CymitQuimica logo
Recettore dell'adenosina

Recettore dell'adenosina

I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.

Trovati 242 prodotti di "Recettore dell'adenosina"

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Norisoboldine hydrochloride

    CAS:
    <p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>
    Formula:C18H20ClNO4
    Colore e forma:Solid
    Peso molecolare:349.81
  • FSCPX

    CAS:
    <p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>
    Formula:C23H27FN4O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:506.55
  • LUF7690

    CAS:
    <p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>
    Formula:C25H24FN5O6S
    Colore e forma:Solid
    Peso molecolare:541.55
  • Adenosine receptor antagonist 1

    CAS:
    <p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>
    Formula:C22H15ClFN7O
    Colore e forma:Solid
    Peso molecolare:447.86
  • N6-Benzyl-5'-ethylcarboxamido adenosine

    CAS:
    <p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>
    Formula:C19H22N6O4
    Colore e forma:Solid
    Peso molecolare:398.42
  • A3AR modulator 1


    <p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>
    Formula:C23H25IN4
    Colore e forma:Solid
    Peso molecolare:484.38
  • Adenosine receptor agonist 1


    <p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>
    Formula:C12H14ClN5O2Se
    Colore e forma:Solid
    Peso molecolare:374.68
  • PSB 0777 ammonium salt

    CAS:
    <p>adenosine A2A receptor full agonist</p>
    Formula:C18H24N6O7S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:500.55
  • Apadenoson TFA


    <p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>
    Formula:C25H31F3N6O8
    Purezza:98.08%
    Colore e forma:Soild
    Peso molecolare:600.55
  • Heterobivalent ligand-1


    <p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>
    Formula:C86H115FN16O21
    Colore e forma:Solid
    Peso molecolare:1727.93
  • GW-328267

    CAS:
    <p>GW-328267 is an agonist of the adenosine A2 receptor.</p>
    Formula:C21H26N10O4
    Colore e forma:Solid
    Peso molecolare:482.5
  • MRS-1706

    CAS:
    <p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>
    Formula:C27H29N5O5
    Purezza:99.00%
    Colore e forma:Solid
    Peso molecolare:503.55
  • Xanthine amine congener trihydrochloride

    CAS:
    <p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>
    Formula:C21H29ClN6O4
    Purezza:98.81%
    Colore e forma:Solid
    Peso molecolare:464.95
  • ABT-702

    CAS:
    <p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>
    Formula:C22H19BrN6O
    Purezza:99.57%
    Colore e forma:Soild
    Peso molecolare:463.33
  • Xanthine amine congener dihydrochloride

    CAS:
    <p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>
    Formula:C21H30Cl2N6O4
    Colore e forma:Solid
    Peso molecolare:501.41
  • A-286501

    CAS:
    <p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>
    Formula:C11H14BrN5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:328.17
  • Danshenol B


    <p>Danshenol B is a natural product that can be used as a reference standard.</p>
    Formula:C22H26O4
    Colore e forma:Solid
    Peso molecolare:354.446
  • AR ligand 40


    <p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>
    Formula:C21H25N5
    Colore e forma:Solid
    Peso molecolare:347.211
  • Theophyllol

    CAS:
    <p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>
    Formula:C9H10N4Na2O4
    Colore e forma:Solid
    Peso molecolare:284.18
  • LUF6096

    CAS:
    <p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>
    Formula:C22H21Cl2N3O
    Purezza:99.5%
    Colore e forma:Solid
    Peso molecolare:414.33