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Recettore dell'adenosina

Recettore dell'adenosina

I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.

Trovati 242 prodotti di "Recettore dell'adenosina"

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  • MRS1220

    CAS:
    <p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>
    Formula:C21H14ClN5O2
    Purezza:98.43%
    Colore e forma:Solid
    Peso molecolare:403.82
  • N 0861

    CAS:
    <p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>
    Formula:C13H17N5
    Purezza:98.78%
    Colore e forma:Solid
    Peso molecolare:243.31
  • Selodenoson

    CAS:
    <p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>
    Formula:C17H24N6O4
    Purezza:99.52%
    Colore e forma:Solid
    Peso molecolare:376.41
  • ISAM-140

    CAS:
    <p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>
    Formula:C19H19N3O3
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:337.37
  • GW-493838

    CAS:
    <p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>
    Formula:C21H21ClFN7O4
    Purezza:99.11% - 99.58%
    Colore e forma:Solid
    Peso molecolare:489.89
  • GS-9667

    CAS:
    <p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>
    Formula:C21H24FN5O4S
    Purezza:99.76% - 99.77%
    Colore e forma:Solid
    Peso molecolare:461.51
  • A2A receptor antagonist 1

    CAS:
    <p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>
    Formula:C16H12FN5O
    Purezza:99.52% - 99.93%
    Colore e forma:Solid
    Peso molecolare:309.3
  • LAS38096

    CAS:
    <p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>
    Formula:C17H12N6O
    Purezza:99.18% - 99.95%
    Colore e forma:Solid
    Peso molecolare:316.32
  • N6-(2-Phenylethyl)adenosine

    CAS:
    <p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>
    Formula:C18H21N5O4
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:371.39
  • 2'-MeCCPA

    CAS:
    2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.
    Formula:C16H22ClN5O4
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:383.83
  • KI-7

    CAS:
    <p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>
    Formula:C23H18N2O2
    Purezza:98.33%
    Colore e forma:Solid
    Peso molecolare:354.4
  • FK-453

    CAS:
    <p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>
    Formula:C23H25N3O2
    Purezza:99.44%
    Colore e forma:Solid
    Peso molecolare:375.46
  • GP3269

    CAS:
    <p>GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.</p>
    Formula:C23H21FN4O3
    Colore e forma:Solid
    Peso molecolare:420.44
  • PSB-1115 potassium salt

    CAS:
    <p>PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].</p>
    Formula:C14H13KN4O5S
    Colore e forma:Solid
    Peso molecolare:388.44
  • MRS3558

    CAS:
    <p>MRS3558 is an agonist of A3 adenosine receptors.</p>
    Formula:C20H20Cl2N6O3
    Colore e forma:Solid
    Peso molecolare:463.32
  • ABT-702 hydrochloride

    CAS:
    <p>ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].</p>
    Formula:C22H20BrClN6O
    Colore e forma:Solid
    Peso molecolare:499.79
  • KFM19

    CAS:
    KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.
    Formula:C16H22N4O3
    Purezza:98.62%
    Colore e forma:Solid
    Peso molecolare:318.37
  • Neladenoson dalanate

    CAS:
    <p>Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.</p>
    Formula:C35H34ClN7O4S2
    Colore e forma:Solid
    Peso molecolare:716.27
  • Sulmazole

    CAS:
    <p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>
    Formula:C14H13N3O2S
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:287.34
  • Xanthine amine congener

    CAS:
    <p>Xanthine amine congener is an Adenosine receptor antagonist.</p>
    Formula:C21H28N6O4
    Purezza:99.7%
    Colore e forma:Solid
    Peso molecolare:428.48