
Recettore dell'adenosina
I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.
Trovati 242 prodotti di "Recettore dell'adenosina"
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FSCPX
CAS:<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Formula:C23H27FN4O6SPurezza:98%Colore e forma:SolidPeso molecolare:506.55N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:<p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>Formula:C19H22N6O4Colore e forma:SolidPeso molecolare:398.42PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Formula:C18H20N5O7S2·NH4·75H2OPurezza:98%Colore e forma:SolidPeso molecolare:532.09AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Formula:C21H25N5Colore e forma:SolidPeso molecolare:347.211Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Formula:C25H31F3N6O8Purezza:98.08%Colore e forma:SoildPeso molecolare:600.55A2A/A3 AR antagonist-1
<p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).</p>Formula:C56H71N15O12S2Colore e forma:SolidPeso molecolare:1210.39MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formula:C17H19N5OC2H2O4Purezza:97.10%Colore e forma:SolidPeso molecolare:354.39(Rac)-Mirabegron-d5
CAS:<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Formula:C21H24N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:401.54GR79236
CAS:<p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>Formula:C15H21N5O5Colore e forma:SolidPeso molecolare:351.36LAS101057
CAS:<p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>Formula:C18H14FN5OPurezza:99.03% - >99.99%Colore e forma:SolidPeso molecolare:335.34Norisoboldine
CAS:<p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>Formula:C18H19NO4Purezza:98.12% - 99.7%Colore e forma:SolidPeso molecolare:313.35Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purezza:99.11%Colore e forma:SolidPeso molecolare:306.125'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formula:C12H16N6O4Purezza:98.95% - ≥95%Colore e forma:PowderPeso molecolare:308.29Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formula:C18H18ClIN6O4Purezza:98.97%Colore e forma:SolidPeso molecolare:544.73N6,N6-Dimethyladenosine
CAS:<p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>Formula:C12H17N5O4Purezza:98.79%Colore e forma:White PowderPeso molecolare:295.29VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Formula:C18H12F3NOSPurezza:99.78%Colore e forma:SolidPeso molecolare:347.35BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Formula:C18H22F3N3O4SPurezza:98.05%Colore e forma:SolidPeso molecolare:433.45Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formula:C25H29N9O3Purezza:98.02% - 99.68%Colore e forma:SolidPeso molecolare:503.56Swertisin
CAS:<p>Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.</p>Formula:C22H22O10Purezza:99.74% - 99.89%Colore e forma:SolidPeso molecolare:446.41-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Formula:C6H9N3O2Purezza:99.29%Colore e forma:SolidPeso molecolare:155.15

