CymitQuimica logo
Recettore dell'adenosina

Recettore dell'adenosina

I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.

Trovati 242 prodotti di "Recettore dell'adenosina"

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • FSCPX

    CAS:
    <p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>
    Formula:C23H27FN4O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:506.55
  • N6-Benzyl-5'-ethylcarboxamido adenosine

    CAS:
    <p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>
    Formula:C19H22N6O4
    Colore e forma:Solid
    Peso molecolare:398.42
  • PSB 0777 ammonium hydrate


    <p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>
    Formula:C18H20N5O7S2·NH4·75H2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:532.09
  • AR ligand 40


    <p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>
    Formula:C21H25N5
    Colore e forma:Solid
    Peso molecolare:347.211
  • Apadenoson TFA


    <p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>
    Formula:C25H31F3N6O8
    Purezza:98.08%
    Colore e forma:Soild
    Peso molecolare:600.55
  • A2A/A3 AR antagonist-1


    <p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) &amp; 31.8 nM (hA3).</p>
    Formula:C56H71N15O12S2
    Colore e forma:Solid
    Peso molecolare:1210.39
  • MRS-3777 hemioxalate

    CAS:
    <p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>
    Formula:C17H19N5OC2H2O4
    Purezza:97.10%
    Colore e forma:Solid
    Peso molecolare:354.39
  • (Rac)-Mirabegron-d5

    CAS:
    <p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>
    Formula:C21H24N4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:401.54
  • GR79236

    CAS:
    <p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>
    Formula:C15H21N5O5
    Colore e forma:Solid
    Peso molecolare:351.36
  • LAS101057

    CAS:
    <p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>
    Formula:C18H14FN5O
    Purezza:99.03% - >99.99%
    Colore e forma:Solid
    Peso molecolare:335.34
  • Norisoboldine

    CAS:
    <p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>
    Formula:C18H19NO4
    Purezza:98.12% - 99.7%
    Colore e forma:Solid
    Peso molecolare:313.35
  • Taminadenant

    CAS:
    <p>Taminadenant is an adenosine receptor antagonist.</p>
    Formula:C10H8BrN7
    Purezza:99.11%
    Colore e forma:Solid
    Peso molecolare:306.12
  • 5'-N-Ethylcarboxamidoadenosine

    CAS:
    <p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>
    Formula:C12H16N6O4
    Purezza:98.95% - ≥95%
    Colore e forma:Powder
    Peso molecolare:308.29
  • Namodenoson

    CAS:
    <p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>
    Formula:C18H18ClIN6O4
    Purezza:98.97%
    Colore e forma:Solid
    Peso molecolare:544.73
  • N6,N6-Dimethyladenosine

    CAS:
    <p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>
    Formula:C12H17N5O4
    Purezza:98.79%
    Colore e forma:White Powder
    Peso molecolare:295.29
  • VPC171

    CAS:
    <p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>
    Formula:C18H12F3NOS
    Purezza:99.78%
    Colore e forma:Solid
    Peso molecolare:347.35
  • BAY-545

    CAS:
    <p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>
    Formula:C18H22F3N3O4S
    Purezza:98.05%
    Colore e forma:Solid
    Peso molecolare:433.45
  • Preladenant

    CAS:
    <p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has &gt;1000-fold selectivity over all other adenosine</p>
    Formula:C25H29N9O3
    Purezza:98.02% - 99.68%
    Colore e forma:Solid
    Peso molecolare:503.56
  • Swertisin

    CAS:
    <p>Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.</p>
    Formula:C22H22O10
    Purezza:99.74% - 99.89%
    Colore e forma:Solid
    Peso molecolare:446.4
  • 1-Ethyl-6-aminouracil

    CAS:
    <p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>
    Formula:C6H9N3O2
    Purezza:99.29%
    Colore e forma:Solid
    Peso molecolare:155.15