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GPCR19

GPCR19

GPCR19, noto anche come GPR19, è un membro della famiglia dei recettori accoppiati alle proteine G, i cui ruoli sono ancora in fase di chiarimento in vari processi fisiologici. Sebbene meno caratterizzato rispetto ad altri GPCR, GPCR19 è di interesse nella ricerca focalizzata sulla scoperta di nuovi bersagli terapeutici per malattie metaboliche, cancro e disturbi neurologici. Presso CymitQuimica, offriamo una selezione di strumenti di ricerca e reagenti per supportare le vostre indagini sulle funzioni e le potenziali applicazioni terapeutiche di GPCR19.

Trovati 33 prodotti di "GPCR19"

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  • BAR501
    Targetmol
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    BAR501

    CAS:
    BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。
    Formula:C26H46O3
    Purezza:99.29% - 99.68%
    Colore e forma:Solid
    Peso molecolare:406.64

    Ref: TM-T4083

  • PEN (human) aceate
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    PEN (human) aceate

    PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.
    Formula:C99H163N27O34
    Purezza:99.25%
    Colore e forma:Solid
    Peso molecolare:2275.51

    Ref: TM-TP1949L

  • Ursodeoxycholic acid sodium
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    Ursodeoxycholic acid sodium

    CAS:
    <p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>
    Formula:C24H40NaO4
    Purezza:99.66% - 99.96%
    Colore e forma:Solid
    Peso molecolare:415.56

    Ref: TM-T29078

  • WB403
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    WB403

    CAS:
    WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.
    Formula:C19H19BrN2OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.34

    Ref: TM-T29154

  • CAY10789
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    CAY10789

    CAS:
    CAY10789: potent CysLT1R antagonist (IC50 2.8 µM), GPBAR1 agonist (EC50 3 µM), reduces U937 cell adhesion, TNF-α, stable with promising pharmacokinetics.
    Formula:C17H15NO2
    Colore e forma:Solid
    Peso molecolare:265.31

    Ref: TM-T60439

  • TGR5 agonist 3
    Targetmol
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    TGR5 agonist 3

    CAS:
    Compound 8, a cholic acid derivative, functions as a selective TGR5 agonist and exhibits an EC50 value of 5 μM [1].
    Formula:C28H48O5
    Colore e forma:Solid
    Peso molecolare:464.68

    Ref: TM-T79424

  • TGR5 Receptor Agonist 4
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    TGR5 Receptor Agonist 4

    CAS:
    TGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM
    Formula:C25H27ClN2O5
    Colore e forma:Solid
    Peso molecolare:470.95

    Ref: TM-T81000

  • INT-777 R-enantiomer
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    INT-777 R-enantiomer

    CAS:
    INT-777 is the R-enantiomer of INT-777, less potent than INT-777,EC50 of 4.79 μM for TGR5.
    Formula:C27H46O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:450.65

    Ref: TM-T11662

  • RO5527239
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    RO5527239

    CAS:
    RO5527239 is a potent, orally available GPBAR1 agonist agent.
    Formula:C28H31N3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:457.56

    Ref: TM-T26108

  • INT-777
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    INT-777

    CAS:
    INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.
    Formula:C27H46O5
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:450.65

    Ref: TM-T11662L

  • Logo CymitQuimica
    Targetmol
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    5-HT7R antagonist 1

    5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.
    Formula:C14H18Cl2N4
    Colore e forma:Solid
    Peso molecolare:313.23

    Ref: TM-T60790

  • TGR5 Receptor Agonist 3
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    TGR5 Receptor Agonist 3

    CAS:
    TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) & 209 nM (mTGR5), ensures gallbladder safety and reduces filling.
    Formula:C29H27N3O6
    Colore e forma:Solid
    Peso molecolare:513.54

    Ref: TM-T63554

  • GPBAR1-IN-3
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    GPBAR1-IN-3

    CAS:
    GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].
    Formula:C21H23NO2
    Colore e forma:Solid
    Peso molecolare:321.41

    Ref: TM-T60863