
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 444 prodotti di "Recettore della dopamina"
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(+)-UH 232 maleate
CAS:D2 antagonistFormula:C18H29NOPurezza:98%Colore e forma:SolidPeso molecolare:275.43A412997
CAS:A412997 is a selective agonist of dopamine D4 receptor.Formula:C19H23N3OPurezza:98%Colore e forma:SolidPeso molecolare:309.41S-3608
CAS:S-3608 is an atypical dopamine agonist.Formula:C16H20ClN3OSColore e forma:SolidPeso molecolare:337.87FR 64822
CAS:FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Formula:C11H14N4OColore e forma:SolidPeso molecolare:218.26SV-156
CAS:SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).Formula:C21H23BrN2O2Colore e forma:SolidPeso molecolare:415.32Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Formula:C22H26ClNPurezza:98%Colore e forma:SolidPeso molecolare:339.9Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Formula:C20H25BrN4OColore e forma:SolidPeso molecolare:417.34SKF-104557
CAS:N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.Formula:C13H18N2OColore e forma:SolidPeso molecolare:218.29A 68930 hydrochloride
CAS:A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].Formula:C16H18ClNO3Colore e forma:Off-White SolidPeso molecolare:307.77SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Formula:C19H22BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:376.29Tau-aggregation-IN-1
CAS:Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).Formula:C28H37N5O2SColore e forma:SolidPeso molecolare:507.69DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurezza:96.7%Colore e forma:SolidPeso molecolare:228.12Octoclothepin maleate salt
CAS:Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.Formula:C23H25ClN2O4SColore e forma:SolidPeso molecolare:460.97RTI 336
CAS:RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.Formula:C24H26Cl2N2OPurezza:98%Colore e forma:SolidPeso molecolare:429.38SKF-75670 Hydrobromide
CAS:SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.Formula:C17H20BrNO2Colore e forma:SolidPeso molecolare:350.25UNC9995
CAS:UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).Formula:C20H21Cl2N3OSPurezza:98%Colore e forma:SolidPeso molecolare:422.37NPEC-caged-dopamine
CAS:Dopamine receptor agonistFormula:C17H18N2O6Purezza:98%Colore e forma:SolidPeso molecolare:346.33RBI-257 Maleate
CAS:RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.Formula:C25H32IN3O5Colore e forma:SolidPeso molecolare:581.44Quinelorane dihydrochloride
CAS:Dopamine D2 and D3 receptor agonistFormula:C14H23ClN4Purezza:98%Colore e forma:SolidPeso molecolare:282.81SKF-83822
CAS:SKF-83822 is an agonist of dopamine D1-like receptor.Formula:C20H22ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:343.85BRD5814
CAS:BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.Formula:C21H23ClF3NO2Colore e forma:SolidPeso molecolare:413.86SB-277011 dihydrochloride
CAS:SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.Formula:C28H32Cl2N4OPurezza:98%Colore e forma:SolidPeso molecolare:511.49PF2562
CAS:PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Formula:C19H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:331.37Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formula:C19H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:329.82Lenperone
CAS:Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic.Formula:C22H23F2NO2Colore e forma:SolidPeso molecolare:371.42BAK2-66
CAS:BAK2-66 is a selective antagonist of the dopamine D3 receptor.Formula:C23H24Cl2FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:464.36Brl 20596
CAS:Brl 20596 is a central dopamine antagonist in the class of anilide.Formula:C20H24ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:373.88FAUC-3019
CAS:FAUC-3019 is a partial agonist of the dopamine D(4) receptor.Formula:C22H24N2OColore e forma:SolidPeso molecolare:332.44Lergotrile
CAS:Lergotrile is used as an enzyme Inhibitor (Prolactin).Formula:C17H18ClN3Purezza:98%Colore e forma:SolidPeso molecolare:299.8CJB-090 2HCl
CAS:CJB-090 2HCl is a partial agonist of the dopamine D3 receptor.Formula:C26H30Cl4N4OColore e forma:SolidPeso molecolare:556.35Gyki 32887
CAS:Gyki 32887 is a dopamine agonist.Formula:C23H28N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:516.57Amitifadine free base
CAS:Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.Formula:C11H11Cl2NColore e forma:SolidPeso molecolare:228.12A 69024
CAS:A 69024 is a highly selective antagonist of dopamine D-1 receptor.Formula:C20H24BrNO4Purezza:98%Colore e forma:SolidPeso molecolare:422.31Seproxetine HCl
CAS:Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.Formula:C16H17ClF3NOPurezza:98%Colore e forma:SolidPeso molecolare:331.76A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurezza:98%Colore e forma:SolidPeso molecolare:337.89Lergotrile mesylate
CAS:Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.Formula:C18H22ClN3O3SColore e forma:SolidPeso molecolare:395.9Bromperidol decanoate
CAS:Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.Formula:C31H41BrFNO3Colore e forma:SolidPeso molecolare:574.56LY 171859
CAS:LY 171859 is an agonist of D2-receptor.Formula:C17H14O5Purezza:98%Colore e forma:SolidPeso molecolare:298.29Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Formula:C22H25NO6Purezza:98%Colore e forma:SolidPeso molecolare:399.44Clothixamide
CAS:Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.Formula:C24H28ClN3OSPurezza:95.51%Colore e forma:SolidPeso molecolare:442.02CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purezza:98%Colore e forma:SolidPeso molecolare:231.33'-Fluorobenzylspiperone maleate
CAS:ligand for the D2 receptorFormula:C34H35F2N3O6Purezza:98%Colore e forma:SolidPeso molecolare:619.66Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Formula:C25H31NOPurezza:98%Colore e forma:SolidPeso molecolare:361.52PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Formula:C11H17N3SPurezza:98%Colore e forma:SolidPeso molecolare:223.34Sch 24518
CAS:Sc h24518 is an antagonist of D1 receptor.Formula:C16H17BrClNOPurezza:98%Colore e forma:SolidPeso molecolare:354.67Trimopam
CAS:Trimopam is a dopamine receptor agonist of the benzazepine group.Formula:C19H23NO2Colore e forma:SolidPeso molecolare:297.39SKF-80723 HBr
CAS:SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.Formula:C16H16BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:334.21TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColore e forma:SolidPeso molecolare:413.68GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Colore e forma:SolidPeso molecolare:530.665Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Colore e forma:SolidPeso molecolare:219.33
