergotrile is used as an enzyme Inhibitor (Prolactin).Formula:C17H18ClN3Purezza:98%Colore e forma:SolidPeso molecolare:299.8CJB-090 2HCl
CAS:CJB-090 2HCl is a partial agonist of the dopamine D3 receptor.Formula:C26H30Cl4N4OColore e forma:SolidPeso molecolare:556.35Oxiperomide
CAS:Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.Formula:C20H23N3O2Purezza:98%Colore e forma:SolidPeso molecolare:337.42Gyki 32887
CAS:Gyki 32887 is a dopamine agonist.Formula:C23H28N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:516.57Amitifadine free base
CAS:Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.Formula:C11H11Cl2NColore e forma:SolidPeso molecolare:228.12A 69024
CAS:A 69024 is a highly selective antagonist of dopamine D-1 receptor.Formula:C20H24BrNO4Purezza:98%Colore e forma:SolidPeso molecolare:422.31Seproxetine HCl
CAS:Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.Formula:C16H17ClF3NOPurezza:98%Colore e forma:SolidPeso molecolare:331.76A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurezza:98%Colore e forma:SolidPeso molecolare:337.89Clopenthixol
CAS:Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.Formula:C22H25ClN2OSColore e forma:SolidPeso molecolare:400.96SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:403.86U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColore e forma:SolidPeso molecolare:325.45PF-06256142
CAS:PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).Formula:C21H16N4O2Purezza:98%Colore e forma:SolidPeso molecolare:356.38Remoxipride
CAS:Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.Formula:C16H23BrN2O3Purezza:98%Colore e forma:SolidPeso molecolare:371.27A68930
CAS:A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.Formula:C16H17NO3Colore e forma:SolidPeso molecolare:271.31Zelandopam free base
CAS:Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.Formula:C15H15NO4Colore e forma:SolidPeso molecolare:273.28PD168,077
CAS:PD168,077 is an agonist of dopamine D4 receptor. It has a facilitatory effect on memory consolidation.Formula:C20H22N4OPurezza:98%Colore e forma:SolidPeso molecolare:334.41Savoxepin mesylate
CAS:Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.Formula:C26H30N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:466.59Nafadotride
CAS:Nafadotride is a dopamine D3 receptor antagonist.Formula:C22H27N3O2Colore e forma:SolidPeso molecolare:365.47WAY-260022
CAS:WAY-260022 is the norepinephrine transporter inhibitor.Formula:C21H31F3N2O2Purezza:97.61% - 99.41%Colore e forma:SolidPeso molecolare:400.48(R)-PF-06256142
CAS:(R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.Formula:C21H16N4O2Colore e forma:SolidPeso molecolare:356.38L 741742 hydrochloride
CAS:L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.Formula:C23H26Cl2N2OPurezza:99.9%Colore e forma:SolidPeso molecolare:417.37SV293
CAS:SV293 is a selective antagonist of D2 dopamine receptor.Formula:C22H26N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:382.52Org-10490
CAS:Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.Formula:C17H19NOPurezza:98%Colore e forma:SolidPeso molecolare:253.34ST-836
CAS:ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H34N4OSPurezza:98%Colore e forma:SolidPeso molecolare:414.61GBR 12783
CAS:GBR 12783 enhances memory, boosts rat hippocampal acetylcholine, and is a potent dopamine uptake inhibitor with IC50s of 1.8/1.2 nM in rats/mice.Formula:C28H32N2OPurezza:98%Colore e forma:SolidPeso molecolare:412.57Foscarbidopa
CAS:Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.Formula:C10H15N2O7PPurezza:96.17% - 97.27%Colore e forma:SolidPeso molecolare:306.21Talipexole
CAS:Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.Formula:C10H15N3SPurezza:98%Colore e forma:SolidPeso molecolare:209.31UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Formula:C23H28Cl2N4O2Purezza:98.78% - 98.78%Colore e forma:SolidPeso molecolare:463.4Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formula:C13H18N2Purezza:98%Colore e forma:SolidPeso molecolare:202.3PD 120697
CAS:PD 120697 is a dopamine antagonist with central dopamine agonist properties.Formula:C11H15N3SPurezza:98%Colore e forma:SolidPeso molecolare:221.32Acetophenazine
CAS:Acetophenazine is an anxiolytic compound that is used in the study of depression.Formula:C23H29N3O2SPurezza:99.30%Colore e forma:SoildPeso molecolare:411.56L-750,667 Trihydrochloride
CAS:L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.Formula:C18H22Cl3IN4Purezza:99.63%Colore e forma:SolidPeso molecolare:527.66Tesofensine
CAS:Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.Formula:C17H23Cl2NOPurezza:98%Colore e forma:SolidPeso molecolare:328.286-Chloromelatonin
CAS:6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.Formula:C13H15ClN2O2Purezza:97.26% - 99.25%Colore e forma:SolidPeso molecolare:266.72Ref: TM-T22530
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€CP-226269
CAS:<p>CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.</p>Formula:C18H19FN4Purezza:99.08%Colore e forma:SolidPeso molecolare:310.37(-)-GSK598809
CAS:(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.Formula:C22H23F4N5OSPurezza:98%Colore e forma:SolidPeso molecolare:481.51Lenperone HCl
CAS:Lenperone HCl is a dopamine antagonist and an antipsychotic agent.Formula:C22H24ClF2NO2Purezza:98%Colore e forma:SolidPeso molecolare:407.88
