Recettore dell'adenosina
I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.
Trovati 242 prodotti di "Recettore dell'adenosina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
L-97-1
CAS:<p>L-97-1 is an antagonist of the adenosine A1 receptor.</p>Formula:C29H38N6O3Purezza:98%Colore e forma:SolidPeso molecolare:518.65CVT-5440
CAS:<p>CVT-5440 is a selective, high-affinity (2B) adenosine receptor antagonist with good selectivity.</p>Formula:C27H28N6O5Colore e forma:SolidPeso molecolare:516.55A1AR antagonist 1
<p>Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).</p>Formula:C18H14N4OColore e forma:SolidPeso molecolare:302.33DMPX
CAS:<p>DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine-like compound capable of crossing the blood-brain barrier. It serves as an A2-selective adenosine receptor (AR) antagonist, effectively and selectively blocking the hypothermia and behavioral inhibition induced by A2 adenosine receptor agonists, such as NECA. DMPX is utilized in research on diseases like Parkinson's disease.</p>Formula:C10H10N4O2Colore e forma:SolidPeso molecolare:218.212A2A receptor antagonist 2
<p>A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).</p>Formula:C25H28FN7O3Colore e forma:SolidPeso molecolare:493.53ADORA2A/PDE4D-IN-1
CAS:<p>ADORA2A/PDE4D-IN-1 (Compound 9) is a dual inhibitor of the adenosine A2a receptor (ADORA2A) and phosphodiesterase 4D (PDE4D). This compound is applicable for research in bronchial asthma.</p>Formula:C14H11N5Colore e forma:SolidPeso molecolare:249.271PSB 36
CAS:<p>A1 adenosine receptor antagonist</p>Formula:C21H30N4O3Purezza:98%Colore e forma:SolidPeso molecolare:386.49LJ-4517
<p>LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.</p>Formula:C19H21N5O3SColore e forma:SolidPeso molecolare:399.47M1069
<p>M1069 is an oral A2A/A2B receptor antagonist, 100x more selective over A1/A3, with antitumor properties by blocking adenosine's immunosuppressive effects.</p>Formula:C25H30N4O8SColore e forma:SolidPeso molecolare:546.59UK-432097
CAS:<p>UK 432097 is an adenosine A2A agonist.</p>Formula:C40H47N11O6Colore e forma:SolidPeso molecolare:777.87YGZ-331
CAS:<p>YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine nucleoside NGBA. It functions through activating A1R and A2aR, and inhibiting the phosphorylation of CaMKII (pCaMKII), thereby exerting its calming effects. Additionally, YGZ-331 reduces spontaneous motor activity in mice.</p>Formula:C19H23N5O4Colore e forma:SolidPeso molecolare:385.42CP-608039
CAS:<p>CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.</p>Formula:C23H25ClN8O5Colore e forma:SolidPeso molecolare:528.95Neladenoson
CAS:<p>Neladenoson is an effective and selective agonist of the Adenosine A1 Receptor (A1R). EGFR-IN-162 shows potential for research in heart failure.</p>Formula:C29H24ClN5O2S2Colore e forma:SolidPeso molecolare:574.12MRS7799
CAS:<p>MRS7799 is a selective A3 Adenosine Receptor antagonist with Kd values of 0.55 nM for humans, 3.74 nM for mice, and 2.80 nM for rats. MRS7799 can be utilized in research related to neurodegenerative diseases, cancer, cardiac and cerebral ischemia, and autoimmune inflammatory diseases.</p>Formula:C22H18N4OSColore e forma:SolidPeso molecolare:386.47Tonapofylline
CAS:<p>Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.</p>Formula:C22H32N4O4Purezza:98.57%Colore e forma:SolidPeso molecolare:416.51A3AR antagonist 5
CAS:<p>A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.</p>Formula:C18H16N2O2SColore e forma:SolidPeso molecolare:324.40hA3AR agonist 1
<p>hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .</p>Formula:C10H14N6OSColore e forma:SolidPeso molecolare:266.32KF26777
CAS:<p>KF26777 is a potent and selective antagonist of adenosine A3 receptor.</p>Formula:C16H16BrN5OPurezza:98%Colore e forma:SolidPeso molecolare:374.23MSX-3
CAS:<p>MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.</p>Formula:C21H23N4Na2O7PPurezza:98%Colore e forma:SolidPeso molecolare:520.389Inupadenant HCl
CAS:<p>Inupadenant (EOS-850) is a selective A2a receptor antagonist, targeting immunosuppression in tumors.</p>Formula:C25H27ClF2N8O4S2Colore e forma:SolidPeso molecolare:641.11
